TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 0.00700nMAssay Description:In vitro inhibition constant of human leukocyte elastase.More data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 0.00800nMAssay Description:Potency of inhibition against human leukocyte elastase (HLE) expressed as an apparent binding constantMore data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 0.00800nMAssay Description:In vitro inhibition constant of human leukocyte elastase.More data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 0.0100nMAssay Description:In vitro inhibition constant of human leukocyte elastase.More data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 0.0110nMAssay Description:Potency of inhibition against human leukocyte elastase (HLE) expressed as an apparent binding constantMore data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 0.0110nMAssay Description:Potency of inhibition against human leukocyte elastase (HLE) expressed as an apparent binding constantMore data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 0.0130nMAssay Description:Potency of inhibition against human leukocyte elastase (HLE) expressed as an apparent binding constantMore data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 0.0130nMAssay Description:Potency of inhibition against human leukocyte elastase (HLE) expressed as an apparent binding constantMore data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 0.0140nMAssay Description:Potency of inhibition against human leukocyte elastase (HLE) expressed as an apparent binding constantMore data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 0.0220nMAssay Description:Inhibition of Human Leukocyte Elastase (HLE) as apparent binding constant (kreact/kinact)More data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 0.0230nMAssay Description:Evaluated for inhibitory activity against Human leukocyte elastase (HLE)More data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 0.0300nMAssay Description:Evaluated for inhibitory activity against Human leukocyte elastase (HLE)More data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 0.0300nMAssay Description:In vitro inhibition constant of human leukocyte elastase.More data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 0.0300nMAssay Description:Evaluated for inhibitory activity against Human leukocyte elastase (HLE)More data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 0.0350nMAssay Description:In vitro inhibitory activity against Human leukocyte elastaseMore data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 0.0490nMAssay Description:Inhibition of Human Leukocyte Elastase (HLE) as apparent binding constant (kreact/kinact)More data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 0.0600nMAssay Description:In vitro inhibition constant of human leukocyte elastase.More data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 0.0700nMAssay Description:In vitro inhibitory activity against Human leukocyte elastaseMore data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 0.0700nMAssay Description:Inhibition of Human Leukocyte Elastase (HLE) as apparent binding constant (kreact/kinact)More data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 0.0800nMAssay Description:Inhibition of Human Leukocyte Elastase (HLE) as apparent binding constant (kreact/kinact)More data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 0.0800nMAssay Description:Inhibition of Human Leukocyte Elastase (HLE) as apparent binding constant (kreact/kinact)More data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 0.100nMAssay Description:In vitro inhibitory activity against Human leukocyte elastaseMore data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 0.110nMAssay Description:Inhibition of Human Leukocyte Elastase (HLE) as apparent binding constant (kreact/kinact)More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Walter Reed Army Institute Of Research
Curated by ChEMBL
Walter Reed Army Institute Of Research
Curated by ChEMBL
Affinity DataKi: 0.165nMAssay Description:Displacement of [3H] N-methylscopolamine from human muscarinic M2 receptor expressed in CHOK1 cells after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 0.170nMAssay Description:Inhibition of Human Leukocyte Elastase (HLE) as apparent binding constant (kreact/kinact)More data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 0.170nMAssay Description:In vitro inhibition constant of human leukocyte elastase.More data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 0.200nMAssay Description:Potency of inhibition against human leukocyte elastase (HLE) expressed as an apparent binding constantMore data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 0.200nMAssay Description:Evaluated for inhibitory activity against Human leukocyte elastase (HLE)More data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 0.240nMAssay Description:Inhibition