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Found 14 Enz. Inhib. hit(s) with all data for entry = 10585
TargetEpidermal growth factor receptor [669-770,'SVD',771-1210](Homo sapiens (Human))
Bayer Aktiengesellschaft

WIPO
LigandPNGBDBM552588(N-[2-({4-[3-(3-chloro-2-methoxyanilino)-4-oxo-4,5,...)
Affinity DataIC50:  0.160nMAssay Description: Inhibitory activity of compounds of the present invention against an Epidermal Growth Factor Receptor (EGFR) with an insertion of the amino acids se...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetEpidermal growth factor receptor [669-770,'SVD',771-1210](Homo sapiens (Human))
Bayer Aktiengesellschaft

WIPO
LigandPNGBDBM552593(N-[2-({4-[3-(3-fluoro-2-methoxyanilino)-4-oxo-4,5,...)
Affinity DataIC50:  0.170nMAssay Description: Inhibitory activity of compounds of the present invention against an Epidermal Growth Factor Receptor (EGFR) with an insertion of the amino acids se...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetEpidermal growth factor receptor [669-770,'SVD',771-1210](Homo sapiens (Human))
Bayer Aktiengesellschaft

WIPO
LigandPNGBDBM552600(3-(3-chloro-2-methoxyanilino)-2-(3-{[(2S)-1-(prop-...)
Affinity DataIC50:  0.210nMAssay Description: Inhibitory activity of compounds of the present invention against an Epidermal Growth Factor Receptor (EGFR) with an insertion of the amino acids se...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetEpidermal growth factor receptor [669-770,'SVD',771-1210](Homo sapiens (Human))
Bayer Aktiengesellschaft

WIPO
LigandPNGBDBM552592(N-[2-({4-[3-(3-chloro-2-methoxyanilino)-4-oxo-4,5,...)
Affinity DataIC50:  0.230nMAssay Description: Inhibitory activity of compounds of the present invention against an Epidermal Growth Factor Receptor (EGFR) with an insertion of the amino acids se...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetEpidermal growth factor receptor [669-770,'SVD',771-1210](Homo sapiens (Human))
Bayer Aktiengesellschaft

WIPO
LigandPNGBDBM552590(N-[2-({4-[3-(3-chloro-2-methylanilino)-4-oxo-4,5,6...)
Affinity DataIC50:  0.270nMAssay Description: Inhibitory activity of compounds of the present invention against an Epidermal Growth Factor Receptor (EGFR) with an insertion of the amino acids se...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetEpidermal growth factor receptor [669-770,'SVD',771-1210](Homo sapiens (Human))
Bayer Aktiengesellschaft

WIPO
LigandPNGBDBM552591(N-[3-({4-[3-(3-chloro-2-methoxyanilino)-4-oxo-4,5,...)
Affinity DataIC50:  0.310nMAssay Description: Inhibitory activity of compounds of the present invention against an Epidermal Growth Factor Receptor (EGFR) with an insertion of the amino acids se...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetEpidermal growth factor receptor [669-770,'SVD',771-1210](Homo sapiens (Human))
Bayer Aktiengesellschaft

WIPO
LigandPNGBDBM552589(N-[2-({4-[3-(3-fluoro-2-methylanilino)-4-oxo-4,5,6...)
Affinity DataIC50:  0.390nMAssay Description: Inhibitory activity of compounds of the present invention against an Epidermal Growth Factor Receptor (EGFR) with an insertion of the amino acids se...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetEpidermal growth factor receptor [669-770,'SVD',771-1210](Homo sapiens (Human))
Bayer Aktiengesellschaft

WIPO
LigandPNGBDBM552598(N-[2-({4-[3'-(3-chloro-2-methoxyanilino)-4'-oxo-1'...)
Affinity DataIC50:  0.460nMAssay Description: Inhibitory activity of compounds of the present invention against an Epidermal Growth Factor Receptor (EGFR) with an insertion of the amino acids se...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetEpidermal growth factor receptor [669-770,'SVD',771-1210](Homo sapiens (Human))
Bayer Aktiengesellschaft

WIPO
LigandPNGBDBM552595((2E)-4-(dimethylamino)-N-[2-({4-[3-(3-fluoro-2-met...)
Affinity DataIC50:  0.550nMAssay Description: Inhibitory activity of compounds of the present invention against an Epidermal Growth Factor Receptor (EGFR) with an insertion of the amino acids se...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetEpidermal growth factor receptor [669-770,'SVD',771-1210](Homo sapiens (Human))
Bayer Aktiengesellschaft

WIPO
LigandPNGBDBM552601(N-(2-{[4-(3-{[2-(difluoromethoxy)phenyl]amino}-4-o...)
Affinity DataIC50:  0.570nMAssay Description: Inhibitory activity of compounds of the present invention against an Epidermal Growth Factor Receptor (EGFR) with an insertion of the amino acids se...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetEpidermal growth factor receptor [669-770,'SVD',771-1210](Homo sapiens (Human))
Bayer Aktiengesellschaft

WIPO
LigandPNGBDBM552599(N-[2-({4-[3-(3-chloro-2-methoxyanilino)-6,6-dimeth...)
Affinity DataIC50:  0.580nMAssay Description: Inhibitory activity of compounds of the present invention against an Epidermal Growth Factor Receptor (EGFR) with an insertion of the amino acids se...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetEpidermal growth factor receptor [669-770,'SVD',771-1210](Homo sapiens (Human))
Bayer Aktiengesellschaft

WIPO
LigandPNGBDBM552594(N-[2-({4-[3-(4-fluoroanilino)-4-oxo-4,5,6,7-tetrah...)
Affinity DataIC50:  1.62nMAssay Description: Inhibitory activity of compounds of the present invention against an Epidermal Growth Factor Receptor (EGFR) with an insertion of the amino acids se...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetEpidermal growth factor receptor [669-770,'SVD',771-1210](Homo sapiens (Human))
Bayer Aktiengesellschaft

WIPO
LigandPNGBDBM552596((2E)-N-[2-({4-[3-(3-chloro-2-methoxyanilino)-4-oxo...)
Affinity DataIC50:  2.48nMAssay Description: Inhibitory activity of compounds of the present invention against an Epidermal Growth Factor Receptor (EGFR) with an insertion of the amino acids se...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetEpidermal growth factor receptor [669-770,'SVD',771-1210](Homo sapiens (Human))
Bayer Aktiengesellschaft

WIPO
LigandPNGBDBM552597((2E)-N-[2-({4-[3'-(3-chloro-2-methoxyanilino)-4'-o...)
Affinity DataIC50:  3.55nMAssay Description: Inhibitory activity of compounds of the present invention against an Epidermal Growth Factor Receptor (EGFR) with an insertion of the amino acids se...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed