BDBM31592 PF-2545920::US9138494, MP-10::substituted pyrazole, 9

SMILES Cn1cc(c(n1)-c1ccc(OCc2ccc3ccccc3n2)cc1)-c1ccncc1

InChI Key InChIKey=AZEXWHKOMMASPA-UHFFFAOYSA-N

Data  1 KI  15 IC50  3 Kd

PDB links: 2 PDB IDs match this monomer.

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 31592   

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM31592(PF-2545920 | US9138494, MP-10 | substituted pyraz...)
Affinity DataIC50:  2.60nMAssay Description:Inhibition of PDE10A (unknown origin)More data for this Ligand-Target Pair