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Report error Found 2409 Enz. Inhib. hit(s) with Target = 'Alpha-1B adrenergic receptor'
TargetAlpha-1B adrenergic receptor(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50265530(CHEMBL4067502)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at recombinant human alpha1B adrenergic receptor expressed in HEK293 cells after 6 hrs by NFAT-luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50118703(N-[5-(4,5-Dihydro-1H-imidazol-2-yl)-2-hydroxy-5,6,...)
Affinity DataEC50:  316nMAssay Description:In vitro agonist potency towards Alpha-1B adrenergic receptor in rat spleenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50470944(CHEMBL336161)
Affinity DataEC50:  186nMAssay Description:In vitro agonist potency towards Alpha-1B adrenergic receptor in rat spleenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM30712(SMR000059324 | Oxymetazoline | cid_66259 | 6-tert-...)
Affinity DataEC50:  339nMAssay Description:In vitro agonist potency towards Alpha-1B adrenergic receptor in rat spleenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50470943(CHEMBL133451)
Affinity DataEC50: <1.00E+5nMAssay Description:In vitro agonist potency towards Alpha-1B adrenergic receptor in rat spleenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50029051(4-[(1R)-2-amino-1-hydroxyethyl]benzene-1,2-diol | ...)
Affinity DataEC50:  1.02E+4nMAssay Description:In vitro agonist potency towards Alpha-1B adrenergic receptor in rat spleenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50067212(CHEBI:8093 | Cyclomydril | Duo-Medihaler | Phenyle...)
Affinity DataEC50:  1.10E+4nMAssay Description:In vitro agonist potency towards Alpha-1B adrenergic receptor in rat spleenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50473669(CHEMBL70692)
Affinity DataEC50:  85nMAssay Description:Agonist potency at Alpha-1B adrenergic receptor expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50473672(CHEMBL72768)
Affinity DataEC50:  1.90nMAssay Description:Agonist potency at Alpha-1B adrenergic receptor expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50473668(CHEMBL70973)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonist potency at Alpha-1B adrenergic receptor expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM30712(SMR000059324 | Oxymetazoline | cid_66259 | 6-tert-...)
Affinity DataEC50: <2.51E+4nMAssay Description:Agonist potency at Alpha-1B adrenergic receptor expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50473677(CHEMBL72441)
Affinity DataEC50:  0.417nMAssay Description:Agonist potency at Alpha-1B adrenergic receptor expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50000215(NS-49)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonist potency at Alpha-1B adrenergic receptor expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50473663(CHEMBL553276)
Affinity DataEC50:  62nMAssay Description:Agonist potency at Alpha-1B adrenergic receptor expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50473684(CHEMBL74467)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonist potency at Alpha-1B adrenergic receptor expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50473666(CHEMBL542402)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonist potency at Alpha-1B adrenergic receptor expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50473681(CHEMBL540035)
Affinity DataEC50:  14nMAssay Description:Agonist potency at Alpha-1B adrenergic receptor expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50473683(CHEMBL72724)
Affinity DataEC50:  6nMAssay Description:Agonist potency at Alpha-1B adrenergic receptor expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50473680(CHEMBL302698)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonist potency at Alpha-1B adrenergic receptor expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50473671(CHEMBL71479)
Affinity DataEC50:  141nMAssay Description:Agonist potency at Alpha-1B adrenergic receptor expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50473670(CHEMBL70740)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonist potency at Alpha-1B adrenergic receptor expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50218593(CHEMBL117094)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonist potency at Alpha-1B adrenergic receptor expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50473682(CHEMBL70691)
Affinity DataEC50:  3.60nMAssay Description:Agonist potency at Alpha-1B adrenergic receptor expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50473678(CHEMBL306792)
Affinity DataEC50:  6nMAssay Description:Agonist potency at Alpha-1B adrenergic receptor expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50473676(CHEMBL70563)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonist potency at alpha-1b adrenoceptors assayed in rat-1 fibroblasts expressing human Alpha-1B adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50473665(CHEMBL70751)
Affinity DataEC50:  0.501nMAssay Description:Agonist potency at Alpha-1B adrenergic receptor expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50473675(CHEMBL74114)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonist potency at Alpha-1B adrenergic receptor expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50218568(CHEMBL71001)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonist potency at Alpha-1B adrenergic receptor expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50473667(CHEMBL419448)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonist potency at Alpha-1B adrenergic receptor expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50473673(CHEMBL74071)
Affinity DataEC50: <1.00E+4nMAssay Description:Agonist potency at Alpha-1B adrenergic receptor expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50473674(CHEMBL70634)
Affinity DataEC50:  62nMAssay Description:Agonist potency at Alpha-1B adrenergic receptor expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50473664(CHEMBL70326)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonist potency at Alpha-1B adrenergic receptor expressed in rat-1 fibroblastsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50421580(CHEMBL117248)
Affinity DataEC50:  2.20nMAssay Description:Agonist potency at alpha-1b adrenoceptors assayed in rat-1 fibroblasts expressing human alpha-1bMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50474671(CHEMBL111554)
Affinity DataEC50:  5.13E+3nMAssay Description:Agonist activity at alpha1B adrenoreceptor in Rattus norvegicus (rat) spleenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article

TargetAlpha-1B adrenergic receptor(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50474654(CHEMBL323402)
Affinity DataEC50:  977nMAssay Description:Agonist activity at alpha1B adrenoreceptor in Rattus norvegicus (rat) spleenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article

TargetAlpha-1B adrenergic receptor(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50487266(CHEMBL2261355)
Affinity DataEC50:  3.80E+3nMAssay Description:Agonist activity at alpha1B adrenoreceptor in Rattus norvegicus (rat) spleenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article

TargetAlpha-1B adrenergic receptor(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50474630(CHEMBL108804)
Affinity DataEC50:  229nMAssay Description:Agonist activity at alpha1B adrenoreceptor in Rattus norvegicus (rat) spleenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article

TargetAlpha-1B adrenergic receptor(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50118703(N-[5-(4,5-Dihydro-1H-imidazol-2-yl)-2-hydroxy-5,6,...)
Affinity DataEC50:  316nMAssay Description:Agonist activity at alpha1B adrenoreceptor in Rattus norvegicus (rat) spleenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article

TargetAlpha-1B adrenergic receptor(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50022722((1R, 2S)-2-Amino-1-phenyl-propan-1-ol | CHEMBL1365...)
Affinity DataEC50:  2.82E+5nMAssay Description:Agonist activity at alpha1B adrenoreceptor in Rattus norvegicus (rat) spleenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article

TargetAlpha-1B adrenergic receptor(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50474648(CHEMBL109848)
Affinity DataEC50:  1.45E+4nMAssay Description:Agonist activity at alpha1B adrenoreceptor in Rattus norvegicus (rat) spleenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article

TargetAlpha-1B adrenergic receptor(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50474650(CHEMBL111537)
Affinity DataEC50:  1.41E+4nMAssay Description:Agonist activity at alpha1B adrenoreceptor in Rattus norvegicus (rat) spleenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article

TargetAlpha-1B adrenergic receptor(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50118702(CHEMBL1076 | Orvaten | 2-Amino-1-(2,5-dimethoxy-ph...)
Affinity DataEC50:  8.51E+4nMAssay Description:Agonist activity at alpha1B adrenoreceptor in Rattus norvegicus (rat) spleenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article

TargetAlpha-1B adrenergic receptor(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50118705(ABT-866 | N-[3-(1H-imidazol-4-ylmethyl)-phenyl]eth...)
Affinity DataEC50:  692nMAssay Description:Agonist activity at alpha1B adrenoreceptor in Rattus norvegicus (rat) spleenMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article

TargetAlpha-1B adrenergic receptor(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50029050(4-[(1R)-1-hydroxy-2-(methylamino)ethyl]benzene-1,2...)
Affinity DataEC50:  75nMAssay Description:Agonist activity at human alpha1 beta adrenergic receptor expressed in CHOK1 cells co-expressing Galpha15 assessed as increase in calcium influx by m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50029050(4-[(1R)-1-hydroxy-2-(methylamino)ethyl]benzene-1,2...)
Affinity DataEC50:  75nMAssay Description:Agonist activity at human alpha1 beta adrenergic receptor expressed in CHOK1 cells co-expressing Galpha15 assessed as increase in calcium influx by m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50118703(N-[5-(4,5-Dihydro-1H-imidazol-2-yl)-2-hydroxy-5,6,...)
Affinity DataEC50:  320nMAssay Description:Effective concentration in vitro against rat spleen Alpha-1B adrenergic receptor indicates EC50 < 15% at a concentration of 10 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50022722((1R, 2S)-2-Amino-1-phenyl-propan-1-ol | CHEMBL1365...)
Affinity DataEC50:  2.80E+5nMAssay Description:Effective concentration in vitro against rat spleen Alpha-1B adrenergic receptor indicates EC50 < 15% at a concentration of 10 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50118702(CHEMBL1076 | Orvaten | 2-Amino-1-(2,5-dimethoxy-ph...)
Affinity DataEC50:  8.50E+4nMAssay Description:Effective concentration in vitro against rat spleen Alpha-1B adrenergic receptor indicates EC50 < 15% at a concentration of 10 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50238822(2-(2,3-dihydro-1H-inden-1-yl)-1H-imidazole | CHEMB...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human cloned adrenergic Alpha-1B receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50259332(2-(2,3-dihydro-1H-inden-2-yl)-1H-imidazole | CHEMB...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human cloned adrenergic Alpha-1B receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
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