Compile Data Set for Download or QSAR
Report error Found 182 for UniProtKB: O95665
TargetNeurotensin receptor type 2(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50553771(CHEMBL4776986)
Affinity DataKi:  0.00300nMAssay Description:Displacement of [125I]-neurotensin from human recombinant NTS2 stably expressed in human 1321N1 cell membranes incubated for 60 mins by gamma counter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50553769(CHEMBL4798887)
Affinity DataKi:  0.0300nMAssay Description:Displacement of [125I]-neurotensin from human recombinant NTS2 stably expressed in human 1321N1 cell membranes incubated for 60 mins by gamma counter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50553767(CHEMBL4789659)
Affinity DataKi:  0.0900nMAssay Description:Displacement of [125I]-neurotensin from human recombinant NTS2 stably expressed in human 1321N1 cell membranes incubated for 60 mins by gamma counter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50553779(CHEMBL4742999)
Affinity DataKi:  0.110nMAssay Description:Displacement of [125I]-neurotensin from human recombinant NTS2 stably expressed in human 1321N1 cell membranes incubated for 60 mins by gamma counter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50553770(CHEMBL4758754)
Affinity DataKi:  0.160nMAssay Description:Displacement of [125I]-neurotensin from human recombinant NTS2 stably expressed in human 1321N1 cell membranes incubated for 60 mins by gamma counter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50133193(Neurotensin analogue | CHEMBL337721)
Affinity DataIC50: 0.230nMAssay Description:Evaluated for binding affinity by inhibiting binding of [125I]Tyr(3)-NT to human Neurotensin receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50124132(CHEMBL3622802)
Affinity DataIC50: 0.260nMAssay Description:Displacement of [125I]-Tyr3-NT from human NTS2 receptor expressed in 1321N1 cell membranes incubated for 30 mins by gamma-counting based competitive ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2016
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50553768(CHEMBL4744531)
Affinity DataKi:  0.290nMAssay Description:Displacement of [125I]-neurotensin from human recombinant NTS2 stably expressed in human 1321N1 cell membranes incubated for 60 mins by gamma counter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50133188(Compound KK17 | CHEMBL336836)
Affinity DataIC50: 0.300nMAssay Description:Evaluated for binding affinity by inhibiting binding of [125I]Tyr(3)-NT to human Neurotensin receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50553772(CHEMBL4749016)
Affinity DataKi:  0.320nMAssay Description:Displacement of [125I]-neurotensin from human recombinant NTS2 stably expressed in human 1321N1 cell membranes incubated for 60 mins by gamma counter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50553775(CHEMBL4745899)
Affinity DataKi:  0.330nMAssay Description:Displacement of [125I]-neurotensin from human recombinant NTS2 stably expressed in human 1321N1 cell membranes incubated for 60 mins by gamma counter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50553777(CHEMBL4597094)
Affinity DataKi:  0.460nMAssay Description:Displacement of [125I]-neurotensin from human recombinant NTS2 stably expressed in human 1321N1 cell membranes incubated for 60 mins by gamma counter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50342242((S)-2-((2S,3S)-2-((S)-2-((S)-1-((S)-6-amino-2-((S)...)
Affinity DataIC50: 0.470nMAssay Description:Inhibition of human NTR2More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetNeurotensin receptor type 2(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50553776(CHEMBL4747286)
Affinity DataKi:  0.5nMAssay Description:Displacement of [125I]-neurotensin from human recombinant NTS2 stably expressed in human 1321N1 cell membranes incubated for 60 mins by gamma counter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50048908(CHEMBL415788)
Affinity DataKi:  0.550nMAssay Description:Displacement of [125I]-neurotensin from human recombinant NTS2 stably expressed in human 1321N1 cell membranes incubated for 60 mins by gamma counter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50342238((S)-2-((2S,3S)-2-((S)-2-((S)-1-((S)-2-((S)-3-amino...)
Affinity DataKi:  0.610nMAssay Description:Displacement of [3H]NT from human NTS2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50133198(Compound KK16 | CHEMBL434227)
Affinity DataIC50: 0.670nMAssay Description:Evaluated for binding affinity by inhibiting binding of [125I]Tyr(3)-NT to human Neurotensin receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50133206(Compound KK1 | CHEMBL337644)
Affinity DataIC50: 0.700nMAssay Description:Evaluated for binding affinity by inhibiting binding of [125I]Tyr(3)-NT to human Neurotensin receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50159155(CHEMBL3786852)
Affinity DataKi:  0.740nMAssay Description:Displacement of [3H]NT(8 to 13 residues) from human NTSR2 expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2017
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50342241((S)-2-((2S,3S)-2-((S)-2-((S)-1-((S)-6-amino-2-(2-(...)
Affinity DataKi:  0.740nMAssay Description:Displacement of [3H]NT from human NTS2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50048908(CHEMBL415788)
Affinity DataKi:  0.741nMAssay Description:Displacement of [3H] UR-MK300 from human neurotensin receptor 2 in HEK293 cells homogenate incubated in dark after 30 mins by liquid scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50133201(Compound KK18 | CHEMBL132524)
Affinity DataIC50: 0.780nMAssay Description:Evaluated for binding affinity by inhibiting binding of [125I]Tyr(3)-NT to human Neurotensin receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50133204(Compound KK15 | CHEMBL132409)
Affinity DataIC50: 0.900nMAssay Description:Evaluated for binding affinity by inhibiting binding of [125I]Tyr(3)-NT to human Neurotensin receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50342242((S)-2-((2S,3S)-2-((S)-2-((S)-1-((S)-6-amino-2-((S)...)