of Human Leukocyte Elastase (HLE) as apparent binding constant (kreact/kinact)More data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 0.270nMAssay Description:Evaluated for inhibitory activity against Human leukocyte elastase (HLE)More data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 0.300nMAssay Description:Ratio of Koff to that of Kon was determined on human leukocyte elastase(HLE)More data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 0.340nMAssay Description:Inhibition of Human Leukocyte Elastase (HLE) as apparent binding constant (kreact/kinact)More data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 0.400nMAssay Description:Binding affinity for human leukocyte elastase (HLE); Kreact/KinactMore data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 0.470nMAssay Description:Inhibition of Human Leukocyte Elastase (HLE) as apparent binding constant (kreact/kinact)More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Walter Reed Army Institute Of Research
Curated by ChEMBL
Walter Reed Army Institute Of Research
Curated by ChEMBL
Affinity DataKi: 0.543nMAssay Description:Displacement of [3H] N-methylscopolamine from human muscarinic M3 receptor expressed in CHOK1 cells after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Walter Reed Army Institute Of Research
Curated by ChEMBL
Walter Reed Army Institute Of Research
Curated by ChEMBL
Affinity DataKi: 0.594nMAssay Description:Displacement of [3H] N-methylscopolamine from human muscarinic M1 receptor expressed in CHOK1 cells after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 0.600nMAssay Description:Ratio of Koff to that of Kon was determined on human leukocyte elastase(HLE)More data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 0.600nMAssay Description:Ratio of Koff to that of Kon was determined on human leukocyte elastase(HLE)More data for this Ligand-Target Pair
TargetProstaglandin E2 receptor EP3 subtype(Homo sapiens (Human))
Merck Frosst Centre For Therapeutic Research
Curated by ChEMBL
Merck Frosst Centre For Therapeutic Research
Curated by ChEMBL
Affinity DataKi: 0.600nMAssay Description:Binding affinity to EP3 receptorMore data for this Ligand-Target Pair
TargetProstaglandin E2 receptor EP3 subtype(Homo sapiens (Human))
Merck Frosst Centre For Therapeutic Research
Curated by ChEMBL
Merck Frosst Centre For Therapeutic Research
Curated by ChEMBL
Affinity DataKi: 0.600nMAssay Description:Binding affinity to EP3 receptorMore data for this Ligand-Target Pair
TargetProstaglandin E2 receptor EP3 subtype(Homo sapiens (Human))
Merck Frosst Centre For Therapeutic Research
Curated by ChEMBL
Merck Frosst Centre For Therapeutic Research
Curated by ChEMBL
Affinity DataKi: 0.700nMAssay Description:Binding affinity to EP3 receptor in presence of HSAMore data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 0.700nMAssay Description:Ratio of Koff to that of Kon was determined on human leukocyte elastase(HLE)More data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 0.800nMAssay Description:Binding affinity for human leukocyte elastase (HLE); Kreact/KinactMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Walter Reed Army Institute Of Research
Curated by ChEMBL
Walter Reed Army Institute Of Research
Curated by ChEMBL
Affinity DataKi: 0.881nMAssay Description:Displacement of [3H] N-methylscopolamine from human muscarinic M1 receptor expressed in CHOK1 cells after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetProstaglandin E2 receptor EP3 subtype(Homo sapiens (Human))
Merck Frosst Centre For Therapeutic Research
Curated by ChEMBL
Merck Frosst Centre For Therapeutic Research
Curated by ChEMBL
Affinity DataKi: 0.900nMAssay Description:Binding affinity to EP3 receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Walter Reed Army Institute Of Research
Curated by ChEMBL
Walter Reed Army Institute Of Research
Curated by ChEMBL
Affinity DataKi: 0.922nMAssay Description:Displacement of [3H] N-methylscopolamine from human muscarinic M1 receptor expressed in CHOK1 cells after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:In vitro inhibition constant of human leukocyte elastase.More data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 1.10nMAssay Description:Evaluated for inhibitory activity against Human leukocyte elastase (HLE)More data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Sterling Winthrop Pharmaceutical Research Division
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:Inhibition of Human Leukocyte Elastase (HLE) as apparent binding constant (kreact/kinact)More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Walter Reed Army Institute Of Research
Curated by ChEMBL
Walter Reed Army Institute Of Research
Curated by ChEMBL
Affinity DataKi: 1.29nMAssay Description:Displacement of [3H] N-methylscopolamine from human muscarinic M1 receptor expressed in CHOK1 cells after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair