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Report error Found 122 Enz. Inhib. hit(s) with Target = 'Aminopeptidase B'
TargetAminopeptidase B(Rat)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50017480(CHEMBL281437 | 5-Amino-8-guanidino-2-(4-hydroxy-be...)
Affinity DataKi:  0.840nMAssay Description:Inhibition of aminopeptidase B or arginyl aminopeptidase purified from rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetAminopeptidase B(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50036831(6-Amino-2-mercapto-hexanoic acid | CHEMBL432852)
Affinity DataKi:  0.900nMAssay Description:Inhibition of arginylaminopeptidase (aminopeptidase B)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/29/2012
Entry Details Article
PubMed
TargetAminopeptidase B(Rat)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50022743(2,6-Diamino-hexane-1-thiol | CHEMBL68509)
Affinity DataKi:  0.910nMAssay Description:Inhibitory activity against aminopeptidase BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetAminopeptidase B(Rat)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50017482(CHEMBL282583 | 5-Amino-2-benzyl-8-guanidino-4-oxo-...)
Affinity DataKi:  2.5nMAssay Description:Inhibition of aminopeptidase B or arginyl aminopeptidase purified from rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetAminopeptidase B(Rat)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50017476(CHEMBL28623 | 5,9-Diamino-2-benzyl-4-oxo-nonanoic ...)
Affinity DataKi:  4nMAssay Description:Non-competitive inhibition of aminopeptidase B or arginyl aminopeptidase purified from rat liver; Ki value reporting the intercept effect(Kii)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetAminopeptidase B(Rat)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50022751(CHEMBL1204264 | 2-(3-Amino-2-mercapto-4-phenyl-but...)
Affinity DataKi:  4.60nMAssay Description:Inhibitory activity against aminopeptidase BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetAminopeptidase B(Rat)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50022751(CHEMBL1204264 | 2-(3-Amino-2-mercapto-4-phenyl-but...)
Affinity DataKi:  6.40nMAssay Description:Inhibitory activity against aminopeptidase BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetAminopeptidase B(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50036829(2-Mercapto-4-methylsulfanyl-butyric acid | CHEMBL2...)
Affinity DataKi:  11nMAssay Description:Inhibition of arginylaminopeptidase (aminopeptidase B)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/29/2012
Entry Details Article
PubMed
TargetAminopeptidase B(Rat)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM23971(CHEMBL29292 | (2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-...)
Affinity DataKi:  14nMAssay Description:Inhibition of aminopeptidase B or arginyl aminopeptidase purified from rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetAminopeptidase B(Rat)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50010219(CHEMBL3251700)
Affinity DataIC50: 28nMAssay Description:Inhibition of rat liver aminopeptidase B using 0.2 mM L-leucine-beta-naphthylamide by colorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetAminopeptidase B(Rat)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50010220(CHEMBL3251704)
Affinity DataIC50: 31nMAssay Description:Inhibition of rat liver aminopeptidase B using 0.2 mM L-leucine-beta-naphthylamide by colorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetAminopeptidase B(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50652793(CHEMBL5653589)
Affinity DataKd:  42nMAssay Description:Binding affinity to human RNPEP incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetAminopeptidase B(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50036814(2-Mercapto-4-methyl-pentanoic acid | CHEMBL27010)
Affinity DataKi:  51nMAssay Description:Inhibition of arginylaminopeptidase (aminopeptidase B)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/29/2012
Entry Details Article
PubMed
TargetAminopeptidase B(Rat)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM23971(CHEMBL29292 | (2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-...)
Affinity DataKi:  60nMAssay Description:Inhibitory activity against aminopeptidase BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetAminopeptidase B(Rat)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50010221(CHEMBL3251689)
Affinity DataIC50: 130nMAssay Description:Inhibition of rat liver aminopeptidase B using 0.2 mM L-leucine-beta-naphthylamide by colorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetAminopeptidase B(Rat)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50022748(2-Amino-4-methyl-pentane-1-thiol | CHEMBL69349)
Affinity DataKi:  130nMAssay Description:Inhibitory activity against aminopeptidase BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetAminopeptidase B(Rat)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50010222(CHEMBL3251673)
Affinity DataIC50: 160nMAssay Description:Inhibition of rat liver aminopeptidase B using 0.2 mM L-leucine-beta-naphthylamide by colorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetAminopeptidase B(Rat)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM23971(CHEMBL29292 | (2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-...)
Affinity DataIC50: 160nMAssay Description:Inhibition of rat liver aminopeptidase B using 0.2 mM L-leucine-beta-naphthylamide by colorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetAminopeptidase B(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50008434(CHEMBL140459 | 5-Amino-2-benzyl-7-methyl-4-oxo-oct...)
Affinity DataKi:  170nMAssay Description:Compound was tested for binding affinity towards arginyl aminopeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAminopeptidase B(Rat)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50008434(CHEMBL140459 | 5-Amino-2-benzyl-7-methyl-4-oxo-oct...)
Affinity DataKi:  170nMAssay Description:Non-competitive inhibition of aminopeptidase B or arginyl aminopeptidase purified from rat liver; Ki value reporting the intercept effect(Kii)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetAminopeptidase B(Rat)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50010224(CHEMBL3251703)
Affinity DataIC50: 200nMAssay Description:Inhibition of rat liver aminopeptidase B using 0.2 mM L-leucine-beta-naphthylamide by colorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetAminopeptidase B(Rat)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50010226(CHEMBL3251701)
Affinity DataIC50: 310nMAssay Description:Inhibition of rat liver aminopeptidase B using 0.2 mM L-leucine-beta-naphthylamide by colorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetAminopeptidase B(Rat)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50339784((S)-2-((2S,3R)-3-amino-2-hydroxy-4-phenylbutanamid...)
Affinity DataIC50: 420nMAssay Description:Inhibition of rat liver aminopeptidase B using 0.2 mM L-leucine-beta-naphthylamide by colorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetAminopeptidase B(Rat)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50010227(CHEMBL3251688)
Affinity DataIC50: 580nMAssay Description:Inhibition of rat liver aminopeptidase B using 0.2 mM L-leucine-beta-naphthylamide by colorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetAminopeptidase B(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50652792(CHEMBL3752910)
Affinity DataKd:  664nMAssay Description:Binding affinity to human RNPEP incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetAminopeptidase B(Rat)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50010228(CHEMBL3251685)
Affinity DataIC50: 670nMAssay Description:Inhibition of rat liver aminopeptidase B using 0.2 mM L-leucine-beta-naphthylamide by colorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetAminopeptidase B(Rat)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50405948(CHEMBL2114365)
Affinity DataKi:  770nMAssay Description:Non-competitive inhibition of aminopeptidase B or arginyl aminopeptidase purified from rat liver; Ki value reporting the intercept effect(Kii)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetAminopeptidase B(Rat)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50010229(CHEMBL3251686)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of rat liver aminopeptidase B using 0.2 mM L-leucine-beta-naphthylamide by colorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetAminopeptidase B(Rat)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50457479(CHEMBL1159812)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of APB in rat testis using ArgbetaNA as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAminopeptidase B(Rat)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50010140(CHEMBL3251702)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of rat liver aminopeptidase B using 0.2 mM L-leucine-beta-naphthylamide by colorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetAminopeptidase B(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50008430(CHEMBL143589 | 3-Amino-N-(3-methyl-butyl)-2-oxo-4-...)
Affinity DataKi:  1.50E+3nMAssay Description:Compound was tested for binding affinity towards arginyl aminopeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAminopeptidase B(Rat)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50010142(CHEMBL476869 | CHEBI:3070)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of rat liver aminopeptidase B using 0.2 mM L-leucine-beta-naphthylamide by colorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetAminopeptidase B(Rat)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50010141(CHEMBL3251687)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of rat liver aminopeptidase B using 0.2 mM L-leucine-beta-naphthylamide by colorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetAminopeptidase B(Rat)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50017479(CHEMBL28708 | 2-(5,9-Diamino-2-methyl-4-oxo-nonano...)
Affinity DataKi:  2.00E+3nMAssay Description:Non-competitive inhibition of aminopeptidase B or arginyl aminopeptidase purified from rat liver; Ki value reporting the intercept effect(Kii)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetAminopeptidase B(Rat)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50017484(CHEMBL282212 | 5,9-Diamino-2-methyl-4-oxo-nonanoic...)
Affinity DataKi:  2.00E+3nMAssay Description:Non-competitive inhibition of aminopeptidase B or arginyl aminopeptidase purified from rat liver; Ki value reporting the intercept effect(Kii)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetAminopeptidase B(Rat)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50022747(CHEMBL68979 | CHEMBL304141 | 2-(3-Amino-2-hydroxy-...)
Affinity DataKi:  2.40E+3nMAssay Description:Inhibitory activity against aminopeptidase BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetAminopeptidase B(Rat)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50010143(CHEMBL3251684)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of rat liver aminopeptidase B using 0.2 mM L-leucine-beta-naphthylamide by colorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetAminopeptidase B(Rat)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50017479(CHEMBL28708 | 2-(5,9-Diamino-2-methyl-4-oxo-nonano...)
Affinity DataKi:  2.80E+3nMAssay Description:Non-competitive inhibition of aminopeptidase B or arginyl aminopeptidase purified from rat liver; Ki value reporting the KidMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetAminopeptidase B(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50008433(CHEMBL140846 | 3-Amino-5-methyl-2-oxo-hexanoic aci...)
Affinity DataKi:  3.20E+3nMAssay Description:Compound was tested for binding affinity towards arginyl aminopeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAminopeptidase B(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50010157(CHEMBL3251698)
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of aminopeptidase B (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2017
Entry Details Article
PubMed
TargetAminopeptidase B(Rat)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50010157(CHEMBL3251698)
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of rat liver aminopeptidase B using 0.2 mM L-leucine-beta-naphthylamide by colorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetAminopeptidase B(Rat)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50010159(CHEMBL3251683)
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of rat liver aminopeptidase B using 0.2 mM L-leucine-beta-naphthylamide by colorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetAminopeptidase B(Rat)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50022744(3-Amino-2-mercapto-N-(3-methyl-butyl)-4-phenyl-but...)
Affinity DataKi:  4.00E+3nMAssay Description:Inhibitory activity against aminopeptidase BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetAminopeptidase B(Rat)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50046325(2-(3-Amino-2-hydroxy-4-phenyl-butyrylamino)-4-meth...)
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of rat liver aminopeptidase B using 0.2 mM L-leucine-beta-naphthylamide by colorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetAminopeptidase B(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM23971(CHEMBL29292 | (2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-...)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of Aminopeptidase B in murine L-cells by Aoyagi method.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetAminopeptidase B(Rat)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM23971(CHEMBL29292 | (2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-...)
Affinity DataIC50: 6.00E+3nMAssay Description:Compound was evaluated for its inhibitory potency against purified membrane bound rat brain Aminopeptidase B using L-lysine-beta napthylamide as subs...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetAminopeptidase B(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50008432(CHEMBL140779 | 3-Amino-5-methyl-2-oxo-hexanoic aci...)
Affinity DataKi:  6.50E+3nMAssay Description:Compound was tested for binding affinity towards arginyl aminopeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAminopeptidase B(Rat)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50022745(3-Amino-5-methyl-hexane-2-thiol | CHEMBL69814)
Affinity DataKi:  7.00E+3nMAssay Description:Inhibitory activity against aminopeptidase BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetAminopeptidase B(Rat)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50017479(CHEMBL28708 | 2-(5,9-Diamino-2-methyl-4-oxo-nonano...)
Affinity DataKi:  8.80E+3nMAssay Description:Non-competitive inhibition of aminopeptidase B or arginyl aminopeptidase purified from rat liver; Ki value reporting the slope effect(Kis)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetAminopeptidase B(Rat)
University of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50010197(CHEMBL3251691)
Affinity DataIC50: 9.20E+3nMAssay Description:Inhibition of rat liver aminopeptidase B using 0.2 mM L-leucine-beta-naphthylamide by colorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
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