Compile Data Set for Download or QSAR
Report error Found 119 Enz. Inhib. hit(s) with Target = 'Pro-cathepsin H'
TargetPro-cathepsin H(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50460481(CHEMBL4228126)
Affinity DataKi:  4.62E+5nMAssay Description:Uncompetitive inhibition of human liver cathepsin H assessed as inhibitory constant for enzyme-substrate-inhibitor complex using R-AMC as substrate i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetPro-cathepsin H(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50425017(CHEMBL2312203)
Affinity DataKi:  3.54E+5nMAssay Description:Uncompetitive inhibition of human liver cathepsin H endopeptidase activity using R-AMC substrate assessed as inhibition constant for enzyme-substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPro-cathepsin H(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50460502(CHEMBL4228576)
Affinity DataKi:  3.29E+5nMAssay Description:Non-competitive inhibition of human liver cathepsin H assessed as inhibitory constant for enzyme-inhibitor complex using R-AMC as substrate in presen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetPro-cathepsin H(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50460502(CHEMBL4228576)
Affinity DataKi:  3.29E+5nMAssay Description:Non-competitive inhibition of human liver cathepsin H assessed as inhibitory constant for enzyme-substrate-inhibitor complex using R-AMC as substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetPro-cathepsin H(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50074049(3-((S)-1-Benzyloxycarbonyl-3-methyl-butylcarbamoyl...)
Affinity DataKi:  2.60E+5nMAssay Description:Inhibition constant for the non time dependent inhibition of cathepsin HMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPro-cathepsin H(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50415097(CHEMBL570897)
Affinity DataKi:  2.51E+5nMAssay Description:Uncompetitive inhibition of human liver cathepsin H endopeptidase activity using R-AMC substrate assessed as inhibition constant for enzyme-substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPro-cathepsin H(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50425024(CHEMBL2312204)
Affinity DataKi:  2.21E+5nMAssay Description:Noncompetitive inhibition of human liver cathepsin H endopeptidase activity using R-AMC substrate assessed as inhibition constant for enzyme-substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPro-cathepsin H(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50425024(CHEMBL2312204)
Affinity DataKi:  2.21E+5nMAssay Description:Noncompetitive inhibition of human liver cathepsin H endopeptidase activity using R-AMC substrate assessed as inhibition constant for enzyme-inhibito...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPro-cathepsin H(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50074048(1-((S)-2-tert-Butoxycarbonylamino-3-phenyl-propion...)
Affinity DataKi:  2.10E+5nMAssay Description:Compound was evaluated for inhibition constant for the non-time dependent inhibition of Cathepsin H.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPro-cathepsin H(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50074052(1-(2-Benzyloxycarbonylamino-propionyl)-aziridine-2...)
Affinity DataKi:  1.60E+5nMAssay Description:Inhibition constant for the non time dependent inhibition of Cathepsin HMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPro-cathepsin H(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50074050(3-(1-Benzyloxycarbonyl-3-methyl-butylcarbamoyl)-1-...)
Affinity DataKi:  1.37E+5nMAssay Description:Inhibition constant for the non time dependent inhibition of cathepsin HMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPro-cathepsin H(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50425030(CHEMBL2312216)
Affinity DataKi:  1.29E+5nMAssay Description:Noncompetitive inhibition of human liver cathepsin H endopeptidase activity using R-AMC substrate assessed as inhibition constant for enzyme-substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPro-cathepsin H(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50425030(CHEMBL2312216)
Affinity DataKi:  1.29E+5nMAssay Description:Noncompetitive inhibition of human liver cathepsin H endopeptidase activity using R-AMC substrate assessed as inhibition constant for enzyme-inhibito...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPro-cathepsin H(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50460493(CHEMBL4228921)
Affinity DataKi:  1.08E+5nMAssay Description:Competitive inhibition of human liver cathepsin H assessed as inhibitory constant for enzyme-inhibitor complex using R-AMC as substrate in presence o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetPro-cathepsin H(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50074051(3-(1-Benzyloxycarbonyl-3-methyl-butylcarbamoyl)-1-...)
Affinity DataKi:  9.30E+4nMAssay Description:Inhibition constant for the non time dependent inhibition of cathepsin HMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPro-cathepsin H(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50460480(CHEMBL4229176)
Affinity DataKi:  8.90E+4nMAssay Description:Non-competitive inhibition of human liver cathepsin H assessed as inhibitory constant for enzyme-inhibitor complex using R-AMC as substrate in presen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetPro-cathepsin H(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50460480(CHEMBL4229176)
Affinity DataKi:  8.90E+4nMAssay Description:Non-competitive inhibition of human liver cathepsin H assessed as inhibitory constant for enzyme-substrate-inhibitor complex using R-AMC as substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetPro-cathepsin H(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50167297((Cyano-methyl-amino)-acetic acid (S)-2-cyclohexyl-...)
Affinity DataKi: >1.30E+4nMAssay Description:Inhibition constant against human cathepsin H using L-Arg-b-naphthalamideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPro-cathepsin H(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50286441(Ac-LLR-CHO | Ac-Leu-Leu-Arg-H | (S)-2-((S)-2-Acety...)
Affinity DataKi:  9.20E+3nMAssay Description:Inhibition of human liver cathepsin HMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2015
Entry Details Article
PubMed
TargetPro-cathepsin H(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50286441(Ac-LLR-CHO | Ac-Leu-Leu-Arg-H | (S)-2-((S)-2-Acety...)
Affinity DataKi:  9.20E+3nMAssay Description:Inhibition of human liver cathepsin HMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2016
Entry Details Article
PubMed
TargetPro-cathepsin H(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50464766(CHEMBL4292287)
Affinity DataKi:  7.00E+3nMAssay Description:Reversible competitive inhibition of human cathepsin H using fluorogenic AMC-derived peptide substrate assessed as reduction in residual activity pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPro-cathepsin H(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50186088((S)-2-amino-N-((S)-2-biphenyl-4-yl-1-cyano-ethyl)-...)
Affinity DataKi:  3.70E+3nMAssay Description:Inhibition of human recombinant cathepsin H by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPro-cathepsin H(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50243232(N~2~-(MORPHOLIN-4-YLCARBONYL)-N~1~-[(1S,2E)-1-(2-P...)
Affinity DataKi:  1.40E+3nMAssay Description:Inhibition of human recombinant cathepsin H by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPro-cathepsin H(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50464764(CHEMBL4287663)
Affinity DataKi:  1.30E+3nMAssay Description:Reversible competitive inhibition of human cathepsin H using fluorogenic AMC-derived peptide substrate assessed as reduction in residual activity pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPro-cathepsin H(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50247192((S)-2-amino-N-((S)-5-phenyl-1-(phenylsulfonyl)pent...)
Affinity DataKi:  137nMAssay Description:Inhibition of human recombinant cathepsin H by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPro-cathepsin H(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50167289((1S)-2-cyclohexyl-1-methylethyl 2-cyano-2-methylhy...)
Affinity DataKi:  1.40nMAssay Description:Inhibition constant against human cathepsin H using L-Arg-b-naphthalamideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPro-cathepsin H(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50167290((1S)-2-cyclohexyl-1-methylethyl 2-cyano-2-isopropy...)
Affinity DataKi:  0.460nMAssay Description:Inhibition constant against human cathepsin H using L-Arg-b-naphthalamideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPro-cathepsin H(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50201707(5-((2,3-dimethylphenoxy)methyl)-3-methyloxazolidin...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant cathepsin HMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPro-cathepsin H(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50201704((3S,4R)-4-(2,3-dimethylphenoxy)piperidin-3-ol | CH...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant cathepsin HMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPro-cathepsin H(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50201706((3R,4R)-4-(2,3-dimethylphenoxy)piperidin-3-ol | CH...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant cathepsin HMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPro-cathepsin H(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50201703((1S,2S)-2-bromo-7-oxa-5-aza-bicyclo[3.2.1]octan-6-...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant cathepsin HMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPro-cathepsin H(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50201702((1R,2S)-2-phenoxy-7-oxa-5-aza-bicyclo[3.2.1]octane...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant cathepsin HMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPro-cathepsin H(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50250153(3-acetyl-2-(4-tert-butylphenylamino)-8-chloro-6-ni...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human liver cathepsin H after 30 mins by fluorometric end-point assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetPro-cathepsin H(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50250190(3-acetyl-6-chloro-2-(2-chloro-4-methylphenylamino)...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human liver cathepsin H after 30 mins by fluorometric end-point assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetPro-cathepsin H(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50249606(3-acetyl-8-bromo-5-chloro-2-(4-chlorophenylamino)q...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human liver cathepsin H after 30 mins by fluorometric end-point assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetPro-cathepsin H(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50249607(3-acetyl-5,8-dichloro-2-(2,4-dichlorophenylamino)q...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human liver cathepsin H after 30 mins by fluorometric end-point assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetPro-cathepsin H(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50073850([(S)-1-(1-Benzyl-2-oxo-ethylcarbamoyl)-2-methyl-pr...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human liver cathepsin H after 30 mins by fluorometric end-point assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetPro-cathepsin H(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM16509(CA074 | CHEMBL490920 | (2S)-1-[(2S,3S)-3-methyl-2-...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human liver cathepsin H after 30 mins by fluorometric end-point assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetPro-cathepsin H(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50249736(benzyl (S)-1-((S)-4-fluoro-3-oxo-1-phenylbutan-2-y...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human liver cathepsin H after 30 mins by fluorometric end-point assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetPro-cathepsin H(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50249605(3-acetyl-5,8-dibromo-2-(4-bromophenylamino)quinoli...)
Affinity DataIC50: 9.18E+4nMAssay Description:Inhibition of human liver cathepsin H after 30 mins by fluorometric end-point assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetPro-cathepsin H(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50249659(3-acetyl-8-chloro-2-(2,4-dibromophenylamino)-5-met...)
Affinity DataIC50: 6.65E+4nMAssay Description:Inhibition of human liver cathepsin H after 30 mins by fluorometric end-point assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetPro-cathepsin H(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50310690(Cis-(S)-2-amino-N-((1R,2R)-1-cyano-2-phenylcyclopr...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human cathepsin HMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetPro-cathepsin H(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50270039((S)-1-((1S,2S)-1-cyano-2-phenylcyclopropylamino)-1...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human recombinant cathepsin H after 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetPro-cathepsin H(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50270040((S)-1-((1R,2R)-1-cyano-2-phenylcyclopropylamino)-1...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human recombinant cathepsin H after 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetPro-cathepsin H(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM19492((2R)-2-{[(1S)-1-(4-bromophenyl)-2,2,2-trifluoroeth...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human recombinant cathepsin H after 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetPro-cathepsin H(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50270031(1-((1R,2R)-1-cyano-2-phenylcyclopropylamino)-3-(3-...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human recombinant cathepsin H after 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2012
Entry Details Article
PubMed
TargetPro-cathepsin H(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50250191(3-acetyl-6-chloro-2-(2,4-dichlorophenylamino)-8-ni...)
Affinity DataIC50: 3.26E+4nMAssay Description:Inhibition of human liver cathepsin H after 30 mins by fluorometric end-point assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetPro-cathepsin H(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50033762(Gallinamide A)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human Cathepsin H using Arg-aminomethylcoumarin as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetPro-cathepsin H(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50033762(Gallinamide A)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human Cathepsin H using Arg-aminomethylcoumarin as substrate preincubated for 30 mins followed by substrate additionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetPro-cathepsin H(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50201698(rac-trans4-(2,3-dimethylphenoxy)-6-oxa-1-aza-bicyc...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human recombinant cathepsin HMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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