TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataKi: 43nMAssay Description:Displacement of Bak BH3 domain peptide from human Bax by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataKi: 800nMAssay Description:Displacement of FITC-BIM from recombinant N-terminal GST-tagged human BAX expressed in Escherichia coli after 30 mins by fluorescence polarization as...More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataKi: 1.00E+3nMAssay Description:Displacement of FITC-BIM from recombinant N-terminal GST-tagged human BAX expressed in Escherichia coli after 30 mins by fluorescence polarization as...More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataKi: 1.10E+3nMAssay Description:Displacement of FITC-BIM from recombinant N-terminal GST-tagged human BAX expressed in Escherichia coli after 30 mins by fluorescence polarization as...More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataKi: 1.20E+3nMAssay Description:Displacement of FITC-BIM from recombinant N-terminal GST-tagged human BAX expressed in Escherichia coli after 30 mins by fluorescence polarization as...More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataKi: 1.30E+3nMAssay Description:Displacement of FITC-BIM from recombinant N-terminal GST-tagged human BAX expressed in Escherichia coli after 30 mins by fluorescence polarization as...More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataKi: 1.30E+3nMAssay Description:Displacement of FITC-BIM from recombinant N-terminal GST-tagged human BAX expressed in Escherichia coli after 30 mins by fluorescence polarization as...More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataKi: 1.70E+3nMAssay Description:Displacement of FITC-BIM from recombinant N-terminal GST-tagged human BAX expressed in Escherichia coli after 30 mins by fluorescence polarization as...More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataKi: 2.50E+3nMAssay Description:Displacement of FITC-BIM from recombinant N-terminal GST-tagged human BAX expressed in Escherichia coli after 30 mins by fluorescence polarization as...More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataKi: 9.10E+3nMAssay Description:Displacement of FITC-BIM from recombinant N-terminal GST-tagged human BAX expressed in Escherichia coli after 30 mins by fluorescence polarization as...More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataKi: 1.26E+4nMAssay Description:Displacement of FITC-BIM from recombinant N-terminal GST-tagged human BAX expressed in Escherichia coli after 30 mins by fluorescence polarization as...More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataKi: 1.29E+4nMAssay Description:Displacement of FITC-BIM from recombinant N-terminal GST-tagged human BAX expressed in Escherichia coli after 30 mins by fluorescence polarization as...More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataKi: 1.35E+4nMAssay Description:Displacement of FITC-BIM from recombinant N-terminal GST-tagged human BAX expressed in Escherichia coli after 30 mins by fluorescence polarization as...More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataKi: 1.58E+4nMAssay Description:Displacement of FITC-BIM from recombinant N-terminal GST-tagged human BAX expressed in Escherichia coli after 30 mins by fluorescence polarization as...More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataKi: 3.09E+4nMAssay Description:Displacement of FITC-BIM from recombinant N-terminal GST-tagged human BAX expressed in Escherichia coli after 30 mins by fluorescence polarization as...More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataKi: 6.31E+4nMAssay Description:Displacement of FITC-BIM from recombinant N-terminal GST-tagged human BAX expressed in Escherichia coli after 30 mins by fluorescence polarization as...More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataKi: 8.51E+4nMAssay Description:Displacement of FITC-BIM from recombinant N-terminal GST-tagged human BAX expressed in Escherichia coli after 30 mins by fluorescence polarization as...More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataIC50: 43nMAssay Description:Displacement of fluorescent Bak BH3 peptide domain from human recombinant Bax by competition fluorescence polarization assayMore data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataIC50: 250nMAssay Description:Activation of BAX (unknown origin)More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:Activation of Bax in human SMMC7721 cellsMore data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataIC50: 3.30E+3nMAssay Description:Activation of BAX (unknown origin)More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataEC50: 700nMAssay Description:Activation of Bax in human HuH7 cells assessed as inhibition of mitochondrial accumulation of fluorescent probe Mitotracker Red after 12 to 72 hrs by...More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataEC50: 719nMAssay Description:Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F...More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataEC50: 809nMAssay Description:Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F...More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataEC50: 1.14E+3nMAssay Description:Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F...More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataEC50: 393nMAssay Description:Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F...More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataEC50: 2.22E+3nMAssay Description:Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F...More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataEC50: 725nMAssay Description:Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F...More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataEC50: 967nMAssay Description:Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F...More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataEC50: 925nMAssay Description:Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F...More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataEC50: 856nMAssay Description:Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F...More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataEC50: 532nMAssay Description:Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F...More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataEC50: 538nMAssay Description:Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F...More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataEC50: 992nMAssay Description:Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F...More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataEC50: 278nMAssay Description:Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F...More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F...More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataEC50: 8.20E+3nMAssay Description:Activation of Bax in human HuH7 cells assessed as inhibition of mitochondrial accumulation of fluorescent probe Mitotracker Red after 12 to 72 hrs by...More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataEC50: 704nMAssay Description:Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F...More data for this Ligand-Target Pair
TargetApoptosis regulator BAX(Homo sapiens (Human))
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
University Of Texas Medical Branch (Utmb)
Curated by ChEMBL
Affinity DataEC50: 874nMAssay Description:Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F...More data for this Ligand-Target Pair