BDBM26474 5-({4-[(2,3-dimethyl-2H-indazol-6-yl)(methyl)amino]pyrimidin-2-yl}amino)-2-methylbenzene-1-sulfonamide::GW-786034::JMC514632 Compound 13::Pazopanib::cid_10113978
SMILES CN(c1ccc2c(C)n(C)nc2c1)c1ccnc(Nc2ccc(C)c(c2)S(N)(=O)=O)n1
InChI Key InChIKey=CUIHSIWYWATEQL-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 26474
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Daegu-Gyeongbuk Medical Innovation Foundation (Dgmif)
Curated by ChEMBL
Daegu-Gyeongbuk Medical Innovation Foundation (Dgmif)
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of GST-tagged human VEGFR2 C-terminal domain using (biotin-aminohexyl-EEEEYFELVAKKKK-NH2 substrate incubated for 60 mins by HTRF assayMore data for this Ligand-Target Pair