Report error Found 1468 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A2a/A2b'
Affinity DataKi: 1.20E+7nMAssay Description:Binding affinity against adenosine A2 receptor in rat striatum by using [3H]NECA as a radioligandMore data for this Ligand-Target Pair
Affinity DataKi: >3.00E+5nMAssay Description:Antagonism of N-ethylcarboxamido adenosine-stimulated adenylate cyclase associated with stimulation of Adenosine A2 receptor of rat PC12 membranesMore data for this Ligand-Target Pair
Affinity DataKi: >3.00E+5nMAssay Description:Antagonism of N-ethylcarboxamido adenosine-stimulated adenylate cyclase associated with stimulation of Adenosine A2 receptor of rat PC12 membranesMore data for this Ligand-Target Pair
Affinity DataKi: >3.00E+5nMAssay Description:Antagonism of N-ethylcarboxamido adenosine-stimulated adenylate cyclase associated with stimulation of Adenosine A2 receptor of rat PC12 membranesMore data for this Ligand-Target Pair
Affinity DataKi: >3.00E+5nMAssay Description:Antagonism of N-ethylcarboxamido adenosine-stimulated adenylate cyclase associated with stimulation of Adenosine A2 receptor of rat PC12 membranesMore data for this Ligand-Target Pair
Affinity DataKi: >3.00E+5nMAssay Description:Antagonism of N-ethylcarboxamido adenosine-stimulated adenylate cyclase associated with stimulation of Adenosine A2 receptor of rat PC12 membranesMore data for this Ligand-Target Pair
Affinity DataKi: >3.00E+5nMAssay Description:Antagonism of N-ethylcarboxamido adenosine-stimulated adenylate cyclase associated with stimulation of Adenosine A2 receptor of rat PC12 membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2.63E+5nMAssay Description:Binding affinity against Adenosine A2 receptor from rat striatal membrane using [3H]NECA as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 2.60E+5nMAssay Description:Antagonism of N-ethylcarboxamido adenosine-stimulated adenylate cyclase associated with stimulation of Adenosine A2 receptor of rat PC12 membranesMore data for this Ligand-Target Pair
Affinity DataKi: >2.50E+5nMAssay Description:Binding affinity for Adenosine A2 receptor from rat striatum using [3H]NECA as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: >2.50E+5nMAssay Description:Binding affinity for Adenosine A2 receptor from rat striatum using [3H]NECA as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 2.50E+5nMAssay Description:Antagonism of N-ethylcarboxamido adenosine-stimulated adenylate cyclase associated with stimulation of Adenosine A2 receptor of rat PC12 membranesMore data for this Ligand-Target Pair
Affinity DataKi: >2.50E+5nMAssay Description:Binding affinity for Adenosine A2 receptor from rat striatum using [3H]NECA as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: >2.50E+5nMAssay Description:Binding affinity for Adenosine A2 receptor from rat striatum using [3H]NECA as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: >2.50E+5nMAssay Description:Binding affinity for Adenosine A2 receptor from rat striatum using [3H]NECA as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: >2.50E+5nMAssay Description:Binding affinity against Adenosine A2 receptor from rat striatal membrane using [3H]NECA as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: >2.50E+5nMAssay Description:Binding affinity against Adenosine A2 receptor from rat striatal membrane using [3H]NECA as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: >2.50E+5nMAssay Description:Binding affinity against Adenosine A2 receptor from rat striatal membrane using [3H]NECA as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: >2.50E+5nMAssay Description:Binding affinity against Adenosine A2 receptor from rat striatal membrane using [3H]NECA as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: >2.50E+5nMAssay Description:Binding affinity against Adenosine A2 receptor from rat striatal membrane using [3H]NECA as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 2.40E+5nMAssay Description:Inhibition of the stimulation by 5'-(N-ethylcarbamoyl) adenosine of adenyl cyclase via adenosine A2 receptor in human platelet membranes.More data for this Ligand-Target Pair
Affinity DataKi: 2.08E+5nMAssay Description:Binding affinity against Adenosine A2 receptor from rat striatal membrane using [3H]NECA as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 2.03E+5nMAssay Description:Binding affinity against Adenosine A2 receptor from rat striatal membrane using [3H]NECA as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: >2.00E+5nMAssay Description:Binding affinity against adenosine A2 receptor of striatal membrane using [3H]CGS-21680 as a radioligandMore data for this Ligand-Target Pair
Affinity DataKi: >2.00E+5nMAssay Description:Binding affinity against adenosine A2 receptor of striatal membrane using [3H]CGS-21680 as a radioligandMore data for this Ligand-Target Pair
Affinity DataKi: >2.00E+5nMAssay Description:Binding affinity against adenosine A2 receptor of striatal membrane using [3H]CGS-21680 as a radioligandMore data for this Ligand-Target Pair
Affinity DataKi: >2.00E+5nMAssay Description:Binding affinity against adenosine A2 receptor of striatal membrane using [3H]CGS-21680 as a radioligandMore data for this Ligand-Target Pair
Affinity DataKi: >2.00E+5nMAssay Description:Binding affinity against adenosine A2 receptor of striatal membrane using [3H]CGS-21680 as a radioligandMore data for this Ligand-Target Pair
Affinity DataKi: >2.00E+5nMAssay Description:Binding affinity against adenosine A2 receptor of striatal membrane using [3H]CGS-21680 as a radioligandMore data for this Ligand-Target Pair
Affinity DataKi: >2.00E+5nMAssay Description:Binding affinity against adenosine A2 receptor of striatal membrane using [3H]CGS-21680 as a radioligandMore data for this Ligand-Target Pair
Affinity DataKi: >2.00E+5nMAssay Description:Binding affinity against adenosine A2 receptor of striatal membrane using [3H]CGS-21680 as a radioligandMore data for this Ligand-Target Pair
Affinity DataKi: >2.00E+5nMAssay Description:Binding affinity against adenosine A2 receptor of striatal membrane using [3H]CGS-21680 as a radioligandMore data for this Ligand-Target Pair
Affinity DataKi: >2.00E+5nMAssay Description:Binding affinity against adenosine A2 receptor of striatal membrane using [3H]CGS-21680 as a radioligandMore data for this Ligand-Target Pair
Affinity DataKi: >2.00E+5nMAssay Description:Binding affinity against adenosine A2 receptor of striatal membrane using [3H]CGS-21680 as a radioligandMore data for this Ligand-Target Pair
Affinity DataKi: >2.00E+5nMAssay Description:Binding affinity against adenosine A2 receptor of striatal membrane using [3H]CGS-21680 as a radioligandMore data for this Ligand-Target Pair
Affinity DataKi: >2.00E+5nMAssay Description:Binding affinity against adenosine A2 receptor of striatal membrane using [3H]CGS-21680 as a radioligandMore data for this Ligand-Target Pair
Affinity DataKi: >2.00E+5nMAssay Description:Binding affinity against adenosine A2 receptor of striatal membrane using [3H]CGS-21680 as a radioligandMore data for this Ligand-Target Pair
Affinity DataKi: >2.00E+5nMAssay Description:Binding affinity against adenosine A2 receptor of striatal membrane using [3H]CGS-21680 as a radioligandMore data for this Ligand-Target Pair
Affinity DataKi: >2.00E+5nMAssay Description:Binding affinity against adenosine A2 receptor of striatal membrane using [3H]CGS-21680 as a radioligandMore data for this Ligand-Target Pair
Affinity DataKi: >2.00E+5nMAssay Description:Binding affinity against adenosine A2 receptor of striatal membrane using [3H]CGS-21680 as a radioligandMore data for this Ligand-Target Pair
Affinity DataKi: >2.00E+5nMAssay Description:Binding affinity against adenosine A2 receptor of striatal membrane using [3H]CGS-21680 as a radioligandMore data for this Ligand-Target Pair
Affinity DataKi: >2.00E+5nMAssay Description:Binding affinity against adenosine A2 receptor of striatal membrane using [3H]CGS-21680 as a radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.76E+5nMAssay Description:Binding affinity against Adenosine A2 receptor from rat striatal membrane using [3H]NECA as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.70E+5nMAssay Description:Antagonism of N-ethylcarboxamido adenosine-stimulated adenylate cyclase associated with stimulation of Adenosine A2 receptor of rat PC12 membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.70E+5nMAssay Description:In vitro binding affinity to Adenosine A2 receptor of human platelets by inhibition of NECA-stimulated adenylate cyclaseMore data for this Ligand-Target Pair
Affinity DataKi: 1.63E+5nMAssay Description:Antagonism of N-ethylcarboxamido adenosine-stimulated adenylate cyclase associated with stimulation of Adenosine A2 receptor of rat PC12 membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.62E+5nMAssay Description:Binding affinity against adenosine A2 receptor of striatal membrane using [3H]CGS-21680 as a radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.57E+5nMAssay Description:Binding affinity against Adenosine A2 receptor from rat striatal membrane using [3H]NECA as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.55E+5nMAssay Description:Binding affinity against Adenosine A2 receptor from rat striatal membrane using [3H]NECA as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.51E+5nMAssay Description:Binding affinity for Adenosine A2 receptor from rat striatum using [3H]NECA as radioligandMore data for this Ligand-Target Pair












































