Found 14 Enz. Inhib. hit(s) with Target = 'Dual specificity tyrosine-phosphorylation-regulated kinase 4'
TargetDual specificity tyrosine-phosphorylation-regulated kinase 4(Homo sapiens (Human))
University Of Canterbury
Curated by ChEMBL
University Of Canterbury
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of DYRK4 (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 4(Homo sapiens (Human))
University Of Canterbury
Curated by ChEMBL
University Of Canterbury
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of Dyrk4 (unknown origin) by quantitative PCRMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 4(Homo sapiens (Human))
University Of Canterbury
Curated by ChEMBL
University Of Canterbury
Curated by ChEMBL
Affinity DataIC50: 520nMAssay Description:Inhibition of human recombinant GST-tagged DYRK4 expressed in Escherichia coli using GRSRSRSRSRSR as substrate and [gamma33P]ATP after 30 mins by sci...More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 4(Homo sapiens (Human))
University Of Canterbury
Curated by ChEMBL
University Of Canterbury
Curated by ChEMBL
Affinity DataIC50: 1.57E+3nMAssay Description:Inhibition of DYRK4 (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 4(Homo sapiens (Human))
University Of Canterbury
Curated by ChEMBL
University Of Canterbury
Curated by ChEMBL
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of DYRK4 (unknown origin) by TR FRET assayMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 4(Homo sapiens (Human))
University Of Canterbury
Curated by ChEMBL
University Of Canterbury
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of DYRK4 (unknown origin) by TR FRET assayMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 4(Homo sapiens (Human))
University Of Canterbury
Curated by ChEMBL
University Of Canterbury
Curated by ChEMBL
Affinity DataIC50: 4.38E+3nMAssay Description:Inhibition of human DYRK4 using RRRFRPASPLRGPPK as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 4(Homo sapiens (Human))
University Of Canterbury
Curated by ChEMBL
University Of Canterbury
Curated by ChEMBL
Affinity DataIC50: 9.50E+3nMAssay Description:Inhibition of human recombinant GST-tagged DYRK4 expressed in Escherichia coli using GRSRSRSRSRSR as substrate and [gamma33P]ATP after 30 mins by sci...More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 4(Homo sapiens (Human))
University Of Canterbury
Curated by ChEMBL
University Of Canterbury
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant GST-tagged DYRK4 expressed in Escherichia coli using GRSRSRSRSRSR as substrate and [gamma33P]ATP after 30 mins by sci...More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 4(Homo sapiens (Human))
University Of Canterbury
Curated by ChEMBL
University Of Canterbury
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human DYRK4 using [RRRFRPASPLRGPPK] as substrateMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 4(Homo sapiens (Human))
University Of Canterbury
Curated by ChEMBL
University Of Canterbury
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of DYRK4 (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 4(Homo sapiens (Human))
University Of Canterbury
Curated by ChEMBL
University Of Canterbury
Curated by ChEMBL
Affinity DataIC50: 7.40E+4nMAssay Description:Inhibition of GST-tagged Dyrk4 (unknown origin) expressed in Escherichia coli using [33P]ATP[gammaP]/DYRKtide as substrate after 5 mins by liquid sci...More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 4(Homo sapiens (Human))
University Of Canterbury
Curated by ChEMBL
University Of Canterbury
Curated by ChEMBL
Affinity DataIC50: 8.00E+4nMAssay Description:Inhibition of full-length recombinant human GST-tagged DYRK4 expressed in baculovirus infected insect cells using DYRKtide as substrate after 5 mins ...More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 4(Homo sapiens (Human))
University Of Canterbury
Curated by ChEMBL
University Of Canterbury
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 using Z-Leu-Arg-AMC as substrate compound treated for 30 min before substrate addition by...More data for this Ligand-Target Pair