Affinity DataIC50: 0.950nMAssay Description:Displacement of 125I-[Tyr3]-NT from human NTS2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2020
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50509508(CHEMBL4534768)
Affinity DataKi:  0.955nMAssay Description:Displacement of [3H] UR-MK300 from human neurotensin receptor 2 in HEK293 cells homogenate incubated in dark after 30 mins by liquid scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50563034(CHEMBL4742223)
Affinity DataKi: >1nMAssay Description:Binding affinity to NTS2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50130880(pGlu-Leu-Tyr-Glu-Asn-Lys-Pro-Arg-Arg-Pro-Tyr-Ile-L...)
Affinity DataIC50: 1.10nMAssay Description:Inhibition of human NTR2More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetNeurotensin receptor type 2(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50509510(CHEMBL4564746)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H] UR-MK300 from human neurotensin receptor 2 in HEK293 cells homogenate incubated in dark after 30 mins by liquid scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50048908(CHEMBL415788)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]NT(8 to 13 residues) from human NTSR2 expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2017
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50048908(CHEMBL415788)
Affinity DataKi:  1.20nMAssay Description:Displacement of [leucine-3H]NT (8 to 13 residues) from human NTS2 receptor expressed in HEK293 cell membranes after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2018
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50342239((S)-2-((2S,3S)-2-((S)-2-((S)-1-((S)-2-((S)-2-amino...)
Affinity DataKd:  1.20nMAssay Description:Displacement of [3H]NT from human NTS2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50048908(CHEMBL415788)
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]NT(8-13) from human NTSR2 expressed in HEK293 cell membranes by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetNeurotensin receptor type 2(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50553773(CHEMBL4742666)
Affinity DataKi:  1.70nMAssay Description:Displacement of [125I]-neurotensin from human recombinant NTS2 stably expressed in human 1321N1 cell membranes incubated for 60 mins by gamma counter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50048908(CHEMBL415788)
Affinity DataKd:  1.80nMAssay Description:Binding affinity to human NTSR2 transfected in HEK293 cells assessed as inhibition constant incubated for 60 mins in the presence of [Leu3H]NT(8-13) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetNeurotensin receptor type 2(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50133196(Compound KK6 | CHEMBL337260)
Affinity DataIC50: 1.80nMAssay Description:Evaluated for binding affinity by inhibiting binding of [125I]Tyr(3)-NT to human Neurotensin receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50133190(Compound KK5 | CHEMBL430910)
Affinity DataIC50: 2.10nMAssay Description:Evaluated for binding affinity by inhibiting binding of [125I]Tyr(3)-NT to human Neurotensin receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50159156(CHEMBL3786291)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]NT(8 to 13 residues) from human NTSR2 expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2017
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50240845(2-{(S)-2-[2-({(S)-1-[(S)-2-((S)-2-Amino-5-guanidin...)
Affinity DataIC50: 2.70nMAssay Description:Evaluated for binding affinity by inhibiting binding of [125I]Tyr(3)-NT to human Neurotensin receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50562998(CHEMBL4786574)
Affinity DataKi:  2.70nMAssay Description:Displacement of [125I]Tyr3-neurotensin from human recombinant NTS2 stably expressed in human 1321N1 cell membranes incubated for 60 mins by gamma cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50133191(Compound KK7 | CHEMBL132507)
Affinity DataIC50: 2.80nMAssay Description:Evaluated for binding affinity by inhibiting binding of [125I]Tyr(3)-NT to human Neurotensin receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50553778(CHEMBL4740539)
Affinity DataKi:  2.90nMAssay Description:Displacement of [125I]-neurotensin from human recombinant NTS2 stably expressed in human 1321N1 cell membranes incubated for 60 mins by gamma counter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50553780(CHEMBL4762684)
Affinity DataKi:  3nMAssay Description:Displacement of [125I]-neurotensin from human recombinant NTS2 stably expressed in human 1321N1 cell membranes incubated for 60 mins by gamma counter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50133199(Compound KK9 | CHEMBL339139)
Affinity DataIC50: 3nMAssay Description:Evaluated for binding affinity by inhibiting binding of [125I]Tyr(3)-NT to human Neurotensin receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50133202(Compound KK4 | CHEMBL132794)
Affinity DataIC50: 3.10nMAssay Description:Evaluated for binding affinity by inhibiting binding of [125I]Tyr(3)-NT to human Neurotensin receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50133205(Compound KK8 | CHEMBL133798)
Affinity DataIC50: 3.20nMAssay Description:Evaluated for binding affinity by inhibiting binding of [125I]Tyr(3)-NT to human Neurotensin receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50133195(Compound KK10 | CHEMBL133340)
Affinity DataIC50: 3.5nMAssay Description:Evaluated for binding affinity by inhibiting binding of [125I]Tyr(3)-NT to human Neurotensin receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50133187(Compound KK3 | CHEMBL133850)
Affinity DataIC50: 3.5nMAssay Description:Evaluated for binding affinity by inhibiting binding of [125I]Tyr(3)-NT to human Neurotensin receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50509513(CHEMBL4537266)
Affinity DataKi:  3.5nMAssay Description:Displacement of [3H] UR-MK300 from human neurotensin receptor 2 in HEK293 cells homogenate incubated in dark after 30 mins by liquid scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50133192(Compound NT | CHEMBL439494)
Affinity DataIC50: 4nMAssay Description:Evaluated for binding affinity by inhibiting binding of [125I]Tyr(3)-NT to human Neurotensin receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50509511(CHEMBL4457798)
Affinity DataKi:  4nMAssay Description:Displacement of [3H] UR-MK300 from human neurotensin receptor 2 in HEK293 cells homogenate incubated in dark after 30 mins by liquid scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
Displayed 1 to 50 (of 182 total ) | Next | Last >>
Jump to: