Affinity DataKi: 0.920nM ΔG°: -47.9kJ/molepH: 7.5 T: 2°CAssay Description:Ki Values were determined by competition of [32P]-S1P binding to stably transfected CHO (S1P1,2,4) or RH7777 (S1P3,5) cells expressing the indicated ...More data for this Ligand-Target Pair
Affinity DataKi: 1.12nMAssay Description:Inhibitory activity against canine skin chymaseMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nM ΔG°: -47.3kJ/molepH: 7.5 T: 2°CAssay Description:Ki Values were determined by competition of [32P]-S1P binding to stably transfected CHO (S1P1,2,4) or RH7777 (S1P3,5) cells expressing the indicated ...More data for this Ligand-Target Pair
Affinity DataKi: 2.10nM ΔG°: -46.0kJ/molepH: 7.5 T: 2°CAssay Description:Ki Values were determined by competition of [32P]-S1P binding to stably transfected CHO (S1P1,2,4) or RH7777 (S1P3,5) cells expressing the indicated ...More data for this Ligand-Target Pair
Affinity DataKi: 2.20nM ΔG°: -45.9kJ/molepH: 7.5 T: 2°CAssay Description:Ki Values were determined by competition of [32P]-S1P binding to stably transfected CHO (S1P1,2,4) or RH7777 (S1P3,5) cells expressing the indicated ...More data for this Ligand-Target Pair
Affinity DataKi: 2.62nMAssay Description:In vitro inhibitory activity was determined against human heart chymaseMore data for this Ligand-Target Pair
Affinity DataKi: 2.70nM ΔG°: -45.5kJ/molepH: 7.5 T: 2°CAssay Description:Ki Values were determined by competition of [32P]-S1P binding to stably transfected CHO (S1P1,2,4) or RH7777 (S1P3,5) cells expressing the indicated ...More data for this Ligand-Target Pair
Affinity DataKi: 3.40nM ΔG°: -44.9kJ/molepH: 7.5 T: 2°CAssay Description:Ki Values were determined by competition of [32P]-S1P binding to stably transfected CHO (S1P1,2,4) or RH7777 (S1P3,5) cells expressing the indicated ...More data for this Ligand-Target Pair
Affinity DataKi: 3.56nMAssay Description:In vitro inhibitory activity was determined against human heart chymaseMore data for this Ligand-Target Pair
Affinity DataKi: 3.68nMAssay Description:Inhibitory activity against canine skin chymaseMore data for this Ligand-Target Pair
Affinity DataKi: 4.10nM ΔG°: -44.5kJ/molepH: 7.5 T: 2°CAssay Description:Ki Values were determined by competition of [32P]-S1P binding to stably transfected CHO (S1P1,2,4) or RH7777 (S1P3,5) cells expressing the indicated ...More data for this Ligand-Target Pair
Affinity DataKi: 4.20nM ΔG°: -44.4kJ/molepH: 7.5 T: 2°CAssay Description:Ki Values were determined by competition of [32P]-S1P binding to stably transfected CHO (S1P1,2,4) or RH7777 (S1P3,5) cells expressing the indicated ...More data for this Ligand-Target Pair
Affinity DataKi: 4.85nMAssay Description:Inhibitory activity evaluated against chymase from human heart.More data for this Ligand-Target Pair
Affinity DataKi: 5.40nM ΔG°: -43.9kJ/molepH: 7.5 T: 2°CAssay Description:Ki Values were determined by competition of [32P]-S1P binding to stably transfected CHO (S1P1,2,4) or RH7777 (S1P3,5) cells expressing the indicated ...More data for this Ligand-Target Pair
Affinity DataKi: 5.57nMAssay Description:Inhibitory activity evaluated against chymase from human heart.More data for this Ligand-Target Pair
Affinity DataKi: 5.60nMAssay Description:In vitro inhibitory activity was determined against human heart chymaseMore data for this Ligand-Target Pair
Affinity DataKi: 5.60nMAssay Description:Inhibitory activity evaluated against chymase from human heart.More data for this Ligand-Target Pair
Affinity DataKi: 5.90nM ΔG°: -43.7kJ/molepH: 7.5 T: 2°CAssay Description:Ki Values were determined by competition of [32P]-S1P binding to stably transfected CHO (S1P1,2,4) or RH7777 (S1P3,5) cells expressing the indicated ...More data for this Ligand-Target Pair
Affinity DataKi: 7.71nMAssay Description:In vitro inhibitory activity was determined against human heart chymaseMore data for this Ligand-Target Pair
Affinity DataKi: 9.32nMAssay Description:In vitro inhibitory activity was determined against human heart chymaseMore data for this Ligand-Target Pair
Affinity DataKi: 9.36nMAssay Description:inhibitory activity against alpha chymotrypsin from bovine pancreas.More data for this Ligand-Target Pair
Affinity DataKi: 9.36nMAssay Description:In vitro inhibitory activity was determined against bovine pancreas chymotrypsinMore data for this Ligand-Target Pair
Affinity DataKi: 9.70nMAssay Description:In vitro inhibitory activity was determined against human heart chymaseMore data for this Ligand-Target Pair
Affinity DataKi: 10.2nMAssay Description:In vitro inhibitory activity was determined against human heart chymaseMore data for this Ligand-Target Pair
Affinity DataKi: 10.2nMAssay Description:In vitro inhibitory activity was determined against human heart chymaseMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:In vitro inhibitory activity was determined against human heart chymaseMore data for this Ligand-Target Pair
Affinity DataKi: 12.6nMAssay Description:In vitro inhibitory activity was determined against bovine pancreas chymotrypsinMore data for this Ligand-Target Pair
Affinity DataKi: 13nM ΔG°: -41.8kJ/molepH: 7.5 T: 2°CAssay Description:Ki Values were determined by competition of [32P]-S1P binding to stably transfected CHO (S1P1,2,4) or RH7777 (S1P3,5) cells expressing the indicated ...More data for this Ligand-Target Pair
Affinity DataKi: 13.1nMAssay Description:inhibitory activity was evaluated against chymase from human heart.More data for this Ligand-Target Pair
Affinity DataKi: 13.1nMAssay Description:In vitro inhibitory activity was determined against human heart chymaseMore data for this Ligand-Target Pair
Affinity DataKi: 13.3nMAssay Description:In vitro inhibitory activity was determined against human heart chymaseMore data for this Ligand-Target Pair
Affinity DataKi: 13.8nMAssay Description:In vitro inhibitory activity was determined against human heart chymaseMore data for this Ligand-Target Pair
Affinity DataKi: 14.3nMAssay Description:Inhibitory activity evaluated against chymase from human heart.More data for this Ligand-Target Pair
Affinity DataKi: 15.7nMAssay Description:In vitro inhibitory activity was determined against human heart chymaseMore data for this Ligand-Target Pair
Affinity DataKi: 16.6nMAssay Description:In vitro inhibitory activity was determined against human heart chymaseMore data for this Ligand-Target Pair
Affinity DataKi: 16.9nMAssay Description:In vitro inhibitory activity was determined against human heart chymaseMore data for this Ligand-Target Pair
Affinity DataKi: 16.9nMAssay Description:In vitro inhibitory activity was determined against human heart chymaseMore data for this Ligand-Target Pair
Affinity DataKi: 18.5nMAssay Description:In vitro inhibitory activity was determined against human heart chymaseMore data for this Ligand-Target Pair
Affinity DataKi: 22.6nMAssay Description:Inhibitory activity evaluated against chymase from human heart.More data for this Ligand-Target Pair
Affinity DataKi: 23nM ΔG°: -40.5kJ/molepH: 7.5 T: 2°CAssay Description:Ki Values were determined by competition of [32P]-S1P binding to stably transfected CHO (S1P1,2,4) or RH7777 (S1P3,5) cells expressing the indicated ...More data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:In vitro inhibitory activity was determined against human heart chymaseMore data for this Ligand-Target Pair
Affinity DataKi: 23.3nMAssay Description:Inhibitory activity against alpha chymotrypsin from bovine pancreas.More data for this Ligand-Target Pair
Affinity DataKi: 26.1nMAssay Description:Inhibitory activity evaluated against chymase from human heart.More data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Inhibitory activity against canine skin chymaseMore data for this Ligand-Target Pair
Affinity DataKi: 28.9nMAssay Description:In vitro inhibitory activity was determined against human heart chymaseMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Inhibitory activity evaluated against chymase from human heart.More data for this Ligand-Target Pair
Affinity DataKi: 32.5nMAssay Description:In vitro inhibitory activity was determined against human heart chymaseMore data for this Ligand-Target Pair
Affinity DataKi: 32.6nMAssay Description:Inhibitory activity against alpha chymotrypsin from bovine pancreas.More data for this Ligand-Target Pair
Affinity DataKi: 33.7nMAssay Description:In vitro inhibitory activity was determined against human heart chymaseMore data for this Ligand-Target Pair
Affinity DataKi: 37nM ΔG°: -39.4kJ/molepH: 7.5 T: 2°CAssay Description:Ki Values were determined by competition of [32P]-S1P binding to stably transfected CHO (S1P1,2,4) or RH7777 (S1P3,5) cells expressing the indicated ...More data for this Ligand-Target Pair