Compile Data Set for Download or QSAR
Report error Found 1199 Enz. Inhib. hit(s) with Target = 'Casein kinase I isoform alpha'
TargetCasein kinase I isoform alpha-like(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM31090((E)-N-[4-(3-chloro-4-fluoroanilino)-3-cyano-7-etho...)
Affinity DataKd:  1.00E+3nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2011
Entry Details
PCBioAssay
TargetCasein kinase I isoform alpha-like(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM31095(5-[(Z)-(5-fluoranyl-2-oxidanylidene-1H-indol-3-yli...)
Affinity DataKd:  1.50E+3nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2011
Entry Details
PCBioAssay
TargetCasein kinase I isoform alpha-like(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM31096(CHEMBL290084 | Staurosporine | cid_451705 | US2024...)
Affinity DataKd:  250nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2011
Entry Details
PCBioAssay
TargetCasein kinase I isoform alpha-like(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM4814(SUNITINIB MALATE | CHEMBL535 | N-[2-(diethylamino)...)
Affinity DataKd:  550nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2011
Entry Details
PCBioAssay
TargetCasein kinase I isoform alpha(Human)
University of Connecticut

Curated by ChEMBL
LigandPNGBDBM50587736(PYRVINIUM | CHEBI:8687 | Pyrvinium | Pyrvinium (ca...)
Affinity DataKd:  1nMAssay Description:Binding affinity to CK1alpha (unknown origin) using casein as substrate by fluorescence based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetCasein kinase I isoform alpha-like(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50284506(4-[5-(4-Fluoro-phenyl)-2-(4-methanesulfonyl-phenyl...)
Affinity DataKd:  1.70E+3nMAssay Description:Binding affinity to CK1a1L (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetCasein kinase I isoform alpha(Human)
University of Connecticut

Curated by ChEMBL
LigandPNGBDBM50643907(CHEMBL5569495)
Affinity DataKd:  5.30nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetCasein kinase I isoform alpha(Human)
University of Connecticut

Curated by ChEMBL
LigandPNGBDBM50643908(CHEMBL5571313)
Affinity DataKd:  9.80nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetCasein kinase I isoform alpha(Human)
University of Connecticut

Curated by ChEMBL
LigandPNGBDBM50649668(CHEMBL5618142)
Affinity DataEC50: >1.00E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetCasein kinase I isoform alpha(Human)
University of Connecticut

Curated by ChEMBL
LigandPNGBDBM50649669(CHEMBL5619691)
Affinity DataEC50: >1.00E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetCasein kinase I isoform alpha(Human)
University of Connecticut

Curated by ChEMBL
LigandPNGBDBM50649670(CHEMBL5619101)
Affinity DataEC50: >1.00E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetCasein kinase I isoform alpha(Human)
University of Connecticut

Curated by ChEMBL
LigandPNGBDBM50649671(CHEMBL5619187)
Affinity DataEC50: >1.00E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetCasein kinase I isoform alpha(Human)
University of Connecticut

Curated by ChEMBL
LigandPNGBDBM50649672(CHEMBL5619864)
Affinity DataEC50: >1.00E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetCasein kinase I isoform alpha(Human)
University of Connecticut

Curated by ChEMBL
LigandPNGBDBM50649673(CHEMBL5619144)
Affinity DataEC50:  220nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetCasein kinase I isoform alpha(Human)
University of Connecticut

Curated by ChEMBL
LigandPNGBDBM50649674(CHEMBL5620287)
Affinity DataEC50: >1.00E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetCasein kinase I isoform alpha(Human)
University of Connecticut

Curated by ChEMBL
LigandPNGBDBM50649675(CHEMBL5618477)
Affinity DataEC50: >1.00E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetCasein kinase I isoform alpha(Human)
University of Connecticut

Curated by ChEMBL
LigandPNGBDBM50649676(CHEMBL5619449)
Affinity DataEC50: >1.00E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetCasein kinase I isoform alpha(Human)
University of Connecticut

Curated by ChEMBL
LigandPNGBDBM50649677(CHEMBL5619015)
Affinity DataEC50: >1.00E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetCasein kinase I isoform alpha(Human)
University of Connecticut

Curated by ChEMBL
LigandPNGBDBM50649678(CHEMBL5619325)
Affinity DataEC50: >1.00E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetCasein kinase I isoform alpha(Human)
University of Connecticut

Curated by ChEMBL
LigandPNGBDBM50649679(CHEMBL5618239)
Affinity DataEC50: >1.00E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetCasein kinase I isoform alpha(Human)
University of Connecticut

Curated by ChEMBL
LigandPNGBDBM50649680(CHEMBL5618808)
Affinity DataEC50:  170nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetCasein kinase I isoform alpha(Human)
University of Connecticut

Curated by ChEMBL
LigandPNGBDBM50649681(CHEMBL5620230)
Affinity DataEC50:  1.50E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetCasein kinase I isoform alpha(Human)
University of Connecticut

Curated by ChEMBL
LigandPNGBDBM50649682(CHEMBL5618970)
Affinity DataEC50:  1.50E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetCasein kinase I isoform alpha(Human)
University of Connecticut

Curated by ChEMBL
LigandPNGBDBM50649683(CHEMBL5619492)
Affinity DataEC50:  2.10E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetCasein kinase I isoform alpha(Human)
University of Connecticut

Curated by ChEMBL
LigandPNGBDBM50649684(CHEMBL5618672)
Affinity DataEC50: >1.00E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetCasein kinase I isoform alpha(Human)
University of Connecticut

Curated by ChEMBL
LigandPNGBDBM50649685(CHEMBL5618646)
Affinity DataEC50:  250nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetCasein kinase I isoform alpha(Human)
University of Connecticut

Curated by ChEMBL
LigandPNGBDBM50649686(CHEMBL5619824)
Affinity DataEC50:  1.20E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetCasein kinase I isoform alpha(Human)
University of Connecticut

Curated by ChEMBL
LigandPNGBDBM50649687(CHEMBL5618377)
Affinity DataEC50:  1.60E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetCasein kinase I isoform alpha(Human)
University of Connecticut

Curated by ChEMBL
LigandPNGBDBM50649688(CHEMBL5618952)
Affinity DataEC50: >1.00E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetCasein kinase I isoform alpha(Human)
University of Connecticut

Curated by ChEMBL
LigandPNGBDBM50649689(CHEMBL5619918)
Affinity DataEC50: >1.00E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetCasein kinase I isoform alpha(Human)
University of Connecticut

Curated by ChEMBL
LigandPNGBDBM50649690(CHEMBL5618357)
Affinity DataEC50: >1.00E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetCasein kinase I isoform alpha(Human)
University of Connecticut

Curated by ChEMBL
LigandPNGBDBM50649691(CHEMBL5619063)
Affinity DataEC50: >1.00E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetCasein kinase I isoform alpha(Human)
University of Connecticut

Curated by ChEMBL
LigandPNGBDBM50652793(CHEMBL5653589)
Affinity DataKd:  1.04E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetCasein kinase I isoform alpha(Human)
University of Connecticut

Curated by ChEMBL
LigandPNGBDBM50273635(1-(4-methyl-2,5-di(pyridin-4-yl)-1H-pyrrol-3-yl)et...)
Affinity DataKd:  225nMAssay Description:Binding affinity to human CK1alpha2More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCasein kinase I isoform alpha(Human)
University of Connecticut

Curated by ChEMBL
LigandPNGBDBM50326053(PKC-412 | CHEMBL608533 | US20240132489, Compound S...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to CSNK1A1LMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2011
Entry Details Article
PubMed
TargetCasein kinase I isoform alpha(Human)
University of Connecticut

Curated by ChEMBL
LigandPNGBDBM50308060(CEP-701 | 16-hydroxy-16-(hydroxymethyl)-15-methyl-...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to CSNK1A1LMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2011
Entry Details Article
PubMed
TargetCasein kinase I isoform alpha(Human)
University of Connecticut

Curated by ChEMBL
LigandPNGBDBM50300690(CHEMBL576982 | N-(5-tert-Butyl-isoxazol-3-yl)-N'-{...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to CSNK1A1LMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2011
Entry Details Article
PubMed
TargetCasein kinase I isoform alpha(Human)
University of Connecticut

Curated by ChEMBL
LigandPNGBDBM50326054(CHEMBL1240703)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to CSNK1A1LMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2011
Entry Details Article
PubMed
TargetCasein kinase I isoform alpha(Human)
University of Connecticut

Curated by ChEMBL
LigandPNGBDBM13535(N-(4-isopropoxyphenyl)-4-[6-methoxy-7-(3-piperidin...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to CSNK1A1LMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2011
Entry Details Article
PubMed
TargetCasein kinase I isoform alpha(Human)
University of Connecticut

Curated by ChEMBL
LigandPNGBDBM16673(Xarelto | BAY439006 | CHEMBL1336 | BAY 43-9006 | 4...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to CSNK1A1LMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2011
Entry Details Article
PubMed
TargetCasein kinase I isoform alpha(Human)
University of Connecticut

Curated by ChEMBL
LigandPNGBDBM4814(SUNITINIB MALATE | CHEMBL535 | N-[2-(diethylamino)...)
Affinity DataKd:  550nMAssay Description:Binding affinity to CSNK1A1LMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2011
Entry Details Article
PubMed
TargetCasein kinase I isoform alpha-like(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50026612(BIBF-1120 | Nintedanib | Vargatef | US10981896, Co...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1A1L kinase domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2012
Entry Details Article
PubMed
TargetCasein kinase I isoform alpha(Human)
University of Connecticut

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataKd:  970nMAssay Description:Binding constant for CSNK1A1 kinase domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2012
Entry Details Article
PubMed
TargetCasein kinase I isoform alpha(Human)
University of Connecticut

Curated by ChEMBL
LigandPNGBDBM50326053(PKC-412 | CHEMBL608533 | US20240132489, Compound S...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1A1 kinase domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2012
Entry Details Article
PubMed
TargetCasein kinase I isoform alpha-like(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50326053(PKC-412 | CHEMBL608533 | US20240132489, Compound S...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1A1L kinase domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2012
Entry Details Article
PubMed
TargetCasein kinase I isoform alpha-like(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50308060(CEP-701 | 16-hydroxy-16-(hydroxymethyl)-15-methyl-...)
Affinity DataKd:  7.10E+3nMAssay Description:Binding constant for CSNK1A1L kinase domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2012
Entry Details Article
PubMed
TargetCasein kinase I isoform alpha(Human)
University of Connecticut

Curated by ChEMBL
LigandPNGBDBM50308060(CEP-701 | 16-hydroxy-16-(hydroxymethyl)-15-methyl-...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1A1 kinase domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2012
Entry Details Article
PubMed
TargetCasein kinase I isoform alpha-like(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataKd:  250nMAssay Description:Binding constant for CSNK1A1L kinase domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2012
Entry Details Article
PubMed
TargetCasein kinase I isoform alpha(Human)
University of Connecticut

Curated by ChEMBL
LigandPNGBDBM50026612(BIBF-1120 | Nintedanib | Vargatef | US10981896, Co...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1A1 kinase domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2012
Entry Details Article
PubMed
TargetCasein kinase I isoform alpha(Human)
University of Connecticut

Curated by ChEMBL
LigandPNGBDBM25919(N-(2-aminoethyl)-3,12-dimethyl-2,5,8-triazatricycl...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1A1 kinase domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/19/2012
Entry Details Article
PubMed
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