BDBM50307254 CHEMBL604990::GWTLNSAGYLLGPPPALALA-CONH2::M40

SMILES CC(C)C[C@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CN)[C@@H](C)O)C(=O)NCC(=O)N1CCC[C@H]1C(=O)N1CCC[C@H]1C(=O)N1CCC[C@H]1C(=O)N[C@@H](C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(N)=O

InChI Key InChIKey=OSGCBUDLRBUEGW-UHFFFAOYSA-N

Data  18 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 18 hits for monomerid = 50307254   

TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50307254(M40 | CHEMBL604990 | GWTLNSAGYLLGPPPALALA-CONH2)
Affinity DataKi:  0.100nMAssay Description:Binding affinity to human GalR1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGalanin receptor type 2(Rat)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50307254(M40 | CHEMBL604990 | GWTLNSAGYLLGPPPALALA-CONH2)
Affinity DataKi:  0.700nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGalanin receptor type 1(Rat)
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50307254(M40 | CHEMBL604990 | GWTLNSAGYLLGPPPALALA-CONH2)
Affinity DataKi:  0.900nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGalanin receptor type 2(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50307254(M40 | CHEMBL604990 | GWTLNSAGYLLGPPPALALA-CONH2)
Affinity DataKi:  1.5nMAssay Description:Displacement of Eu-labeled galanin from human GalR2 by DELFIA competitive assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGalanin receptor type 2(Rat)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50307254(M40 | CHEMBL604990 | GWTLNSAGYLLGPPPALALA-CONH2)
Affinity DataKi:  1.90nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50307254(M40 | CHEMBL604990 | GWTLNSAGYLLGPPPALALA-CONH2)
Affinity DataKi:  2.40nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGalanin receptor type 2(Rat)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50307254(M40 | CHEMBL604990 | GWTLNSAGYLLGPPPALALA-CONH2)
Affinity DataKi:  2.88nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGalanin receptor type 2(Rat)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50307254(M40 | CHEMBL604990 | GWTLNSAGYLLGPPPALALA-CONH2)
Affinity DataKi:  3.55nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGalanin receptor type 1(Rat)
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50307254(M40 | CHEMBL604990 | GWTLNSAGYLLGPPPALALA-CONH2)
In DepthDetails Article
PubMed
TargetGalanin receptor type 2(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50307254(M40 | CHEMBL604990 | GWTLNSAGYLLGPPPALALA-CONH2)
Affinity DataKi:  4.07nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGalanin receptor type 1(Rat)
Merck Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50307254(M40 | CHEMBL604990 | GWTLNSAGYLLGPPPALALA-CONH2)
Affinity DataKi:  6.76nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGalanin receptor type 2(Rat)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50307254(M40 | CHEMBL604990 | GWTLNSAGYLLGPPPALALA-CONH2)
Affinity DataKi:  18nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGalanin receptor type 3(Rat)
Schering-Plough Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM50307254(M40 | CHEMBL604990 | GWTLNSAGYLLGPPPALALA-CONH2)
Affinity DataKi:  54nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGalanin receptor type 3(Rat)
Schering-Plough Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM50307254(M40 | CHEMBL604990 | GWTLNSAGYLLGPPPALALA-CONH2)
Affinity DataKi:  79.4nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50307254(M40 | CHEMBL604990 | GWTLNSAGYLLGPPPALALA-CONH2)
Affinity DataKi:  109nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetGalanin receptor type 3(Human)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50307254(M40 | CHEMBL604990 | GWTLNSAGYLLGPPPALALA-CONH2)
Affinity DataKi:  288nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGalanin receptor type 3(Human)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50307254(M40 | CHEMBL604990 | GWTLNSAGYLLGPPPALALA-CONH2)
Affinity DataKi:  288nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50307254(M40 | CHEMBL604990 | GWTLNSAGYLLGPPPALALA-CONH2)
Affinity DataKi:  713nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed