9185 SMILES Strings for Mitogen-activated protein kinase kinase kinase kinase 1

Compound Name
SMILES String
Cc1ccc(F)c(NC(=O)Nc2ccc(cc2)-c2cccc3[nH]nc(N)c23)c1
CCN1CCN(Cc2ccc(NC(=O)Nc3ccc(Oc4cc(NC)ncn4)cc3)cc2C(F)(F)F)CC1
CN1CCN(CC1)c1ccc2nc([nH]c2c1)-c1c(N)c2c(F)cccc2[nH]c1=O
Cc1cccc(c1NC(=O)c2cnc(s2)Nc3cc(nc(n3)C)N4CCN(CC4)CCO)Cl
CCOc1cc2c(cc1NC(=O)/C=C/CN(C)C)c(c(cn2)C#N)Nc3ccc(c(c3)Cl)F
CN1CCC([C@H](O)C1)c1c(O)cc(O)c2c1oc(cc2=O)-c1ccccc1Cl
CN(c1ccc2c(C)n(C)nc2c1)c1ccnc(Nc2ccc(C)c(c2)S(N)(=O)=O)n1
c1cc(c(c(c1)F)C(=O)n2c(nc(n2)Nc3ccc(cc3)S(=O)(=O)N)N)F
CN(C)C[C@@H]1CCn2cc(C3=C(C(=O)NC3=O)c3cn(CCO1)c1ccccc31)c1ccccc21 |r,t:10|
[H][C@@]12C[C@@H]([C@H](OC)[C@@](C)(O1)n1c3ccccc3c3c4CNC(=O)c4c4c5ccccc5n2c4c13)N(C)C(=O)c1ccccc1 |TLB:11:10:9:4.3.2,17:33:9:4.3.2,THB:24:32:9:4.3.2,5:4:9:10.31.33.32,30:31:9:4.3.2|
Cc1[nH]c(\C=C2/C(=O)Nc3ccc(F)cc23)c(C)c1C(=O)NC[C@H](O)CN1CCOCC1
CN[C@H]1C[C@@H]2O[C@](C)([C@H]1OC)n1c3ccccc3c3c4CNC(=O)c4c4c5ccccc5n2c4c13
CCN(CC)CCNC(=O)c1c(C)[nH]c(\C=C2/C(=O)Nc3ccc(F)cc23)c1C
CN1CCN(CC1)c1cc(Nc2cc(C)n[nH]2)nc(Sc2ccc(NC(=O)C3CC3)cc2)n1
CN(C)Cc1nc(Nc2cnc(-c3ccnc4c3c3c(n4C)CCC3)c3c2C(=O)NC3)ccc1C1CCOCC1
CN(C)Cc1nc(Nc2ccc(-c3ccnc4c3c3c(n4C)CCC3)c3c2C(=O)NC3)ccc1C1CCOC1
CN(C)Cc1nc(Nc2cnc(-c3ccnc4c3c3c(n4C)CCC3)c3c2C(=O)NC3)ccc1C1(O)CCOCC1
CN(C)Cc1nc(Nc2ccc(-c3cnn4ccc5ccoc5c34)c3c2C(=O)NC3)ccc1C1CCOCC1
CN(C)Cc1nc(Nc2ccc(-c3ccnc4c3c3c(n4C)CCC3)c3c2C(=O)NC3)ccc1N1CC[C@@H](O)C1
CN(C)Cc1nc(Nc2cnc(-c3ccnc4c3c3c(n4C)CCC3)c3c2C(=O)NC3)ccc1N1CCOCC1
[2H]C([2H])([2H])N(CC1=NC(Nc2cnc(-c3ccnc4c3c3c(n4C)CCC3)c3c2C(=O)NC3)=CCC1C1CCOCC1)C([2H])([2H])[2H]
[2H]C([2H])([2H])N(Cc1nc(Nc2cnc(-c3ccnc4c3c3c(n4C([2H])([2H])[2H])CCC3)c3c2C(=O)NC3)ccc1C1CCOCC1)C([2H])([2H])[2H]
[2H]C([2H])(c1nc(Nc2ccc(-c3ccnc4c3c3c(n4C)CCC3)c3c2C(=O)NC3)ccc1C1CCOCC1)N(C)C
[2H]C([2H])(c1nc(Nc2cnc(-c3ccnc4c3c3c(n4C)CCC3)c3c2C(=O)NC3)ccc1C1CCOCC1)N(C)C
CN(C)Cc1nc(Nc2ccc(-c3nnc4ccc5c(n34)CCC5)c3c2C(=O)NC3)ccc1C1CCOCC1
CN(C)Cc1nc(Nc2ccc(-c3ncnc4c3c3c(n4C)CCC3)c3c2C(=O)NC3)ccc1C1CCOCC1
CN(C)Cc1nc(Nc2ccc(-c3ncnc4[nH]c5ccccc5c34)c3c2C(=O)NC3)ccc1C1CCOCC1
CN(C)Cc1nc(Nc2ccc(-c3ncnc4[nH]c5c(c34)CCC5)c3c2C(=O)NC3)ccc1C1CCOCC1
CN(C)Cc1nc(Nc2cnc(-c3nnc4ccc5c(n34)CCC5)c3c2C(=O)NC3)ccc1C1CCOCC1
CN(C)Cc1nc(Nc2ccc(-c3nnc4cc5c(nn34)CCC5)c3c2C(=O)NC3)ccc1C1CCOCC1
CN(C)Cc1nc(Nc2ccc(-c3nnc4cc5c(cn34)CCC5)c3c2C(=O)NC3)ccc1C1CCOCC1
CN(C)Cc1nc(Nc2ccc(-c3cnc4ccc5c(n34)CCO5)c3c2C(=O)NC3)ccc1C1CCOCC1
CN(C)Cc1nc(Nc2ccc(-c3cnc4ccc5c(n34)CCC5)c3c2C(=O)NC3)ccc1C1CCOCC1
CN(C)Cc1nc(Nc2ccc(-c3cnn4cc5c(nc34)CCC5)c3c2C(=O)NC3)ccc1C1CCOCC1
CN(C)Cc1nc(Nc2ccc(-c3cnc4ccc5c(ccn5C)n34)c3c2C(=O)NC3)ccc1C1CCOCC1
CN(C)Cc1nc(Nc2ccc(-c3nnc4ccc5occc5n34)c3c2C(=O)NC3)ccc1C1CCOCC1
CN(C)Cc1nc(Nc2ccc(-c3cnn4c3CC3(CC3)C4)c3c2C(=O)NC3)ccc1C1CCOCC1
CN(C)Cc1nc(Nc2ccc(-c3cnc4ccc5c(n34)CCO5)c3c2C(=O)NC3)ccc1C1CCOCC1
CN(C)Cc1nc(Nc2ccc(-c3nnc4ccc5c(n34)OCC5)c3c2C(=O)NC3)ccc1C1CCOCC1
CN(C)Cc1nc(Nc2ccc(-c3cnn4ccc5occc5c34)c3c2C(=O)NC3)ccc1C1CCOCC1
CN(C)Cc1nc(Nc2ccc(-c3cnn4ccc5c(c34)CCO5)c3c2C(=O)NC3)ccc1C1CCOCC1
CN(C)Cc1nc(Nc2cnc(-c3cnc4ccc5sccc5n34)c3c2C(=O)NC3)ccc1C1CCOCC1
CN(C)Cc1nc(Nc2ccc(-c3cnc4n3C3CC3C4)c3c2C(=O)NC3)ccc1C1CCOCC1
CN(C)Cc1nc(Nc2ccc(-c3cnc4ccc5c(n34)OCC5)c3c2C(=O)NC3)ccc1C1CCOCC1
CN(C)Cc1nc(Nc2ccc(-c3cnc4ccc5occc5n34)c3c2C(=O)NC3)ccc1C1(O)CCOCC1
CN(C)Cc1nc(Nc2cnc(-c3cnn4ccc5occc5c34)c3c2C(=O)NC3)ccc1C1CCOCC1
CN(C)Cc1nc(Nc2cnc(-c3cnn4ccc5occc5c34)c3c2C(=O)NC3)ccc1N1CCOCC1
CN(C)Cc1nc(Nc2ccc(-c3cnc4cnc5occc5n34)c3c2C(=O)NC3)ccc1C1CCOCC1
CN(C)Cc1nc(Nc2ccc(-c3cnn4ccc5occc5c34)c3c2C(=O)NC3)ccc1N1CCN(C)C1=O
CN(C)Cc1nc(Nc2ccc(-c3cnc4ccc5occc5n34)c3c2C(=O)NC3)ccc1N1CCN(C)C1=O
CN(C)Cc1nc(Nc2ccc(-c3cnn4ccc5occc5c34)c3c2C(=O)NC3)ccc1N1CCCC1=O
CN(C)Cc1nc(Nc2ccc(-c3cnc4ccc5occc5n34)c3c2C(=O)NC3)ccc1N1CCCC1=O
[2H]C([2H])(c1nc(Nc2ccc(-c3cnn4c3CC3(CC3)C4)c3c2C(=O)NC3)ccc1C1CCOCC1)N(C)C
CN(C)Cc1nc(Nc2ccc(-c3cnc4cnc5occc5n34)c3c2C(=O)NC3)ccc1C1CCOC1
CN(C)Cc1nc(Nc2cnc(-c3cnn4c3CC3(CC3)C4)c3c2C(=O)NC3)ccc1C1CCOCC1
O=C1NCc2c(-c3cnn4ccc5occc5c34)ccc(Nc3ccc(N4CCOCC4)c([C@H]4CCCN4)n3)c21
CN(C)Cc1nc(Nc2ccc(-c3cnc4cnc5occc5n34)c3c2C(=O)NC3)ccc1C1CC(=O)N(C)C1
CN(C)Cc1nc(Nc2ccc(-c3cnn4ccc5occc5c34)c3c2C(=O)NC3)ccc1C1CC(=O)N(C)C1
CN(C)Cc1nc(Nc2ccc(-c3cnn4ccc5occc5c34)c3c2C(=O)NC3)ccc1C1CCN(C)C(=O)C1
CN(C)Cc1nc(Nc2ccc(-c3cnc4cnc5occc5n34)c3c2C(=O)NC3)ccc1C1CCN(C)C(=O)C1
CN(C)Cc1nc(Nc2ccc(-c3cnn4ccc5occc5c34)c3c2C(=O)NC3)ccc1C1CCCO1
CN(C)Cc1nc(Nc2ccc(-c3cnc4cnc5occc5n34)c3c2C(=O)NC3)ccc1C1CCCO1
CN(C)Cc1nc(Nc2ccc(-c3cnc4ccc5occc5n34)c3c2C(=O)NC3)ccc1C1CCN(C)C(=O)C1
CN(C)Cc1nc(Nc2ccc(-c3cnn4c3CC3(CC3)C4)c3c2C(=O)NC3)ccc1C1CCN(C)C(=O)C1
CN(C)Cc1nc(Nc2ccc(-c3cnc4cnc5occc5n34)c3c2C(=O)NC3)ccc1[C@@H]1CCN(C)C(=O)C1
CN(C)Cc1nc(Nc2ccc(-c3cnc4cnc5occc5n34)c3c2C(=O)NC3)ccc1[C@H]1CCN(C)C(=O)C1
CC(=O)N(C)c1ccc(Nc2ccc(-c3cnn4ccc5occc5c34)c3c2C(=O)NC3)nc1CN(C)C
CN(C)Cc1nc(Nc2ccc(-c3cnn4c3CC3(CC4)CC3)c3c2C(=O)NC3)ccc1[C@@H]1CCN(C)C(=O)C1
CN(C)Cc1nc(Nc2ccc(-c3cnc4ccc5occc5n34)c3c2C(=O)NC3)ccc1[C@H]1CCN(C)C(=O)C1
CN(C)Cc1nc(Nc2ccc(-c3cnc4ccc5occc5n34)c3c2C(=O)NC3)ccc1[C@@H]1CCN(C)C(=O)C1
CN(C)Cc1nc(Nc2ccc(C3=C4C5=C(C=CC4N=C3)OCC5)c3c2C(=O)NC3)ccc1C1CCN(C)C(=O)C1
CN(C)Cc1nc(Nc2ccc(-c3cnn4c3CC3(CC3)C4)c3c2C(=O)NC3)ccc1N1CCN(C)C(=O)C1
CN(C)Cc1nc(Nc2ccc(-c3cnn4ccc5occc5c34)c3c2C(=O)NC3)ccc1N1CCN(C)C(=O)C1
CN(C)Cc1nc(Nc2ccc(-c3cnc4ccc5occc5n34)c3c2C(=O)NC3)ccc1-c1ccn(C)c(=O)c1
CN(C)Cc1nc(Nc2ccc(-c3cnn4c3CC3(CC3)C4)c3c2C(=O)NC3)ccc1C1CCN(C)CC1
CCCc1nc(Nc2ccc(-c3cnn4ccc5occc5c34)c3c2C(=O)NC3)ccc1C1CCOC1
CN(C)Cc1nc(Nc2ccc(-c3cnc4cnc5occc5n34)c3c2C(=O)NC3)ccc1C1CCN(C)CC1
CN(C)Cc1nc(Nc2ccc(-c3cnn4ccc5occc5c34)c3c2C(=O)NC3)ccc1-c1ccn(C)c(=O)c1
CN(C)Cc1nc(Nc2ccc(-c3ccnc4c3cc3n4CCC3)c3c2C(=O)NC3)ccc1C1CCN(C)C(=O)C1
CN(C)Cc1nc(Nc2ccc(-c3cnn4ccc5occc5c34)c3c2C(=O)NC3)ccc1C1CCN(C)CC1
CN(C)Cc1nc(Nc2ccc(-c3ccnc4c3c3c(n4C)CCC3)c3c2C(=O)NC3)ccc1C1CCN(C)C(=O)C1
CNCc1nc(Nc2ccc(-c3cnn4ccc5occc5c34)c3c2C(=O)NC3)sc1C1CCOCC1
Clc1cccc(Cl)c1-c1ccc2cnc(Nc3ccncn3)cc2c1
CN1CCC(Cn2cc(Nc3cc4cc(-c5c(Cl)cccc5Cl)ccc4cn3)cn2)C1
Clc1cccc(Cl)c1-c1ccc2cnc(Nc3cnn(C4CCOC4)c3)cc2c1
Fc1cccc(Cl)c1-c1ccc2cnc(Nc3ccncn3)cc2c1
CCc1ccnc(Nc2cc3cc(-c4cnccc4C)ccc3cn2)c1
Cc1ccncc1-c1ccc2cnc(Nc3cc(C(F)F)ccn3)cc2c1
Cc1cc(Nc2cc3cc(-c4cnccc4C)ccc3cn2)ncn1
Cc1ccnc(Nc2cc3cc(-c4cnccc4C)ccc3cn2)c1
Cc1c(-c2cc3cc(Nc4ccn([C@H](C)C#N)n4)ncc3cc2F)cnc2c1NCCO2
Cc1c(-c2cc3cc(Nc4ccn([C@@H](C)C#N)n4)ncc3cc2F)cnc2c1NCCO2
Cc1ccncc1-c1cc2cc(Nc3cc4n(n3)CC(=O)N(C)CC4)ncc2c(Cl)c1F
Cc1c(N)cncc1-c1cc2cc(Nc3cc4n(n3)CC(=O)N(C)CC43CC3)ncc2cc1F
Cc1c(N)cncc1-c1cc2cc(Nc3cc4n(n3)CS(=O)(=O)N(C)CC4C)ncc2cc1F
Cc1ccncc1-c1cc2cc(Nc3cn4c(n3)CC(=O)N(C)CC4)ncc2c(Cl)c1F
Cc1c(-c2cc3cc(Nc4cc5n(n4)CC(=O)N(C(C)C)CC5)ncc3c(Cl)c2F)cnc2c1NCCO2
Cc1c(-c2cc3cc(Nc4cc5n(n4)CC(=O)N(C(C)C)CC5)ncc3cc2F)cnc2c1NCCO2
Cc1c(N)cncc1-c1cc(Cl)c2cnc(Nc3cc4n(n3)CC(=O)N(C(C)C)CC4)cc2c1
Cc1c(N)cncc1-c1cc2cc(Nc3cc4n(n3)CC(=O)N(C(C)C)CC4)ncc2c(F)c1F
CC(C)N1CCc2cc(Nc3cc4cc(c(F)cc4cn3)-c3cncc(N)c3C)nn2CC1=O
Cc1c(N)cncc1-c1cc2cc(Nc3cc4n(n3)CC(=O)N(C)C(C)(C)C4)ncc2cc1F
Cc1c(N)cncc1-c1cc2cc(Nc3cc4n(n3)CC(=O)N(C(C)C)CC4)ncc2c(C)c1F
Cc1ccncc1-c1ccc2cnc(Nc3cc4n(n3)CC(=O)N(C(C)C)CC4)cc2c1
Cc1c(-c2cc3cc(Nc4cc5n(n4)CC(=O)N(C(C)C)CC5)ncc3cc2F)cnc2c1NC(=O)CO2
CC(C)N1CCc2cc(Nc3cc4cc(C(=O)N5CCN(C)CC5)c(F)cc4cn3)nn2CC1=O
Cc1c(N)cncc1-c1cc2cc(Nc3cc4n(n3)Cc3nccn3CC4)ncc2cc1F
Cc1ncc(-c2cc3cc(Nc4cc5n(n4)CC(=O)N(C(C)C)CC5)ncc3cc2F)c(C)c1N
Cc1c(N)cncc1-c1cc2cc(Nc3cc4n(n3)CC(=O)N(C)CC4(F)F)ncc2cc1F
Cc1c(-c2cc3cc(Nc4cc5n(n4)CC(=O)N(C)CC5)ncc3cc2F)cnc2c1NCCO2
Cc1c(N)cncc1-c1ccc2cnc(Nc3cc4n(n3)CC(=O)N(C(C)C)CC4)cc2c1
Cc1c(N)cncc1-c1cc2cc(Nc3cc4n(n3)CC(=O)N(C(C)C)CC4)ncc2c(C)c1C#N
Cc1ccncc1-c1cc2cc(Nc3cc4n(n3)CC(=O)N(C(C)C)CC4)ncc2cc1F
Cc1c(-c2cc3cc(Nc4cc5n(n4)CC(=O)N(CCN4CCOCC4)CC5)ncc3cc2F)cnc2c1NCCO2
Cc1ncc(-c2cc3cc(Nc4cc5n(n4)CC(=O)N(C(C)C)CC5)ncc3c(O)c2F)c(C)c1N
Cc1ccncc1-c1cc2cc(Nc3cc4n(n3)CC3=NOC(C)(C)N3CC4)ncc2cc1F
Cc1c(-c2cc3cc(Nc4cc5n(n4)CC(=O)N(C(C)C)CC5)ncc3c(F)c2F)cnc2c1NCCO2
Cc1c(N)cncc1-c1cc2cc(Nc3cc4n(n3)CC(=O)N(CCN3CCOCC3)CC4)ncc2cc1F
COc1cc(C)c(-c2cc3cc(Nc4cc5n(n4)CC(=O)N(C)CC5)ncc3cc2F)cn1
Cc1c(-c2cc3cc(Nc4cc5n(n4)CC(=O)N(C)CC5)ncc3c(F)c2F)cnc2c1NCCO2
Cc1c(N)cncc1-c1cc2cc(Nc3cc4n(n3)Cc3nncn3CC4)ncc2cc1F
Cc1c(N)cncc1-c1cc2cc(Nc3cc4n(n3)CC(=O)N(C(C)C)CC4)ncc2cc1Cl
Cc1c(-c2cc3cc(Nc4cc5n(n4)CC(=O)N(C(C)C)C[C@H]5O)ncc3cc2F)cnc2c1NCCO2
Cc1c(-c2cc3cc(Nc4cc5n(n4)CC(=O)N(C(C)C)CC5O)ncc3cc2F)cnc2c1NCCO2
Cc1c(-c2cc3cc(Nc4cc5n(n4)CC(=O)N(C(C)C)CC5)ncc3cc2F)cnc2oc(=O)[nH]c12
Cc1c(-c2cc3cc(Nc4cc5n(n4)Cc4nccn4CC5)ncc3cc2F)cnc2c1NCCO2
Cc1c(N)cncc1-c1cc2cc(Nc3cc4n(n3)CC(=O)NCC4)ncc2cc1F
Cc1c(-c2cc3cc(Nc4cc5n(n4)CC(=O)N(CCO)CC5)ncc3cc2F)cnc2c1NCCO2
Cc1c(-c2ccc3cnc(Nc4cc5n(n4)CC(=O)N(CCO)CC5)cc3c2F)cnc2c1NCCO2
Cc1c(-c2cc3cc(Nc4cc5n(n4)CC(=O)N([C@@H](C)C#N)CC5)ncc3cc2F)cnc2c1NCCO2
Cc1c(-c2cc3cc(Nc4cc5n(n4)CC(=O)N(C(C)C#N)CC5)ncc3cc2F)cnc2c1NCCO2
Cc1c(-c2cc3cc(Nc4cc5n(n4)CC(=O)N([C@@H](C)CO)CC5)ncc3cc2F)cnc2c1NCCO2
Cc1c(-c2cc3cc(Nc4cc5n(n4)CC(=O)N(C(C)CO)CC5)ncc3cc2F)cnc2c1NCCO2
Cc1c(N)cncc1-c1cc2cc(Nc3cc4n(n3)CC(=O)N([C@@H](C)CO)CC4)ncc2cc1F
Cc1c(N)cncc1-c1cc2cc(Nc3cc4n(n3)CC(=O)N(C(C)CO)CC4)ncc2cc1F
Cc1ncc(-c2cc3cc(Nc4cc5n(n4)CC(=O)N(C(C)C)CC5F)ncc3cc2F)c(C)c1N
Cc1c(-c2cc3cc(Nc4cc5n(n4)Cc4nncn4CC5)ncc3cc2F)cnc2c1NCCO2
Cc1c(N)cncc1-c1ccc2cnc(Nc3cc4n(n3)CC(=O)N(C(C)C)CC4)cc2c1Cl
Cc1c(N)cncc1-c1cc2cc(Nc3cc4n(n3)CC(=O)N(C(C)C)C[C@H]4O)ncc2cc1F
Cc1c(N)cncc1-c1cc2cc(Nc3cc4n(n3)CC(=O)N(C(C)C)CC4O)ncc2cc1F
Cc1c(N)cncc1-c1cc2cc(Nc3cc4n(n3)CC(=O)N([C@@H](C)C#N)CC4)ncc2cc1F
Cc1c(N)cncc1-c1cc2cc(Nc3cc4n(n3)CC(=O)N(C(C)C#N)CC4)ncc2cc1F
COCCN1CCc2cc(Nc3cc4cc(-c5cnc6c(c5C)NCCO6)c(F)cc4cn3)nn2CC1=O
COCCN1CCc2cc(Nc3cc4cc(-c5cncc(N)c5C)c(F)cc4cn3)nn2CC1=O
Cc1c(N)cncc1-c1cc2cc(Nc3cc4n(n3)Cc3nccn3CC4)ncc2c(F)c1F
Cc1c(N)cncc1-c1cc2cc(Nc3cc4n(n3)CC(=O)N(CC(C)(C)O)CC4)ncc2cc1F
Cc1c(N)cncc1-c1cc2cc(Nc3cc4n(n3)CC(=O)N(CCO)CC4)ncc2cc1F
Cc1c(-c2cc3cc(Nc4cc5n(n4)CC(=O)NCC5)ncc3cc2F)cnc2c1NCCO2
Cc1c(-c2cc3cc(Nc4cc5n(n4)Cc4nccn4CC5)ncc3c(F)c2F)cnc2c1NCCO2
Cc1c(-c2cc3cc(Nc4cc5n(n4)CC(=O)N(C)CC5)ncc3cc2F)cnc2c1N(C)CCO2
Cc1c(N)cncc1-c1cc2cc(Nc3cc4n(n3)Cc3ncc(C)n3CC4)ncc2cc1F
Cc1c(N)cncc1-c1cc2cc(Nc3cc4n(n3)CC(=O)N(CCN3CC(F)C3)CC4)ncc2cc1F
Cc1c(N)cncc1-c1cc2cc(Nc3cc4n(n3)CC(=O)N(CCN3CC(O)C3)CC4)ncc2cc1F
Cc1c(N)cncc1-c1cc2cc(Nc3cc4n(n3)CC3=NOC(C)(C)N3CC4)ncc2cc1F
Cc1c(N)cncc1-c1cc2cc(Nc3cc4n(n3)CC(=O)N(C(C)(C)C)C[C@H]4F)ncc2cc1F
Cc1c(N)cncc1-c1cc2cc(Nc3cc4n(n3)CC(=O)N(C(C)(C)C)CC4F)ncc2cc1F
Cc1c(N)cncc1-c1cc(F)c2cnc(Nc3cc4n(n3)Cc3nccn3CC4)cc2c1
Cc1c(N)cncc1-c1cc2cc(Nc3cc4n(n3)CC(=O)N(C(C)C)CC4)ncc2cc1C#N
Cc1c(N)cncc1-c1cc2cc(Nc3cc4n(n3)Cc3nccn3CC4O)ncc2c(F)c1F
CC(=O)Nc1cncc(-c2cc3cc(Nc4cc5n(n4)CC(=O)N(C)CC5)ncc3cc2F)c1C
Cc1c(NS(C)(=O)=O)cncc1-c1cc2cc(Nc3cc4n(n3)CC(=O)N(C)CC4)ncc2cc1F
Cc1c(-c2ccc3cnc(Nc4cc5n(n4)CC(=O)N(C)CC5)cc3c2F)cnc2c1NCCO2
Cc1c(-c2cc3cc(Nc4cc5n(n4)CC(=O)N(C)CC5)ncc3cc2F)cnc2nc[nH]c12
Cc1c(-c2cc3cc(Nc4cc5n(n4)CC(=O)NCC5)ncc3cc2F)cnc2c1NCC(F)(F)O2
Cc1c(-c2cc3cc(Nc4cc5n(n4)CC(=O)N(C)CC5)ncc3cc2F)cnc2c1NCCS2(=O)=O
Cc1cc(S(C)(=N)=O)ncc1-c1cc2cc(Nc3cc4n(n3)CC(=O)N(C)CC4)ncc2cc1F
Cc1c(NC2CNC2)cncc1-c1cc2cc(Nc3cc4n(n3)Cc3nccn3CC4)ncc2cc1F
Cc1c(-c2cc3cc(Nc4cc5n(n4)CC(=O)N(C)CC5)ncc3cc2F)cnc2c1C(O)CCO2
Cc1c(-c2cc3cc(Nc4cc5n(n4)CC(=O)N(C)CC5)ncc3cc2F)cnc2c1C(O)CCO2
CNc1cncc(-c2cc3cc(Nc4cc5n(n4)CC(=O)NCC5)ncc3cc2F)c1C
Cc1c(-c2cc3cc(Nc4cc5n(n4)CC(=O)NCC5)ncc3cc2F)cnc2c1NC(C)CO2
Cc1c(-c2cc3cc(Nc4cc5n(n4)Cc4nccn4CC5)ncc3cc2F)cnc2c1NCCCO2
Cc1c(-c2cc3cc(Nc4cc5n(n4)CC(=O)NCC5)ncc3cc2F)cnc2c1NCC(C)O2
Cc1c(N)cncc1-c1cc2cc(Nc3cc4n(n3)CC(=O)N(C)C[C@@]4(C)O)ncc2cc1F
Cc1c(N)cncc1-c1cc2cc(Nc3cc4n(n3)CC(=O)N(C)CC4(C)O)ncc2cc1F
Cc1c(-c2cc3cc(Nc4cc5n(n4)CC(=O)N(C)CC5)ncc3cc2F)cnc2cn[nH]c12
Cc1c(-c2cc3cc(Nc4cc5n(n4)CC(=O)N(C)CC5)ncc3cc2F)cnc2c1NCN(C)C2=O
Cc1c(-c2cc3cc(Nc4cc5n(n4)Cc4nccn4CC5)ncc3cc2F)cnc2c1NCCS2=O
Cc1c(-c2cc3cc(Nc4cc5n(n4)CC(=O)N(C)CC5)ncc3cc2F)cnc2c1CCCO2
Cc1c(N)cncc1-c1cc2cc(Nc3cc4n(n3)CS(=O)CC4)ncc2cc1F
Cc1c(-c2cc3cc(Nc4cc5n(n4)CC(=O)NCC5)ncc3cc2F)cnc2c1NCCC2
Cc1c(-c2cc3cc(Nc4cc5n(n4)CC(=O)N(C)CC5)ncc3cc2F)cnc2c1NS(=O)(=O)CO2
Cc1c(-c2cc3cc(Nc4cc5n(n4)CC(=O)N(C)CC5)ncc3cc2F)cnnc1N
Cc1c[nH]c2c(C)c(-c3cc4cc(Nc5cc6n(n5)CC(=O)N(C)CC6)ncc4cc3F)cnc12
Cc1c(-c2cc3cc(Nc4cc5n(n4)CC(=O)NCC5)ncc3cc2F)cnc2c1NCCC2=O
Cc1c(NS(=O)(=O)C2CC2)cncc1-c1cc2cc(Nc3cc4n(n3)CC(=O)N(C)CC4)ncc2cc1F
Cc1cc(N2CCNCC2)ncc1-c1cc2cc(Nc3cc4n(n3)CC(=O)N(C)CC4)ncc2cc1F
CNC1CCN(c2cc(C)c(-c3cc4cc(Nc5cc6n(n5)CC(=O)N(C)CC6)ncc4cc3F)cn2)CC1
CN1CCc2cc(Nc3cc4cc(-c5cccc6c5CCNC6)c(F)cc4cn3)nn2CC1=O
Cc1c(-c2cc3cc(Nc4cc5n(n4)CC(=O)NCC5)ncc3cc2F)cnc2c1NCCC2O
Cc1[nH]ncc1-c1cc2cc(Nc3cc4n(n3)CC(=O)N(C)CC4)ncc2c(O)c1F
Cc1c(-c2cc3cc(Nc4cc5n(n4)CC(=O)N(C)CC5)ncc3cc2F)cnc(=O)n1C
Cc1c(CS(C)(=O)=O)cncc1-c1cc2cc(Nc3cc4n(n3)CC(=O)N(C)CC4)ncc2cc1F
Cc1c(-c2cc3cc(Nc4cc5n(n4)CC(=O)N(C)CC54CC4)ncc3cc2F)cnc2c1NCC[C@H]2O
Cc1c(-c2cc3cc(Nc4cc5n(n4)CC(=O)N(C)CC54CC4)ncc3cc2F)cnc2c1NCC[C@@H]2O
CN[C@@H]1CCN(c2cc(C)c(-c3cc4cc(Nc5cc6n(n5)CC(=O)N(C)CC6)ncc4cc3F)cn2)C1
CN[C@H]1CCN(c2cc(C)c(-c3cc4cc(Nc5cc6n(n5)CC(=O)N(C)CC6)ncc4cc3F)cn2)C1
Cc1c(CN)cncc1-c1cc2cc(Nc3cc4n(n3)CC(=O)N(C)CC4)ncc2cc1F
Cc1c(-c2cc3cc(Nc4cc5n(n4)CC(=O)N(C)CC5)ncc3cc2F)cnc2c1NCCC2(F)F
Cc1c(-c2cc3cc(Nc4cc5n(n4)CC(=O)N(C)CC5)ncc3cc2F)cnc2c(=O)n(C)[nH]c12
CNCc1cncc(-c2cc3cc(Nc4cc5n(n4)CC(=O)N(C)CC5)ncc3cc2F)c1C
Cc1c(CN)cncc1-c1cc2cc(Nc3cc4n(n3)CC(=O)N(C)CC4)ncc2cc1F
Cc1cc(CN)ncc1-c1cc2cc(Nc3cc4n(n3)CC(=O)N(C)CC4)ncc2cc1F
Cc1cc(CN)ccc1-c1cc2cc(Nc3cc4n(n3)CC(=O)N(C)CC4)ncc2cc1F
CN1CCc2cc(Nc3cc4cc(-c5cncc6c5CCC6O)c(F)cc4cn3)nn2CC1=O
CN1CCc2cc(Nc3cc4cc(-c5cccc6c5CNC6)c(F)cc4cn3)nn2CC1=O
Cc1c(N)cnnc1-c1cc2cc(Nc3cc4n(n3)CC(=O)N(C)CC4)ncc2cc1F
CNCc1cccc(-c2cc3cc(Nc4cc5n(n4)CC(=O)N(C)CC5)ncc3cc2F)c1C
Cc1cc(C2CCCCO2)ncc1-c1cc2cc(Nc3cc4n(n3)CC(=O)N(C)CC4)ncc2cc1F
CNCc1ccc(F)c(-c2ccc3cnc(Nc4cc5n(n4)CC(=O)N(C)CC5)cc3c2)c1C
CNCc1cc(-c2ccc3cnc(Nc4cc5n(n4)CC(=O)N(C)CC5)cc3c2)c(F)cc1C
Cc1c(-c2cc3cc(Nc4cc5n(n4)CC(=O)N(C)CC5)ncc3cc2F)ccc2c1CNC2
CNCc1cc(C)c(-c2ccc3cnc(Nc4cc5n(n4)CC(=O)N(C)CC5)cc3c2)c(F)c1
Cc1c(-c2c(F)cc3cnc(Nc4cc5n(n4)CC(=O)N(C)CC5)cc3c2F)cnc2c1NCCO2
Cc1c(N)cncc1-c1cc2cc(Nc3cc4n(n3)CC(=O)NCC43CC3)ncc2cc1F
Cc1c(N)cncc1-c1cc(F)c2cnc(Nc3cc4n(n3)CC(=O)NCC43CC3)cc2c1
Cc1c(-c2cc3cc(Nc4cc5n(n4)CC(=O)N(C)CC5)ncc3cc2F)cnc2c1[C@@](C)(O)CCO2
Cc1c(-c2cc3cc(Nc4cc5n(n4)CC(=O)N(C)CC5)ncc3cc2F)cnc2c1[C@](C)(O)CCO2
CN1CCc2cc(Nc3cc4cc(-c5cncc(N)c5C(F)(F)F)c(F)cc4cn3)nn2CC1=O
CN[C@@H]1CCc2c(-c3cc4cc(Nc5cc6n(n5)CC(=O)N(C)CC6)ncc4cc3F)cncc21
CN[C@H]1CCc2c(-c3cc4cc(Nc5cc6n(n5)CC(=O)N(C)CC6)ncc4cc3F)cncc21
Cc1c(-c2cc3cc(Nc4cc5n(n4)CC(=O)N(C)CC54CC4)ncc3cc2F)cnc2c1NCC[C@]2(C)O
Cc1c(-c2cc3cc(Nc4cc5n(n4)CC(=O)N(C)CC54CC4)ncc3cc2F)cnc2c1NCC[C@@]2(C)O
Cc1c(-c2cc3cc(Nc4cc5n(n4)CC(=O)NCC5)ncc3cc2F)cnc2c1NCCOC2
Cc1c(-c2cc(F)c3cnc(Nc4cc5n(n4)CC(=O)N(C)CC5)cc3c2)cnc2c1NCC[C@@]2(C)O
Cc1c(-c2cc(F)c3cnc(Nc4cc5n(n4)CC(=O)N(C)CC5)cc3c2)cnc2c1NCC[C@]2(C)O
Cc1c(-c2cc3cc(Nc4cc5n(n4)CC(=O)N(C)CC5)ncc3cc2F)cnc2c1CNCCO2
Cc1ncc(-c2cc(F)c3cnc(Nc4cc5n(n4)CC(=O)NCC5)cc3c2)c(C)c1N
CO[C@H]1CCNc2c1ncc(-c1cc(F)c3cnc(Nc4cc5n(n4)CC(=O)N(C)CC5)cc3c1)c2C
CO[C@@H]1CCNc2c1ncc(-c1cc(F)c3cnc(Nc4cc5n(n4)CC(=O)N(C)CC5)cc3c1)c2C
Cc1c(-c2cc3cc(Nc4cc5n(n4)CC(=O)N(C)CC5)ncc3cc2F)cnc2c1[C@@H](F)CCO2
Cc1c(-c2cc3cc(Nc4cc5n(n4)CC(=O)N(C)CC5)ncc3cc2F)cnc2c1[C@H](F)CCO2
Cc1c(-c2cc3cc(Nc4cc5n(n4)CC(=O)N(C)CC5)ncc3cc2F)cnc2c1NCC[C@@H]2O
Cc1c(-c2cc3cc(Nc4cc5n(n4)CC(=O)N(C)CC5)ncc3cc2F)cnc2c1NCC[C@H]2O
Cc1c(-c2cc(F)c3cnc(Nc4cc5n(n4)CC(=O)N(C)CC54CC4)cc3c2)cnc2c1NCC[C@@H]2O
Cc1c(-c2cc(F)c3cnc(Nc4cc5n(n4)CC(=O)N(C)CC54CC4)cc3c2)cnc2c1NCC[C@H]2O
Cc1c(CC#N)cncc1-c1cc(F)c2cnc(Nc3cc4n(n3)CC(=O)NCC4)cc2c1
Cc1c(NCC(F)(F)F)cncc1-c1cc2cc(Nc3cc4n(n3)CC(=O)NCC4)ncc2cc1F
Cc1c(-c2cc3cc(Nc4cc5n(n4)CC(=O)N(C)CC5)ncc3cc2F)cnc2c1NCC(C)(C)C2=O
Cc1c(-c2cc3cc(Nc4cc5n(n4)CC(=O)N(C)CC5)ncc3cc2F)cnc2c1NCC(C)(C)[C@H]2O
Cc1c(-c2cc3cc(Nc4cc5n(n4)CC(=O)N(C)CC5)ncc3cc2F)cnc2c1NCC(C)(C)[C@@H]2O
Cc1c(-c2cc3cc(Nc4cc5n(n4)CS(=O)(=O)N(C)C5)ncc3cc2F)cnc2c1NCC[C@@H]2O
Cc1c(-c2cc3cc(Nc4cc5n(n4)CS(=O)(=O)N(C)C5)ncc3cc2F)cnc2c1NCC[C@H]2O
Cc1c(-c2cc3cc(Nc4cc5n(n4)Cc4nccn4CC5)ncc3cc2F)cnc2c1NCC[C@@H]2O
Cc1c(-c2cc3cc(Nc4cc5n(n4)Cc4nccn4CC5)ncc3cc2F)cnc2c1NCC[C@H]2O
Cc1c(-c2cc3cc(Nc4cc5n(n4)CC(=O)N(C)OC5)ncc3cc2F)cnc2c1NCCO2
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2cc(=O)n(cc12)-c1ccccc1
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2cc(=O)n(cc12)-c1ccccc1F
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2cc(=O)n(cc12)-c1ccccc1C
COc1ccccc1-n1cc2c(n[nH]c2cc1=O)-c1ccc(cc1)N1CCN(C)CC1
COc1cccc(F)c1-n1cc2c(n[nH]c2cc1=O)-c1ccc(cc1)N1CCN(C)CC1 |(-1.11,2.37,;-2.44,1.6,;-3.78,2.37,;-3.78,3.91,;-5.11,4.68,;-6.45,3.91,;-6.45,2.37,;-7.78,1.6,;-5.11,1.6,;-5.11,.06,;-3.78,-.71,;-3.78,-2.25,;-2.63,-3.28,;-3.26,-4.68,;-4.79,-4.52,;-5.11,-3.02,;-6.45,-2.25,;-6.45,-.71,;-7.78,.06,;-1.15,-2.88,;-.06,-3.97,;1.43,-3.57,;1.83,-2.08,;.74,-.99,;-.75,-1.39,;3.32,-1.68,;4.41,-2.77,;5.89,-2.37,;6.29,-.89,;7.78,-.49,;5.2,.2,;3.72,-.19,)|
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2cc(=O)n(cc12)-c1cccc2CNCCc12
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2cc(=O)n(cc12)-c1cccc2OCCOc12
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2cc(=O)n(cc12)-c1ncccc1F
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2cc(=O)n(cc12)C1CCCCC1
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2cc(=O)n(cc12)C1CCOC1
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2cc(=O)n(Cc3ccccc3)cc12
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2cc(=O)n(CC3CCCCC3)cc12
CC(c1ccccc1C(F)(F)F)n1cc2c(n[nH]c2cc1=O)-c1ccc(cc1)N1CCN(C)CC1
CC(c1ccccc1)n1cc2c(n[nH]c2cc1=O)-c1ccc(cc1)N1CCN(C)CC1
CN1CCC(C1=O)n1cc2c(n[nH]c2cc1=O)-c1ccc(cc1)N1CCN(C)CC1
CC1OCCCC1n1cc2c(n[nH]c2cc1=O)-c1ccc(cc1)N1CCN(C)CC1
NC(=O)c1ccc2cc(Cc3cc(ccn3)C(=O)NCc3cc4c(Cl)c[nH]c4cc3F)ccc2n1
Cc1cc(N)nc(C)c1CNC(=O)c1ccnc(Cc2ccc3nc(ccc3c2)C(N)=O)c1
Nc1nccc2cc(CNC(=O)c3ccnc(Cc4ccc5nc(ccc5c4)C#N)c3)ccc12
NC(=O)c1ccc2cc(Cc3cc(ccn3)C(=O)NCc3ccc4c(N)nccc4c3)ccc2n1
Fc1cc2[nH]cc(Cl)c2cc1CNC(=O)c1ccnc(Cc2ccc3ncc(cc3c2)C#N)c1
Nc1nccc2cc(CNC(=O)c3ccnc(Cc4ccc5ncc(cc5c4)C#N)c3)ccc12
Cc1cc(N)nc(C)c1CNC(=O)c1ccnc(Cc2ccc3ncc(cc3c2)C#N)c1
Nc1nccc2cc(CNC(=O)c3ccnc(Cc4cnc5ccc(F)cc5n4)c3)ccc12
CC(=O)NCc1ccc2cc(Cc3cc(ccn3)C(=O)NCc3cc4c(Cl)c[nH]c4cc3F)ccc2n1
CC(=O)NCc1ccc2cc(Cc3cc(ccn3)C(=O)NCc3ccc4c(N)nccc4c3)ccc2n1
CC(=O)NCc1ccc2cc(Cc3cc(ccn3)C(=O)NCc3c(C)cc(N)nc3C)ccc2n1
CS(=O)(=O)c1ccc2ncc(Cc3cc(ccn3)C(=O)NCc3cc4c(Cl)c[nH]c4cc3F)cc2c1
CS(=O)(=O)c1ccc2ncc(Cc3cc(ccn3)C(=O)NCc3ccc4c(N)nccc4c3)cc2c1
Cc1cc(N)nc(C)c1CNC(=O)c1ccnc(Cc2cnc3ccc(cc3c2)S(C)(=O)=O)c1
Cc1cnc2c(cc(Cc3cc(ccn3)C(=O)NCc3c(C)cc(N)nc3C)cc2c1)S(C)(=O)=O
Cc1cnc2c(cc(Cc3cc(ccn3)C(=O)NCc3ccc4c(N)nccc4c3)cc2c1)S(C)(=O)=O
Cc1cnc2c(cc(Cc3cc(ccn3)C(=O)NCc3cc4c(Cl)c[nH]c4cc3F)cc2c1)S(C)(=O)=O
Cc1cnc2c(cc(Cc3cc(ccn3)C(=O)NCc3cc4cc[nH]c4cc3F)cc2c1)S(C)(=O)=O
Cc1cnc2c(cc(Cc3cc(ccn3)C(=O)NCc3cnc4[nH]cc(Cl)c4c3)cc2c1)S(C)(=O)=O
Cc1cnc2c(cc(Cc3cc(ccn3)C(=O)NCc3n[nH]c4ccc(Cl)cc34)cc2c1)S(C)(=O)=O
Cc1cnc2c(cc(Cc3cc(ccn3)C(=O)NCc3ccc4[nH]cc(Cl)c4c3F)cc2c1)S(C)(=O)=O
Cc1cc(N)nc(C)c1CNC(=O)c1ccnc(Cn2ccc3c(Cl)cccc3c2=O)c1
Cc1cc(N)nc(C)c1CNC(=O)c1ccnc(Cn2ccc3cc(Cl)ccc3c2=O)c1
Cc1cc(N)nc(C)c1CNC(=O)c1ccnc(Cc2ccc3[nH]cc(Cl)c3c2)c1
Cc1c[nH]c2ccc(Cc3cc(ccn3)C(=O)NCc3c(C)cc(N)nc3C)cc12
Cc1nc(N)c(cc1CNC(=O)c1ccnc(Cc2ccc3ncc(Cl)cc3c2)c1)C#N
Cc1nc(N)c(cc1CNC(=O)c1ccnc(Cc2ccc3ncc(Cl)cc3c2)c1)C(N)=O
Cc1nc(N)c(Cl)cc1CNC(=O)c1ccnc(Cc2ccc3ncc(Cl)cc3c2)c1
Cc1cc(N)ncc1CNC(=O)c1ccnc(Cc2ccc3ncc(Cl)cc3c2)c1
Nc1ccc(CNC(=O)c2ccnc(Cc3ccc4ncc(Cl)cc4c3)c2)c(n1)C(F)(F)F
Nc1nccc2cc(CNC(=O)c3ccnc(Cc4ccc5ncc(Cl)cc5c4)c3)ccc12
Fc1cc2[nH]ncc2cc1CNC(=O)c1ccnc(Cc2ccc3ncc(Cl)cc3c2)c1
Fc1cc2[nH]cc(Cl)c2cc1CNC(=O)c1ccnc(Cc2ccc3ncc(Cl)cc3c2)c1
Cc1nc(N)ccc1CNC(=O)c1ccnc(Cc2ccc3ncc(Cl)cc3c2)c1
Cc1cc(N)nc(C)c1CNC(=O)c1ccnc(Cc2ccc3ncc(Cl)cc3c2)c1
Nc1noc2cc(CNC(=O)c3ccnc(Cc4ccc5ncc(Cl)cc5c4)c3)ccc12
Clc1ccc2[nH]nc(CNC(=O)c3ccnc(Cc4ccc5ncc(Cl)cc5c4)c3)c2c1
Clc1c[nH]c2ncc(CNC(=O)c3ccnc(Cc4ccc5ncc(Cl)cc5c4)c3)cc12
Fc1c(CNC(=O)c2ccnc(Cc3ccc4ncc(Cl)cc4c3)c2)ccc2[nH]cc(Cl)c12
Fc1cc2[nH]ccc2cc1CNC(=O)c1ccnc(Cc2ccc3ncc(Cl)cc3c2)c1
CNc1ccc(CNC(=O)c2ccnc(Cc3ccc4ncc(Cl)cc4c3)c2)c(C)n1
Nc1ccc(CNC(=O)c2ccnc(Cc3ccc4ncc(Cl)cc4c3)c2)c(n1)C1CC1
CN(C)c1ccc(CNC(=O)c2ccnc(Cc3ccc4ncc(Cl)cc4c3)c2)c(C)n1
NCc1ccc2cc(Cc3cc(ccn3)C(=O)NCc3cc4c(Cl)c[nH]c4cc3F)ccc2n1
Cc1cc(N)nc(C)c1CNC(=O)c1ccnc(Cc2ccc3nc(CN)ccc3c2)c1
Cc1cnc2ccc(Cc3cc(ccn3)C(=O)NCc3ccc4c(N)noc4c3)cc2c1
Cc1ccc2ncc(Cc3cc(ccn3)C(=O)NCc3ccc4c(N)noc4c3)cc2c1
Fc1cc2[nH]cc(Cl)c2cc1CNC(=O)c1ccnc(Cc2cc(C#N)c3ncc(Cl)cc3c2)c1
Cc1cc(N)nc(C)c1CNC(=O)c1ccnc(Cc2cc(C#N)c3ncc(Cl)cc3c2)c1
Fc1c(CNC(=O)c2ccnc(Cc3cc(C#N)c4ncc(Cl)cc4c3)c2)ccc2[nH]cc(Cl)c12
Fc1cc2[nH]ccc2cc1CNC(=O)c1ccnc(Cc2cc(C#N)c3ncc(Cl)cc3c2)c1
Cc1cc(N)ncc1CNC(=O)c1ccnc(Cc2cc(C#N)c3ncc(Cl)cc3c2)c1
Clc1ccc2[nH]nc(CNC(=O)c3ccnc(Cc4cc(C#N)c5ncc(Cl)cc5c4)c3)c2c1
Clc1c[nH]c2ncc(CNC(=O)c3ccnc(Cc4cc(C#N)c5ncc(Cl)cc5c4)c3)cc12
Cc1nc(N)ccc1CNC(=O)c1ccnc(Cc2cc(C#N)c3ncc(Cl)cc3c2)c1
Nc1nccc2cc(CNC(=O)c3ccnc(Cc4cc(C#N)c5ncc(Cl)cc5c4)c3)ccc12
Cc1cc(N)nc(C)c1CNC(=O)c1ccnc(Cc2cc(C(N)=O)c3ncc(Cl)cc3c2)c1
Cc1cc2[nH]cc(Cl)c2cc1CNC(=O)c1ccnc(Cc2cc(C(N)=O)c3ncc(Cl)cc3c2)c1
NC(=O)c1cc(Cc2cc(ccn2)C(=O)NCc2n[nH]c3ccc(Cl)cc23)cc2cc(Cl)cnc12
NC(=O)c1cc(Cc2cc(ccn2)C(=O)NCc2cnc3[nH]cc(Cl)c3c2)cc2cc(Cl)cnc12
Cc1nc(N)ccc1CNC(=O)c1ccnc(Cc2cc(C(N)=O)c3ncc(Cl)cc3c2)c1
Cc1cc(N)ncc1CNC(=O)c1ccnc(Cc2cc(C(N)=O)c3ncc(Cl)cc3c2)c1
NC(=O)c1cc(Cc2cc(ccn2)C(=O)NCc2ccc3c(N)nccc3c2)cc2cc(Cl)cnc12
NC(=O)c1cc(Cc2cc(ccn2)C(=O)NCc2ccc3[nH]cc(Cl)c3c2F)cc2cc(Cl)cnc12
NC(=O)c1cc(Cc2cc(ccn2)C(=O)NCc2cc3cc[nH]c3cc2F)cc2cc(Cl)cnc12
Cc1cc(N)nc(C)c1CNC(=O)c1ccnc(Cc2cc(c3ncc(Cl)cc3c2)S(C)(=O)=O)c1
CS(=O)(=O)c1cc(Cc2cc(ccn2)C(=O)NCc2cc3c(Cl)c[nH]c3cc2F)cc2cc(Cl)cnc12
Cc1nc(N)ccc1CNC(=O)c1ccnc(Cc2cc(c3ncc(Cl)cc3c2)S(C)(=O)=O)c1
Cc1cnc2c(cc(Cc3cc(ccn3)C(=O)NCc3c(C)cc(N)nc3C)cc2c1)C#N
Cc1cnc2c(cc(Cc3cc(ccn3)C(=O)NCc3ccc4c(N)nccc4c3)cc2c1)C#N
Cc1cnc2c(cc(Cc3cc(ccn3)C(=O)NCc3cc4c(Cl)c[nH]c4cc3F)cc2c1)C#N
Cc1cnc2c(cc(Cc3cc(ccn3)C(=O)NCc3cnc4[nH]cc(Cl)c4c3)cc2c1)C#N
Cc1cnc2c(cc(Cc3cc(ccn3)C(=O)NCc3ccc4[nH]cc(Cl)c4c3F)cc2c1)C#N
Cc1cnc2c(cc(Cc3cc(ccn3)C(=O)NCc3n[nH]c4ccc(Cl)cc34)cc2c1)C#N
Cc1cnc2c(cc(Cc3cc(ccn3)C(=O)NCc3cc4cc[nH]c4cc3F)cc2c1)C#N
Cc1cnc2c(cc(Cc3cc(ccn3)C(=O)NCc3c(C)cc(N)nc3C)cc2c1)C(N)=O
Cc1cnc2c(cc(Cc3cc(ccn3)C(=O)NCc3cc4c(Cl)c[nH]c4cc3F)cc2c1)C(N)=O
Cc1cnc2c(cc(Cc3cc(ccn3)C(=O)NCc3ccc4c(N)nccc4c3)cc2c1)C(N)=O
Cc1cnc2c(cc(Cc3cc(ccn3)C(=O)NCc3cnc4[nH]cc(Cl)c4c3)cc2c1)C(N)=O
Cc1cnc2c(cc(Cc3cc(ccn3)C(=O)NCc3ccc4[nH]cc(Cl)c4c3F)cc2c1)C(N)=O
Cc1cnc2c(cc(Cc3cc(ccn3)C(=O)NCc3n[nH]c4ccc(Cl)cc34)cc2c1)C(N)=O
Cc1cnc2c(cc(Cc3cc(ccn3)C(=O)NCc3cc4cc[nH]c4cc3F)cc2c1)C(N)=O
Cc1cnc2c(cc(Cc3cc(ccn3)C(=O)NCc3c(C)cc(N)nc3C)cc2c1)C(O)=O
Cc1cc(N)ncc1CNC(=O)c1ccnc(Cn2cc3cc(Cl)ccc3cc2=O)c1
Cc1nc(N)ccc1CNC(=O)c1ccnc(Cn2cc3cc(Cl)ccc3cc2=O)c1
Cc1cc(N)nc(C)c1CNC(=O)c1ccnc(Cn2cc3cc(Cl)ccc3cc2=O)c1
Fc1cc2[nH]cc(Cl)c2cc1CNC(=O)c1ccnc(Cn2cc3cc(Cl)ccc3cc2=O)c1
Cc1cc(N)nc(C)c1CNC(=O)c1ccnc(Cc2cc(F)c3ncc(Cl)cc3c2)c1
Fc1cc2[nH]cc(Cl)c2cc1CNC(=O)c1ccnc(Cc2cc(F)c3ncc(Cl)cc3c2)c1
Cc1nc(N)ccc1CNC(=O)c1ccnc(Cc2cc(F)c3ncc(Cl)cc3c2)c1
COC(=O)c1cc(Cc2cc(ccn2)C(=O)NCc2c(C)cc(N)nc2C)cc2cc(Cl)cnc12
Cc1cc(N)nc(C)c1CNC(=O)c1ccnc(Cc2cc(C(O)=O)c3ncc(Cl)cc3c2)c1
Cc1cc(N)nc(C)c1CNC(=O)c1ccnc(Cc2cc(CO)c3ncc(Cl)cc3c2)c1
COC(=O)c1cc(Cc2cc(ccn2)C(=O)NCc2ccc(N)nc2C)cc2cc(Cl)cnc12
Cc1nc(N)ccc1CNC(=O)c1ccnc(Cc2cc(C(O)=O)c3ncc(Cl)cc3c2)c1
Cc1nc(N)ccc1CNC(=O)c1ccnc(Cc2cc(CO)c3ncc(Cl)cc3c2)c1
Cc1cc(N)[n+]([O-])c(C)c1CNC(=O)c1ccnc(Cc2ccc3ncc(Cl)cc3c2)c1
Cc1cc(N)nc(C)c1CNC(=O)c1ccnc(Cc2ccc3[n+]([O-])cc(Cl)cc3c2)c1
Cc1cc(N)nc(C)c1CNC(=O)c1ccnc(Cc2cc(Cl)c3ncc(Cl)cc3c2)c1
Cc1nc(N)ccc1CNC(=O)c1ccnc(Cc2cc(Cl)c3ncc(Cl)cc3c2)c1
Cc1cc(N)nc(C)c1CNC(=O)c1ccnc(Cc2ccc3ncc(Cl)cc3c2F)c1
Cc1nc(N)ccc1CNC(=O)c1ccnc(Cc2ccc3ncc(Cl)cc3c2F)c1
Cc1cc(cc(Cc2ccc3ncc(Cl)cc3c2)n1)C(=O)NCc1c(C)cc(N)nc1C
Cc1cc(N)nc(C)c1CNC(=O)c1ccnc(Cn2ncc3cc(Cl)ccc23)c1
Cc1cc(N)nc(C)c1CNC(=O)c1ccnc(Cn2cc3cc(Cl)ccc3n2)c1
Cc1ccc2nn(Cc3cc(ccn3)C(=O)NCc3c(C)cc(N)nc3C)cc2c1
Cc1ccc2n(Cc3cc(ccn3)C(=O)NCc3c(C)cc(N)nc3C)ncc2c1
Cc1ccc2nc(c(Cc3cc(ccn3)C(=O)NCc3cc4c(Cl)c[nH]c4cc3F)cc2c1)S(C)(=O)=O
Cc1ccc2cc(Cc3cc(ccn3)C(=O)NCc3cc4c(Cl)c[nH]c4cc3F)ccc2n1
Cc1ccc2cc(Cc3cc(ccn3)C(=O)NCc3ccc4c(N)nccc4c3)ccc2n1
Cc1ccc2cc(Cc3cc(ccn3)C(=O)NCc3ccc(N)nc3C)ccc2n1
Cc1ccc2cc(Cc3cc(ccn3)C(=O)NCc3c(C)cc(N)nc3C)ccc2n1
Cc1ccc2ncc(Cc3cc(ccn3)C(=O)NCc3c(C)cc(N)nc3C)cc2c1
Cc1ccc2ncc(Cc3cc(ccn3)C(=O)NCc3ccc4c(N)nccc4c3)cc2c1
Cc1ccc2ncc(Cc3cc(ccn3)C(=O)NCc3cc4c(Cl)c[nH]c4cc3F)cc2c1
Cc1ccc2ncc(Cc3cc(ccn3)C(=O)NCc3ccc(N)nc3C)cc2c1
Nc1nccc2cc(CNC(=O)c3ccnc(Cc4cnc5ccc(F)cc5c4)c3)ccc12
Cc1cc(N)nc(C)c1CNC(=O)c1ccnc(Cc2cnc3ccc(F)cc3c2)c1
Fc1ccc2ncc(Cc3cc(ccn3)C(=O)NCc3cc4c(Cl)c[nH]c4cc3F)cc2c1
Cc1nc(N)ccc1CNC(=O)c1ccnc(Cc2cnc3ccc(F)cc3c2)c1
Cc1cc(N)nc(C)c1CNC(=O)c1ccnc(Cc2cnc3cc(F)ccc3c2)c1
Fc1ccc2cc(Cc3cc(ccn3)C(=O)NCc3cc4c(Cl)c[nH]c4cc3F)cnc2c1
Nc1nccc2cc(CNC(=O)c3ccnc(Cc4cnc5cc(F)ccc5c4)c3)ccc12
Fc1cc2[nH]cc(Cl)c2cc1CNC(=O)c1ccnc(Cc2cnc3ccccc3c2)c1
Fc1cc2[nH]cc(Cl)c2cc1CNC(=O)c1ccnc(Cc2cnc3ccc(Cl)cc3c2)c1
Cc1ccc2ccc(Cc3cc(ccn3)C(=O)NCc3ccc4c(N)nccc4c3)cc2n1
Cc1ccc2ccc(Cc3cc(ccn3)C(=O)NCc3cc4c(Cl)c[nH]c4cc3F)cc2n1
Cc1ccc2ccc(Cc3cc(ccn3)C(=O)NCc3c(C)cc(N)nc3C)cc2n1
Fc1cc2[nH]cc(Cl)c2cc1CNC(=O)c1ccnc(Cc2ccc3nc(ccc3c2)C#N)c1
Cc1cc(N)nc(C)c1CNC(=O)c1ccnc(Cc2ccc3nc(ccc3c2)C#N)c1
Cc1cc2cc(Cc3cc(ccn3)C(=O)NCc3ccc4c(N)nccc4c3)ccc2cn1
Cc1cc2cc(Cc3cc(ccn3)C(=O)NCc3cc4c(Cl)c[nH]c4cc3F)ccc2cn1
CS(=O)(=O)c1ccc2cc(Cc3cc(ccn3)C(=O)NCc3ccc4c(N)nccc4c3)ccc2n1
CS(=O)(=O)c1ccc2cc(Cc3cc(ccn3)C(=O)NCc3cc4c(Cl)c[nH]c4cc3F)ccc2n1
Nc1nccc2cc(CNC(=O)c3ccnc(Cc4ccc5nccc(C#N)c5c4)c3)ccc12
Fc1cc2[nH]cc(Cl)c2cc1CNC(=O)c1ccnc(Cc2ccc3nccc(C#N)c3c2)c1
Cc1cc(N)nc(C)c1CNC(=O)c1ccnc(Cc2ccc3nccc(C#N)c3c2)c1
Nc1nccc2cc(CNC(=O)c3ccnc(Cc4cnc5cc(Cl)ccc5c4)c3)ccc12
Fc1cc2[nH]cc(Cl)c2cc1CNC(=O)c1ccnc(Cc2cnc3cc(Cl)ccc3c2)c1
Cc1cc(N)nc(C)c1CNC(=O)c1ccnc(Cc2cnc3cc(Cl)ccc3c2)c1
Cc1cnc2ccc(Cc3cc(ccn3)C(=O)NCc3ccc4c(N)nccc4c3)cc2c1
Cc1cnc2ccc(Cc3cc(ccn3)C(=O)NCc3cc4c(Cl)c[nH]c4cc3F)cc2c1
Cc1cnc2ccc(Cc3cc(ccn3)C(=O)NCc3c(C)cc(N)nc3C)cc2c1
Cc1cc2cc(Cc3cc(ccn3)C(=O)NCc3c(C)cc(N)nc3C)ccc2cn1
NCc1ccc2cc(Cc3cc(ccn3)C(=O)NCc3ccc4c(N)nccc4c3)ccc2n1
Cc1cc(N)nc(C)c1CNC(=O)c1ccnc(Cc2cc3cc(Cl)ccc3[nH]2)c1
Cc1cc(N)nc(C)c1CNC(=O)c1ccnc(Cc2cc3cc(Cl)cnc3cn2)c1
Cc1nc(N)ccc1CNC(=O)c1ccnc(Cc2cc3cc(Cl)cnc3cn2)c1
Cc1cc(N)nc(C)c1CNC(=O)c1ccnc(Cc2cnc3[nH]c(Cl)cc3c2)c1
Cc1cc(N)nc(C)c1CNC(=O)c1ccnc(Cc2cc3cc(ccc3[nH]2)C(F)(F)F)c1
Cc1cc(N)nc(C)c1CNC(=O)c1ccnc(Cc2cnc3[nH]c(cc3c2)C(F)(F)F)c1
Cc1cc(N)nc(C)c1CNC(=O)c1ccnc(Cc2cc3cc(Cl)cn3cn2)c1
Clc1ccc2nnc(CNC(=O)c3ccnc(Cc4ccc5ncc(Cl)cc5c4)c3)n2c1
Cc1ccn2nnc(CNC(=O)c3ccnc(Cc4ccc5ncc(Cl)cc5c4)c3)c2c1
Cc1ccn2cnc(CNC(=O)c3ccnc(Cc4ccc5ncc(Cl)cc5c4)c3)c2c1
Clc1ccc2ncc(CNC(=O)c3ccnc(Cc4ccc5ncc(Cl)cc5c4)c3)n2c1
Cc1nc(CNC(=O)c2ccnc(Cc3ccc4ncc(Cl)cc4c3)c2)c2cc(C)ccn12
Cc1nc(CNC(=O)c2ccnc(Cc3ccc4ncc(cc4c3)C(F)(F)F)c2)c2cc(C)ccn12
Cc1ccn2c(nc(CNC(=O)c3ccnc(Cc4ccc5ncc(Cl)cc5c4)c3)c2c1)C(F)(F)F
Cc1nc2NCCc2cc1CNC(=O)c1ccnc(Cc2ccc3ncc(Cl)cc3c2)c1
Cc1nc2NCCc2cc1CNC(=O)c1ccnc(Cc2ccc3ncc(cc3c2)C(F)(F)F)c1
Cc1nc2CNCc2cc1CNC(=O)c1ccnc(Cc2ccc3ncc(Cl)cc3c2)c1
Cc1nc2CNCc2cc1CNC(=O)c1ccnc(Cc2ccc3ncc(cc3c2)C(F)(F)F)c1
Cc1nc(N)cc(c1CNC(=O)c1ccnc(Cc2ccc3ncc(Cl)cc3c2)c1)C(F)(F)F
COc1cc(N)nc(C)c1CNC(=O)c1ccnc(Cc2ccc3ncc(Cl)cc3c2)c1
Cc1nc(N)cc(C#N)c1CNC(=O)c1ccnc(Cc2ccc3ncc(Cl)cc3c2)c1
NCc1ccc(CNC(=O)c2ccnc(Cc3ccc4ncc(Cl)cc4c3)c2)cc1
NCc1ccc(CNC(=O)c2ccnc(Cc3ccc4ncc(Cl)cc4c3)c2)cn1
NCc1ccc(CNC(=O)c2ccnc(Cc3ccc4ncc(Cl)cc4c3)c2)nc1
Cc1cc(CN)nc(C)c1CNC(=O)c1ccnc(Cc2ccc3ncc(Cl)cc3c2)c1
Cc1cc(CN)nc(C)c1CNC(=O)c1ccnc(Cc2ccc3ncc(cc3c2)C(F)(F)F)c1
CC(N)c1cc(C)c(CNC(=O)c2ccnc(Cc3ccc4ncc(Cl)cc4c3)c2)c(C)n1
Cc1cc(nc(C)c1CNC(=O)c1ccnc(Cc2ccc3ncc(cc3c2)C(F)(F)F)c1)C(C)(C)O
Cc1nc2NCCc2c(C)c1CNC(=O)c1ccnc(Cc2ccc3ncc(Cl)cc3c2)c1
Cc1nc2NCCc2c(C)c1CNC(=O)c1ccnc(Cc2ccc3ncc(cc3c2)C(F)(F)F)c1
Cc1c(CNC(=O)c2ccnc(Cc3ccc4ncc(Cl)cc4c3)c2)ccc2c(N)nccc12
Nc1nccc2c(F)c(CNC(=O)c3ccnc(Cc4ccc5ncc(Cl)cc5c4)c3)ccc12
Nc1nccc2cc(CNC(=O)c3ccnc(Cc4ccc5ncc(Cl)cc5c4)c3)c(F)cc12
Cc1cc2c(N)nccc2cc1CNC(=O)c1ccnc(Cc2ccc3ncc(Cl)cc3c2)c1
Nc1nccc2cc(CNC(=O)c3ccnc(Cc4ccc5ncc(cc5c4)C(F)(F)F)c3)c(F)cc12
Cc1cc2c(N)nccc2cc1CNC(=O)c1ccnc(Cc2ccc3ncc(cc3c2)C(F)(F)F)c1
Cc1c(CNC(=O)c2ccnc(Cc3ccc4ncc(cc4c3)C(F)(F)F)c2)ccc2c(N)nccc12
FC(F)(F)c1ncc2ccc(CNC(=O)c3ccnc(Cc4ccc5ncc(Cl)cc5c4)c3)cn12
Nc1nc(n2cc(CNC(=O)c3ccnc(Cc4ccc5ncc(Cl)cc5c4)c3)ccc12)C(F)(F)F
Nc1ncc2cc(CNC(=O)c3ccnc(Cc4ccc5ncc(Cl)cc5c4)c3)ccn12
Cc1cc2cncn2cc1CNC(=O)c1ccnc(Cc2ccc3ncc(Cl)cc3c2)c1
Cc1c(CNC(=O)c2ccnc(Cc3ccc4ncc(Cl)cc4c3)c2)cnc2[nH]cc(Cl)c12
Cc1cc2[nH]cc(Cl)c2cc1CNC(=O)c1ccnc(Cc2ccc3ncc(Cl)cc3c2)c1
Cc1nc2[nH]cc(Cl)c2cc1CNC(=O)c1ccnc(Cc2ccc3ncc(Cl)cc3c2)c1
Cc1nc2[nH]cc(Cl)c2c(C)c1CNC(=O)c1ccnc(Cc2ccc3ncc(Cl)cc3c2)c1
CC(=O)Nc1cc(C)c(CNC(=O)c2ccnc(Cc3ccc4ncc(Cl)cc4c3)c2)c(C)n1
Cc1cc(C)c(CNC(=O)c2ccnc(Cc3ccc4ncc(Cl)cc4c3)c2)c(C)n1
Cc1nc2NCCCc2c(C)c1CNC(=O)c1ccnc(Cc2ccc3ncc(Cl)cc3c2)c1
Cc1cc(N)nc(C)c1CNC(=O)c1cc(Cc2ccc3ncc(Cl)cc3c2)nc(c1)-c1n[nH]c(=O)[nH]1
CC1=CC2C=NN(Cc3cc(ccn3)C(=O)NCc3c(C)cc(N)nc3C)C2C=C1 |c:4,31,t:1|
Cc1cc(N)nc(C)c1CNC(=O)c1ccnc(Cn2cc3cc(Cl)cnc3n2)c1
Cc1cc(N)nc(C)c1CNC(=O)c1ccnc(Cc2cnc3ncc(Cl)cc3c2)c1
Cc1nc(N)ccc1CNC(=O)c1ccnc(Cc2cnc3ncc(Cl)cc3c2)c1
Clc1cnc2ccc(Cc3cc(ccn3)C(=O)NCc3ccc4ncc(Cl)cn34)cc2c1
Cc1cc(N)nc(C)c1CNC(=O)c1cc(Cc2ccc3ncc(Cl)cc3c2)nc(c1)C#N
Cc1cc(N)nc(C)c1CNC(=O)c1cc(Cc2ccc3ncc(Cl)cc3c2)nc(c1)C(N)=O
Cc1cc(N)nc(C)c1CNC(=O)c1cc(Cc2ccc3ncc(Cl)cc3c2)nc(c1)C(O)=O
Cc1cc(N)nc(C)c1CNC(=O)c1cc(Cc2ccc3ncc(Cl)cc3c2)nc(c1)C(C)(C)O
Cc1cc(N)nc(C)c1CNC(=O)c1cc(CN)nc(Cc2ccc3ncc(Cl)cc3c2)c1
Cc1cc(N)nc(C)c1CNC(=O)c1cc(CO)nc(Cc2ccc3ncc(Cl)cc3c2)c1
Cc1cc(N)nc(C)c1CNC(=O)c1cc(CC#N)nc(Cc2ccc3ncc(Cl)cc3c2)c1
Cc1cc(N)nc(C)c1CNC(=O)c1cc(CC(N)=O)nc(Cc2ccc3ncc(Cl)cc3c2)c1
Cc1cc(N)nc(C)c1CNC(=O)c1ccnc(Cc2cc3cc(cnc3[nH]2)C(F)(F)F)c1
Cc1nc(N)ccc1CNC(=O)c1cc(Cc2cnc3ncc(Cl)cc3c2)ncc1C#N
Cc1cc(N)nc(C)c1CNC(=O)c1ccnc(Cc2cc(N)c3ncc(Cl)cc3c2)c1
Cc1nc(N)ccc1CNC(=O)c1ccnc(Cc2cc(N)c3ncc(Cl)cc3c2)c1
Cc1cc(N)nc(C)c1CNC(=O)c1ccnc(Cc2cc(c3ncc(Cl)cc3c2)C(C)(C)O)c1
Cc1nc(N)ccc1CNC(=O)c1ccnc(Cc2cc(c3ncc(Cl)cc3c2)C(C)(C)O)c1
CC(C)(O)c1cc(Cc2cc(ccn2)C(=O)NCc2cc3c(Cl)c[nH]c3cc2F)cc2cc(Cl)cnc12
CC(C)(O)c1cc(Cc2cc(ccn2)C(=O)NCc2ccc3[nH]cc(Cl)c3c2F)cc2cc(Cl)cnc12
CC(C)(O)c1cc(Cc2cc(ccn2)C(=O)NCc2cnc3[nH]cc(Cl)c3c2)cc2cc(Cl)cnc12
CC(C)(O)c1cc(Cc2cc(ccn2)C(=O)NCc2ccc3c(N)nccc3c2)cc2cc(Cl)cnc12
CC(C)(O)c1cc(Cc2cc(ccn2)C(=O)NCc2n[nH]c3ccc(Cl)cc23)cc2cc(Cl)cnc12
Cc1cc(N)nc(C)c1CNC(=O)c1ccnc(Cc2cnc3cc(F)c(Cl)cc3c2)c1
Cc1nc(N)ccc1CNC(=O)c1ccnc(Cc2cnc3cc(F)c(Cl)cc3c2)c1
Cc1cc(N)nc(C)c1CNC(=O)c1ccnc(Cc2ccc3ncc(cc3c2)C(F)(F)F)c1
Cc1nc(N)ccc1CNC(=O)c1ccnc(Cc2ccc3ncc(cc3c2)C(F)(F)F)c1
Fc1nc2[nH]cc(Cl)c2cc1CNC(=O)c1ccnc(Cc2ccc3ncc(cc3c2)C(F)(F)F)c1
FC(F)(F)c1cnc2ccc(Cc3cc(ccn3)C(=O)NCc3cnc4[nH]cc(Cl)c4c3)cc2c1
Nc1nccc2cc(CNC(=O)c3ccnc(Cc4ccc5ncc(cc5c4)C(F)(F)F)c3)ccc12
FC(F)(F)c1cnc2ccc(Cc3cc(ccn3)C(=O)NCc3n[nH]c4ccc(Cl)cc34)cc2c1
Fc1c(CNC(=O)c2ccnc(Cc3ccc4ncc(cc4c3)C(F)(F)F)c2)ccc2[nH]cc(Cl)c12
Cc1cc(N)nc(C)c1CNC(=O)c1ccnc(Cc2cc(c3ncc(Cl)cc3c2)S(N)(=O)=O)c1
Cc1nc(N)ccc1CNC(=O)c1ccnc(Cc2cc(c3ncc(Cl)cc3c2)S(N)(=O)=O)c1
CC(NC(=O)c1ccnc(Cc2ccc3ncc(Cl)cc3c2)c1)c1ccc(N)nc1C
Cc1cc(N)nc(C)c1CNC(=O)c1ccnc(Cc2ccc3nc(C)c(Cl)cc3c2)c1
Cc1nc2ccc(Cc3cc(ccn3)C(=O)NCc3ccc(N)nc3C)cc2cc1Cl
Cc1cc(N)nc(C)c1CNC(=O)c1ccnc(Cc2cccc(c2)-c2noc(=O)[nH]2)c1
Cc1cc(N)nc(C)c1CNC(=O)c1ccnc(Cc2cc(CN)c3ncc(Cl)cc3c2)c1
COCCNc1ccc(CNC(=O)c2ccnc(Cc3ccc4ncc(Cl)cc4c3)c2)c(C)n1
Cc1cc(N)nc(C)c1CNC(=O)c1ccnc(Cc2ccc3ncc(cc3c2)C2CC2)c1
Cc1nc(N)ccc1CNC(=O)c1ccnc(Cc2ccc3ncc(cc3c2)C2CC2)c1
Fc1cc2[nH]cc(Cl)c2cc1CNC(=O)c1ccnc(Cc2ccc3ncc(cc3c2)C2CC2)c1
Clc1c[nH]c2ncc(CNC(=O)c3ccnc(Cc4ccc5ncc(cc5c4)C4CC4)c3)cc12
Nc1nccc2cc(CNC(=O)c3ccnc(Cc4ccc5ncc(cc5c4)C4CC4)c3)ccc12
Fc1c(CNC(=O)c2ccnc(Cc3ccc4ncc(cc4c3)C3CC3)c2)ccc2[nH]cc(Cl)c12
Clc1ccc2[nH]nc(CNC(=O)c3ccnc(Cc4ccc5ncc(cc5c4)C4CC4)c3)c2c1
Cc1cc(N)nc(C)c1CNC(=O)c1ccnc(Cc2ccc3ncc(cc3c2)C(N)=O)c1
Cc1nc(N)ccc1CNC(=O)c1ccnc(Cc2ccc3ncc(cc3c2)C(N)=O)c1
Cc1nc(NCCO)ccc1CNC(=O)c1ccnc(Cc2ccc3ncc(Cl)cc3c2)c1
Cc1nc(N)ccc1CNC(=O)c1ccnc(Cc2cc(CN)c3ncc(Cl)cc3c2)c1
CC(C)c1cnc2ccc(Cc3cc(ccn3)C(=O)NCc3c(C)cc(N)nc3C)cc2c1
CCCc1cnc2ccc(Cc3cc(ccn3)C(=O)NCc3c(C)cc(N)nc3C)cc2c1
Clc1cnc2ccc(Cc3cc(ccn3)C(=O)NCc3cnc4ncc(Cl)cn34)cc2c1
Cc1cc(N)nc(C)c1CNC(=O)c1ccnc(Cc2ccc3ncc(CO)cc3c2)c1
Cc1nc(N)ccc1CNC(=O)c1ccnc(Cc2ccc3ncc(CO)cc3c2)c1
Cc1n[nH]c2ccc(CNC(=O)c3ccnc(Cc4ccc5ncc(Cl)cc5c4)c3)cc12
CC(O)c1cnc2ccc(Cc3cc(ccn3)C(=O)NCc3c(C)cc(N)nc3C)cc2c1
CC(O)c1cnc2ccc(Cc3cc(ccn3)C(=O)NCc3ccc(N)nc3C)cc2c1
COc1cnc2ccc(Cc3cc(ccn3)C(=O)NCc3c(C)cc(N)nc3C)cc2c1
COc1cnc2ccc(Cc3cc(ccn3)C(=O)NCc3ccc(N)nc3C)cc2c1
Cc1n[nH]c2ncc(CNC(=O)c3ccnc(Cc4ccc5ncc(Cl)cc5c4)c3)cc12
FC(F)(F)c1n[nH]c2ccc(CNC(=O)c3ccnc(Cc4ccc5ncc(Cl)cc5c4)c3)cc12
Clc1ccc2[nH]cc(CNC(=O)c3ccnc(Cc4ccc5ncc(Cl)cc5c4)c3)c2c1
Clc1cnc2[nH]cc(CNC(=O)c3ccnc(Cc4ccc5ncc(Cl)cc5c4)c3)c2c1
Cc1[nH]c2ccc(Cl)cc2c1CNC(=O)c1ccnc(Cc2ccc3ncc(Cl)cc3c2)c1
FC(F)(F)c1n[nH]c2ncc(CNC(=O)c3ccnc(Cc4ccc5ncc(Cl)cc5c4)c3)cc12
Cc1cc(N)nc(C)c1CNC(=O)c1ccnc(Cc2cc(-c3nnn[nH]3)c3ncc(Cl)cc3c2)c1
Cc1nc(N)ccc1CNC(=O)c1ccnc(Cc2cc(-c3nnn[nH]3)c3ncc(Cl)cc3c2)c1
Cc1cc(N)nc(C)c1CNC(=O)c1ccnc(c1)C(=O)c1ccc2ncc(Cl)cc2c1
Cc1cc(N)nc(C)c1CNC(=O)c1ccnc(c1)C(O)c1ccc2ncc(Cl)cc2c1
Cc1cc(N)nc(C)c1CNC(=O)c1ccnc(c1)C(N)c1ccc2ncc(Cl)cc2c1
Cc1cc(N)nc(C)c1CNC(=O)c1ccnc(c1)C(C)(O)c1ccc2ncc(Cl)cc2c1
Cc1cc(N)nc(C)c1CNC(=O)c1ccnc(Cc2ccc3ncc(CC(F)F)cc3c2)c1
Cc1nc(N)ccc1CNC(=O)c1ccnc(Cc2ccc3ncc(CC(F)F)cc3c2)c1
CCc1cnc2ccc(Cc3cc(ccn3)C(=O)NCc3cc4c(Cl)c[nH]c4cc3F)cc2c1
CCc1cnc2ccc(Cc3cc(ccn3)C(=O)NCc3cnc4[nH]cc(Cl)c4c3)cc2c1
CCc1cnc2ccc(Cc3cc(ccn3)C(=O)NCc3ccc4[nH]cc(Cl)c4c3F)cc2c1
CCc1cnc2ccc(Cc3cc(ccn3)C(=O)NCc3ccc4c(N)nccc4c3)cc2c1
CCc1cnc2ccc(Cc3cc(ccn3)C(=O)NCc3n[nH]c4ccc(Cl)cc34)cc2c1
CCc1cnc2ccc(Cc3cc(ccn3)C(=O)NCc3ccc(N)nc3C)cc2c1
CCc1cnc2ccc(Cc3cc(ccn3)C(=O)NCc3c(C)cc(N)nc3C)cc2c1
Cc1cnc2c(cc(Cc3cc(ccn3)C(=O)NCc3cc4c(Cl)c[nH]c4cc3F)cc2c1)S(N)(=O)=O
Cc1cnc2c(cc(Cc3cc(ccn3)C(=O)NCc3n[nH]c4ccc(Cl)cc34)cc2c1)S(N)(=O)=O
Cc1cnc2c(cc(Cc3cc(ccn3)C(=O)NCc3ccc4c(N)nccc4c3)cc2c1)S(N)(=O)=O
Cc1cnc2c(cc(Cc3cc(ccn3)C(=O)NCc3ccc4[nH]cc(Cl)c4c3F)cc2c1)S(N)(=O)=O
Cc1cnc2c(cc(Cc3cc(ccn3)C(=O)NCc3cnc4[nH]cc(Cl)c4c3)cc2c1)S(N)(=O)=O
Fc1cc2[nH]cc(Cl)c2cc1CNC(=O)c1ccnc(Cc2ccc3ncc(cc3c2)N2CCOCC2)c1
Nc1nccc2cc(CNC(=O)c3ccnc(Cc4ccc5ncc(cc5c4)N4CCOCC4)c3)ccc12
Clc1c[nH]c2ncc(CNC(=O)c3ccnc(Cc4ccc5ncc(cc5c4)N4CCOCC4)c3)cc12
Clc1ccc2[nH]nc(CNC(=O)c3ccnc(Cc4ccc5ncc(cc5c4)N4CCOCC4)c3)c2c1
COC(c1ccc2ncc(Cl)cc2c1)c1cc(ccn1)C(=O)NCc1c(C)cc(N)nc1C
Nc1cnc2ccc(Cc3cc(ccn3)C(=O)NCc3cc4c(Cl)c[nH]c4cc3F)cc2c1
Nc1cnc2ccc(Cc3cc(ccn3)C(=O)NCc3ccc4c(N)nccc4c3)cc2c1
Nc1cnc2ccc(Cc3cc(ccn3)C(=O)NCc3n[nH]c4ccc(Cl)cc34)cc2c1
Nc1cnc2ccc(Cc3cc(ccn3)C(=O)NCc3cnc4[nH]cc(Cl)c4c3)cc2c1
Nc1cnc2ccc(Cc3cc(ccn3)C(=O)NCc3ccc4[nH]cc(Cl)c4c3F)cc2c1
Fc1cc2[nH]cc(Cl)c2cc1CNC(=O)c1ccnc(Cc2ccc3ncc(cc3c2)N2CCCCC2)c1
Nc1nccc2cc(CNC(=O)c3ccnc(Cc4ccc5ncc(cc5c4)N4CCCCC4)c3)ccc12
Fc1c(CNC(=O)c2ccnc(Cc3ccc4ncc(cc4c3)N3CCCCC3)c2)ccc2[nH]cc(Cl)c12
Clc1c[nH]c2ncc(CNC(=O)c3ccnc(Cc4ccc5ncc(cc5c4)N4CCCCC4)c3)cc12
Fc1cc2[nH]cc(Cl)c2cc1CNC(=O)c1ccnc(Cc2ccc3ncc(cc3c2)N2CCCC2)c1
Nc1nccc2cc(CNC(=O)c3ccnc(Cc4ccc5ncc(cc5c4)N4CCCC4)c3)ccc12
Clc1ccc2[nH]nc(CNC(=O)c3ccnc(Cc4ccc5ncc(cc5c4)N4CCCC4)c3)c2c1
Clc1c[nH]c2ncc(CNC(=O)c3ccnc(Cc4ccc5ncc(cc5c4)N4CCCC4)c3)cc12
Fc1c(CNC(=O)c2ccnc(Cc3ccc4ncc(cc4c3)N3CCCC3)c2)ccc2[nH]cc(Cl)c12
Clc1ccc2[nH]nc(CNC(=O)c3ccnc(Cc4ccc5ncc(cc5c4)N4CCNCC4)c3)c2c1
Fc1cc2[nH]cc(Cl)c2cc1CNC(=O)c1ccnc(Cc2ccc3ncc(cc3c2)N2CCNCC2)c1
Cc1cnc2c(cc(Cc3cc(ccn3)C(=O)NCc3cc4c(Cl)c[nH]c4cc3F)cc2c1)C(C)(C)O
Cc1cnc2c(cc(Cc3cc(ccn3)C(=O)NCc3ccc4[nH]cc(Cl)c4c3F)cc2c1)C(C)(C)O
Cc1cnc2c(cc(Cc3cc(ccn3)C(=O)NCc3cnc4[nH]cc(Cl)c4c3)cc2c1)C(C)(C)O
Cc1cnc2c(cc(Cc3cc(ccn3)C(=O)NCc3n[nH]c4ccc(Cl)cc34)cc2c1)C(C)(C)O
Cc1cnc2c(cc(Cc3cc(ccn3)C(=O)NCc3c(C)cc(N)nc3C)cc2c1)C(C)(C)O
Cc1cnc2c(cc(Cc3cc(ccn3)C(=O)NCc3ccc4c(N)nccc4c3)cc2c1)C(C)(C)O
Fc1cc2[nH]cc(Cl)c2cc1CNC(=O)c1ccnc(Cc2ccc3ncc(cc3c2)N2CCC2)c1
COc1cccc(F)c1-c1cc2c(NC(=O)c3ccccc3)n[nH]c2cn1
COc1cccc(F)c1-c1cc2c(NC(=O)c3ccc(C)cc3)n[nH]c2cn1
COc1cccc(F)c1-c1cc2c(NC(=O)c3ccc(Br)cc3)n[nH]c2cn1
COc1cccc(F)c1-c1cc2c(NC(=O)c3cccc(Br)c3)n[nH]c2cn1
COc1cccc(F)c1-c1cc2c(NC(=O)c3ccc(F)cc3)n[nH]c2cn1
COc1cccc(F)c1-c1cc2c(NC(=O)c3cccc(F)c3)n[nH]c2cn1
COc1cccc(F)c1-c1cc2c(NC(=O)c3cccc(c3)C#N)n[nH]c2cn1
CCc1ccc(cc1)C(=O)Nc1n[nH]c2cnc(cc12)-c1c(F)cccc1OC
COc1cccc(c1)C(=O)Nc1n[nH]c2cnc(cc12)-c1c(F)cccc1OC
COc1cccc(F)c1-c1cc2c(NC(=O)c3ccc(F)c(C)c3)n[nH]c2cn1
COc1cccc(F)c1-c1cc2c(NC(=O)c3cc(F)cc(F)c3)n[nH]c2cn1
COc1cccc(F)c1-c1cc2c(NC(=O)c3ccc(F)c(F)c3)n[nH]c2cn1
COc1cccc(F)c1-c1cc2c(NC(=O)c3ccc4OCOc4c3)n[nH]c2cn1
COc1cccc(F)c1-c1cc2c(NC(=O)c3cnn(C)c3)n[nH]c2cn1
COc1cccc(F)c1-c1cc2c(NC(=O)c3ccn(C)n3)n[nH]c2cn1
COc1cccc(F)c1-c1cc2c(NC(=O)c3cccc(c3)N3CCOCC3)n[nH]c2cn1
COc1cccc(F)c1-c1cc2c(NC(=O)c3cccc(c3)N3CCNC(=O)C3)n[nH]c2cn1
COc1cccc(F)c1-c1cc2c(NC(=O)c3cccc(c3)N3CCN(C)CC3)n[nH]c2cn1
COc1cccc(F)c1-c1cc2c(NC(=O)c3cccc(c3)N3CCN(C)C(=O)C3)n[nH]c2cn1
CCN1CCN(CC1)c1cccc(c1)C(=O)Nc1n[nH]c2cnc(cc12)-c1c(F)cccc1OC
COc1cccc(F)c1-c1cc2c(NC(=O)c3cccc(c3)N3CCN(CC(F)(F)F)C(=O)C3)n[nH]c2cn1
COc1cccc(F)c1-c1cc2c(NC(=O)c3cccc(c3)N3CCN(CC3)S(C)(=O)=O)n[nH]c2cn1
COc1cccc(F)c1-c1cc2c(NC(=O)c3cccc(c3)N3CCNCC3)n[nH]c2cn1
COc1cccc(F)c1-c1cc2c(NC(=O)c3ccc(cc3)N3CCOCC3)n[nH]c2cn1
COc1cccc(F)c1-c1cc2c(NC(=O)c3ccc(cc3)N3CCNC(=O)C3)n[nH]c2cn1
COc1cccc(F)c1-c1cc2c(NC(=O)c3ccc(cc3)N3CCN(C)CC3)n[nH]c2cn1
COc1cccc(F)c1-c1cc2c(NC(=O)c3ccc(cc3)N3CCN(C)C(=O)C3)n[nH]c2cn1
CCN1CCN(CC1)c1ccc(cc1)C(=O)Nc1n[nH]c2cnc(cc12)-c1c(F)cccc1OC
COc1cccc(F)c1-c1cc2c(NC(=O)c3ccc(cc3)N3CCN(CC(F)(F)F)C(=O)C3)n[nH]c2cn1
COc1cccc(F)c1-c1cc2c(NC(=O)c3ccc(cc3)N3CCN(CC3)C(C)C)n[nH]c2cn1
COc1cccc(F)c1-c1cc2c(NC(=O)c3ccc(cc3)N3CCN(C4CC4)C(=O)C3)n[nH]c2cn1
COc1cccc(F)c1-c1cc2c(NC(=O)c3ccc(cc3)N3CCN(CC3)S(C)(=O)=O)n[nH]c2cn1
COc1cccc(F)c1-c1cc2c(NC(=O)c3ccc(cc3)N3CCNCC3)n[nH]c2cn1
COc1cccc(F)c1-c1cc2c(n[nH]c2cn1)-c1cnc(s1)N1CCOCC1
COc1cccc(F)c1-c1cc2c(n[nH]c2cn1)-c1cc(C)no1
COc1cccc(F)c1-c1cc2c(n[nH]c2cn1)-c1cnc(C)s1
COc1cccc(F)c1-c1cc2c(n[nH]c2cn1)N1CCN(C(=O)C1)c1ccc(Br)cc1
COc1cccc(F)c1-c1cc2c(n[nH]c2cn1)N1CCc2ccc(cc2C1)C#N
COc1cccc(F)c1-c1cc2c(n[nH]c2cn1)N1CCN(CC1)c1ccc(cc1)C#N
COc1cccc(F)c1-c1cc2c(n[nH]c2cn1)N1CCN(CC1)c1ccncc1
COc1cccc(F)c1-c1cc2c(NCc3ccc(cc3)N3CCN(C)CC3)n[nH]c2cn1
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2cnc(cc12)-c1cc(F)cc(c1)C1(CN)CC1
COc1cccc(F)c1-c1cc2c(n[nH]c2cn1)-c1ccc(cc1)N1CCN(C)CC1
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2cnc(cc12)-c1c(F)cccc1F
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2cnc(cc12)-c1c(C)cccc1C
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2cnc(cc12)-c1c(F)cc(F)cc1F
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2cnc(cc12)-c1c(F)cccc1Cl
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2cnc(cc12)-c1c(F)cc(O)cc1F
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2cnc(cc12)-c1c(C)cccc1F
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2cnc(cc12)-c1c(Cl)cccc1C(F)(F)F
CCOc1cccc(F)c1-c1cc2c(n[nH]c2cn1)-c1ccc(cc1)N1CCN(C)CC1
COc1cccc(Cl)c1-c1cc2c(n[nH]c2cn1)-c1ccc(cc1)N1CCN(C)CC1
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2cnc(cc12)-c1c(F)cccc1C(F)(F)F
COc1cccc(F)c1-c1cc2c(n[nH]c2cn1)C(=O)Nc1ccc(cc1)N1CCN(C)CC1
COc1cccc(F)c1-c1cc2c(n[nH]c2cn1)C(=O)Nc1ccc(cc1)N1CCOCC1
CCN1CCN(CC1)c1ccc(NC(=O)c2n[nH]c3cnc(cc23)-c2c(F)cccc2OC)cc1
COCCNC(=O)c1cc(F)c(c(F)c1)-c1cc2c(n[nH]c2cn1)-c1cnn(C)c1
COC1CN(C1)C(=O)c1cc(F)c(c(F)c1)-c1cc2c(n[nH]c2cn1)-c1cnn(C)c1
Cn1cc(cn1)-c1n[nH]c2cnc(cc12)-c1c(F)ccc(NC(=O)C2CCC2)c1F
Cn1cc(cn1)-c1n[nH]c2cnc(cc12)-c1c(F)ccc(NC(=O)Cc2ccccc2)c1F
CNc1ccc(F)c(-c2cc3c(n[nH]c3cn2)-c2cnn(C)c2)c1F
CN(C)c1ccc(F)c(-c2cc3c(n[nH]c3cn2)-c2cnn(C)c2)c1F
CN(C)c1cc(F)c(c(F)c1)-c1cc2c(n[nH]c2cn1)-c1cnn(C)c1
Cn1cc(cn1)-c1n[nH]c2cnc(cc12)-c1c(F)cc(NC(=O)CN2CCCC2)cc1F
Cn1cc(cn1)C(=O)Nc1cc(F)c(c(F)c1)-c1cc2c(n[nH]c2cn1)-c1cnn(C)c1
Cn1cc(cn1)-c1n[nH]c2cnc(cc12)-c1c(F)cc(NC(=O)CC2CCCC2)cc1F
Cn1cc(cn1)-c1n[nH]c2cnc(cc12)-c1c(F)cc(NC(=O)Cc2cccnc2)cc1F
Cn1cc(cn1)-c1n[nH]c2cnc(cc12)-c1c(F)cc(NC(=O)CN2C3CCC2CC3)cc1F
Cn1cc(cn1)-c1n[nH]c2cnc(cc12)-c1c(F)cc(NC(=O)CN2CC3(C2)CCOCC3)cc1F
CC(N1CCCC1)C(=O)Nc1cc(F)c(c(F)c1)-c1cc2c(n[nH]c2cn1)-c1cnn(C)c1
COCCNC(=O)Nc1cc(F)c(c(F)c1)-c1cc2c(n[nH]c2cn1)-c1cnn(C)c1
Cn1cc(cn1)-c1n[nH]c2cnc(cc12)-c1c(F)cc(NC(=O)CN2CCC2)cc1OC(F)F
Cn1cc(cn1)-c1n[nH]c2cnc(cc12)-c1c(F)cc(NC(=O)CN2CCCC2)cc1Cl
COc1cc(NC(=O)CN2CCCC2)cc(F)c1-c1cc2c(n[nH]c2cn1)-c1cnn(C)c1
COc1cc(NC(=O)CN2CC(C)(C)C2)cc(F)c1-c1cc2c(n[nH]c2cn1)-c1cnn(C)c1
COc1cc(NC(=O)OC2CCN(C)CC2)cc(F)c1-c1cc2c(n[nH]c2cn1)-c1cnn(C)c1
Cn1cc(cn1)-c1n[nH]c2cnc(cc12)-c1c(F)cc(NC(=O)CN2CCC2)c(F)c1F
CN(C)CC(=O)Nc1cc(C)c(c(Cl)c1)-c1cc2c(n[nH]c2cn1)-c1cnn(C)c1
Cc1cc(NC(=O)CN2C[C@H]3CC[C@@H]2C3)ccc1-c1cc2c(n[nH]c2cn1)-c1cnn(C)c1 |r|
Cc1cc(NC(=O)CN2CCCC2)cc(F)c1-c1cc2c(n[nH]c2cn1)-c1cnn(C)c1
CN(C)CC(=O)Nc1cc(C)c(c(F)c1)-c1cc2c(n[nH]c2cn1)-c1cnn(C)c1
Cc1cc(NC(=O)CN2C3CCC2CC3)cc(F)c1-c1cc2c(n[nH]c2cn1)-c1cnn(C)c1
Cc1cc(NC(=O)CN2C[C@H]3CC[C@@H]2C3)cc(F)c1-c1cc2c(n[nH]c2cn1)-c1cnn(C)c1 |r|
CN(C)CCC(=O)Nc1cc(C)c(c(F)c1)-c1cc2c(n[nH]c2cn1)-c1cnn(C)c1
Cc1cc(NC(=O)CC#N)cc(F)c1-c1cc2c(n[nH]c2cn1)-c1cnn(C)c1
CNCc1cccc(c1C)-c1cc2c(n[nH]c2cn1)-c1cnn(C)c1
CNCc1ccc(C)c(c1)-c1cc2c(n[nH]c2cn1)-c1cnn(C)c1
CNCc1cccc(-c2cc3c(n[nH]c3cn2)-c2cnn(C)c2)c1C(F)(F)F
Cn1cc(cn1)-c1n[nH]c2cnc(cc12)-c1cccc(CN2CCC2)c1C(F)(F)F
Cn1cc(cn1)-c1n[nH]c2cnc(cc12)-c1cccc(CNC2CCOCC2)c1C(F)(F)F
CC(C)NCc1cccc(-c2cc3c(n[nH]c3cn2)-c2cnn(C)c2)c1C(F)(F)F
CNCc1ccc(F)c(c1C)-c1cc2c(n[nH]c2cn1)-c1cnn(C)c1
CC(C)NCc1ccc(F)c(c1C)-c1cc2c(n[nH]c2cn1)-c1cnn(C)c1
Cc1c(CN2CCC2)ccc(F)c1-c1cc2c(n[nH]c2cn1)-c1cnn(C)c1
CC(C)NC1CC(C1)c1cc(F)c(c(F)c1)-c1cc2c(n[nH]c2cn1)-c1cnn(C)c1 |(-3.59,8.47,;-3.59,6.93,;-4.92,6.16,;-2.25,6.16,;-2.25,4.62,;-1.16,3.53,;-2.25,2.44,;-3.34,3.53,;-2.25,.9,;-.92,.13,;-.92,-1.41,;.41,-2.18,;-2.25,-2.18,;-3.59,-1.41,;-4.92,-2.18,;-3.59,.13,;-2.25,-3.72,;-.92,-4.49,;-.92,-6.03,;.23,-7.06,;-.4,-8.47,;-1.93,-8.31,;-2.25,-6.8,;-3.59,-6.03,;-3.59,-4.49,;1.73,-6.74,;2.88,-7.77,;4.21,-7,;3.89,-5.49,;4.92,-4.35,;2.36,-5.33,)|
CNCCc1cc(F)c(c(F)c1)-c1cc2c(n[nH]c2cn1)-c1cnn(C)c1
CNCCc1ccc(F)c(c1F)-c1cc2c(n[nH]c2cn1)-c1cnn(C)c1
Cn1cc(cn1)-c1n[nH]c2cnc(cc12)-c1c(F)ccc(CCNC2CCOCC2)c1F
CC(C)N1CC(C1)NCCc1cc(F)c(c(F)c1)-c1cc2c(n[nH]c2cn1)-c1cnn(C)c1
CNC(=O)c1ccc(cc1F)-c1n[nH]c2cnc(cc12)-c1c(F)cccc1OC
CNC(=O)c1ccc(cn1)-c1n[nH]c2cnc(cc12)-c1c(F)cccc1OC
CNC(=O)c1ccc(cc1OC)-c1n[nH]c2cnc(cc12)-c1c(F)cccc1OC
CNC(=O)c1ccc(cc1C)-c1n[nH]c2cnc(cc12)-c1c(F)cccc1OC
COc1cccc(F)c1-c1cc2c(n[nH]c2cn1)-n1cnc(c1)C(=O)NC(C)C
CNC(=O)c1cn(cn1)-c1n[nH]c2cnc(cc12)-c1c(F)cccc1OC
Cn1cc(cn1)-c1n[nH]c2cnc(cc12)-c1c(F)cc(OCC2CCN2)cc1F
Cn1cc(cn1)-c1n[nH]c2cnc(cc12)-c1c(F)cc(OC2CCOCC2)cc1F
Cn1cc(cn1)-c1n[nH]c2cnc(cc12)-c1c(F)cc(OCc2ccncc2)cc1F
CN(C)C(=O)Oc1cc(F)c(c(F)c1)-c1cc2c(n[nH]c2cn1)-c1cnn(C)c1
Cn1cc(cn1)-c1n[nH]c2cnc(cc12)-c1c(F)cc(OC(=O)N2CCOCC2)cc1F
CNCc1ccc(c(C)c1)-c1cc2c(n[nH]c2cn1)-c1cnn(C)c1
CNCc1ccc(-c2cc3c(n[nH]c3cn2)-c2cnn(C)c2)c(c1)C(F)(F)F
CNCc1cc(C)c(c(F)c1)-c1cc2c(n[nH]c2cn1)-c1ccc(nc1)N1CCC(O)C1
CNCc1cc(C)c(c(F)c1)-c1cc2c(n[nH]c2cn1)-c1ccc(nc1)N1CCCC(C1)OC
COc1cccc(F)c1-c1cc2c(n[nH]c2cn1)-c1cccc(n1)C1CCN(C)CC1
COc1cccc(F)c1-c1cc2c(\C=C\c3ccc(Br)cc3)n[nH]c2cn1
CNCc1cc(C)c(c(F)c1)-c1cc2c(n[nH]c2cn1)-c1cccc(n1)N1CCOCC1
CCN(C)c1cccc(n1)-c1n[nH]c2cnc(cc12)-c1c(C)cc(CNC)cc1F
CNCc1cc(F)c(-c2cc3c(n[nH]c3cn2)-c2ccc(nc2)N2CCN(C)CC2)c(c1)C(F)(F)F
CNCc1cc(F)c(-c2cc3c(n[nH]c3cn2)-c2ccc(nc2)C2CC2)c(c1)C(F)(F)F
CNCc1cc(F)c(-c2cc3c(n[nH]c3cn2)-c2ccc(nc2)N2CCOCC2)c(c1)C(F)(F)F
CNCc1cc(F)c(c(F)c1)-c1cc2c(n[nH]c2cn1)-c1cnn(C)c1
CC(C)NCc1cc(F)c(c(F)c1)-c1cc2c(n[nH]c2cn1)-c1cnn(C)c1
Cn1cc(cn1)-c1n[nH]c2cnc(cc12)-c1c(F)cc(CNc2ccccn2)cc1F
Cn1ccc(NCc2cc(F)c(c(F)c2)-c2cc3c(n[nH]c3cn2)-c2cnn(C)c2)n1
Cn1cc(cn1)-c1n[nH]c2cnc(cc12)-c1c(F)cc(CNCCO)cc1F
CNCc1ccc(F)c(c1F)-c1cc2c(n[nH]c2cn1)-c1cnn(C)c1
CC(C)NCc1ccc(F)c(-c2cc3c(n[nH]c3cn2)-c2cnn(C)c2)c1F
Cn1cc(cn1)-c1n[nH]c2cnc(cc12)-c1c(F)ccc(CNC2CC2)c1F
COC1CCCN(Cc2ccc(F)c(c2F)-c2cc3c(n[nH]c3cn2)-c2cnn(C)c2)C1
CNCc1cc(F)c(-c2cc3c(n[nH]c3cn2)-c2cnn(C)c2)c(c1)C(F)(F)F
CNCc1cc(F)c(-c2cc3c(n[nH]c3cn2)-c2ccc(cc2)N2CCN(C)CC2)c(c1)C(F)(F)F
CCn1cc(cn1)-c1n[nH]c2cnc(cc12)-c1c(C)cc(CNC)cc1F
CNCc1cc(C)c(c(F)c1)-c1cc2c(n[nH]c2cn1)-c1cnn(c1)C1CC1
CNCc1cc(C)c(c(F)c1)-c1cc2c(n[nH]c2cn1)-c1cnn(c1)-c1ccccc1C#N
CNCc1cc(C)c(c(F)c1)-c1cc2c(n[nH]c2cn1)-c1cnn(c1)C1CCOCC1
CNC1(CC1)c1cc(F)c(c(F)c1)-c1cc2c(n[nH]c2cn1)-c1cnn(C)c1
CNCc1ccc(F)c(-c2cc3c(n[nH]c3cn2)-c2cnn(C)c2)c1OC
CCNCc1ccc(F)c(-c2cc3c(n[nH]c3cn2)-c2cnn(C)c2)c1OC
CC(C)NCc1cc(F)c(c(F)c1)-c1cc2c(NC(=O)c3ccc(cc3)N3CCN(C)CC3)n[nH]c2cn1
CN1CCN(CC1)c1ccc(cc1)C(=O)Nc1n[nH]c2cnc(cc12)-c1c(F)cc(CN2CCCC2)cc1F
CN1CCN(CC1)c1ccc(cc1)C(=O)Nc1n[nH]c2cnc(cc12)-c1c(F)cc(CN2CCC2)cc1F
COC1CN(Cc2cc(F)c(c(F)c2)-c2cc3c(NC(=O)c4ccc(cc4)N4CCN(C)CC4)n[nH]c3cn2)C1
CNCc1cc(F)c(c(F)c1)-c1cc2c(NC(=O)c3cnn(C)c3)n[nH]c2cn1
CNCc1cc(F)c(c(F)c1)-c1cc2c(NC(=O)c3cccc(c3)N3CCN(C)CC3)n[nH]c2cn1
COc1cccc(c1)C(=O)Nc1n[nH]c2cnc(cc12)-c1c(F)cc(CNC(C)C)cc1F
COC(=O)N1CCN(CC1)c1ccc(cc1)C(=O)Nc1n[nH]c2cnc(cc12)-c1c(F)cc(CNC(C)C)cc1F
COC(=O)N1CCN(CC1)c1ccc(C(=O)Nc2n[nH]c3cnc(cc23)-c2c(F)cc(CNC(C)C)cc2F)c(F)c1
COc1cc(ccc1C(=O)Nc1n[nH]c2cnc(cc12)-c1c(F)cc(CNC(C)C)cc1F)N1CCN(C)CC1
CC(C)NCc1cc(F)c(c(F)c1)-c1cc2c(NC(=O)c3cccc(N4CCN(C)CC4)c3F)n[nH]c2cn1
CC(C)NCc1cc(F)c(c(F)c1)-c1cc2c(NC(=O)c3ccc(F)c(c3)N3CCN(C)CC3)n[nH]c2cn1
CN1CCN(CC1)c1ccc(cc1)C(=O)Nc1n[nH]c2cnc(cc12)-c1c(C)cccc1F
CN1CCN(CC1)c1ccc(cc1)C(=O)Nc1n[nH]c2cnc(cc12)-c1c(F)cccc1C(F)(F)F
CCNCc1cc(F)c(-c2cc3c(NC(=O)c4ccc(cc4)N4CCN(C)CC4)n[nH]c3cn2)c(c1)C(F)(F)F
CC(C)NCc1cc(F)c(c(F)c1)-c1cc2c(n[nH]c2cn1)C(=O)Nc1ccc(cc1)N1CCN(C)CC1
CN1CCN(CC1)c1ccc(cc1)C(=O)Nc1n[nH]c2cnc(cc12)-c1c(F)cc(NC(=O)CN2CCCC2)cc1F
CN1CCN(CC1)c1ccc(C(=O)Nc2n[nH]c3cnc(cc23)-c2c(C)cccc2F)c(N)c1
CC(O)CNc1cc(ccc1C(=O)Nc1n[nH]c2cnc(cc12)-c1c(C)cccc1F)N1CCN(C)CC1
CN1CCN(CC1)c1ccc(C(=O)Nc2n[nH]c3cnc(cc23)-c2c(C)cccc2F)c(NCc2ccnn2C)c1
CN1CCN(CC1)c1ccc(C(=O)Nc2n[nH]c3cnc(cc23)-c2c(C)cccc2F)c(NC2CCC(C2)C#N)c1
CNCc1cc(F)c(c(F)c1)-c1cc2c(n[nH]c2cn1)-c1cnn(c1)-c1ccccc1C#N
CNCc1cc(F)c(c(F)c1)-c1cc2c(n[nH]c2cn1)-c1cnn(c1)C1CNC1
CNCc1cc(F)c(c(F)c1)-c1cc2c(n[nH]c2cn1)-c1ccnc(c1)N1CCN(C)CC1
CNCc1cc(F)c(c(F)c1)-c1cc2c(n[nH]c2cn1)-c1cnn(CCO)c1
CNCc1cc(F)c(c(F)c1)-c1cc2c(n[nH]c2cn1)-c1ccc(OC)cc1
CNCc1cc(F)c(c(F)c1)-c1cc2c(n[nH]c2cn1)-c1ccc(nc1)N1CCC(O)CC1
CNCc1cc(F)c(c(F)c1)-c1cc2c(n[nH]c2cn1)-c1ccc(cn1)N1CCC(F)C1
CNCc1cc(C)c(c(F)c1)-c1cc2c(n[nH]c2cn1)-c1cnn(C)c1
CNCc1cc(C)c(c(F)c1)-c1cc2c(n[nH]c2cn1)-c1ccc(cc1)C(=O)NC
CNC(=O)c1ccc(cc1)-c1n[nH]c2cnc(cc12)-c1c(C)cc(cc1F)C1CCCN1
Cc1cc(cc(F)c1-c1cc2c(n[nH]c2cn1)-c1cnn(C)c1)C1CCCN1
CN1CCCC1c1cc(C)c(c(F)c1)-c1cc2c(n[nH]c2cn1)-c1cnn(C)c1
Cc1cc(cc(F)c1-c1cc2c(n[nH]c2cn1)-c1cnn(C)c1)C1CCCCN1
CCNCc1cc(C)c(c(F)c1)-c1cc2c(n[nH]c2cn1)-c1cnn(C)c1
Cc1cc(CNC2CC2)cc(F)c1-c1cc2c(n[nH]c2cn1)-c1cnn(C)c1
CC(C)NCc1cc(C)c(c(F)c1)-c1cc2c(n[nH]c2cn1)-c1cnn(C)c1
Cc1cc(CNCC(F)(F)F)cc(F)c1-c1cc2c(n[nH]c2cn1)-c1cnn(C)c1
Cc1cc(CNCCO)cc(F)c1-c1cc2c(n[nH]c2cn1)-c1cnn(C)c1
Cc1cc(CNC2CC(O)C2)cc(F)c1-c1cc2c(n[nH]c2cn1)-c1cnn(C)c1 |(.63,.45,;-.71,1.22,;-.71,2.76,;-2.04,3.53,;-2.04,5.07,;-.71,5.84,;.63,5.07,;1.02,3.58,;2.51,3.98,;3.85,3.21,;2.11,5.47,;-3.38,2.76,;-3.38,1.22,;-4.71,.45,;-2.04,.45,;-2.04,-1.09,;-.71,-1.86,;-.71,-3.4,;.44,-4.43,;-.19,-5.84,;-1.72,-5.68,;-2.04,-4.17,;-3.38,-3.4,;-3.38,-1.86,;1.92,-4.03,;3.17,-4.94,;4.42,-4.03,;3.94,-2.57,;4.71,-1.23,;2.4,-2.57,)|
Cc1cc(CN2CCC2)cc(F)c1-c1cc2c(n[nH]c2cn1)-c1cnn(C)c1
Cc1cc(CN2CCC(O)C2)cc(F)c1-c1cc2c(n[nH]c2cn1)-c1cnn(C)c1
Cc1cc(CNCC(C)(C)O)cc(F)c1-c1cc2c(n[nH]c2cn1)-c1cnn(C)c1
COC1CN(Cc2cc(C)c(c(F)c2)-c2cc3c(n[nH]c3cn2)-c2cnn(C)c2)C1
Cc1cc(CNCc2cn(C)cn2)cc(F)c1-c1cc2c(n[nH]c2cn1)-c1cnn(C)c1
Cc1cc(CNCc2cocn2)cc(F)c1-c1cc2c(n[nH]c2cn1)-c1cnn(C)c1
Cc1cc(CNCC#N)cc(F)c1-c1cc2c(n[nH]c2cn1)-c1cnn(C)c1
CNC(C)c1cc(C)c(c(F)c1)-c1cc2c(n[nH]c2cn1)-c1cnn(C)c1
CC(=O)NCc1cc(C)c(c(F)c1)-c1cc2c(n[nH]c2cn1)-c1cnn(C)c1
COC(=O)NCc1cc(C)c(c(F)c1)-c1cc2c(n[nH]c2cn1)-c1cnn(C)c1
CNCc1cc(F)c(c(OC(F)F)c1)-c1cc2c(n[nH]c2cn1)-c1ccc(cn1)N1CCN(CC1)C(C)=O
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2cnc(cc12)-c1c(F)cccc1CC#N
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2cnc(cc12)-c1c(F)cccc1CN
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2cnc(cc12)-c1c(F)cccc1CO
CNC1CCc2c1cc(F)c(-c1cc3c(n[nH]c3cn1)-c1ccc(cc1)N1CCN(C)CC1)c2F
CNC1CCc2c1cc(F)c(c2F)-c1cc2c(n[nH]c2cn1)-c1cnn(C)c1
CNC1CCc2cc(F)c(-c3cc4c(n[nH]c4cn3)-c3ccc(cc3)N3CCN(C)CC3)c(F)c2C1
CNC1CCc2cc(F)c(-c3cc4c(n[nH]c4cn3)-c3cnn(C)c3)c(F)c2C1
CNC1CCCc2c(F)c(c(F)cc12)-c1cc2c(n[nH]c2cn1)-c1ccc(cc1)C(=O)NC
CNC1CCCc2c(F)c(c(F)cc12)-c1cc2c(n[nH]c2cn1)-c1cnn(C)c1
CN1CCN(CC1)c1ccc(cn1)-c1n[nH]c2cnc(cc12)-c1c(F)cc2C(N)CCCc2c1F
CNC1CCc2cc(F)c(-c3cc4c(n[nH]c4cn3)-c3ccc(cc3)C(=O)NC)c(F)c12
CNC1CCc2cc(F)c(-c3cc4c(n[nH]c4cn3)-c3ccc(cc3)N3CCN(C)CC3)c(F)c12
COc1c2C(N)CCc2cc(F)c1-c1cc2c(n[nH]c2cn1)-c1ccc(cc1)N1CCN(C)CC1
COc1c2C(N)CCc2cc(F)c1-c1cc2c(n[nH]c2cn1)-c1cnn(C)c1
CNC1CCCc2c1ccc(F)c2-c1cc2c(n[nH]c2cn1)-c1ccc(nc1)C(=O)NC
CNC1CCCc2c1ccc(F)c2-c1cc2c(n[nH]c2cn1)-c1ccc(cc1)N1CCN(C)CC1
Cn1cc(cn1)-c1n[nH]c2cnc(cc12)-c1c(F)ccc2C(N)CCCc12
CN1CCN(CC1)c1ncc(cn1)-c1n[nH]c2cnc(cc12)-c1c(F)cc(CC#N)cc1F
Cn1cc(cn1)-c1n[nH]c2cnc(cc12)-c1c(F)cc2CCC(O)c2c1F
CN1CCN(CC1)c1ccc(cn1)-c1n[nH]c2cnc(cc12)-c1c(F)cc2CCC(O)c2c1F
CNC1CCc2cc(F)c(c(F)c2C1)-c1ncc2[nH]nc(-c3cnn(C)c3)c2c1OC |(1.57,5.64,;.08,6.04,;-1.01,4.95,;-2.5,5.35,;-3.59,4.26,;-3.19,2.77,;-4.28,1.68,;-3.88,.2,;-4.97,-.89,;-2.39,-.2,;-1.3,.89,;.18,.49,;-1.7,2.37,;-.61,3.46,;-1.99,-1.69,;-3.08,-2.78,;-2.68,-4.27,;-1.2,-4.67,;-.5,-6.04,;1.02,-5.8,;1.26,-4.28,;2.6,-3.51,;4.06,-3.98,;4.97,-2.74,;4.06,-1.49,;4.83,-.16,;2.6,-1.97,;-.11,-3.58,;-.51,-2.09,;.58,-1,;2.07,-1.4,)|
CNCc1cc(F)c(c(F)c1)-c1ncc2[nH]nc(-c3cnn(C)c3)c2c1OC |(-1.01,5.29,;-2.5,5.69,;-3.59,4.6,;-3.19,3.12,;-4.28,2.03,;-3.88,.54,;-4.97,-.55,;-2.39,.14,;-1.3,1.23,;.18,.83,;-1.7,2.72,;-1.99,-1.35,;-3.08,-2.43,;-2.68,-3.92,;-1.2,-4.32,;-.5,-5.69,;1.02,-5.45,;1.26,-3.93,;2.6,-3.16,;4.06,-3.64,;4.97,-2.39,;4.06,-1.15,;4.83,.19,;2.6,-1.62,;-.11,-3.23,;-.51,-1.74,;.58,-.66,;2.07,-1.05,)|
Cn1cc(cn1)-c1n[nH]c2cnc(c(F)c12)-c1c(F)cc2CCC(N)c2c1F |(4.82,.45,;4.05,-.88,;2.59,-1.36,;2.59,-2.9,;4.05,-3.38,;4.96,-2.13,;1.25,-3.67,;1.01,-5.19,;-.51,-5.43,;-1.21,-4.06,;-2.7,-3.66,;-3.09,-2.17,;-2,-1.08,;-.52,-1.48,;.57,-.39,;-.12,-2.97,;-2.4,.4,;-3.87,.88,;-4.96,-.21,;-4.19,2.39,;-3.04,3.42,;-3.04,4.96,;-1.58,5.43,;-.67,4.19,;.87,4.19,;-1.58,2.94,;-1.26,1.43,;.23,1.03,)|
CNCc1cc(F)c(c(F)c1)-c1cc2c(n[nH]c2cn1)-c1cnc(nc1)N1CCN(C)CC1
CNCc1cc(F)c(c(F)c1)-c1cc2c(n[nH]c2cn1)-c1cnc(nc1)N1CCC(O)CC1
CNCc1cc(F)c(c(F)c1)-c1cc2c(n[nH]c2cn1)-c1cncc(c1)N1CCN(C)CC1
CNC1CCc2c1cc(C)c(c2F)-c1cc2c(n[nH]c2cn1)-c1cnn(C)c1
Cc1c(CN2CC(C)(C)C2)ccc(F)c1-c1cc2c(n[nH]c2cn1)-c1cnn(C)c1
CO[C@H]1C[C@@H](C1)NCc1ccc(F)c(c1C)-c1cc2c(n[nH]c2cn1)-c1cnn(C)c1 |r,wU:4.6,wD:2.1,(5.63,6.39,;5.63,4.85,;4.3,4.08,;2.79,4.47,;2.39,2.98,;3.88,2.59,;1.06,2.21,;-.28,2.98,;-1.61,2.21,;-2.94,2.98,;-4.28,2.21,;-4.28,.67,;-5.61,-.1,;-2.94,-.1,;-1.61,.67,;-.28,-.1,;-2.94,-1.64,;-1.61,-2.41,;-1.61,-3.95,;-.47,-4.98,;-1.09,-6.38,;-2.62,-6.22,;-2.94,-4.72,;-4.28,-3.95,;-4.28,-2.41,;1.02,-4.58,;2.06,-5.71,;3.46,-5.08,;3.29,-3.55,;4.38,-2.46,;1.78,-3.24,)|
Cc1c(CNC2CC(C)(C)C2)ccc(F)c1-c1cc2c(n[nH]c2cn1)-c1cnn(C)c1
Cc1c(CNCC2(C)CC2)ccc(F)c1-c1cc2c(n[nH]c2cn1)-c1cnn(C)c1
CNCc1ccc(F)c(-c2cc3c(n[nH]c3cn2)-c2cnn(C)c2)c1C(F)(F)F
Cn1cc(cn1)-c1n[nH]c2cnc(cc12)-c1c(F)cc(cc1C(F)(F)F)[C@@H]1CCCN1 |r|
Cn1cc(cn1)-c1n[nH]c2cnc(cc12)-c1c(F)cc(cc1C(F)(F)F)[C@H]1CCCN1 |r|
CN[C@H](C)c1cc(C)c(c(F)c1)-c1cc2c(n[nH]c2cn1)-c1cnn(c1)C1CC1 |r|
CN[C@@H](C)c1cc(C)c(c(F)c1)-c1cc2c(n[nH]c2cn1)-c1cnn(c1)C1CC1 |r|
CCn1cc(cn1)-c1n[nH]c2cnc(cc12)-c1c(C)cc(cc1F)[C@@H]1CCCCN1 |r|
CCn1cc(cn1)-c1n[nH]c2cnc(cc12)-c1c(C)cc(cc1F)[C@H]1CCCCN1 |r|
Cc1cc(cc(F)c1-c1cc2c(n[nH]c2cn1)-c1cnn(c1)C1CC1)[C@H]1CCCCN1 |r|
Cc1cc(cc(F)c1-c1cc2c(n[nH]c2cn1)-c1cnn(C)c1)C1COCCN1
CNCc1cc(F)c(-c2cc3c(n[nH]c3cn2)-c2cnn(C)c2)c(c1)C(F)F
CCNCc1ccc(F)c(c1C)-c1cc2c(n[nH]c2cn1)-c1cnn(C)c1
CCNCc1cccc(-c2cc3c(n[nH]c3cn2)-c2cnn(C)c2)c1C(F)(F)F
CNC1CCCc2c1ccc(F)c2-c1cc2c(n[nH]c2cn1)-c1ccc(nc1)N1CCN(C)CC1
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2cnc(cc12)-c1c(F)ccc2C(N)CCCc12
CCn1cc(cn1)-c1n[nH]c2cc(C#N)c(cc12)-c1c(C)cc(CNC)cc1F |(6.28,-1.88,;4.79,-1.48,;3.7,-2.57,;2.16,-2.57,;1.69,-4.03,;2.93,-4.94,;4.18,-4.03,;.2,-4.43,;-.43,-5.84,;-1.96,-5.68,;-2.28,-4.17,;-3.61,-3.4,;-3.66,-1.83,;-4.99,-1.06,;-6.33,-.29,;-2.28,-1.09,;-.94,-1.86,;-.94,-3.4,;-2.28,.45,;-.94,1.22,;.39,.45,;-.94,2.76,;-2.28,3.53,;-2.28,5.07,;-.94,5.84,;.39,5.07,;-3.61,2.76,;-3.61,1.22,;-4.95,.45,)|
CNCc1cc(C)c(c(F)c1)-c1cc2c(n[nH]c2cc1C#N)-c1cnn(c1)C1CC1 |(.47,5.07,;-.87,5.84,;-2.2,5.07,;-2.2,3.53,;-.87,2.76,;-.87,1.22,;.47,.45,;-2.2,.45,;-3.54,1.22,;-4.87,.45,;-3.54,2.76,;-2.2,-1.09,;-.87,-1.86,;-.87,-3.4,;.28,-4.43,;-.35,-5.84,;-1.88,-5.68,;-2.2,-4.17,;-3.54,-3.4,;-3.58,-1.83,;-4.92,-1.06,;-6.25,-.29,;1.76,-4.03,;3.01,-4.94,;4.26,-4.03,;3.78,-2.57,;2.24,-2.57,;4.87,-1.48,;6.2,-.71,;4.87,.06,)|
CNCc1cc(C)c(c(F)c1)-c1cc2c(n[nH]c2cc1C#N)-c1cnn(CC(F)(F)F)c1 |(-.35,5.07,;-1.69,5.84,;-3.02,5.07,;-3.02,3.53,;-1.69,2.76,;-1.69,1.22,;-.35,.45,;-3.02,.45,;-4.36,1.22,;-5.69,.45,;-4.36,2.76,;-3.02,-1.09,;-1.69,-1.86,;-1.69,-3.4,;-.54,-4.43,;-1.17,-5.84,;-2.7,-5.68,;-3.02,-4.17,;-4.36,-3.4,;-4.4,-1.83,;-5.74,-1.06,;-7.07,-.29,;.94,-4.03,;2.19,-4.94,;3.44,-4.03,;2.96,-2.57,;3.86,-1.32,;3.24,.08,;2.61,1.49,;4.64,.71,;1.83,-.54,;1.42,-2.57,)|
CNCc1cc(C)c(c(F)c1)-c1cc2c(n[nH]c2cc1C#N)-c1cn[nH]c1 |(1.45,5.07,;.11,5.84,;-1.22,5.07,;-1.22,3.53,;.11,2.76,;.11,1.22,;1.45,.45,;-1.22,.45,;-2.56,1.22,;-3.89,.45,;-2.56,2.76,;-1.22,-1.09,;.11,-1.86,;.11,-3.4,;1.26,-4.43,;.63,-5.84,;-.9,-5.68,;-1.22,-4.17,;-2.56,-3.4,;-2.56,-1.86,;-3.89,-1.09,;-5.22,-.32,;2.76,-4.11,;3.85,-5.2,;5.22,-4.5,;4.98,-2.98,;3.46,-2.74,)|
CNCc1cc(C)c(c(F)c1)-c1cc2c(n[nH]c2cc1C#N)-c1cnn(c1)-c1ccccc1Cl |(-.27,5.07,;-1.6,5.84,;-2.93,5.07,;-2.93,3.53,;-1.6,2.76,;-1.6,1.22,;-.27,.45,;-2.93,.45,;-4.27,1.22,;-5.6,.45,;-4.27,2.76,;-2.93,-1.09,;-1.6,-1.86,;-1.6,-3.4,;-.46,-4.43,;-1.08,-5.84,;-2.61,-5.68,;-2.93,-4.17,;-4.27,-3.4,;-4.27,-1.86,;-5.6,-1.09,;-6.94,-.32,;1.05,-4.11,;2.14,-5.2,;3.51,-4.5,;3.27,-2.98,;1.75,-2.74,;4.36,-1.89,;3.96,-.4,;5.05,.69,;6.54,.29,;6.94,-1.2,;5.85,-2.29,;6.25,-3.78,)|
CNCc1cc(C)c(c(F)c1)-c1cc2c(n[nH]c2cc1C#N)-c1cnn(c1)C(C)C |(.28,5.07,;-1.06,5.84,;-2.39,5.07,;-2.39,3.53,;-1.06,2.76,;-1.06,1.22,;.28,.45,;-2.39,.45,;-3.72,1.22,;-5.06,.45,;-3.72,2.76,;-2.39,-1.09,;-1.06,-1.86,;-1.06,-3.4,;.09,-4.43,;-.54,-5.84,;-2.07,-5.68,;-2.39,-4.17,;-3.72,-3.4,;-3.72,-1.86,;-5.06,-1.09,;-6.39,-.32,;1.59,-4.11,;2.68,-5.2,;4.06,-4.5,;3.81,-2.98,;2.29,-2.74,;4.9,-1.89,;4.51,-.4,;6.39,-2.29,)|
CNCc1cc(C)c(c(F)c1)-c1cc2c(n[nH]c2cc1C#N)-c1ccc(CO)cc1 |(.22,5.07,;-1.12,5.84,;-2.45,5.07,;-2.45,3.53,;-1.12,2.76,;-1.12,1.22,;.22,.45,;-2.45,.45,;-3.78,1.22,;-5.12,.45,;-3.78,2.76,;-2.45,-1.09,;-1.12,-1.86,;-1.12,-3.4,;.03,-4.43,;-.6,-5.84,;-2.13,-5.68,;-2.45,-4.17,;-3.78,-3.4,;-3.78,-1.86,;-5.12,-1.09,;-6.45,-.32,;1.53,-4.11,;2.56,-5.26,;4.07,-4.94,;4.55,-3.47,;6.05,-3.15,;6.45,-1.66,;3.52,-2.33,;2.01,-2.65,)|
CNCc1cc(C)c(c(F)c1)-c1cc2c(n[nH]c2cc1C#N)-c1ccc(cc1)C(=O)NC |(-.84,5.07,;-2.18,5.84,;-3.51,5.07,;-3.51,3.53,;-2.18,2.76,;-2.18,1.22,;-.84,.45,;-3.51,.45,;-4.84,1.22,;-6.18,.45,;-4.84,2.76,;-3.51,-1.09,;-2.18,-1.86,;-2.18,-3.4,;-1.03,-4.43,;-1.66,-5.84,;-3.19,-5.68,;-3.51,-4.17,;-4.84,-3.4,;-4.84,-1.86,;-6.18,-1.09,;-7.51,-.32,;.47,-4.11,;1.5,-5.26,;3.01,-4.94,;3.49,-3.47,;2.46,-2.33,;.95,-2.65,;4.99,-3.15,;5.47,-1.69,;6.02,-4.3,;7.51,-3.9,)|
CNCc1cc(C)c(c(F)c1)-c1cc2c(n[nH]c2cc1C#N)-c1ccc(cc1)C(=O)N(C)C |(-.84,5.07,;-2.18,5.84,;-3.51,5.07,;-3.51,3.53,;-2.18,2.76,;-2.18,1.22,;-.84,.45,;-3.51,.45,;-4.84,1.22,;-6.18,.45,;-4.84,2.76,;-3.51,-1.09,;-2.18,-1.86,;-2.18,-3.4,;-1.03,-4.43,;-1.66,-5.84,;-3.19,-5.68,;-3.51,-4.17,;-4.84,-3.4,;-4.84,-1.86,;-6.18,-1.09,;-7.51,-.32,;.47,-4.11,;1.5,-5.26,;3.01,-4.94,;3.49,-3.47,;2.46,-2.33,;.95,-2.65,;4.99,-3.15,;5.47,-1.69,;6.02,-4.3,;7.51,-3.9,;5.63,-5.78,)|
CNCc1cc(C)c(c(F)c1)-c1cc2c(n[nH]c2cc1C#N)-c1ccc(NC(C)=O)cc1 |(-.53,5.07,;-1.86,5.84,;-3.19,5.07,;-3.19,3.53,;-1.86,2.76,;-1.86,1.22,;-.53,.45,;-3.19,.45,;-4.53,1.22,;-5.86,.45,;-4.53,2.76,;-3.19,-1.09,;-1.86,-1.86,;-1.86,-3.4,;-.72,-4.43,;-1.34,-5.84,;-2.87,-5.68,;-3.19,-4.17,;-4.53,-3.4,;-4.53,-1.86,;-5.86,-1.09,;-7.2,-.32,;.79,-4.11,;1.82,-5.26,;3.33,-4.94,;3.8,-3.47,;5.31,-3.15,;5.71,-1.66,;7.2,-1.27,;4.62,-.57,;2.77,-2.33,;1.27,-2.65,)|
CNCc1cc(C)c(c(F)c1)-c1cc2c(n[nH]c2cc1C#N)-c1ccc(C)cc1 |(.42,5.07,;-.92,5.84,;-2.25,5.07,;-2.25,3.53,;-.92,2.76,;-.92,1.22,;.42,.45,;-2.25,.45,;-3.58,1.22,;-4.92,.45,;-3.58,2.76,;-2.25,-1.09,;-.92,-1.86,;-.92,-3.4,;.23,-4.43,;-.4,-5.84,;-1.93,-5.68,;-2.25,-4.17,;-3.58,-3.4,;-3.58,-1.86,;-4.92,-1.09,;-6.25,-.32,;1.73,-4.11,;2.76,-5.26,;4.27,-4.94,;4.75,-3.47,;6.25,-3.15,;3.72,-2.33,;2.21,-2.65,)|
CNCc1cc(C)c(c(F)c1)-c1cc2c(n[nH]c2cc1C#N)-c1cccc(OC)c1 |(1.17,5.07,;-.16,5.84,;-1.5,5.07,;-1.5,3.53,;-.16,2.76,;-.16,1.22,;1.17,.45,;-1.5,.45,;-2.83,1.22,;-4.17,.45,;-2.83,2.76,;-1.5,-1.09,;-.16,-1.86,;-.16,-3.4,;.98,-4.43,;.35,-5.84,;-1.18,-5.68,;-1.5,-4.17,;-2.83,-3.4,;-2.83,-1.86,;-4.17,-1.09,;-5.5,-.32,;2.49,-4.11,;3.52,-5.26,;5.02,-4.94,;5.5,-3.47,;4.49,-2.27,;4.96,-.81,;3.93,.33,;2.96,-2.65,)|
CNCc1cc(C)c(c(F)c1)-c1cc2c(n[nH]c2cc1C#N)-c1ccc(OC)cc1 |(.18,5.07,;-1.16,5.84,;-2.49,5.07,;-2.49,3.53,;-1.16,2.76,;-1.16,1.22,;.18,.45,;-2.49,.45,;-3.82,1.22,;-5.16,.45,;-3.82,2.76,;-2.49,-1.09,;-1.16,-1.86,;-1.16,-3.4,;-.01,-4.43,;-.64,-5.84,;-2.17,-5.68,;-2.49,-4.17,;-3.82,-3.4,;-3.82,-1.86,;-5.16,-1.09,;-6.49,-.32,;1.5,-4.11,;2.53,-5.26,;4.03,-4.94,;4.56,-3.46,;6.07,-3.14,;6.54,-1.68,;3.48,-2.33,;1.97,-2.65,)|
CNCc1cc(C)c(c(F)c1)-c1cc2c(n[nH]c2cc1C#N)-c1ccc(cc1)C(F)(F)F |(-.34,5.07,;-1.67,5.84,;-3,5.07,;-3,3.53,;-1.67,2.76,;-1.67,1.22,;-.34,.45,;-3,.45,;-4.34,1.22,;-5.67,.45,;-4.34,2.76,;-3,-1.09,;-1.67,-1.86,;-1.67,-3.4,;-.53,-4.43,;-1.15,-5.84,;-2.68,-5.68,;-3,-4.17,;-4.34,-3.4,;-4.34,-1.86,;-5.67,-1.09,;-7.01,-.32,;.98,-4.11,;2.01,-5.26,;3.52,-4.94,;4.05,-3.46,;2.96,-2.33,;1.46,-2.65,;5.55,-3.14,;7.06,-2.82,;5.87,-4.65,;5.23,-1.63,)|
CNCc1cc(C)c(c(F)c1)-c1cc2c(n[nH]c2cc1C#N)-c1ccc(cc1)C1CC1 |(-.33,5.07,;-1.66,5.84,;-3,5.07,;-3,3.53,;-1.66,2.76,;-1.66,1.22,;-.33,.45,;-3,.45,;-4.33,1.22,;-5.66,.45,;-4.33,2.76,;-3,-1.09,;-1.66,-1.86,;-1.66,-3.4,;-.52,-4.43,;-1.14,-5.84,;-2.67,-5.68,;-3,-4.17,;-4.33,-3.4,;-4.33,-1.86,;-5.66,-1.09,;-7,-.32,;.99,-4.11,;2.02,-5.26,;3.53,-4.94,;4,-3.47,;2.97,-2.33,;1.47,-2.65,;5.51,-3.15,;7,-3.55,;6.6,-2.06,)|
CNCc1cc(C)c(c(F)c1)-c1cc2c(n[nH]c2cc1C#N)-c1ccc(CC#N)cc1 |(-.06,5.07,;-1.39,5.84,;-2.73,5.07,;-2.73,3.53,;-1.39,2.76,;-1.39,1.22,;-.06,.45,;-2.73,.45,;-4.06,1.22,;-5.39,.45,;-4.06,2.76,;-2.73,-1.09,;-1.39,-1.86,;-1.39,-3.4,;-.25,-4.43,;-.88,-5.84,;-2.41,-5.68,;-2.73,-4.17,;-4.06,-3.4,;-4.06,-1.86,;-5.39,-1.09,;-6.73,-.32,;1.26,-4.11,;2.29,-5.26,;3.79,-4.94,;4.27,-3.47,;5.78,-3.15,;6.25,-1.69,;6.73,-.22,;3.24,-2.33,;1.73,-2.65,)|
CNCc1cc(C)c(c(F)c1)-c1cc2c(n[nH]c2cc1C#N)-c1ccc(C(=O)NC)c(F)c1 |(-.81,5.07,;-2.14,5.84,;-3.48,5.07,;-3.48,3.53,;-2.14,2.76,;-2.14,1.22,;-.81,.45,;-3.48,.45,;-4.81,1.22,;-6.14,.45,;-4.81,2.76,;-3.48,-1.09,;-2.14,-1.86,;-2.14,-3.4,;-1,-4.43,;-1.62,-5.84,;-3.16,-5.68,;-3.48,-4.17,;-4.81,-3.4,;-4.81,-1.86,;-6.14,-1.09,;-7.48,-.32,;.51,-4.11,;1.54,-5.26,;3.04,-4.94,;3.52,-3.47,;5.03,-3.15,;6.06,-4.3,;5.5,-1.69,;7.48,-1.29,;2.49,-2.33,;2.97,-.86,;.98,-2.65,)|
CNCc1cc(C)c(c(F)c1)-c1cc2c(n[nH]c2cc1C#N)-c1ccc(cc1)S(C)(=O)=O |(-.34,5.07,;-1.67,5.84,;-3,5.07,;-3,3.53,;-1.67,2.76,;-1.67,1.22,;-.34,.45,;-3,.45,;-4.34,1.22,;-5.67,.45,;-4.34,2.76,;-3,-1.09,;-1.67,-1.86,;-1.67,-3.4,;-.53,-4.43,;-1.15,-5.84,;-2.68,-5.68,;-3,-4.17,;-4.34,-3.4,;-4.34,-1.86,;-5.67,-1.09,;-7.01,-.32,;.98,-4.11,;2.01,-5.26,;3.52,-4.94,;4.05,-3.46,;2.96,-2.33,;1.46,-2.65,;5.55,-3.14,;5.23,-1.63,;7.06,-2.82,;5.87,-4.65,)|
CNCc1cc(C)c(c(F)c1)-c1cc2c(n[nH]c2cc1C#N)-c1ccc(cc1)C(C)(C)C#N |(8.37,-2.47,;7.03,-1.7,;5.7,-2.47,;4.37,-1.7,;4.37,-.16,;3.03,.61,;3.03,2.15,;1.7,-.16,;1.7,-1.7,;.37,-2.47,;3.03,-2.47,;.37,.61,;-.97,-.16,;-2.3,.61,;-3.77,.14,;-4.67,1.38,;-3.77,2.63,;-2.3,2.15,;-.97,2.92,;.37,2.15,;1.7,2.92,;3.03,3.69,;-4.24,-1.33,;-3.21,-2.47,;-3.69,-3.94,;-5.19,-4.26,;-6.22,-3.11,;-5.75,-1.65,;-5.67,-5.72,;-7.13,-5.24,;-4.21,-6.2,;-6.15,-7.18,;-6.62,-8.65,)|
CNCc1cc(C)c(c(F)c1)-c1cc2c(n[nH]c2cc1C#N)-c1ccc(cc1)C1(CC1)C#N |(8.24,-2.48,;6.91,-1.71,;5.57,-2.48,;4.24,-1.71,;4.24,-.17,;2.91,.6,;2.91,2.14,;1.57,-.17,;1.57,-1.71,;.24,-2.48,;2.91,-2.48,;.24,.6,;-1.1,-.17,;-2.43,.6,;-3.89,.12,;-4.8,1.37,;-3.89,2.61,;-2.43,2.14,;-1.1,2.91,;.24,2.14,;1.57,2.91,;2.91,3.68,;-4.37,-1.34,;-3.34,-2.49,;-3.82,-3.95,;-5.32,-4.27,;-6.35,-3.13,;-5.88,-1.66,;-5.8,-5.74,;-6.75,-6.95,;-7.32,-5.52,;-4.44,-6.46,;-3.08,-7.18,)|
CNCc1cc(C)c(c(F)c1)-c1cc2c(n[nH]c2cc1C#N)-c1ccc(C(=O)N(C)C)c(F)c1 |(-.83,5.07,;-2.17,5.84,;-3.5,5.07,;-3.5,3.53,;-2.17,2.76,;-2.17,1.22,;-.83,.45,;-3.5,.45,;-4.84,1.22,;-6.17,.45,;-4.84,2.76,;-3.5,-1.09,;-2.17,-1.86,;-2.17,-3.4,;-1.02,-4.43,;-1.65,-5.84,;-3.18,-5.68,;-3.5,-4.17,;-4.84,-3.4,;-4.84,-1.86,;-6.17,-1.09,;-7.5,-.32,;.46,-4.03,;1.55,-5.12,;3.04,-4.72,;3.44,-3.24,;4.93,-2.84,;5.33,-1.35,;6.02,-3.93,;7.5,-3.53,;5.62,-5.41,;2.35,-2.15,;2.75,-.66,;.86,-2.55,)|
CNCc1cc(C)c(c(F)c1)-c1cc2c(n[nH]c2cc1C#N)-c1ccc(cc1Cl)C(=O)NC(C)C |(-1.38,5.07,;-2.71,5.84,;-4.05,5.07,;-4.05,3.53,;-2.71,2.76,;-2.71,1.22,;-1.38,.45,;-4.05,.45,;-5.38,1.22,;-6.71,.45,;-5.38,2.76,;-4.05,-1.09,;-2.71,-1.86,;-2.71,-3.4,;-1.57,-4.43,;-2.19,-5.84,;-3.73,-5.68,;-4.05,-4.17,;-5.38,-3.4,;-5.38,-1.86,;-6.71,-1.09,;-8.05,-.32,;-.08,-4.03,;1.01,-5.12,;2.5,-4.72,;2.89,-3.24,;1.81,-2.15,;.32,-2.55,;-.77,-1.46,;4.38,-2.84,;4.78,-1.35,;5.47,-3.93,;6.96,-3.53,;8.05,-4.62,;7.36,-2.04,)|
CNCc1cc(C)c(c(F)c1)-c1cc2c(n[nH]c2cc1C#N)-c1ccc(c(F)c1)S(C)(=O)=O |(-.29,5.07,;-1.62,5.84,;-2.96,5.07,;-2.96,3.53,;-1.62,2.76,;-1.62,1.22,;-.29,.45,;-2.96,.45,;-4.29,1.22,;-5.62,.45,;-4.29,2.76,;-2.96,-1.09,;-1.62,-1.86,;-1.62,-3.4,;-.48,-4.43,;-1.11,-5.84,;-2.64,-5.68,;-2.96,-4.17,;-4.29,-3.4,;-4.29,-1.86,;-5.62,-1.09,;-6.96,-.32,;1.01,-4.03,;2.1,-5.12,;3.58,-4.72,;4.04,-3.22,;2.89,-2.15,;3.29,-.66,;1.41,-2.55,;5.52,-2.82,;5.13,-1.34,;7.01,-2.42,;5.92,-4.31,)|
CNCc1cc(C)c(c(F)c1)-c1cc2c(n[nH]c2cc1C#N)-c1ccc(cc1Cl)S(C)(=O)=O |(-.29,5.07,;-1.62,5.84,;-2.96,5.07,;-2.96,3.53,;-1.62,2.76,;-1.62,1.22,;-.29,.45,;-2.96,.45,;-4.29,1.22,;-5.62,.45,;-4.29,2.76,;-2.96,-1.09,;-1.62,-1.86,;-1.62,-3.4,;-.48,-4.43,;-1.11,-5.84,;-2.64,-5.68,;-2.96,-4.17,;-4.29,-3.4,;-4.29,-1.86,;-5.62,-1.09,;-6.96,-.32,;1.01,-4.03,;2.1,-5.12,;3.58,-4.72,;4.04,-3.22,;2.89,-2.15,;1.41,-2.55,;.32,-1.46,;5.52,-2.82,;5.13,-1.34,;7.01,-2.42,;5.92,-4.31,)|
CNCc1cc(C)c(c(F)c1)-c1cc2c(n[nH]c2cc1C#N)-c1ccc(cc1)S(=O)(=O)C(C)C |(-.83,5.07,;-2.17,5.84,;-3.5,5.07,;-3.5,3.53,;-2.17,2.76,;-2.17,1.22,;-.83,.45,;-3.5,.45,;-4.84,1.22,;-6.17,.45,;-4.84,2.76,;-3.5,-1.09,;-2.17,-1.86,;-2.17,-3.4,;-1.02,-4.43,;-1.65,-5.84,;-3.18,-5.68,;-3.5,-4.17,;-4.84,-3.4,;-4.84,-1.86,;-6.17,-1.09,;-7.5,-.32,;.46,-4.03,;1.55,-5.12,;3.04,-4.72,;3.44,-3.24,;2.35,-2.15,;.86,-2.55,;4.93,-2.84,;5.32,-1.35,;4.53,-4.33,;6.02,-3.93,;7.5,-3.53,;5.62,-5.41,)|
CNCc1cc(C)c(c(F)c1)-c1cc2c(n[nH]c2cc1C#N)-c1cnn(C)c1 |(1.03,5.07,;-.3,5.84,;-1.64,5.07,;-1.64,3.53,;-.3,2.76,;-.3,1.22,;1.03,.45,;-1.64,.45,;-2.97,1.22,;-4.3,.45,;-2.97,2.76,;-1.64,-1.09,;-.3,-1.86,;-.3,-3.4,;.84,-4.43,;.21,-5.84,;-1.32,-5.68,;-1.64,-4.17,;-2.97,-3.4,;-2.97,-1.86,;-4.3,-1.09,;-5.64,-.32,;2.33,-4.03,;3.42,-5.12,;4.79,-4.42,;4.55,-2.9,;5.64,-1.81,;3.03,-2.66,)|
CNCc1cc(C)c(c(F)c1)-c1cc2c(n[nH]c2cc1C#N)-c1cnc(nc1)N1CCN(C)CC1 |(-1.78,5.07,;-3.11,5.84,;-4.44,5.07,;-4.44,3.53,;-3.11,2.76,;-3.11,1.22,;-1.78,.45,;-4.44,.45,;-5.78,1.22,;-7.11,.45,;-5.78,2.76,;-4.44,-1.09,;-3.11,-1.86,;-3.11,-3.4,;-1.97,-4.43,;-2.59,-5.84,;-4.12,-5.68,;-4.44,-4.17,;-5.78,-3.4,;-5.78,-1.86,;-7.11,-1.09,;-8.45,-.32,;-.48,-4.03,;.61,-5.12,;2.1,-4.72,;2.5,-3.24,;1.41,-2.15,;-.08,-2.55,;3.98,-2.84,;5.07,-3.93,;6.56,-3.53,;6.96,-2.04,;8.45,-1.64,;5.87,-.95,;4.38,-1.35,)|
CNCc1cc(C)c(c(F)c1)-c1cc2c(n[nH]c2cc1C#N)-c1ccc(nc1)N1CCOCC1 |(-1.03,5.07,;-2.37,5.84,;-3.7,5.07,;-3.7,3.53,;-2.37,2.76,;-2.37,1.22,;-1.03,.45,;-3.7,.45,;-5.03,1.22,;-6.37,.45,;-5.03,2.76,;-3.7,-1.09,;-2.37,-1.86,;-2.37,-3.4,;-1.22,-4.43,;-1.85,-5.84,;-3.38,-5.68,;-3.7,-4.17,;-5.03,-3.4,;-5.03,-1.86,;-6.37,-1.09,;-7.7,-.32,;.26,-4.03,;.66,-2.55,;2.15,-2.15,;3.24,-3.24,;2.84,-4.72,;1.35,-5.12,;4.73,-2.84,;5.82,-3.93,;7.3,-3.53,;7.7,-2.04,;6.61,-.95,;5.13,-1.35,)|
CNCc1cc(C)c(c(F)c1)-c1cc2c(n[nH]c2cc1C#N)-c1ccc(NC(C)=O)nc1 |(-.49,5.07,;-1.82,5.84,;-3.16,5.07,;-3.16,3.53,;-1.82,2.76,;-1.82,1.22,;-.49,.45,;-3.16,.45,;-4.49,1.22,;-5.82,.45,;-4.49,2.76,;-3.16,-1.09,;-1.82,-1.86,;-1.82,-3.4,;-.68,-4.43,;-1.3,-5.84,;-2.84,-5.68,;-3.16,-4.17,;-4.49,-3.4,;-4.49,-1.86,;-5.82,-1.09,;-7.16,-.32,;.81,-4.03,;1.21,-2.55,;2.7,-2.15,;3.78,-3.24,;5.27,-2.84,;5.67,-1.35,;7.16,-.95,;4.58,-.26,;3.39,-4.72,;1.9,-5.12,)|
CNCc1cc(C)c(c(F)c1)-c1cc2c(n[nH]c2cc1C#N)-c1ccc(nc1)N1CCN(CC1)C(C)=O |(-2.32,5.07,;-3.66,5.84,;-4.99,5.07,;-4.99,3.53,;-3.66,2.76,;-3.66,1.22,;-2.32,.45,;-4.99,.45,;-6.32,1.22,;-7.66,.45,;-6.32,2.76,;-4.99,-1.09,;-3.66,-1.86,;-3.66,-3.4,;-2.51,-4.43,;-3.14,-5.84,;-4.67,-5.68,;-4.99,-4.17,;-6.32,-3.4,;-6.32,-1.86,;-7.66,-1.09,;-8.99,-.32,;-1.02,-4.03,;-.63,-2.55,;.86,-2.15,;1.95,-3.24,;1.55,-4.72,;.07,-5.12,;3.44,-2.84,;4.53,-3.93,;6.02,-3.53,;6.41,-2.04,;5.33,-.95,;3.84,-1.35,;7.9,-1.64,;8.99,-2.73,;8.3,-.15,)|
CNCc1cc(C)c(c(F)c1)-c1cc2c(n[nH]c2cc1C#N)-c1ccnc(C)c1 |(1.2,5.07,;-.14,5.84,;-1.47,5.07,;-1.47,3.53,;-.14,2.76,;-.14,1.22,;1.2,.45,;-1.47,.45,;-2.8,1.22,;-4.14,.45,;-2.8,2.76,;-1.47,-1.09,;-.14,-1.86,;-.14,-3.4,;1.01,-4.43,;.38,-5.84,;-1.15,-5.68,;-1.47,-4.17,;-2.8,-3.4,;-2.8,-1.86,;-4.14,-1.09,;-5.47,-.32,;2.5,-4.03,;3.58,-5.12,;5.07,-4.72,;5.47,-3.24,;4.38,-2.15,;4.78,-.66,;2.89,-2.55,)|
CNCc1cc(C)c(c(F)c1)-c1cc2c(n[nH]c2cc1C#N)-c1ccc(nc1)C1CCOCC1 |(-1.03,5.07,;-2.37,5.84,;-3.7,5.07,;-3.7,3.53,;-2.37,2.76,;-2.37,1.22,;-1.03,.45,;-3.7,.45,;-5.03,1.22,;-6.37,.45,;-5.03,2.76,;-3.7,-1.09,;-2.37,-1.86,;-2.37,-3.4,;-1.22,-4.43,;-1.85,-5.84,;-3.38,-5.68,;-3.7,-4.17,;-5.03,-3.4,;-5.03,-1.86,;-6.37,-1.09,;-7.7,-.32,;.26,-4.03,;.66,-2.55,;2.15,-2.15,;3.24,-3.24,;2.84,-4.72,;1.35,-5.12,;4.73,-2.84,;5.82,-3.93,;7.3,-3.53,;7.7,-2.04,;6.61,-.95,;5.13,-1.35,)|
CNCc1cc(C)c(c(F)c1)-c1cc2c(n[nH]c2cc1C#N)-c1ccc(nc1)C(C)(C)O |(-.29,5.07,;-1.62,5.84,;-2.96,5.07,;-2.96,3.53,;-1.62,2.76,;-1.62,1.22,;-.29,.45,;-2.96,.45,;-4.29,1.22,;-5.62,.45,;-4.29,2.76,;-2.96,-1.09,;-1.62,-1.86,;-1.62,-3.4,;-.48,-4.43,;-1.11,-5.84,;-2.64,-5.68,;-2.96,-4.17,;-4.29,-3.4,;-4.29,-1.86,;-5.62,-1.09,;-6.96,-.32,;1.01,-4.03,;1.41,-2.55,;2.89,-2.15,;3.98,-3.24,;3.58,-4.72,;2.1,-5.12,;5.47,-2.84,;6.56,-3.93,;6.96,-2.44,;5.87,-1.35,)|
CNCc1cc(C)c(c(F)c1)-c1cc2c(n[nH]c2cc1C#N)-c1ccc(C)nc1 |(.45,5.07,;-.88,5.84,;-2.21,5.07,;-2.21,3.53,;-.88,2.76,;-.88,1.22,;.45,.45,;-2.21,.45,;-3.55,1.22,;-4.88,.45,;-3.55,2.76,;-2.21,-1.09,;-.88,-1.86,;-.88,-3.4,;.26,-4.43,;-.36,-5.84,;-1.89,-5.68,;-2.21,-4.17,;-3.55,-3.4,;-3.55,-1.86,;-4.88,-1.09,;-6.21,-.32,;1.75,-4.03,;2.15,-2.55,;3.64,-2.15,;4.73,-3.24,;6.21,-2.84,;4.33,-4.72,;2.84,-5.12,)|
CNCc1cc(C)c(c(F)c1)-c1cc2c(n[nH]c2cc1C#N)-c1cnc(OC)nc1 |(.25,5.07,;-1.08,5.84,;-2.41,5.07,;-2.41,3.53,;-1.08,2.76,;-1.08,1.22,;.25,.45,;-2.41,.45,;-3.75,1.22,;-5.08,.45,;-3.75,2.76,;-2.41,-1.09,;-1.08,-1.86,;-1.08,-3.4,;.07,-4.43,;-.56,-5.84,;-2.09,-5.68,;-2.41,-4.17,;-3.75,-3.4,;-3.75,-1.86,;-5.08,-1.09,;-6.41,-.32,;1.55,-4.03,;2.64,-5.12,;4.13,-4.72,;4.58,-3.22,;6.07,-2.82,;6.47,-1.34,;3.44,-2.15,;1.95,-2.55,)|
CNCc1cc(C)c(c(F)c1)-c1cc2c(n[nH]c2cc1C#N)-c1cnco1 |(1.45,5.07,;.12,5.84,;-1.21,5.07,;-1.21,3.53,;.12,2.76,;.12,1.22,;1.45,.45,;-1.21,.45,;-2.55,1.22,;-3.88,.45,;-2.55,2.76,;-1.21,-1.09,;.12,-1.86,;.12,-3.4,;1.27,-4.43,;.64,-5.84,;-.89,-5.68,;-1.21,-4.17,;-2.55,-3.4,;-2.55,-1.86,;-3.88,-1.09,;-5.21,-.32,;2.75,-4.03,;3.84,-5.12,;5.21,-4.42,;4.97,-2.9,;3.45,-2.66,)|
CNCc1cc(C)c(c(F)c1)-c1cc2c(n[nH]c2cc1C#N)-c1cnsc1 |(1.45,5.07,;.12,5.84,;-1.21,5.07,;-1.21,3.53,;.12,2.76,;.12,1.22,;1.45,.45,;-1.21,.45,;-2.55,1.22,;-3.88,.45,;-2.55,2.76,;-1.21,-1.09,;.12,-1.86,;.12,-3.4,;1.27,-4.43,;.64,-5.84,;-.89,-5.68,;-1.21,-4.17,;-2.55,-3.4,;-2.55,-1.86,;-3.88,-1.09,;-5.21,-.32,;2.75,-4.03,;3.45,-2.66,;4.97,-2.9,;5.21,-4.42,;3.84,-5.12,)|
CNCc1cc(C)c(c(F)c1)-c1cc2c(n[nH]c2cc1C#N)-c1cnoc1 |(1.45,5.07,;.12,5.84,;-1.21,5.07,;-1.21,3.53,;.12,2.76,;.12,1.22,;1.45,.45,;-1.21,.45,;-2.55,1.22,;-3.88,.45,;-2.55,2.76,;-1.21,-1.09,;.12,-1.86,;.12,-3.4,;1.27,-4.43,;.64,-5.84,;-.89,-5.68,;-1.21,-4.17,;-2.55,-3.4,;-2.55,-1.86,;-3.88,-1.09,;-5.21,-.32,;2.75,-4.03,;3.45,-2.66,;4.97,-2.9,;5.21,-4.42,;3.84,-5.12,)|
CNCc1cc(C)c(c(F)c1)-c1cc2c(n[nH]c2cc1C#N)-c1ccc(cc1)C1CCOCC1 |(-1.03,5.07,;-2.37,5.84,;-3.7,5.07,;-3.7,3.53,;-2.37,2.76,;-2.37,1.22,;-1.03,.45,;-3.7,.45,;-5.03,1.22,;-6.37,.45,;-5.03,2.76,;-3.7,-1.09,;-2.37,-1.86,;-2.37,-3.4,;-1.22,-4.43,;-1.85,-5.84,;-3.38,-5.68,;-3.7,-4.17,;-5.03,-3.4,;-5.03,-1.86,;-6.37,-1.09,;-7.7,-.32,;.26,-4.03,;1.35,-5.12,;2.84,-4.72,;3.24,-3.24,;2.15,-2.15,;.66,-2.55,;4.73,-2.84,;5.82,-3.93,;7.3,-3.53,;7.7,-2.04,;6.61,-.95,;5.13,-1.35,)|
CNCc1cc(C)c(c(F)c1)-c1cc2c(n[nH]c2cc1C#N)-c1cnc(C)o1 |(1.03,5.07,;-.3,5.84,;-1.64,5.07,;-1.64,3.53,;-.3,2.76,;-.3,1.22,;1.03,.45,;-1.64,.45,;-2.97,1.22,;-4.3,.45,;-2.97,2.76,;-1.64,-1.09,;-.3,-1.86,;-.3,-3.4,;.84,-4.43,;.21,-5.84,;-1.32,-5.68,;-1.64,-4.17,;-2.97,-3.4,;-2.97,-1.86,;-4.3,-1.09,;-5.64,-.32,;2.33,-4.03,;3.42,-5.12,;4.79,-4.42,;4.55,-2.9,;5.64,-1.81,;3.03,-2.66,)|
CNCc1cc(C)c(c(F)c1)-c1cc2c(n[nH]c2cc1C#N)-c1ccc(nc1)N1CC[C@H](F)C1 |r,wU:31.35,(-1.21,5.07,;-2.54,5.84,;-3.88,5.07,;-3.88,3.53,;-2.54,2.76,;-2.54,1.22,;-1.21,.45,;-3.88,.45,;-5.21,1.22,;-6.54,.45,;-5.21,2.76,;-3.88,-1.09,;-2.54,-1.86,;-2.54,-3.4,;-1.4,-4.43,;-2.02,-5.84,;-3.56,-5.68,;-3.88,-4.17,;-5.21,-3.4,;-5.21,-1.86,;-6.54,-1.09,;-7.88,-.32,;.09,-4.03,;1.18,-5.12,;2.67,-4.72,;3.06,-3.24,;1.98,-2.15,;.49,-2.55,;4.55,-2.84,;5.66,-3.93,;7.03,-3.23,;6.79,-1.71,;7.88,-.62,;5.27,-1.47,)|
CNCc1cc(C)c(c(F)c1)-c1cc2c(n[nH]c2cc1C#N)-c1ccc(nc1)N1CCC(O)CC1 |(-1.78,5.07,;-3.11,5.84,;-4.44,5.07,;-4.44,3.53,;-3.11,2.76,;-3.11,1.22,;-1.78,.45,;-4.44,.45,;-5.78,1.22,;-7.11,.45,;-5.78,2.76,;-4.44,-1.09,;-3.11,-1.86,;-3.11,-3.4,;-1.97,-4.43,;-2.59,-5.84,;-4.12,-5.68,;-4.44,-4.17,;-5.78,-3.4,;-5.78,-1.86,;-7.11,-1.09,;-8.45,-.32,;-.48,-4.03,;.61,-5.12,;2.1,-4.72,;2.5,-3.24,;1.41,-2.15,;-.08,-2.55,;3.98,-2.84,;5.07,-3.93,;6.56,-3.53,;6.96,-2.04,;8.45,-1.64,;5.87,-.95,;4.38,-1.35,)|
CC[C@@H](C)Nc1ccc(cn1)-c1n[nH]c2cc(C#N)c(cc12)-c1c(C)cc(CNC)cc1F |r,wD:2.2,(7.7,-2.04,;6.61,-.95,;5.13,-1.35,;4.04,-.26,;4.73,-2.84,;3.24,-3.24,;2.84,-4.72,;1.35,-5.12,;.26,-4.03,;.66,-2.55,;2.15,-2.15,;-1.22,-4.43,;-1.85,-5.84,;-3.38,-5.68,;-3.7,-4.17,;-5.03,-3.4,;-5.03,-1.86,;-6.37,-1.09,;-7.7,-.32,;-3.7,-1.09,;-2.37,-1.86,;-2.37,-3.4,;-3.7,.45,;-2.37,1.22,;-1.03,.45,;-2.37,2.76,;-3.7,3.53,;-3.7,5.07,;-2.37,5.84,;-1.03,5.07,;-5.03,2.76,;-5.03,1.22,;-6.37,.45,)|
CNCc1cc(C)c(c(F)c1)-c1cc2c(n[nH]c2cc1C#N)-c1ccc(nc1)N1CC(CO)C1 |(-1.55,5.07,;-2.88,5.84,;-4.22,5.07,;-4.22,3.53,;-2.88,2.76,;-2.88,1.22,;-1.55,.45,;-4.22,.45,;-5.55,1.22,;-6.88,.45,;-5.55,2.76,;-4.22,-1.09,;-2.88,-1.86,;-2.88,-3.4,;-1.74,-4.43,;-2.37,-5.84,;-3.9,-5.68,;-4.22,-4.17,;-5.55,-3.4,;-5.55,-1.86,;-6.88,-1.09,;-8.22,-.32,;-.25,-4.03,;.84,-5.12,;2.33,-4.72,;2.72,-3.24,;1.64,-2.15,;.15,-2.55,;4.21,-2.84,;5.56,-3.61,;6.33,-2.27,;7.82,-1.88,;8.22,-.39,;5,-1.5,)|
CNCc1cc(C)c(c(F)c1)-c1cc2c(n[nH]c2cc1C#N)-c1cccc(n1)N1CCC(O)CC1 |(.6,5.07,;-.73,5.84,;-2.07,5.07,;-2.07,3.53,;-.73,2.76,;-.73,1.22,;.6,.45,;-2.07,.45,;-3.4,1.22,;-4.73,.45,;-3.4,2.76,;-2.07,-1.09,;-.73,-1.86,;-.73,-3.4,;.41,-4.43,;-.22,-5.84,;-1.75,-5.68,;-2.07,-4.17,;-3.4,-3.4,;-3.4,-1.86,;-4.73,-1.09,;-6.07,-.32,;1.9,-4.03,;2.99,-5.12,;4.47,-4.72,;4.87,-3.24,;3.78,-2.15,;2.3,-2.55,;4.18,-.66,;5.67,-.26,;6.07,1.23,;4.98,2.32,;5.38,3.8,;3.49,1.92,;3.09,.43,)|
CNCc1cc(C)c(c(F)c1)-c1cc2c(n[nH]c2cc1C#N)-c1cccc(n1)N1CCN(C)CC1 |(.6,5.07,;-.73,5.84,;-2.07,5.07,;-2.07,3.53,;-.73,2.76,;-.73,1.22,;.6,.45,;-2.07,.45,;-3.4,1.22,;-4.73,.45,;-3.4,2.76,;-2.07,-1.09,;-.73,-1.86,;-.73,-3.4,;.41,-4.43,;-.22,-5.84,;-1.75,-5.68,;-2.07,-4.17,;-3.4,-3.4,;-3.4,-1.86,;-4.73,-1.09,;-6.07,-.32,;1.9,-4.03,;2.99,-5.12,;4.47,-4.72,;4.87,-3.24,;3.78,-2.15,;2.3,-2.55,;4.18,-.66,;5.67,-.26,;6.07,1.23,;4.98,2.32,;5.38,3.8,;3.49,1.92,;3.09,.43,)|
CNCc1cc(C)c(c(F)c1)-c1cc2c(n[nH]c2cc1C#N)-c1cccc(n1)N1CC[C@@H](C1)N(C)C |r,wD:31.37,(-.48,5.07,;-1.81,5.84,;-3.15,5.07,;-3.15,3.53,;-1.81,2.76,;-1.81,1.22,;-.48,.45,;-3.15,.45,;-4.48,1.22,;-5.81,.45,;-4.48,2.76,;-3.15,-1.09,;-1.81,-1.86,;-1.81,-3.4,;-.67,-4.43,;-1.29,-5.84,;-2.83,-5.68,;-3.15,-4.17,;-4.48,-3.4,;-4.48,-1.86,;-5.81,-1.09,;-7.15,-.32,;.82,-4.03,;1.91,-5.12,;3.4,-4.72,;3.8,-3.24,;2.71,-2.15,;1.22,-2.55,;3.11,-.66,;2.2,.59,;3.11,1.83,;4.57,1.36,;4.57,-.18,;5.66,2.45,;7.15,2.05,;5.26,3.93,)|
Cc1ccccc1-c1cc2c(n[nH]c2cc1C#N)-c1cnn(C)c1
Cn1cc(cn1)-c1n[nH]c2cc(C#N)c(cc12)-c1ccccc1F
COc1cccc(F)c1-c1cc2c(n[nH]c2cc1C#N)-c1cnn(C)c1 |(-5.48,2.59,;-4.3,1.6,;-2.97,2.37,;-2.97,3.91,;-1.64,4.68,;-.3,3.91,;-.3,2.37,;1.03,1.6,;-1.64,1.6,;-1.64,.06,;-.3,-.71,;-.3,-2.25,;.84,-3.28,;.21,-4.68,;-1.32,-4.52,;-1.64,-3.02,;-2.97,-2.25,;-2.97,-.71,;-4.3,.06,;-5.64,.83,;2.33,-2.88,;3.42,-3.97,;4.79,-3.27,;4.55,-1.75,;5.64,-.66,;3.03,-1.51,)|
Cc1cccc(F)c1-c1cc2c(n[nH]c2cc1C#N)-c1cnn(C)c1 |(-4.3,1.6,;-2.97,2.37,;-2.97,3.91,;-1.64,4.68,;-.3,3.91,;-.3,2.37,;1.03,1.6,;-1.64,1.6,;-1.64,.06,;-.3,-.71,;-.3,-2.25,;.84,-3.28,;.21,-4.68,;-1.32,-4.52,;-1.64,-3.02,;-2.97,-2.25,;-2.97,-.71,;-4.3,.06,;-5.64,.83,;2.33,-2.88,;3.42,-3.97,;4.79,-3.27,;4.55,-1.75,;5.64,-.66,;3.03,-1.51,)|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2nn(C)cc2c1N(C)CCO
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2n(C)ncc2c1N(C)CCO
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2n(C)ncc2c1N(C)C1CCN(C)CC1
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2n(C)ncc2c1N(C)C1CC1
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2n(C)ncc2c1N(C)C
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2n(C)ncc2c1N(C)Cc1ccccc1
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2n(C)ncc2c1N(C)Cc1cccnc1
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2n(C)ncc2c1N(C)C1CCOCC1
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2n(C)ncc2c1N(C)CC(C)(C)O
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2n(C)ncc2c1N(C)CC1CCCO1
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2n(C)ncc2c1N(C)CC1(O)COC1
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2n(C)ncc2c1N(C)C1CCNC1
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2n(C)ncc2c1N(C)[C@H]1CCN(C1)C(C)=O |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2n(C)ncc2c1N(C)[C@H]1CCN(C1)S(C)(=O)=O |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2n(C)ncc2c1N(C)[C@H]1CCN(C1)C(=O)N(C)C |r|
CNCc1ccccc1-c1c(NC(=O)c2ccnc(n2)-c2c(F)cccc2OC)ccc2n(C)ncc12 |(7.34,.2,;6,.97,;4.67,.2,;3.33,.97,;3.33,2.51,;2,3.28,;.67,2.51,;.67,.97,;2,.2,;2,-1.34,;.67,-2.11,;-.67,-1.34,;-2,-2.11,;-2,-3.65,;-3.33,-1.34,;-4.67,-2.11,;-6,-1.34,;-6,.2,;-4.67,.97,;-3.33,.2,;-4.67,2.51,;-6,3.28,;-7.34,2.51,;-6,4.82,;-4.67,5.59,;-3.33,4.82,;-3.33,3.28,;-2,2.51,;-.67,3.28,;.67,-3.65,;2,-4.42,;3.33,-3.65,;4.8,-4.13,;5.27,-5.59,;5.7,-2.88,;4.8,-1.63,;3.33,-2.11,)|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c2nn(C)cc2c1N1C[C@@H]2C[C@H]1CN2 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c2n(C)ncc2c1N1C[C@@H]2C[C@H]1CN2 |r|
CCNC(=O)N1C[C@@H]2C[C@H]1CN2c1c(NC(=O)c2ccnc(n2)-c2c(F)cccc2OC)cc(F)c2n(C)ncc12 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c2n(C)ncc2c1N1C[C@@H](N)C[C@H]1CO |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c2nn(C)cc2c1N1C[C@@H](N)C[C@H]1CO |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c2n(C)ncc2c1N1CC[C@@H](N)C1 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c2nn(C)cc2c1N1CC[C@@H](N)C1 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c2n(C)ncc2c1N1C[C@@H]2CC[C@H]1CN2 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c2nn(C)cc2c1N1C[C@@H]2CC[C@H]1CN2 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c2n(C)ncc2c1N1CCC[C@@H]1CO |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c2nn(C)cc2c1N1CCC[C@@H]1CO |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c2n(C)ncc2c1N1CCOCC1
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c2nn(C)cc2c1N1CCOCC1
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c2n(C)ncc2c1N1CCC2(CCNC2=O)C1
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c2nn(C)cc2c1N1CCC2(CCNC2=O)C1
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c2n(C)ncc2c1N1CC(N)C1
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c2n(C)ncc2c1N1CCC[C@@H]1CN |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c2nn(C)cc2c1N1CCC[C@@H]1CN |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c2n(C)ncc2c1C1CCNC1
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c2n(C)ncc2c1N1CCCC1=O
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c2n(C)ncc2c1-n1cccn1
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c2n(C)ncc2c1-c1ccccc1C |(-.62,-3.29,;-1.95,-4.06,;-3.29,-3.29,;-3.29,-1.75,;-4.62,-.98,;-5.96,-1.75,;-5.96,-3.29,;-7.29,-4.06,;-4.62,-4.06,;-4.62,-5.6,;-5.96,-6.37,;-5.96,-7.91,;-4.62,-8.68,;-3.29,-7.91,;-3.29,-6.37,;-1.95,-8.68,;-1.95,-10.22,;-.62,-7.91,;.71,-8.68,;.71,-10.22,;2.05,-10.99,;2.05,-12.53,;3.38,-10.22,;4.84,-10.69,;5.32,-12.16,;5.75,-9.45,;4.84,-8.2,;3.38,-8.68,;2.05,-7.91,;2.05,-6.37,;.71,-5.6,;.71,-4.06,;2.05,-3.29,;3.38,-4.06,;3.38,-5.6,;4.71,-6.37,)|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c2nn(C)cc2c1-c1ccccc1C |(-.62,-3.29,;-1.95,-4.06,;-3.29,-3.29,;-3.29,-1.75,;-4.62,-.98,;-5.96,-1.75,;-5.96,-3.29,;-7.29,-4.06,;-4.62,-4.06,;-4.62,-5.6,;-5.96,-6.37,;-5.96,-7.91,;-4.62,-8.68,;-3.29,-7.91,;-3.29,-6.37,;-1.95,-8.68,;-1.95,-10.22,;-.62,-7.91,;.71,-8.68,;.71,-10.22,;2.05,-10.99,;2.05,-12.53,;3.38,-10.22,;4.84,-10.69,;5.75,-9.45,;7.29,-9.45,;4.84,-8.2,;3.38,-8.68,;2.05,-7.91,;2.05,-6.37,;.71,-5.6,;.71,-4.06,;2.05,-3.29,;3.38,-4.06,;3.38,-5.6,;4.71,-6.37,)|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(C#N)c2n(C)ncc2c1N1CCC[C@@H](N)C1 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(C#N)c2nn(C)cc2c1N1CCC[C@@H](N)C1 |r|
CNC(=O)c1cc(NC(=O)c2ccnc(n2)-c2c(F)cccc2OC)c(N2CCC[C@@H](N)C2)c2cnn(C)c12 |r|
CNC(=O)c1cc(NC(=O)c2ccnc(n2)-c2c(F)cccc2OC)c(N2CCC[C@@H](N)C2)c2cn(C)nc12 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c2n(CCO)ncc2c1N1CC[C@@H](N)C1 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(C)c2n(C)ncc2c1N1CCNCC1
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(C)c2nn(C)cc2c1N1CCNCC1
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(C)c2nn(C)cc2c1N1CC[C@@H](N)C1 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c2n(C)ncc2c1-c1cccnc1
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c2n(C)ncc2c1-c1cnn(C)c1
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c2n(C)ncc2c1-c1cccc(CO)c1
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c2n(C)ncc2c1-c1ccccc1CO |(,3.47,;-1.33,2.69,;-2.67,3.47,;-2.67,5,;-4,5.78,;-5.33,5,;-5.33,3.47,;-6.67,2.69,;-4,2.69,;-4,1.15,;-5.33,.38,;-5.33,-1.15,;-4,-1.93,;-2.67,-1.15,;-2.67,.38,;-1.33,-1.93,;-1.33,-3.47,;,-1.15,;1.33,-1.93,;1.33,-3.47,;2.67,-4.23,;2.67,-5.78,;4,-3.47,;5.47,-3.94,;5.94,-5.41,;6.37,-2.69,;5.47,-1.45,;4,-1.93,;2.67,-1.15,;2.67,.38,;1.33,1.16,;1.33,2.7,;2.67,3.47,;4,2.7,;4,1.16,;5.33,.39,;6.67,1.16,)|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c2n(C)ncc2c1-c1cccc(CN(C)C)c1
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c2n(CCO)ncc2c1N1C[C@@H]2C[C@H]1CN2 |r|
COCCn1ncc2c(N3C[C@@H]4C[C@H]3CN4)c(NC(=O)c3ccnc(n3)-c3c(F)cccc3OC)cc(F)c12 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2n(C)nc(I)c2c1N1CCC(CC1)N(C)C
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2n(C)nc(C)c2c1N1CCC(CC1)N(C)C
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2n(C)nc(-c3ccccc3)c2c1N1CCC(CC1)N(C)C
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2n(C)nc(-c3cnn(C)c3)c2c1N1CCC(CC1)N(C)C
COCCn1ncc2c(N3C[C@@H](N)C[C@H]3CO)c(NC(=O)c3ccnc(n3)-c3c(F)cccc3OC)cc(F)c12 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c2n(ncc2c1N1C[C@@H](N)C[C@H]1CO)[C@@H]1CCOC1 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c2nn(C)cc2c1N1CCN[C@@H](CO)C1 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c2n(ncc2c1N1C[C@@H](N)C[C@H]1CO)-c1ccncc1C#N |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c2n(C)ncc2c1N1C[C@@H](O)C[C@H]1CN |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c2n(CCF)ncc2c1N1C[C@@H]2C[C@H]1CN2 |r|
COCCn1ncc2c(N3C[C@@H](N)C[C@H]3CO)c(NC(=O)c3ccnc(n3)-c3c(F)c(C)ccc3OC)cc(F)c12 |r|
COCCn1ncc2c(N3C[C@@H](N)C[C@H]3CO)c(NC(=O)c3ccnc(n3)-c3c(F)cc(N)cc3OC)cc(F)c12 |r|
CNC(=O)c1ccc(OC)c(c1F)-c1nccc(n1)C(=O)Nc1cc(F)c2n(CCOC)ncc2c1N1C[C@@H](N)C[C@H]1CO |r|
COCCn1ncc2c(N3C[C@@H](N)C[C@H]3CO)c(NC(=O)c3ccnc(n3)-c3c(OC)ccc(-c4cnn(C)c4)c3F)cc(F)c12 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c2n(C)ncc2c1N(C)[C@@H]1CCCNC1 |r|
COCCn1ncc2c(N3C[C@@H](N)C[C@H]3CO)c(NC(=O)c3cccc(n3)-c3c(F)cccc3OC)cc(F)c12 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)ccc1N1C[C@H]2C[C@@H]1CN2 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)ccc1N1CC[C@H](N)C1 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)ccc1N1CCC[C@@H]1CN |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)ccc1N1CCC[C@@H]1CO |r|
COC[C@H]1CCCN1c1ccc(F)cc1NC(=O)c1ccnc(n1)-c1c(F)cccc1OC |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)ccc1N1C[C@@H](N)C[C@H]1CO |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)ccc1N1C[C@@H](O)C[C@@H]1C |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)ccc1N1CCCC1c1ccccn1
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)ccc1N1CCC2CNCC12
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)ccc1N1CCNC[C@H]1C |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)ccc1N1CCNC[C@@H]1CO |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)ccc1N1CCOCC1CO
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)cc(Br)c1N1C[C@H]2C[C@@H]1CN2 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cccc(C#N)c1N1C[C@H]2C[C@@H]1CN2 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)cc(-c2cccnc2)c1N1C[C@H]2C[C@@H]1CN2 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)cc(-c2cnn(C)c2)c1N1C[C@H]2C[C@@H]1CN2 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c(CO)cc1N1C[C@@H]2C[C@H]1CN2 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c(Br)cc1N1C[C@@H]2C[C@H]1CN2 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c(cc1N1C[C@@H]2C[C@H]1CN2)-c1cnn(C)c1 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c(cc1N1C[C@@H]2C[C@H]1CN2)-c1ccc(CO)nc1 |r|
CNC(=O)c1ccc(cn1)-c1cc(N2C[C@@H]3C[C@H]2CN3)c(NC(=O)c2ccnc(n2)-c2c(F)cccc2OC)cc1F |r,TLB:12:13:18.19:16|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c(cc1N1C[C@@H]2C[C@H]1CN2)-c1ccc(=O)n(C)c1 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c(cc1N1C[C@@H]2C[C@H]1CN2)-c1cccnc1C |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc(cc1N1C[C@@H]2C[C@H]1CN2)-c1cccnc1C |r|
COc1ccncc1-c1ccc(NC(=O)c2ccnc(n2)-c2c(F)cccc2OC)c(c1)N1C[C@@H]2C[C@H]1CN2 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc(cc1N1C[C@@H]2C[C@H]1CN2)-c1cnccc1C#N |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc(cc1N1C[C@@H]2C[C@H]1CN2)-c1c(C)nn(C)c1C |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c(cc1N1C[C@@H]2C[C@H]1CN2)N1CCOCC1 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c(cc1N1C[C@@H]2C[C@H]1CN2)N1CCC1 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c(CN2CCOCC2)cc1N1C[C@@H]2C[C@H]1CN2 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c(CNC2CCC2)cc1N1C[C@@H]2C[C@H]1CN2 |r|
CCN1C[C@H]2C[C@@H]1CN2c1ccc(F)cc1NC(=O)c1ccnc(n1)-c1c(F)cccc1OC |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)ccc1N1C[C@H]2C[C@@H]1CN2CCO |r|
CCCNC(=O)N1C[C@H]2C[C@@H]1CN2c1ccc(F)cc1NC(=O)c1ccnc(n1)-c1c(F)cccc1OC |r|
COc1ccc(N2C[C@H]3C[C@@H]2CN3)c(NC(=O)c2ccnc(n2)-c2c(F)cccc2OC)c1 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(CO)ccc1N1C[C@H]2C[C@@H]1CN2 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(ccc1N1C[C@H]2C[C@@H]1CN2)C#N |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc(cc1N1C[C@@H]2C[C@H]1CN2)N1CCC1 |r|
COC[C@@H]1CCN1c1ccc(NC(=O)c2ccnc(n2)-c2c(F)cccc2OC)c(c1)N1C[C@@H]2C[C@H]1CN2 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc(c(F)c1N1C[C@@H]2C[C@H]1CN2)-c1ccncc1C#N |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc(cc1N1C[C@@H](N)C[C@H]1CO)-c1ccncc1C#N |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc(cc1N1C[C@@H](N)C[C@H]1CO)-c1cnccc1C#N |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc(cc1N1C[C@@H](N)C[C@H]1CO)-c1cccnc1C |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc(cc1N1C[C@@H](N)C[C@H]1CO)-c1ccncc1OC |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc(cc1N1C[C@@H](N)C[C@H]1CO)-c1c(F)cccc1C#N |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc(cc1N1C[C@@H](N)C[C@H]1CO)-c1ncccc1C#N |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc(cc1N1C[C@@H](N)C[C@H]1CO)-c1c(cnn1C)C#N |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc(cc1N1C[C@@H](N)C[C@H]1CO)C(C)C |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc(cc1N1C[C@@H](O)C[C@H]1CO)-c1ccncc1C#N |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc(cc1N1C[C@@H](C)NC[C@H]1CO)-c1cnccc1C#N |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc(cc1N1C[C@H](C)NC[C@H]1CO)-c1cnccc1C#N |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc(cc1N1CC2(CC2)NC[C@H]1CO)-c1cnccc1C#N |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc(cc1N1C[C@@H](N)C[C@H]1C1(O)CC1)-c1cnccc1C#N |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc(cc1N1C[C@@H](N)C[C@H]1C(C)(C)O)-c1cnccc1C#N |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc(cc1N1[C@@H]2CN[C@@H](C2)[C@@H]1CO)-c1cnccc1C#N |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc(cc1N1C[C@@H]2C[C@@]1(CO)CN2)-c1cnccc1C#N |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc(cc1N1CC[C@H](N)C[C@@H]1C)-c1cnccc1C#N |r|
COc1cccc(F)c1-c1cccc(n1)C(=O)Nc1ccc(cc1N1C[C@@H](N)C[C@H]1CO)-c1cnccc1C#N |r|
COc1cccc(F)c1-c1nc(ccc1C#N)C(=O)Nc1ccc(cc1N1C[C@@H](N)C[C@H]1CO)-c1cnccc1C#N |r,wU:28.31,31.35,(.05,4.21,;-1.29,3.44,;-2.62,4.21,;-2.67,5.78,;-4,6.55,;-5.33,5.78,;-5.33,4.24,;-6.67,3.47,;-4,3.47,;-4,1.93,;-2.67,1.16,;-2.67,-.38,;-4,-1.15,;-5.33,-.38,;-5.33,1.16,;-6.67,1.93,;-8,2.7,;-1.33,-1.15,;-1.33,-2.69,;,-.39,;1.33,-1.16,;1.33,-2.7,;2.67,-3.47,;4,-2.7,;4,-1.16,;2.67,-.39,;2.67,1.15,;1.42,2.06,;1.9,3.52,;1.13,4.86,;3.44,3.52,;3.91,2.06,;5.25,1.29,;6.58,2.06,;5.33,-3.47,;6.67,-2.7,;8,-3.47,;8,-5.01,;6.67,-5.78,;5.29,-5.03,;3.95,-5.8,;2.62,-6.57,)|
COc1ccc(nc1-c1c(F)cccc1OC)C(=O)Nc1ccc(cc1N1C[C@@H](N)C[C@H]1CO)-c1cnccc1C#N |r,wU:28.31,31.35,(-8,1.16,;-6.67,1.93,;-5.33,1.16,;-5.33,-.38,;-4,-1.15,;-2.67,-.38,;-2.67,1.16,;-4,1.93,;-4,3.47,;-5.33,4.24,;-6.67,3.47,;-5.33,5.78,;-4,6.55,;-2.67,5.78,;-2.62,4.21,;-1.29,3.44,;.05,4.21,;-1.33,-1.15,;-1.33,-2.69,;,-.39,;1.33,-1.16,;1.33,-2.7,;2.67,-3.47,;4,-2.7,;4,-1.16,;2.67,-.39,;2.67,1.15,;1.42,2.06,;1.9,3.52,;1.13,4.86,;3.44,3.52,;3.91,2.06,;5.25,1.29,;6.58,2.06,;5.33,-3.47,;6.67,-2.7,;8,-3.47,;8,-5.01,;6.67,-5.78,;5.29,-5.03,;3.95,-5.8,;2.62,-6.57,)|
N[C@H]1C[C@@H](CO)N(C1)c1cc(ccc1NC(=O)c1ccnc(n1)-c1c(F)cccc1F)-c1cnccc1C#N |r|
Cc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc(cc1N1C[C@@H](N)C[C@H]1CO)-c1cnccc1C#N |r|
N[C@H]1C[C@@H](CO)N(C1)c1cc(ccc1NC(=O)c1ccnc(n1)-c1c(F)cccc1Cl)-c1cnccc1C#N |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc(nc1N1C[C@@H](N)C[C@H]1CO)-c1c(C)nn(C)c1C |r|
N[C@H]1C[C@@H](CO)N(C1)c1ccc(F)cc1NC(=O)c1ccnc(n1)-c1c(F)cccc1F |r|
COc1ccc(C#N)c(F)c1-c1nccc(n1)C(=O)Nc1cc(F)ccc1N1C[C@@H](N)C[C@H]1CO |r|
COc1ccc(F)c(F)c1-c1nccc(n1)C(=O)Nc1cc(F)ccc1N1C[C@@H](N)C[C@H]1CO |r|
COc1ccc(C)c(F)c1-c1nccc(n1)C(=O)Nc1cc(F)ccc1N1C[C@@H](N)C[C@H]1CO |r|
COc1cc(C)cc(F)c1-c1nccc(n1)C(=O)Nc1ccc(cc1N1C[C@@H](N)C[C@H]1CO)-c1cnccc1C#N |r|
Cc1c(F)ccc(F)c1-c1nccc(n1)C(=O)Nc1ccc(cc1N1C[C@@H](N)C[C@H]1CO)-c1cnccc1C#N |r|
COc1ccc(F)c(F)c1-c1nccc(n1)C(=O)Nc1ccc(cc1N1C[C@@H](N)C[C@H]1CO)-c1cnccc1C#N |r|
COc1c(F)ccc(F)c1-c1nccc(n1)C(=O)Nc1ccc(cc1N1C[C@@H](N)C[C@H]1CO)-c1cnccc1C#N |r|
COc1ccc(C#N)c(F)c1-c1nccc(n1)C(=O)Nc1ccc(cc1N1C[C@@H](N)C[C@H]1CO)-c1cnccc1C#N |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccccc1C1CCNCC1
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccccc1[C@@H]1CC[C@H](N)CC1 |r,wU:24.26,27.30,(-6,8.25,;-4.67,7.48,;-3.33,8.25,;-3.33,9.79,;-2,10.56,;-.67,9.79,;-.67,8.25,;.67,7.48,;-2,7.48,;-2,5.94,;-3.33,5.17,;-3.33,3.63,;-2,2.86,;-.67,3.63,;-.67,5.17,;.67,2.86,;.67,1.32,;2,3.63,;3.33,2.86,;3.33,1.32,;4.67,.55,;6,1.32,;6,2.86,;4.67,3.63,;4.67,5.17,;6,5.94,;6,7.48,;4.67,8.25,;4.67,9.79,;3.33,7.48,;3.33,5.94,)|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccccc1C1CCCC(N)C1
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccccc1C1CCC(N)C1
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc(cc1[C@H]1CC[C@H](N)CC1)-c1cnccc1C#N |r,wU:24.26,wD:27.30,(-8,-5.4,;-6.67,-6.17,;-5.33,-5.4,;-5.33,-3.86,;-4,-3.09,;-2.67,-3.86,;-2.67,-5.4,;-1.33,-6.17,;-4,-6.17,;-4,-7.71,;-5.33,-8.48,;-5.33,-10.02,;-4,-10.79,;-2.67,-10.02,;-2.67,-8.48,;-1.33,-10.79,;-1.33,-12.33,;,-10.02,;1.33,-10.79,;1.33,-12.33,;2.67,-13.1,;4,-12.33,;4,-10.79,;2.67,-10.02,;2.67,-8.48,;1.33,-7.71,;1.33,-6.17,;2.67,-5.4,;2.67,-3.86,;4,-6.17,;4,-7.71,;5.33,-13.1,;6.67,-12.33,;8,-13.1,;8,-14.64,;6.67,-15.41,;5.29,-14.66,;3.95,-15.43,;2.62,-16.2,)|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc(cc1[C@@H]1CC[C@H](N)CC1)-c1c(cnn1C)C#N |r,wU:24.26,27.30,(-7.89,11.41,;-6.55,10.64,;-5.22,11.41,;-5.22,12.95,;-3.89,13.72,;-2.55,12.95,;-2.55,11.41,;-1.22,10.64,;-3.89,10.64,;-3.89,9.1,;-5.22,8.33,;-5.22,6.79,;-3.89,6.02,;-2.55,6.79,;-2.55,8.33,;-1.22,6.02,;-1.22,4.48,;.11,6.79,;1.45,6.02,;1.45,4.48,;2.78,3.71,;4.12,4.48,;4.12,6.02,;2.78,6.79,;2.78,8.33,;4.12,9.1,;4.12,10.64,;2.78,11.41,;2.78,12.95,;1.45,10.64,;1.45,9.1,;5.45,3.71,;5.58,2.15,;7.12,1.85,;7.89,3.19,;6.86,4.33,;7.18,5.84,;4.44,1.12,;3.29,.09,)|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc(cc1[C@@H]1CC[C@H](N)CC1)-c1c(C)nn(C)c1C |r,wU:24.26,27.30,(-8.65,3.98,;-7.32,3.21,;-5.99,3.98,;-5.99,5.52,;-4.65,6.29,;-3.32,5.52,;-3.32,3.98,;-1.98,3.21,;-4.65,3.21,;-4.65,1.67,;-5.99,.9,;-5.99,-.64,;-4.65,-1.41,;-3.32,-.64,;-3.32,.9,;-1.98,-1.41,;-1.98,-2.95,;-.65,-.64,;.68,-1.41,;.68,-2.95,;2.02,-3.72,;3.35,-2.95,;3.35,-1.41,;2.02,-.64,;2.02,.9,;3.35,1.67,;3.35,3.21,;2.02,3.98,;2.02,5.52,;.68,3.21,;.68,1.67,;4.68,-3.72,;4.84,-5.26,;3.7,-6.29,;6.35,-5.58,;7.12,-4.24,;8.65,-4.08,;6.09,-3.1,;6.41,-1.59,)|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc(cc1N1C[C@@H](N)C[C@H]1CO)S(C)(=O)=O |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccccc1N1C[C@@H](N)C[C@H]1CO |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(C)ccc1N1C[C@@H](N)C[C@H]1CO |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)ccc1N1C[C@H](C[C@H]1CO)N(C)C |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)ccc1N1C[C@H](C[C@H]1CO)NC(C)C |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc(cc1N1C[C@@H](N)C[C@H]1CO)C1CCOCC1 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc(Cl)cc1N1C[C@@H](N)C[C@H]1CO |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc(F)cc1N1C[C@@H](N)C[C@H]1CO |r|
N[C@H]1C[C@@H](CO)N(C1)c1cc(ccc1NC(=O)c1ccnc(n1)-c1c(F)cccc1F)-c1cc(ncc1C#N)N1CCCC1 |r|
N[C@H]1C[C@@H](CO)N(C1)c1cc(ccc1NC(=O)c1ccnc(n1)-c1c(F)cccc1F)C1(CC1)C#N |r|
N[C@H]1C[C@@H](CO)N(C1)c1cc(ccc1NC(=O)c1ccnc(n1)-c1c(F)cccc1OC(F)F)-c1cnccc1C#N |r|
N[C@H]1C[C@@H](CO)N(C1)c1cc(ccc1NC(=O)c1ccnc(n1)-c1c(F)cccc1C1CC1)-c1cnccc1C#N |r|
CCOc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc(cc1N1C[C@@H](N)C[C@H]1CO)-c1cnccc1C#N |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc(cc1N1C[C@]2(CO)C[C@H]1CN2C)-c1cnccc1C#N |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc(cc1N1CCO[C@H](CO)C1)-c1cnccc1C#N |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc(cc1N1CCO[C@@H](CN(C)C)C1)-c1cnccc1C#N |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc(cc1N1CCO[C@H](CC#N)C1)-c1cnccc1C#N |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc(cc1N1CCN2[C@@H](COC2=O)C1)-c1cnccc1C#N |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)ccc1N1CCN[C@H](CO)C1 |r|
COCC1CN(C1)c1cc(ccc1NC(=O)c1ccnc(n1)-c1c(F)cccc1OC)-c1cnccc1C#N
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc(cc1N1CC[C@H]1CO)-c1cnccc1C#N |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc(cc1N1CC[C@@H]1CN(C)C)-c1cnccc1C#N |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc(cc1N1CCN(C)CC1)-c1cnccc1C#N
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc(cc1N1CCN(CCO)CC1)-c1cnccc1C#N
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c(cc1N1CCN[C@H](CO)C1)C(C)C |r|
Cc1nc2c(N3CC[C@@H](N)C3)c(NC(=O)c3ccnc(n3)-c3c(F)cccc3F)ccc2s1 |r|
Cc1nc2c(N3CC[C@@H](N)C3)c(NC(=O)c3ccnc(n3)-c3c(C)cccc3F)ccc2s1 |r|
Cc1nc2c(N3CC[C@@H](N)C3)c(NC(=O)c3ccnc(n3)-c3c(F)cccc3C(F)(F)F)ccc2s1 |r|
CNCc1cc(C)c(c(F)c1)-c1nccc(n1)C(=O)Nc1ccc2sc(C)nc2c1N1CC[C@@H](N)C1 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(Cl)c2sc(C)nc2c1N1CC[C@H](N)C1 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(Br)c2sc(C)nc2c1N1CC[C@H](N)C1 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(C)c2sc(C)nc2c1N1CC[C@H](N)C1 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(C#N)c2sc(C)nc2c1N1CC[C@H](N)C1 |r|
COCc1nc2c(N3CCC[C@H]3CN)c(NC(=O)c3ccnc(n3)-c3c(F)cccc3OC)ccc2s1 |r|
COCCc1nc2c(N3CCC[C@H]3CN)c(NC(=O)c3ccnc(n3)-c3c(F)cccc3OC)ccc2s1 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2sc(C)nc2c1N1C[C@H](N)C[C@H]1CO |r|
CCc1nc2c(N3C[C@@H](N)C[C@H]3CO)c(NC(=O)c3ccnc(n3)-c3c(F)cccc3OC)ccc2s1 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2sc(nc2c1N1C[C@@H](N)C[C@H]1CO)C(C)C |r|
COc1cccc(C(N)=O)c1-c1nccc(n1)C(=O)Nc1ccc2sc(C)nc2c1N1C[C@H](N)C[C@H]1CO |r|
COc1ccc(-c2cnn(C)c2)c(F)c1-c1nccc(n1)C(=O)Nc1ccc2sc(C)nc2c1N1C[C@H](N)C[C@H]1CO |r|
COc1ccc(F)c(F)c1-c1nccc(n1)C(=O)Nc1ccc2sc(C)nc2c1N1C[C@H](N)C[C@H]1CO |r|
COc1ccc(C#N)c(F)c1-c1nccc(n1)C(=O)Nc1ccc2sc(C)nc2c1N1C[C@H](N)C[C@H]1CO |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2sc(C)nc2c1N1C[C@@H](C[C@H]1CO)NC(C)C |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2sc(C)nc2c1N1C[C@@H](C[C@H]1CO)NC1CCOCC1 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2sc(C)nc2c1N1C[C@@H](C[C@H]1CO)NC(C)=O |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2sc(C)nc2c1N1C[C@@H](C[C@H]1CO)NS(C)(=O)=O |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2sc(C)nc2c1N1C[C@H]2C[C@@H]1CO2 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2sc(C)nc2c1N1C[C@@H](N)C[C@H]1CO |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2sc(C)nc2c1N(C)CC1CCN(C)C1
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2sc(C)nc2c1N1C[C@H]2C[C@@H]1CN2C(=O)N1CCOCC1 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2sc(C)nc2c1N1CCOC[C@@H]1CN |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2sc(C)nc2c1N(C)[C@@H]1CCCNC1 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2sc(C)nc2c1N1CCC2CCNCC12
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2sc(C)nc2c1N1CCC(C1)c1ccccn1
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2sc(C)nc2c1N1CC(F)(F)C[C@H]1CO |r|
Cc1nc2c(N3C[C@@H]4CC[C@H]3CN4)c(NC(=O)c3ccnc(n3)-c3c(F)cccc3F)ccc2s1 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2sc(CN(C)C)nc2c1N1C[C@H](N)C[C@H]1CO |r|
COc1cccc(F)c1-c1cc2c(NC(=O)c3ccc(cc3)N3CCN(C(=O)C3)S(C)(=O)=O)n[nH]c2cn1
CNCCCc1cc(F)c(c(F)c1)-c1cc2c(n[nH]c2cn1)-c1cnn(C)c1
Cn1cc(cn1)-c1n[nH]c2cnc(cc12)-c1c(F)cc(CCCNC2CCOCC2)cc1F
CNCc1cc(C)c(c(F)c1)-c1cc2c(noc2cn1)-c1ccc(nc1)N1CCCC(C1)OC
Cc1cc(cc(F)c1-c1cc2c(n[nH]c2cn1)-c1cnn(c1)C1CC1)[C@@H]1CCCCN1 |r|
CCc1c(Cl)[nH]c2ncc(cc12)-c1cccc(c1)N1CCOCC1=O
CCc1c(Cl)[nH]c2ncc(cc12)-c1ccc(N)c(n1)C(=O)N(C)C
CCc1c(Cl)[nH]c2ncc(cc12)-c1ccc(N)c(c1)C(=O)N(C)C
CCc1c(C)[nH]c2ncc(cc12)-c1ccc(N)c(c1)C(=O)N(C)C
CCc1c(Cl)[nH]c2ncc(cc12)-c1cccc(n1)N1CCOCC1=O
CCc1c(Cl)[nH]c2ncc(cc12)-c1ccc(N)c(n1)C(=O)N1CC(O)C1
CCc1c(Cl)[nH]c2ncc(cc12)-c1ccnc(n1)N1CCOC1=O
Cc1[nH]c2ncc(cc2c1C(F)(F)F)-c1cccc(n1)N1CCOCC1=O
CN(C)C(=O)c1nc(ccc1N)-c1cnc2[nH]c(C)c(c2c1)C(F)(F)F
CN(C)C(=O)c1cc(ccc1N)-c1cnc2[nH]c(C)c(c2c1)C(F)(F)F
Cc1[nH]c2ncc(cc2c1C(F)(F)F)-c1ccc(N)c(n1)N1CCOCC1=O
Cc1[nH]c2ncc(cc2c1C(F)(F)F)-c1cc(N)cc(c1)-c1ncccc1CO
OCc1[nH]c2ncc(cc2c1C(F)(F)F)-c1cccc(c1)N1CCOCC1=O
FCCc1c(Cl)[nH]c2ncc(cc12)-c1cccc(c1)N1CCOCC1=O
Cc1[nH]c2ncc(cc2c1C(F)(F)F)-c1cccc(n1)N1CCOCC1CO
Cc1[nH]c2ncc(cc2c1C(F)(F)F)-c1cccc(n1)N1CCCNC1=O
CN(C)C(=O)c1cc(ccc1N)-c1cnc2[nH]c(C)cc2c1
CCc1c(F)[nH]c2ncc(cc12)-c1cccc(c1)N1CCOCC1=O
CCc1c(F)[nH]c2ncc(cc12)-c1ccc(N)c(C(=O)N(C)C)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3[nH]c(Cl)c(CCO)c3c2)c1F
OCCc1c(Cl)[nH]c2ncc(cc12)-c1cccc(c1)N1CCOCC1=O
CN(C)C(=O)c1cc(ccc1N)-c1cnc2[nH]c(Cl)c(CCO)c2c1Cl
COCc1c(Cl)[nH]c2ncc(cc12)-c1ccc(N)c(C(=O)N(C)C)c1F
CCc1c(Cl)[nH]c2ncc(cc12)-c1ccc(cc1)C1NCCNC1=O
CCc1c(Cl)[nH]c2ncc(cc12)-c1cccc(c1)C1NCCNC1=O
CN(C)C(=O)c1c(N)ccc(c1F)-c1cnc2[nH]c(Cl)c(CCO)c2c1Cl
CCc1c(Cl)[nH]c2ncc(cc12)-c1ccc(N)c(C(=O)N(C)C)c1F
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc3c(c2)OCC2CN(C)CCN32)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C)CC3)cc2F)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc3c(c2)OCO3)cnc2c1NCCO2
COCCN1CCC(c2ccc(NC(=O)c3c(Nc4cnc5c(c4C)NCCO5)cc[nH]c3=O)cc2F)CC1
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C(C)C)CC3)cc2)cnc2c1NCC(C)O2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C)CC3)c(C(=O)N(C)C)c2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2cccc(S(=O)(=O)CCO)c2)cnc2c1NCCO2
COCCCN1CCN(c2ccc(NC(=O)c3c(Nc4cnc5c(c4C)NCCO5)cc[nH]c3=O)cc2)CC1
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(CC(C)O)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc3c(c2)NCCC3)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCC(O)CC3)cc2)cnc2c1NCCO2
COCCN1CCN(c2ccc(NC(=O)c3c(Nc4cnc5c(c4C)NCC(C)O5)cc[nH]c3=O)cc2)CC1
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(NC3CCN(C)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCC(C(N)=O)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(-c3ccccn3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C)CC3)cc2)cnc2c1NCC(C)(C)O2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(S(N)(=O)=O)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc3ncsc3c2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(C3CCN(C(C)C)CC3)cc2)cnc2c1NCCO2
COCCN1CCN(c2ccc(NC(=O)c3c(Nc4cnc5c(c4C)NCC(C)(C)O5)cc[nH]c3=O)cc2)CC1
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C)CC3)c(-n3cnnc3)c2)cnc2c1NCCO2
Cc1nc2ccc(NC(=O)c3c(Nc4cnc5c(c4C)NCCO5)cc[nH]c3=O)cc2s1
COc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(Cc4ccn[nH]4)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCCC(C(C)(C)O)C3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc3c(c2)CCC(=O)N3C)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(C3CCOCC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(CCCO)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(CN3CCN(C)CC3)c(C(F)(F)F)c2)cnc2c1NCCO2
CCC(=O)N1CCN(c2ccc(NC(=O)c3c(Nc4cnc5c(c4C)NCCO5)cc[nH]c3=O)cc2)CC1
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C(C)C)CC3)c(F)c2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(CC4CCC(=O)N4)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCC(F)(F)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C)CC3)cc2)cnc2c1N(C)CCO2
CCN1CCN(c2ccc(NC(=O)c3c(Nc4cnc5c(c4C)NCCO5)cc[nH]c3=O)cc2F)CC1
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C(C)C)CC3)cc2)cnc2c1NCC(C)(C)O2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(C3CCCN(C)C3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc3c(c2)CCC(=O)N3)cnc2c1NCCO2
CCN1CCN(c2ccc(NC(=O)c3c(Nc4cnc5c(c4C)NCCO5)cc[nH]c3=O)cc2)CC1
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(CCC#N)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C)CC3)c(C(=O)O)c2)cnc2c1NCCO2
COc1ccc(Oc2ccc(NC(=O)c3c(Nc4cnc5c(c4C)NCCO5)cc[nH]c3=O)cc2)cc1
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C(=O)N(C)C)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C4CCC4)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCC(C(=O)O)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C)CC3)c(F)c2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCS(=O)(=O)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc3c(c2)CN(C)C(=O)C3)cnc2c1NCCO2
Cc1cc(NS(C)(=O)=O)ccc1NC(=O)c1c(Nc2cnc3c(c2C)NCCO3)cc[nH]c1=O
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(C3CCN(C)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCNCC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CC4CCC(C3)N4C)cc2)cnc2c1NCC(C)O2
CCN1C(=O)C(C)(C)c2cc(NC(=O)c3c(Nc4cnc5c(c4C)NCCO5)cc[nH]c3=O)ccc21
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc3c(c2)CCCN3)cnc2c1NCCO2
COCCN1CCN(c2ccc(NC(=O)c3c(Nc4cnc5c(c4C)NCCO5)cc[nH]c3=O)cc2)CC1
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C(=O)N(C)C)CC3)cc2)cnc2c1NCC(C)O2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C)[C@@H](C)C3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(-n3ccnc3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCC(C)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C(C)C)CC3)c(F)c2)cnc2c1NCC(C)O2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C)[C@H](C)C3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C4COC4)CC3)cc2)cnc2c1NCCO2
CCCCC(CC)CNC(=O)c1ccc(NC(=O)c2c(Nc3cnc4c(c3C)NCCO4)cc[nH]c2=O)cc1
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(C3CC(=O)N(C)C3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc3c(c2)NC(=O)CO3)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc3nc[nH]c3c2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C(=O)N4CCC(F)(F)C4)CC3)cc2)cnc2c1NCCO2
COCCN1CCN(c2ccc(NC(=O)c3c(Nc4cnc5c(c4C)NCC(C)O5)cc[nH]c3=O)cc2F)CC1
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2cnc(nc12)-c1ccccc1F
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2cnc(nc12)-c1ccccc1C
COc1ccccc1-c1ncc2[nH]nc(-c3ccc(cc3)N3CCN(C)CC3)c2n1
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2cnc(nc12)-c1c(F)cccc1Cl
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2cnc(nc12)-c1cccnc1
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2cnc(nc12)-c1cncc(C)c1
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2cnc(nc12)-c1ccc2CNC(=O)c2c1
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2cnc(nc12)-c1cncc(c1)C(=O)N1CCOCC1
CNC(=O)c1cncc(c1)-c1ncc2[nH]nc(-c3ccc(cc3)N3CCN(C)CC3)c2n1
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2cnc(nc12)-c1cccc2CNCCc12
COc1cccc(F)c1-c1ncc2[nH]nc(-c3ccc(cc3)N3CCN(C)CC3)c2n1
COc1cccc(F)c1-c1ncc2[nH]nc(-c3ccccc3)c2n1
COc1cccc(F)c1-c1ncc2[nH]nc(-c3ccccc3F)c2n1
COc1cccc(F)c1-c1ncc2[nH]nc(-c3cnn(C)c3)c2n1
COc1cccc(F)c1-c1ncc2[nH]nc(-c3ccncc3)c2n1
COc1cccc(F)c1-c1ncc2[nH]nc(-c3cncnc3)c2n1
COc1cccc(F)c1-c1ncc2[nH]nc(-c3ccc(cc3)C#N)c2n1
COc1cccc(F)c1-c1ncc2[nH]nc(-c3ccc(cc3)C(F)(F)F)c2n1
COc1cccc(c1)-c1n[nH]c2cnc(nc12)-c1c(F)cccc1OC
COc1cccc(F)c1-c1ncc2[nH]nc(-c3ccccc3C)c2n1
COc1cccc(F)c1-c1ncc2[nH]nc(-c3ccsc3)c2n1
COc1cccc(F)c1-c1ncc2[nH]nc(-c3ccc(cc3)C(=O)N(C)C)c2n1
COc1cccc(F)c1-c1ncc2[nH]nc(-c3ccc(CN4CCN(C)CC4)cc3)c2n1
COc1cccc(F)c1-c1ncc2[nH]nc(-c3ccc(CN4CCOCC4)cc3)c2n1
COc1cccc(F)c1-c1ncc2[nH]nc(-c3cccc(CN4CCN(C)CC4)c3)c2n1
COc1cccc(F)c1-c1ncc2[nH]nc(-c3ccc(cc3)N3CCOCC3)c2n1
COc1cccc(F)c1-c1ncc2[nH]nc(-c3cccc(c3)N3CCNCC3)c2n1
COc1cccc(F)c1-c1ncc2[nH]nc(-c3cccc(c3)N3CCCC3)c2n1
COc1cccc(F)c1-c1ncc2[nH]nc(-c3cccc(c3)N3CCOCC3)c2n1
COc1cccc(F)c1-c1ncc2[nH]nc(-c3cccc(c3)N(C)C)c2n1
COc1cccc(F)c1-c1ncc2[nH]nc(-c3ccc(cc3)C(=O)N3CCOCC3)c2n1
COc1cccc(F)c1-c1ncc2[nH]nc(-c3ccc(cc3)C(=O)NC3CCCC3)c2n1
COc1cccc(F)c1-c1ncc2[nH]nc(-c3ccc(cc3)C3(CC3)N3CCOCC3)c2n1
COc1cccc(F)c1-c1ncc2[nH]nc(-c3ccc(CC#N)cc3)c2n1
COc1ccc(cc1)-c1n[nH]c2cnc(nc12)-c1c(F)cccc1OC
COc1cccc(F)c1-c1ncc2[nH]nc(-c3ccc(F)cc3)c2n1
CCN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2cnc(nc12)-c1c(F)cccc1OC
CNC(=O)c1ccc(cc1)-c1n[nH]c2cnc(nc12)-c1c(F)cccc1OC
COc1cccc(F)c1-c1ncc2[nH]nc(-c3ccc(cc3)C3CC3)c2n1
COc1cccc(F)c1-c1ncc2[nH]nc(-c3ccc(cc3)N3CCCCC3)c2n1
COc1cccc(F)c1-c1ncc2[nH]nc(-c3ccc(CN)cc3)c2n1
COc1cccc(F)c1-c1ncc2[nH]nc(-c3ccc(cc3)C(C)(C)C#N)c2n1
COc1cccc(F)c1-c1ncc2[nH]nc(-c3ccc(cc3)C3CCOCC3)c2n1
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2cnc(nc12)-c1cccc(F)c1F
COc1ccc(F)c(F)c1-c1ncc2[nH]nc(-c3ccc(cc3)N3CCN(C)CC3)c2n1
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2cnc(nc12)-c1cccc(C(N)=O)c1F
CNC(=O)c1cccc(c1F)-c1ncc2[nH]nc(-c3ccc(cc3)N3CCN(C)CC3)c2n1
COc1cccc(F)c1-c1ncc2[nH]nc(-c3cnn(c3)-c3ccccc3)c2n1
COc1cccc(F)c1-c1ncc2[nH]nc(-c3ccn(C)c(=O)c3)c2n1
COc1cccc(F)c1-c1ncc2[nH]nc(-c3ccnc(c3)N3CCNCC3)c2n1
COc1cccc(F)c1-c1ncc2[nH]nc(-c3ccnc(c3)N3CCN(C)CC3)c2n1
COc1cccc(F)c1-c1ncc2[nH]nc(-c3ccc(nc3)N3CCNCC3)c2n1
COc1cccc(F)c1-c1ncc2[nH]nc(-c3ccc(nc3)N3CCOCC3)c2n1
COc1cccc(F)c1-c1ncc2[nH]nc(-c3ccc(nc3)N3CCN(CC3)C(C)=O)c2n1
COc1cccc(F)c1-c1ncc2[nH]nc(\C=C\c3ccc(cc3)N3CCN(C)CC3)c2n1
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2cnc(nc12)-c1c(F)ccc2CNCCc12
Cc1cccc(F)c1-c1ncc2[nH]nc(-c3ccc(cc3)N3CCCC(O)C3)c2n1
Cc1cccc(F)c1-c1ncc2[nH]nc(-c3ccc(cc3)N3CCC(CC3)C#N)c2n1
Cc1cccc(F)c1-c1ncc2[nH]nc(-c3ccc(cc3)N3CCNCC3)c2n1
Cc1cccc(F)c1-c1ncc2[nH]nc(-c3ccc(cc3)N3CCC(O)C3)c2n1
CNCc1cc(F)c(c(F)c1)-c1ncc2[nH]nc(-c3ccc(nc3)C(=O)NC)c2n1
CNCc1cc(F)c(c(F)c1)-c1ncc2[nH]nc(-c3ccc(C(=O)NC)c(F)c3)c2n1
CNCc1cc(F)c(c(F)c1)-c1ncc2[nH]nc(-c3ccc(OC)cc3)c2n1
CNCc1cc(F)c(c(F)c1)-c1ncc2[nH]nc(-c3cccc(c3)C#N)c2n1
CNCc1cc(F)c(c(F)c1)-c1ncc2[nH]nc(-c3ccc(cc3)C3CCNCC3)c2n1
CNCc1cc(F)c(c(F)c1)-c1ncc2[nH]nc(-c3ccc(cc3)C3CCOCC3)c2n1
CCN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2cnc(nc12)-c1c(F)cc(CNC)cc1F
CNCc1cc(F)c(c(F)c1)-c1ncc2[nH]nc(-c3cnc(N4CCOCC4)c(c3)C#N)c2n1
CNCc1cc(F)c(c(F)c1)-c1ncc2[nH]nc(-c3ccnc(N4CCOCC4)c3F)c2n1
CNCc1cc(F)c(c(F)c1)-c1ncc2[nH]nc(-c3ccc(nc3)N3CCN(CC(C)(C)O)CC3)c2n1
CNCc1cc(F)c(c(F)c1)-c1ncc2[nH]nc(-c3ccc(nc3)N3CCCC(C)(CO)C3)c2n1
CNCc1cc(F)c(c(F)c1)-c1ncc2[nH]nc(-c3ccc(NC4CCN(CC4)S(C)(=O)=O)nc3)c2n1
CNCc1cc(F)c(c(F)c1)-c1ncc2[nH]nc(-c3ccc(cc3)N3CCN(CCO)CC3)c2n1
CNCc1cc(F)c(c(F)c1)-c1ncc2[nH]nc(-c3ccc(nc3)N3CCN(CC3)S(C)(=O)=O)c2n1
CCN(C)C(=O)N1CCN(CC1)c1ccc(cn1)-c1n[nH]c2cnc(nc12)-c1c(F)cc(CNC)cc1F
CNCc1cc(F)c(c(F)c1)-c1ncc2[nH]nc(-c3ccc(nc3)N3CCCCC3)c2n1
CNCc1cc(F)c(-c2ncc3[nH]nc(-c4ccc(nc4)N4CCN(CC4)C(C)=O)c3n2)c(c1)C(F)(F)F
CNCc1cc(C)c(c(F)c1)-c1ncc2[nH]nc(-c3cnn(C)c3)c2n1
CNCc1cc(C)c(c(F)c1)-c1ncc2[nH]nc(-c3cnn(c3)-c3ccccc3C#N)c2n1
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2cnc(nc12)-c1c(C)cc(cc1F)C1CCCN1
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2cnc(nc12)-c1c(C)cc(cc1F)C1CCCCN1
Cn1cc(cn1)-c1n[nH]c2cnc(nc12)-c1c(F)cc(NC(=O)CN2CCCC2)cc1F
CN(C)CC(=O)Nc1cc(F)c(c(F)c1)-c1ncc2[nH]nc(-c3cnn(C)c3)c2n1
CNCc1cc(F)c(c(F)c1)-c1ncc2[nH]nc(-c3cnn(C)c3)c2n1
CNC(C)c1cc(F)c(c(F)c1)-c1ncc2[nH]nc(-c3cnn(C)c3)c2n1
CNCc1cc(F)c(c(OC)c1)-c1ncc2[nH]nc(-c3cnn(C)c3)c2n1
CCNCc1cc(F)c(c(OC)c1)-c1ncc2[nH]nc(-c3cnn(C)c3)c2n1
COc1cccc(F)c1-c1ncc2[nH]nc(-c3cc(C)n[nH]3)c2n1
COc1cccc(F)c1-c1ncc2[nH]nc(OCc3ccccc3)c2n1
CN1CCN(CC1)c1cc(ccn1)-c1n[nH]c2cnc(nc12)-c1c(F)cc2CCNCc2c1F
OCCNc1ncc(cn1)-c1n[nH]c2cnc(nc12)-c1c(F)cc2CCNCc2c1F
CN1CCN(CC1)c1ncc(cn1)-c1n[nH]c2cnc(nc12)-c1c(F)cc2CCNCc2c1F
CN(C)c1ncc(cn1)-c1n[nH]c2cnc(nc12)-c1c(F)cc2CCNCc2c1F
CNc1ncc(cn1)-c1n[nH]c2cnc(nc12)-c1c(F)cc2CCNCc2c1F
CS(=O)(=O)NCc1ccc(cc1)-c1n[nH]c2cnc(nc12)-c1c(F)cc2CCNCc2c1F
Fc1cc2CCNCc2c(F)c1-c1ncc2[nH]nc(-c3ccc(cc3)S(=O)(=O)N3CCC3)c2n1
FC(F)Oc1ccc(cn1)-c1n[nH]c2cnc(nc12)-c1c(F)cc2CCNCc2c1F
Fc1cc2CCNCc2c(F)c1-c1ncc2[nH]nc(-c3ccc(nc3)N3CCOCC3)c2n1
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2cnc(nc12)-c1c(F)cc2CCNCc2c1F
COc1ccc(c2CCNCc12)-c1ncc2[nH]nc(-c3ccc(cc3)N3CCN(C)CC3)c2n1
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2cnc(nc12)-c1ccc2cccnc2c1F
COc1ccncc1-c1ncc2[nH]nc(-c3ccc(cc3)N3CCN(C)CC3)c2n1
COc1ccncc1-c1ncc2[nH]nc(-c3ccc(nc3)N3CCN(C)CC3)c2n1
CNCc1cc(C)c(cn1)-c1ncc2[nH]nc(-c3ccc(cc3)N3CCN(C)CC3)c2n1
CN1CCN(CC1)c1ncc(cn1)-c1n[nH]c2cnc(nc12)-c1c(C)cc(CC#N)cc1F
CN1CCN(Cc2ccc(cc2)-c2n[nH]c3cnc(nc23)-c2c(F)ccc3CNCCc23)CC1
CN1CCN(CC1)c1cc(ccn1)-c1n[nH]c2cnc(nc12)-c1c(F)cc2CCNCc2c1C
CC(=O)N1CCN(CC1)c1ccc(cc1)-c1n[nH]c2cnc(nc12)-c1c(F)cc2CCNCc2c1C
Cc1c2CNCCc2cc(F)c1-c1ncc2[nH]nc(-c3ccc(nc3)N3CCOCC3)c2n1
CN1CCN(CC1)c1ccc(cn1)-c1n[nH]c2cnc(nc12)-c1c(F)cc2CCNCc2c1C
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2cnc(nc12)-c1c(F)cc2CCNCc2c1C
CN1CCN(CC1)c1ccc(cn1)-c1n[nH]c2cnc(nc12)-c1c(C)cc2CCNCc2c1F
CNC1CCc2c1cc(F)c(c2F)-c1ncc2[nH]nc(-c3ccc(nc3)N3CCOCC3)c2n1
CNC1CCc2c1cc(F)c(c2F)-c1ncc2[nH]nc(-c3cnc(nc3)N3CCN(C)CC3)c2n1
CNC1CCc2cc(F)c(c(F)c2C1)-c1ncc2[nH]nc(-c3ccc(nc3)N3CCOCC3)c2n1
CNC1CCCc2c(F)c(c(F)cc12)-c1ncc2[nH]nc(-c3ccc(nc3)N3CCOCC3)c2n1
NC1CCCc2c(F)c(c(F)cc12)-c1ncc2[nH]nc(-c3ccc(nc3)N3CCOCC3)c2n1
NC1CCc2cc(F)c(c(F)c12)-c1ncc2[nH]nc(-c3ccc(nc3)N3CCOCC3)c2n1
COc1c2C(N)CCc2cc(F)c1-c1ncc2[nH]nc(-c3ccc(nc3)N3CCOCC3)c2n1
CNC1CCCc2c1ccc(F)c2-c1ncc2[nH]nc(-c3ccc(nc3)N3CCN(C)CC3)c2n1
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2cnc(nc12)-c1c(F)ccc2C(N)CCCc12
CNCc1cc(F)c(c(F)c1)-c1ncc2[nH]nc(-c3ccc(nc3)N3CCC(C)(O)CC3)c2n1
CNCc1cc(F)c(c(F)c1)-c1ncc2[nH]nc(-c3ccc(cc3)N3CCN(CCOC)CC3)c2n1
CCN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2cnc(nc12)-c1c(F)cc(CNC)cc1C(F)(F)F
CCN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2cnc(nc12)-c1c(C)cc(cc1F)C1CCCCN1
CNCc1cc(F)c(-c2ncc3[nH]nc(-c4ccc(nc4)N4CCO[C@@H](COC)C4)c3n2)c(c1)C(F)(F)F |r|
O=C1NCc2c1c(Nc1ccc(cn1)N1CCNCC1)cnc2-c1c[nH]c2ccccc12
CN1CCN(CC1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2c[nH]c3ccccc23)nc1
O=C1NCc2c1c(Nc1ccc(cn1)N1CCOCC1)cnc2-c1c[nH]c2ccccc12
COc1ccc2c(c[nH]c2c1)-c1ncc(Nc2ccc(cn2)N2CCN(C)CC2)c2C(=O)NCc12
CN1CCN(CC1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2c[nH]c3c(C)cccc23)nc1
CN1CCN(CC1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2c[nH]c3ncccc23)nc1
COc1cccc2c(c[nH]c12)-c1ncc(Nc2ccc(cn2)N2CCN(C)CC2)c2C(=O)NCc12
CN1CCN(CC1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2c[nH]c3cc(C)ccc23)nc1
COc1ccc2[nH]cc(-c3ncc(Nc4ccc(cn4)N4CCN(C)CC4)c4C(=O)NCc34)c2c1
O=C1NCc2c1c(Nc1ccc(cn1)N1CC3CCC(C1)O3)cnc2-c1c[nH]c2ccccc12
CN1CCN(CC1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2c(C)[nH]c3ccccc23)nc1 |(-6.56,7.53,;-5.23,6.76,;-3.89,7.53,;-2.56,6.76,;-2.56,5.22,;-3.89,4.45,;-5.23,5.22,;-1.22,4.45,;.11,5.22,;1.44,4.45,;1.44,2.91,;2.78,2.14,;2.78,.6,;1.44,-.17,;1.44,-1.71,;2.78,-2.48,;4.11,-1.71,;5.57,-2.18,;6.48,-.94,;5.57,.31,;6.05,1.77,;4.11,-.17,;2.78,-4.02,;1.53,-4.92,;.07,-4.45,;2.01,-6.39,;3.55,-6.39,;4.58,-7.53,;6.08,-7.21,;6.56,-5.75,;5.53,-4.6,;4.02,-4.92,;.11,2.14,;-1.22,2.91,)|
FC1(F)CCN(CC1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2c[nH]c3ccccc23)nc1
CN1CCN(CC1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2c[nH]c3ccncc23)nc1
CN1CCN(CC1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2cn(C)c3ncccc23)nc1
CN1CCN(CC1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2c(C)[nH]c3ncccc23)nc1 |(-6.52,7.53,;-5.19,6.76,;-3.85,7.53,;-2.52,6.76,;-2.52,5.22,;-3.85,4.45,;-5.19,5.22,;-1.18,4.45,;-1.18,2.91,;.15,2.14,;1.48,2.91,;2.82,2.14,;2.82,.6,;1.48,-.17,;1.48,-1.71,;2.82,-2.48,;4.15,-1.71,;5.61,-2.18,;6.52,-.94,;5.61,.31,;6.09,1.77,;4.15,-.17,;2.82,-4.02,;4.06,-4.92,;5.53,-4.45,;3.59,-6.39,;2.05,-6.39,;1.02,-7.53,;-.49,-7.21,;-.97,-5.75,;.06,-4.6,;1.57,-4.92,;1.48,4.45,;.15,5.22,)|
CN1CCN(CC1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2c(C)[nH]c3nc(C)ccc23)nc1 |(-6.52,7.94,;-5.19,7.17,;-3.85,7.94,;-2.52,7.17,;-2.52,5.63,;-3.85,4.86,;-5.19,5.63,;-1.18,4.86,;-1.18,3.32,;.15,2.55,;1.48,3.32,;2.82,2.55,;2.82,1.01,;1.48,.24,;1.48,-1.3,;2.82,-2.07,;4.15,-1.3,;5.61,-1.77,;6.52,-.53,;5.61,.72,;6.09,2.18,;4.15,.24,;2.82,-3.61,;4.06,-4.51,;5.53,-4.03,;3.59,-5.98,;2.05,-5.98,;1.02,-7.12,;-.49,-6.8,;-1.52,-7.94,;-.97,-5.34,;.06,-4.19,;1.57,-4.51,;1.48,4.86,;.15,5.63,)|
CN1CCN(CC1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)nc1
CN1CCN(CC1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2ccnc3[nH]cc(C)c23)nc1
CN1CCN(CC1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2ccnc3[nH]ccc23)nc1
CN1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2c[nH]c3ncccc23)nc1
CN1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cn(C)c3ncccc23)nc1
CN1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2c[nH]c3cc(C)ccc23)nc1
CN1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2c[nH]c3ccncc23)nc1
CN1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cccc3nccn23)nc1
CN1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2c[nH]c3cccnc23)nc1
CN1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2c(C)[nH]c3ncccc23)nc1 |(-6.56,7.53,;-5.23,6.76,;-3.89,7.53,;-2.56,6.76,;-2.56,5.22,;-3.89,4.45,;-5.23,5.22,;-1.22,4.45,;-1.22,2.91,;.11,2.14,;1.44,2.91,;2.78,2.14,;2.78,.6,;1.44,-.17,;1.44,-1.71,;2.78,-2.48,;4.11,-1.71,;5.57,-2.18,;6.48,-.94,;5.57,.31,;6.05,1.77,;4.11,-.17,;2.78,-4.02,;1.53,-4.92,;.07,-4.45,;2.01,-6.39,;3.55,-6.39,;4.58,-7.53,;6.08,-7.21,;6.56,-5.75,;5.53,-4.6,;4.02,-4.92,;1.44,4.45,;.11,5.22,)|
COc1ccc2c(c[nH]c2c1)-c1ccc(Nc2ccc(cn2)N2CCN(C)CC2)c2C(=O)NCc12
CN1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2c[nH]c3nc(C)ccc23)nc1
CN1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2c[nH]c3ncc(C)cc23)nc1
CN1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2ccnc3[nH]ccc23)nc1
CN1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2c[nH]c3cc(F)ccc23)nc1
CN1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)nc1
CCc1[nH]c2ccccc2c1-c1ccc(Nc2ccc(cn2)N2CCN(C)CC2)c2C(=O)NCc12 |(-1.08,-5.48,;.07,-4.45,;1.53,-4.92,;2.01,-6.39,;3.55,-6.39,;4.58,-7.53,;6.08,-7.21,;6.56,-5.75,;5.53,-4.6,;4.02,-4.92,;2.78,-4.02,;2.78,-2.48,;1.44,-1.71,;1.44,-.17,;2.78,.6,;2.78,2.14,;1.44,2.91,;.11,2.14,;-1.22,2.91,;-1.22,4.45,;.11,5.22,;1.44,4.45,;-2.56,5.22,;-2.56,6.76,;-3.89,7.53,;-5.23,6.76,;-6.56,7.53,;-5.23,5.22,;-3.89,4.45,;4.11,-.17,;5.57,.31,;6.05,1.77,;6.48,-.94,;5.57,-2.18,;4.11,-1.71,)|
CN1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2ccn3ccnc3c2)nc1
CN1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2ccn3ncnc3c2)nc1
CN1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2c[nH]c3cc(C)ncc23)nc1
CN1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2ccnc3[nH]c(C)cc23)nc1
CN1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3ccccn23)nc1
CN1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2c([nH]c3ccccc23)-c2ccccc2)nc1 |(-6.56,7.53,;-5.23,6.76,;-3.89,7.53,;-2.56,6.76,;-2.56,5.22,;-3.89,4.45,;-5.23,5.22,;-1.22,4.45,;-1.22,2.91,;.11,2.14,;1.44,2.91,;2.78,2.14,;2.78,.6,;1.44,-.17,;1.44,-1.71,;2.78,-2.48,;4.11,-1.71,;5.57,-2.18,;6.48,-.94,;5.57,.31,;6.05,1.77,;4.11,-.17,;2.78,-4.02,;1.53,-4.92,;2.01,-6.39,;3.55,-6.39,;4.58,-7.53,;6.08,-7.21,;6.56,-5.75,;5.53,-4.6,;4.02,-4.92,;.07,-4.45,;-.25,-2.94,;-1.72,-2.46,;-2.86,-3.5,;-2.54,-5,;-1.08,-5.48,;1.44,4.45,;.11,5.22,)|
CN1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cccc3[nH]ccc23)nc1
CN1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2ccnc3[nH]cc(C)c23)nc1
Cn1ccc2c(ccnc12)-c1ccc(Nc2ccc(cn2)N2CCNCC2)c2C(=O)NCc12
CN1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3n(C)ccc3c2)nc1
CN1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3[nH]ccc3c2)nc1
CN1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2c[nH]c3ccccc23)nc1
COCCn1ccc2c(ccnc12)-c1ccc(Nc2ccc(cn2)N2CCN(C)CC2)c2C(=O)NCc12
CC(C)n1ccc2c(ccnc12)-c1ccc(Nc2ccc(cn2)N2CCN(C)CC2)c2C(=O)NCc12
CCn1ccc2c(ccnc12)-c1ccc(Nc2ccc(cn2)N2CCN(C)CC2)c2C(=O)NCc12
CN1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2c(C)nc3ccccn23)nc1 |(-6.56,7.53,;-5.23,6.76,;-3.89,7.53,;-2.56,6.76,;-2.56,5.22,;-3.89,4.45,;-5.23,5.22,;-1.22,4.45,;.11,5.22,;1.44,4.45,;1.44,2.91,;2.78,2.14,;2.78,.6,;1.44,-.17,;1.44,-1.71,;2.78,-2.48,;4.11,-1.71,;5.57,-2.18,;6.48,-.94,;5.57,.31,;6.05,1.77,;4.11,-.17,;2.78,-4.02,;1.53,-4.92,;.07,-4.45,;2.01,-6.39,;3.55,-6.39,;4.58,-7.53,;6.08,-7.21,;6.56,-5.75,;5.53,-4.6,;4.02,-4.92,;.11,2.14,;-1.22,2.91,)|
CN1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3ccc(C)cn23)nc1
CN1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3c(C)cccn23)nc1
CN1CCN(CC1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2c[nH]c3cc(F)ccc23)nc1
CN1CCN(CC1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2ccnc3[nH]c(C)cc23)nc1
CN1CCN(CC1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2cnc3ccccn23)nc1
CNC1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2ccnc3[nH]ccc23)nc1
CNC1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3ccccn23)nc1
CN1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cccnn23)nc1
O=C1NCc2c1c(Nc1ccc(cn1)N1CCNCC1)ccc2-c1cnc2ccccn12
CN1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2ccnc3n(C)ncc23)nc1
CNC1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)nc1
O=C1NCc2c1c(Nc1ccc(cn1)N1CCNCC1)cnc2-c1cnc2ccccn12
CN1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(C)ccn23)nc1
CN1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnn3cc(C)ccc23)nc1
CN1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2ccnc3ccn(C)c23)nc1
CN1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2c(F)cnc3n(C)ccc23)nc1 |(-6.52,7.9,;-5.19,7.13,;-3.85,7.9,;-2.52,7.13,;-2.52,5.59,;-3.85,4.82,;-5.19,5.59,;-1.18,4.82,;.15,5.59,;1.48,4.82,;1.48,3.28,;2.82,2.51,;2.82,.97,;1.48,.2,;1.48,-1.34,;2.82,-2.11,;4.15,-1.34,;5.61,-1.82,;6.52,-.57,;5.61,.68,;6.09,2.14,;4.15,.2,;2.82,-3.65,;1.48,-4.42,;.15,-3.65,;1.48,-5.96,;2.82,-6.73,;4.15,-5.96,;5.61,-6.44,;6.09,-7.9,;6.52,-5.19,;5.61,-3.94,;4.15,-4.42,;.15,2.51,;-1.18,3.28,)|
CN1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2ccnc3NCCc23)nc1
CN1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnn3c(C)cccc23)nc1
Cn1ccc2c(ccnc12)-c1ccc(Nc2ccc(cn2)N2CC3CCC(C2)N3)c2C(=O)NCc12
CNC1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(C)ccn23)nc1
Cc1ccn2c(cnc2c1)-c1ccc(Nc2ccc(cn2)N2CCNCC2)c2C(=O)NCc12
CN1CCN(CC1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2cnc3cc(C)ccn23)nc1
CN1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3c(cccn23)C#N)nc1
Cn1ccc2c(ccnc12)-c1ccc(Nc2ccc(cn2)N2CCC(O)CC2)c2C(=O)NCc12
CN1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cnccn23)nc1
CN1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cc(C)nc3[nH]ccc23)nc1
CN1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2c(C)cnc3[nH]ccc23)nc1 |(-6.52,7.31,;-5.19,6.54,;-3.85,7.31,;-2.52,6.54,;-2.52,5,;-3.85,4.23,;-5.19,5,;-1.18,4.23,;.15,5,;1.48,4.23,;1.48,2.69,;2.82,1.93,;2.82,.38,;1.48,-.38,;1.48,-1.93,;2.82,-2.69,;4.15,-1.93,;5.61,-2.4,;6.52,-1.15,;5.61,.09,;6.09,1.56,;4.15,-.38,;2.82,-4.23,;1.48,-5,;.15,-4.23,;1.48,-6.54,;2.82,-7.31,;4.15,-6.54,;5.61,-7.02,;6.52,-5.78,;5.61,-4.53,;4.15,-5,;.15,1.93,;-1.18,2.69,)|
Cn1ccc2c(ccnc12)-c1ccc(Nc2ccc(cn2)N2CCCNCC2)c2C(=O)NCc12
O=C1NCc2c1c(Nc1ccc(cn1)N1CCNCC1)ccc2-c1cnc2CCCCn12
CN1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2ccnc3cc[nH]c23)nc1
O=C1NCc2c1c(Nc1ccc(cn1)N1CCNCC1)ccc2-c1cnc2cccnn12
CN1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2ncnc3n(C)ccc23)nc1
Cc1cccc2c(cnn12)-c1ccc(Nc2ccc(cn2)N2CCNCC2)c2C(=O)NCc12
CN1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2nnc3ccccn23)nc1
Cc1ccc2ncc(-c3ccc(Nc4ccc(cn4)N4CCNCC4)c4C(=O)NCc34)n2c1
O=C1NCc2c1c(Nc1ccc(cn1)N1CCNCC1)ccc2-c1cnc2ncccn12
Fc1cccn2c(cnc12)-c1ccc(Nc2ccc(cn2)N2CCNCC2)c2C(=O)NCc12
O=C1NCc2c1c(Nc1ccc(cn1)N1CCNCC1)ccc2-c1cnn2ccccc12
CNC1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cccnn23)nc1
CN1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3CNCCn23)nc1
Cn1ccc2c(ccnc12)-c1ccc(Nc2ccc(cn2)N2CCC[C@H](N)C2)c2C(=O)NCc12 |r|
Cn1ccc2c(ccnc12)-c1ccc(Nc2ccc(cn2)N2CCC[C@@H](N)C2)c2C(=O)NCc12 |r|
CN[C@H]1CCCN(C1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)nc1 |r|
Cc1cn(C)c2nccc(-c3ccc(Nc4ccc(cn4)N4CCNCC4)c4C(=O)NCc34)c12
Cc1cnc2n(C)ccc2c1-c1ccc(Nc2ccc(cn2)N2CCNCC2)c2C(=O)NCc12 |(-.52,-3.65,;.82,-4.42,;.82,-5.96,;2.15,-6.73,;3.48,-5.96,;4.95,-6.44,;5.42,-7.9,;5.85,-5.19,;4.95,-3.94,;3.48,-4.42,;2.15,-3.65,;2.15,-2.11,;.82,-1.34,;.82,.2,;2.15,.97,;2.15,2.51,;.82,3.28,;-.52,2.51,;-1.85,3.28,;-1.85,4.82,;-.52,5.59,;.82,4.82,;-3.19,5.59,;-3.19,7.13,;-4.52,7.9,;-5.85,7.13,;-5.85,5.59,;-4.52,4.82,;3.48,.2,;4.95,.68,;5.42,2.14,;5.85,-.57,;4.95,-1.82,;3.48,-1.34,)|
CN[C@@H]1CCCN(C1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)nc1 |r|
O=C1NCc2c1c(Nc1ccc(cn1)N1CC3CCC(C1)N3)ccc2-c1cnc2ccccn12
Cn1ccc2c(cccc12)-c1ccc(Nc2ccc(cn2)N2CCNCC2)c2C(=O)NCc12
Cc1cc(-c2ccc(Nc3ccc(cn3)N3CCNCC3)c3C(=O)NCc23)c2ccn(C)c2n1
O=C1NCc2c1c(Nc1ccc(cn1)N1CCCNCC1)ccc2-c1cnc2ccccn12
CN1CCOc2c(ccnc12)-c1ccc(Nc2ccc(cn2)N2CCNCC2)c2C(=O)NCc12
Cn1ccc2c(ccnc12)-c1ccc(Nc2ccc(cn2)S(C)(=O)=O)c2C(=O)NCc12
O=C1NCc2c1c(Nc1ccc(cn1)N1CCNCC1)ccc2-c1ccnc2ccsc12
Cn1ccc2c(ccnc12)-c1ccc(Nc2ccc(cn2)C2CCOC2)c2C(=O)NCc12
CCNC(=O)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)nc1
Cn1ccc2c(ccnc12)-c1ccc(Nc2ccc(cn2)N2CCOCC2)c2C(=O)NCc12
CN1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnn3cc(C)cnc23)nc1
CN1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnn3cccnc23)nc1
CN1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnn3ccncc23)nc1
Cn1cnc2nccc(-c3ccc(Nc4ccc(cn4)N4CCNCC4)c4C(=O)NCc34)c12
Cn1ccc2c(ccnc12)-c1ccc(Nc2cc(n[nH]2)C2CCNCC2)c2C(=O)NCc12
Cn1ccc2c(ccnc12)-c1ccc(Nc2ccc(cn2)N2CCC[C@H](O)C2)c2C(=O)NCc12 |r|
O=C1NCc2c1c(Nc1ccc(cn1)N1CCNCC1)ccc2-c1cnn2cccnc12
CN1CCCc2c(ccnc12)-c1ccc(Nc2ccc(cn2)N2CCNCC2)c2C(=O)NCc12
FC(F)n1ccc2c(ccnc12)-c1ccc(Nc2ccc(cn2)N2CCNCC2)c2C(=O)NCc12
O=C1NCc2c1c(Nc1ccc(cn1)N1CCNCC1)ccc2-c1cnc2cc(ccn12)C#N
Cn1ccc2c(ccnc12)-c1ccc(Nc2ccc(cn2)N2CCC[C@@H](O)C2)c2C(=O)NCc12 |r|
Cn1cnc2c(cccc12)-c1ccc(Nc2ccc(cn2)N2CCNCC2)c2C(=O)NCc12
Cn1ccc2c(ncnc12)-c1ccc(Nc2ccc(cn2)N2CCNCC2)c2C(=O)NCc12
Cc1ccn2c(cnc2c1)-c1ncc(Nc2ccc(cn2)N2CCNCC2)c2C(=O)NCc12
Cc1ccn2c(cnc2c1)-c1ccc(Nc2ccc(cn2)N2CCC(O)CC2)c2C(=O)NCc12
O=C1NCc2c1c(Nc1ccc(cn1)N1CCNCC1)ccc2-c1ccnc2ccnn12
CN1CCN(CC1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2c(F)cnc3n(C)ccc23)nc1 |(-6.52,7.9,;-5.19,7.13,;-3.85,7.9,;-2.52,7.13,;-2.52,5.59,;-3.85,4.82,;-5.19,5.59,;-1.18,4.82,;.15,5.59,;1.48,4.82,;1.48,3.28,;2.82,2.51,;2.82,.97,;1.48,.2,;1.48,-1.34,;2.82,-2.11,;4.15,-1.34,;5.61,-1.82,;6.52,-.57,;5.61,.68,;6.09,2.14,;4.15,.2,;2.82,-3.65,;1.48,-4.42,;.15,-3.65,;1.48,-5.96,;2.82,-6.73,;4.15,-5.96,;5.61,-6.44,;6.09,-7.9,;6.52,-5.19,;5.61,-3.94,;4.15,-4.42,;.15,2.51,;-1.18,3.28,)|
Cn1nc(Nc2ccc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)cc1C1CCOCC1
OC1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3c(F)cccn23)nc1
OC1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnn3ccccc23)nc1
OC1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3ccc(cn23)C(F)(F)F)nc1
OC1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cnccn23)nc1
Cc1ccc2ncc(-c3ccc(Nc4ccc(cn4)N4CCC(O)CC4)c4C(=O)NCc34)n2c1
Cc1cccn2c(cnc12)-c1ccc(Nc2ccc(cn2)N2CCC(O)CC2)c2C(=O)NCc12
Cc1cccc2c(cnn12)-c1ccc(Nc2ccc(cn2)N2CCC(O)CC2)c2C(=O)NCc12
Cc1ccc2c(cnn2c1)-c1ccc(Nc2ccc(cn2)N2CCC(O)CC2)c2C(=O)NCc12
OC1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnn3cc(F)ccc23)nc1
Cn1ccc2c(ccnc12)-c1ncc(Nc2ccc(cn2)N2CCC(O)CC2)c2C(=O)NCc12
OC1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(ccn23)C(F)(F)F)nc1
CN1CCN(CC1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2c([nH]c3ccccc23)-c2ccccc2)nc1 |(-7.49,7.53,;-6.15,6.76,;-4.82,7.53,;-3.49,6.76,;-3.49,5.22,;-4.82,4.45,;-6.15,5.22,;-2.15,4.45,;-2.15,2.91,;-.82,2.14,;.51,2.91,;1.85,2.14,;1.85,.6,;.51,-.17,;.51,-1.71,;1.85,-2.48,;3.18,-1.71,;4.65,-2.18,;5.55,-.94,;4.65,.31,;5.12,1.77,;3.18,-.17,;1.85,-4.02,;3.09,-4.92,;2.62,-6.39,;1.08,-6.39,;.05,-7.53,;-1.46,-7.21,;-1.93,-5.75,;-.9,-4.6,;.6,-4.92,;4.56,-4.45,;5.7,-5.48,;7.17,-5,;7.49,-3.5,;6.34,-2.46,;4.88,-2.94,;.51,4.45,;-.82,5.22,)|
COc1ccc2ncc(-c3ccc(Nc4ccc(cn4)N4CCC(O)CC4)c4C(=O)NCc34)n2c1
OC1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3COCCn23)nc1
Cn1ccc2C(NC=Nc12)c1ccc(Nc2ccc(cn2)N2CCC(O)CC2)c2C(=O)NCc12 |c:7|
Cc1ccn2c(cnc2c1)-c1ccc(Nc2ccc(cn2)N2CCOCC2)c2C(=O)NCc12
CCNC(=O)C(C)(C)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)nc1
Cn1ccc2c(ccnc12)-c1ccc(Nc2cccc(n2)N2CCC(O)CC2)c2C(=O)NCc12
Cc1ccn2c(cnc2c1)-c1ccc(Nc2ccc(cn2)S(C)(=O)=O)c2C(=O)NCc12
OC1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3c(cccn23)C(F)(F)F)nc1
OC1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnn3CC(CCc23)C(=O)NC2CC2)nc1
Cc1ccn2c(cnc2c1F)-c1ccc(Nc2ccc(cn2)N2CCC(O)CC2)c2C(=O)NCc12
Cn1cnc2c(ccnc12)-c1ccc(Nc2ccc(cn2)N2CCC(O)CC2)c2C(=O)NCc12
O=C1NCc2c1c(Nc1ccc(cn1)N1CCOCC1)ccc2-c1cnc2cnccn12
Cc1ccn2c(cnc2c1)-c1ncc(Nc2ccc(cn2)N2CCC(O)CC2)c2C(=O)NCc12
Cc1ccn2c(cnc2c1)-c1ccc(Nc2ccc(cn2)C2CCOC2)c2C(=O)NCc12
Fc1cccn2c(cnc12)-c1ccc(Nc2ccc(cn2)N2CCOCC2)c2C(=O)NCc12
OC1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnn3cccnc23)nc1
Cc1nccn2c(cnc12)-c1ccc(Nc2ccc(cn2)N2CCC(O)CC2)c2C(=O)NCc12
Fc1ccn2c(cnc2c1)-c1ccc(Nc2ccc(cn2)N2CCOCC2)c2C(=O)NCc12
OC1CCN(CC1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2cnc3ccccn23)nc1
Cn1ccc2c(cccc12)-c1ccc(Nc2ccc(cn2)N2CCC(O)CC2)c2C(=O)NCc12
OC1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cccnn23)nc1
Cc1ccn2c(cnc2c1)-c1ncc(Nc2ccc(cn2)N2CCOCC2)c2C(=O)NCc12
COc1ccn2c(cnc2c1)-c1ccc(Nc2ccc(cn2)N2CCC(O)CC2)c2C(=O)NCc12
Cc1cnn2c(ccnc12)-c1ccc(Nc2ccc(cn2)N2CCC(O)CC2)c2C(=O)NCc12
COc1cccn2c(cnc12)-c1ccc(Nc2ccc(cn2)N2CCC(O)CC2)c2C(=O)NCc12
OC1CCN(CC1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1
Cn1ccn2c(cnc2c1=O)-c1ccc(Nc2ccc(cn2)N2CCC(O)CC2)c2C(=O)NCc12
O[C@H]1CCCN(C1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cnccn23)nc1 |r|
Cc1ccn2c(cnc2c1)-c1ccc(Nc2ccc(cn2)N2CCC[C@H](O)C2)c2C(=O)NCc12 |r|
O[C@@H]1CCCN(C1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cnccn23)nc1 |r|
Cc1ccn2c(cnc2c1)-c1ccc(Nc2ccc(cn2)N2CCC[C@@H](O)C2)c2C(=O)NCc12 |r|
Cn1cnc2c(cccc12)-c1ccc(Nc2ccc(cn2)N2CCC(O)CC2)c2C(=O)NCc12
O[C@@H]1CCCN(C1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1 |r|
O[C@H]1CCCN(C1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1 |r|
Cc1ccn2c(cnc2c1C)-c1ccc(Nc2ccc(cn2)N2CCC(O)CC2)c2C(=O)NCc12
[#8][I][#6]-c1ccn2c(cnc2c1)-c1ccc(-[#7]-c2ccc(cn2)-[#7]-2-[#6]-[#6]-[#6](-[#8])-[#6]-[#6]-2)c2-[#6](=O)-[#7]-[#6]-c12
Cn1ccc2c(ccnc12)-c1ncc(Nc2ccc(cn2)N2CCC[C@@H](O)C2)c2C(=O)NCc12 |r|
Cn1ccc2c(ccnc12)-c1ncc(Nc2ccc(cn2)N2CCC[C@H](O)C2)c2C(=O)NCc12 |r|
Cc1ncc2c(cccn12)-c1ccc(Nc2ccc(cn2)N2CCC(O)CC2)c2C(=O)NCc12
OC1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(ccn23)C2CC2)nc1
OC1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(ccn23)C#N)nc1
O=C1NCc2c1c(Nc1ccc(cn1)N1CCOCC1)ccc2-c1cnc2cc(ccn12)C#N
Cc1cnn2c(cnc2c1)-c1ccc(Nc2ccc(cn2)N2CCC(O)CC2)c2C(=O)NCc12
CCOc1c(ccn2c(cnc12)-c1ccc(Nc2ccc(cn2)N2CCC(O)CC2)c2C(=O)NCc12)C#N
OC1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(Cl)ccn23)nc1
OC1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3c(F)c(ccn23)C#N)nc1
O=C1NCc2c1c(Nc1ccc(cn1)N1CCOCC1)cnc2-c1cnc2cc(ccn12)C#N
Cn1ccc2c(ccnc12)-c1c2CNC(=O)c2c(Nc2ccc(cn2)N2CCC(O)CC2)cc1Cl |(6.09,-7.9,;5.61,-6.44,;6.52,-5.19,;5.61,-3.94,;4.15,-4.42,;2.82,-3.65,;1.48,-4.42,;1.48,-5.96,;2.82,-6.73,;4.15,-5.96,;2.82,-2.11,;4.15,-1.34,;5.61,-1.82,;6.52,-.57,;5.61,.68,;6.09,2.14,;4.15,.2,;2.82,.97,;2.82,2.51,;1.48,3.28,;1.48,4.82,;.15,5.59,;-1.18,4.82,;-1.18,3.28,;.15,2.51,;-2.52,5.59,;-2.52,7.13,;-3.85,7.9,;-5.19,7.13,;-6.52,7.9,;-5.19,5.59,;-3.85,4.82,;1.48,.2,;1.48,-1.34,;.15,-2.11,)|
Cc1ccn2c(cnc2c1)-c1ccc(Nc2ccc(cn2)[C@H]2CCOC2)c2C(=O)NCc12 |r|
Cc1ccn2c(cnc2c1)-c1ccc(Nc2ccc(cn2)[C@@H]2CCOC2)c2C(=O)NCc12 |r|
OC1CCN(CC1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2ccnc3[nH]ccc23)nc1
OC1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(ccn23)C(F)F)nc1
CCNC(=O)c1ccn2c(cnc2c1)-c1ccc(Nc2ccc(cn2)N2CCC(O)CC2)c2C(=O)NCc12
OCc1ccn2c(cnc2c1)-c1ccc(Nc2ccc(cn2)N2CCOCC2)c2C(=O)NCc12
Cn1ccc2c(ccnc12)-c1c2CNC(=O)c2c(Nc2ccc(cn2)N2CCC(O)CC2)cc1F |(6.09,-7.9,;5.61,-6.44,;6.52,-5.19,;5.61,-3.94,;4.15,-4.42,;2.82,-3.65,;1.48,-4.42,;1.48,-5.96,;2.82,-6.73,;4.15,-5.96,;2.82,-2.11,;4.15,-1.34,;5.61,-1.82,;6.52,-.57,;5.61,.68,;6.09,2.14,;4.15,.2,;2.82,.97,;2.82,2.51,;1.48,3.28,;1.48,4.82,;.15,5.59,;-1.18,4.82,;-1.18,3.28,;.15,2.51,;-2.52,5.59,;-2.52,7.13,;-3.85,7.9,;-5.19,7.13,;-6.52,7.9,;-5.19,5.59,;-3.85,4.82,;1.48,.2,;1.48,-1.34,;.15,-2.11,)|
OC1CCN(CC1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2cnc3cccnn23)nc1
OC1CCN(CC1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2ccnc3n(ccc23)C(F)F)nc1
OCCOc1ccn2c(cnc2c1)-c1ccc(Nc2ccc(cn2)N2CCOCC2)c2C(=O)NCc12
CC(C)(O)[C@@H]1CCCN(C1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1 |r|
OC(=O)C1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1
OCC1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1
COCCNc1ccn2c(cnc2c1)-c1ccc(Nc2ccc(cn2)N2CCC(O)CC2)c2C(=O)NCc12
COCCNc1ccn2c(cnc2c1)-c1ccc(Nc2ccc(cn2)N2CCOCC2)c2C(=O)NCc12
CCNC(=O)c1ccn2c(cnc2c1)-c1ccc(Nc2ccc(cn2)N2CCOCC2)c2C(=O)NCc12
OC1CCN(CC1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2cnc3cnccn23)nc1
Cc1c(F)ccn2c(cnc12)-c1ccc(Nc2ccc(cn2)N2CCC(O)CC2)c2C(=O)NCc12
CC(C)(O)[C@H]1CCCN(C1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2cnc3ccccn23)nc1 |r|
Cn1ccc2c(ccnc12)-c1ncc(Nc2ccc(cn2)N2CCC[C@@H](C2)C(C)(C)O)c2C(=O)NCc12 |r|
Cn1ccc2c(ccnc12)-c1ncc(Nc2ccc(cn2)N2CCC[C@H](C2)C(C)(C)O)c2C(=O)NCc12 |r|
CC(C)(O)[C@H]1CCCN(C1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1 |r|
C[C@H](O)C1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1 |r|
Cc1cnc2c(cccn12)-c1ccc(Nc2ccc(cn2)N2CCC(O)CC2)c2C(=O)NCc12
Cn1ccc2c(cccc12)-c1ncc(Nc2ccc(cn2)N2CCC[C@@H](C2)C(C)(C)O)c2C(=O)NCc12 |r|
Cn1ccc2c(ccnc12)-c1ncc(Nc2ccc(cn2)[C@H]2CCOC2)c2C(=O)NCc12 |r|
Fc1ccn2c(cnc2c1)-c1ccc(Nc2ccc(cn2)[C@H]2CCOC2)c2C(=O)NCc12 |r|
Cn1ccc2c(ccnc12)-c1ncc(Nc2ccc(cn2)[C@@H]2CCOC2)c2C(=O)NCc12 |r|
CC(C)(O)[C@@H]1CCCN(C1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2cnc3ccccn23)nc1 |r|
Cn1ccc2c(cccc12)-c1ncc(Nc2ccc(cn2)N2CCOCC2)c2C(=O)NCc12
Fc1ccn2c(cnc2c1)-c1ccc(Nc2ccc(cn2)[C@@H]2CCOC2)c2C(=O)NCc12 |r|
Cn1ccc2c(cccc12)-c1ncc(Nc2ccc(cn2)N2CCC[C@H](C2)C(C)(C)O)c2C(=O)NCc12 |r|
CC(C)(O)C1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1
Cc1ccn2c(cnc2n1)-c1ccc(Nc2ccc(cn2)N2CCC[C@@H](C2)C(C)(C)O)c2C(=O)NCc12 |r|
CC(C)(O)[C@@H]1CCCN(C1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1 |r|
CN(C)CCNC(=O)C(C)(C)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1
CNC1CCN(CC1)c1cccc(Nc2cnc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)n1
Cc1cc2c(ccnc2n1C)-c1ncc(Nc2ccc(cn2)N2CCC[C@@H](C2)C(C)(C)O)c2C(=O)NCc12 |r|
CN1CCN(CC1)c1cccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)n1
Cn1ccc2c(ccnc12)-c1ncc(Nc2cccc(n2)N2CCC[C@@H](N)C2)c2C(=O)NCc12 |r|
Cn1ccc2c(ccnc12)-c1ncc(Nc2cccc(n2)N2CCNCC2)c2C(=O)NCc12
Cc1ccn2c(cnc2n1)-c1ccc(Nc2ccc(cn2)N2CCC[C@H](C2)C(C)(C)O)c2C(=O)NCc12 |r|
CN1CCN(CC1)c1cccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cnccn23)n1
COCCN(C)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1
CN1CCN(CC1)c1cccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(Cl)ccn23)n1
Cc1cc2c(ccnc2n1C)-c1ncc(Nc2ccc(cn2)N2CCC[C@H](C2)C(C)(C)O)c2C(=O)NCc12 |r|
Fc1ccn2c(cnc2c1)-c1ccc(Nc2ccc(CN3CCOCC3)cn2)c2C(=O)NCc12
CN[C@@H]1CCCN(C1)c1cccc(Nc2cnc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)n1 |r|
Cn1ccc2c(ccnc12)-c1ncc(Nc2cccc(n2)N2CCCNCC2)c2C(=O)NCc12
Cc1cccn2c(cnc12)-c1ncc(Nc2ccc(cn2)N2CCC[C@@H](C2)C(C)(C)O)c2C(=O)NCc12 |r|
COc1c(F)ccn2c(cnc12)-c1ccc(Nc2ccc(cn2)N2CCC(O)CC2)c2C(=O)NCc12
CC(C)(O)[C@H]1CCCN(C1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2cnc3c(F)cccn23)nc1 |r|
CNC1(C)CCN(CC1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)nc1
CN[C@H]1CCN(C1)c1cccc(Nc2cnc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)n1 |r|
CN(C)CCN(C)c1cccc(Nc2cnc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)n1
CN1CCN(CC1)c1cccc(Nc2ccc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)n1
Cc1nc2ccccn2c1-c1ncc(Nc2ccc(cn2)N2CCC(O)CC2)c2C(=O)NCc12 |(.07,-4.45,;1.53,-4.92,;2.01,-6.39,;3.55,-6.39,;4.58,-7.53,;6.08,-7.21,;6.56,-5.75,;5.53,-4.6,;4.02,-4.92,;2.78,-4.02,;2.78,-2.48,;1.44,-1.71,;1.44,-.17,;2.78,.6,;2.78,2.14,;1.44,2.91,;1.44,4.45,;.11,5.22,;-1.22,4.45,;-1.22,2.91,;.11,2.14,;-2.56,5.22,;-3.89,4.45,;-5.23,5.22,;-5.23,6.76,;-6.56,7.53,;-3.89,7.53,;-2.56,6.76,;4.11,-.17,;5.57,.31,;6.05,1.77,;6.48,-.94,;5.57,-2.18,;4.11,-1.71,)|
CN(C)CCOc1ccn2c(cnc2c1)-c1ccc(Nc2ccc(cn2)N2CCC(F)C(O)C2)c2C(=O)NCc12
CN1CCN(CC1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2c[nH]c3cc(O)ccc23)nc1
CN1CCN(CC1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2cccc3n(C)ccc23)nc1
CN1CCN(CC1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2cccc3[nH]ccc23)nc1
CN1CCN(CC1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2c[nH]c3nc(ccc23)C(F)(F)F)nc1
CN1CCN(CC1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2cnn3CCCc23)nc1
CN1CCN(CC1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2cnn3CCCCc23)nc1
CN1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2ccn3ncccc23)nc1
CN1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2ccnc3n(Cc4ccccc4)ccc23)nc1
Cn1ccc2c(ccnc12)-c1ncc(Nc2ccc(cn2)N2CCNCC2)c2C(=O)NCc12
C[C@@H]1COc2c(cnn2C1)-c1ccc(Nc2ccc(cn2)N2CCN(C)CC2)c2C(=O)NCc12 |r|
CN1CCN(CC1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2c[nH]c3cc(OCc4ccccc4)ccc23)nc1
Cn1ccc2c(ccnc12)-c1ncc(Nc2ccc(cn2)N2CC3CCC(C2)N3)c2C(=O)NCc12
C[C@@H]1CCn2ncc(c2C1)-c1ccc(Nc2ccc(cn2)N2CCN(C)CC2)c2C(=O)NCc12 |r|
C[C@H]1CCn2ncc(c2C1)-c1ccc(Nc2ccc(cn2)N2CCN(C)CC2)c2C(=O)NCc12 |r|
CN1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2ccnc3n(ccc23)C2CC2)nc1
COc1cc(cnc1Nc1ccc(c2CNC(=O)c12)-c1ccnc2n(C)ccc12)N1CCC(O)CC1
CN1CCN(CC1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2cnc3CCCn23)nc1
CN1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2ccnc3n(CC(N)=O)ccc23)nc1
CN1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2ccnc3ocnc23)nc1
CN1CCC(CC1=O)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)nc1
Cn1ccc2c(ccnc12)-c1ccc(Nc2ccc(cn2)C2(C)CCNCC2)c2C(=O)NCc12
Cn1ccc2c(ccnc12)-c1ccc(Nc2ccc(cn2)N2CCNCC2)c2C(=O)NC(C)(C)c12
CN1CCC(O)(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)nc1
CN1CCC(C)(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)nc1
Cn1ccc2c(ccnc12)-c1ncc(Nc2ccc(cn2)N2CCOCC2)c2C(=O)NCc12
Cn1ccc2c(ccnc12)-c1ccc(Nc2ccc(cn2)N2CC[C@@H](O)C2)c2C(=O)NCc12 |r|
Cn1ccc2c(cccc12)-c1ncc(Nc2ccc(cn2)N2CCC(O)CC2)c2C(=O)NCc12
Cn1ccc2c(ccnc12)-c1ccc(Nc2ccc(cn2)N2CCC[C@@H](C2)C(C)(C)O)c2C(=O)NCc12 |r|
Cn1ccc2c(ccnc12)-c1ccc(Nc2ccc(cn2)N2CCC[C@H](C2)C(C)(C)O)c2C(=O)NCc12 |r|
Cn1ccc2c(ccnc12)-c1ccc(Nc2ccc(cn2)N2CCC(O)CC2)c2C(=O)NC(C)(C)c12
OC1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnn3CCCCCc23)nc1
OC1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnn3CCCCc23)nc1
Cn1ccc2c(ccnc12)-c1ccc(Nc2ccc(cn2)N2CC[C@H](O)C2)c2C(=O)NCc12 |r|
C[C@H]1NC(=O)c2c1c(ccc2Nc1ccc(cn1)N1CCC(O)CC1)-c1ccnc2N(C)CCc12 |r|
C[C@@H]1NC(=O)c2c1c(ccc2Nc1ccc(cn1)N1CCC(O)CC1)-c1ccnc2N(C)CCc12 |r|
OC1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3CCCCCn23)nc1
Cn1ccc2c(ccnc12)-c1ncc(Nc2ccc(cn2)N2C[C@H]3C[C@@H]2CO3)c2C(=O)NCc12 |r|
CN1CCc2cc(nn2CC1=O)-c1ccc(Nc2ccc(cn2)N2CCC(O)CC2)c2C(=O)NCc12
Cn1ccc2c(ccnc12)-c1ccc(Nc2ccc(cn2)N2CCC(O)(CN3CCOCC3)CC2)c2C(=O)NCc12
Cc1cc(Nc2ccc(cn2)N2CCC(O)CC2)c2C(=O)NCc2c1-c1cccc2n(C)ccc12 |(-.18,-2.07,;-1.51,-1.3,;-1.51,.24,;-2.84,1.01,;-2.84,2.55,;-1.47,3.24,;-.14,2.47,;1.2,3.24,;1.2,4.78,;-.14,5.55,;-1.47,4.78,;2.53,5.55,;3.88,4.78,;5.21,5.55,;5.21,7.09,;6.55,7.86,;3.88,7.86,;2.55,7.09,;-4.18,.24,;-5.64,.71,;-6.12,2.18,;-6.55,-.53,;-5.64,-1.78,;-4.18,-1.3,;-2.84,-2.07,;-2.84,-3.61,;-1.51,-4.38,;-1.51,-5.92,;-2.84,-6.69,;-4.18,-5.92,;-5.64,-6.4,;-6.12,-7.86,;-6.55,-5.15,;-5.64,-3.91,;-4.18,-4.38,)|
Cn1ccc2c(ccnc12)-c1ccc(Nc2ccc(CS(C)(=O)=O)cn2)c2C(=O)NCc12
CN1CCc2cc(Nc3ccc(c4CNC(=O)c34)-c3ccnc4n(C)ccc34)nn2CC1=O
COc1cc(Nc2ccc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)ncc1N1CCC(O)CC1
OC1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3CCCCn23)nc1
Cn1ccc2c(ccnc12)-c1ccc(Nc2ccc(cn2)N2CC3(CC(O)C3)C2)c2C(=O)NCc12
COCC1(O)CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)nc1
Cn1ccc2c(ccnc12)-c1ccc(Nc2ccc(cn2)N2CCC3(COC3)CC2)c2C(=O)NCc12
O=C1NCc2c1c(Nc1ccc(cn1)N1CCCOCC1)ccc2-c1cnc2cnccn12
OC1CCCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cnccn23)nc1
C[C@@H]1CCn2c(C1)ncc2-c1ccc(Nc2ccc(cn2)N2CCC(O)CC2)c2C(=O)NCc12 |r|
C[C@H]1CCn2c(C1)ncc2-c1ccc(Nc2ccc(cn2)N2CCC(O)CC2)c2C(=O)NCc12 |r|
Cc1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cnccn23)nc1
Cn1ccc2c(ccnc12)-c1ccc(c2C(=O)NCc12)-n1ccc(n1)N1CCC[C@@](C)(O)C1 |r|
Cn1ccc2c(ccnc12)-c1ccc(c2C(=O)NCc12)-n1ccc(n1)N1CCC[C@](C)(O)C1 |r|
O=C1NCc2c1c(Nc1ccc(cn1)S(=O)(=O)N1CCC1)ccc2-c1cnc2cnccn12
Cn1ccc2c(ccnc12)-c1ccc(c2C(=O)NCc12)-n1ccc(n1)N1CCC(O)CC1
Cn1ccc2c(ccnc12)-c1ncc(Nc2ccc(cn2)N2C[C@@H]3C[C@H]2CO3)c2C(=O)NCc12 |r|
CC(C)(O)[C@H]1CCCN(C1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cnccn23)nc1 |r|
CC(C)(O)[C@@H]1CCCN(C1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cnccn23)nc1 |r|
O=C1NCc2c1c(Nc1ccc(cn1)N1CC3(COC3)C1)ccc2-c1cnc2cnccn12
CC1(O)CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cnccn23)nc1
C[C@H]1COCCN1c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cnccn23)nc1 |r|
OC1CN(C1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cnccn23)nc1
C[C@@H]1NC(=O)c2c1c(ccc2Nc1ccc(cn1)N1CCC(O)CC1)-c1cnc2ccccn12 |r|
C[C@H]1NC(=O)c2c1c(ccc2Nc1ccc(cn1)N1CCC(O)CC1)-c1cnc2ccccn12 |r|
O=C1NCc2c1c(Nc1ccc(cn1)N1C[C@@H]3COC[C@@H]3C1)ccc2-c1cnc2cnccn12 |r|
CC(C)N1CCN(CC1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)nc1
Fc1ccn2c(cnc2c1)-c1ccc(Nc2ccc(cn2)S(=O)(=O)CC2CCC2)c2C(=O)NCc12
OC1CN(C1)c1cccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)n1
OC1CCN(CC1)c1ccnc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cnccn23)c1
CN1C[C@H](CCC1=O)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cnccn23)nc1 |r|
CN1C[C@@H](CCC1=O)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cnccn23)nc1 |r|
CN1CCN(CC1)c1cccc(Nc2cnc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)n1
O[C@H]1CCCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cnccn23)nc1 |r|
O[C@@H]1CCCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cnccn23)nc1 |r|
OC1CCN(CC1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2cnn3CCCCc23)nc1
CN1CC(CC1=O)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cnccn23)nc1
COC[C@H]1CN(CCO1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cnccn23)nc1 |r|
COC[C@@H]1CN(CCO1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cnccn23)nc1 |r|
Fc1ccn2c(cnc2c1)-c1ccc(Nc2ccc(cn2)N2CCOCC22CC2)c2C(=O)NCc12
CN1CCC(C1=O)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1
O[C@H]1COCCN(C1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1 |r|
O[C@@H]1COCCN(C1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1 |r|
Fc1ccn2c(cnc2c1)-c1ccc(Nc2cccc(n2)N2CCCC2=O)c2C(=O)NCc12
Cn1ccc2c(ccnc12)-c1ncc(Nc2ccc(cn2)N2CCC(O)(CN3CCOCC3)CC2)c2C(=O)NCc12
CC(C)(O)[C@@H]1CN(CCO1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1 |r|
CC(C)(O)[C@H]1CN(CCO1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1 |r|
O[C@H]1CN(CC[C@@H]1F)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1 |r|
O[C@@H]1CN(CC[C@H]1F)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1 |r|
OC1(CN2CCOCC2)CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1
C[C@H]1C[C@@H](O)CCN1c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cnccn23)nc1 |r|
C[C@@H]1C[C@H](O)CCN1c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cnccn23)nc1 |r|
C[C@@H]1C[C@@H](O)CCN1c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cnccn23)nc1 |r|
C[C@H]1C[C@H](O)CCN1c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cnccn23)nc1 |r|
O[C@H]1CCC[C@H]1Oc1cccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)n1 |r|
O[C@@H]1CCC[C@@H]1Oc1cccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)n1 |r|
CC(C)(O)[C@H]1CCCN(C1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2cnn3CCCCc23)nc1 |r|
C[C@H](O)[C@H]1CCCN(C1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1 |r|
C[C@@H](O)[C@@H]1CCCN(C1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1 |r|
OCC1CN(CCO1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cnccn23)nc1
O[C@@H]1CN(CC[C@@H]1F)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1 |r|
Cc1csc2c(ccnc12)-c1ccc(Nc2ccc(cn2)N2CCC(O)CC2)c2C(=O)NCc12
Cn1ccc2c(cnc2c1)-c1ccc(Nc2ccc(cn2)N2CCC(O)CC2)c2C(=O)NCc12
C[C@H](O)[C@@H]1CCCN(C1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1 |r|
C[C@@H](O)[C@H]1CCCN(C1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1 |r|
CN1CCN(CC2(O)CCN(CC2)c2ccc(Nc3ccc(c4CNC(=O)c34)-c3cnc4cc(F)ccn34)nc2)CC1
CN(C)CC1(O)CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1
O=C1NCc2c1c(Nc1ccc(cn1)N1CCOCC1)cnc2-c1cnn2CCCCc12
OC1CCN(CC1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2cccc3ccnn23)nc1
OC1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2ccc3cnccn23)nc1
OC1CCN(CC1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2cccn3nccc23)nc1
OC1(CCOCC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1
COc1cc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ncc1N1CCC(O)CC1
Cc1csc2c(ccnc12)-c1ncc(Nc2ccc(cn2)N2CCC(O)CC2)c2C(=O)NCc12
Cn1cc(-c2ccc(Nc3ccc(cn3)N3CCC(O)CC3)c3C(=O)NCc23)c2ccnnc12
Cn1nccc2c(cnc12)-c1ccc(Nc2ccc(cn2)N2CCC(O)CC2)c2C(=O)NCc12
OC1CCN(CC1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2cncc3nccn23)nc1
Fc1ccn2c(cnc2c1)-c1ccc(Nc2ccc(cn2)S(=O)(=O)CC2COC2)c2C(=O)NCc12
OC1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(CN4CC(F)C4)ccn23)nc1
Fc1ccn2c(cnc2c1)-c1ccc(Nc2cnn(c2)C2CCOCC2)c2C(=O)NCc12
CN(C)Cc1ccn2c(cnc2c1)-c1ccc(Nc2ccc(cn2)N2CCC(O)CC2)c2C(=O)NCc12
Fc1ccn2c(cnc2c1)-c1ccc(Nc2cc([nH]n2)C2CCOCC2)c2C(=O)NCc12
O=C1NCc2c1c(Cc1ccn(n1)C1CCOCC1)ccc2-c1cnc2ccccn12
CN(C)CC1CN(CCO1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1
OC1CCN(CC1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2cccn3ccnc23)nc1
CN(C)CC1(O)CCCN(C1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1
CN(C)CCN1CCC(CC1=O)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)nc1
OC1(CN2CCCC2)CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1
CN1CCN(CC2(O)CCCN(C2)c2ccc(Nc3ccc(c4CNC(=O)c34)-c3cnc4cc(F)ccn34)nc2)CC1
Cc1cc(Nc2ccc(cn2)N2CCC(O)CC2)c2C(=O)NCc2c1-c1cnc2cc(F)ccn12 |(1.77,-3.18,;.27,-2.85,;-.2,-1.38,;-1.71,-1.05,;-2.16,.42,;-1.12,1.56,;.38,1.21,;1.43,2.34,;.98,3.81,;-.52,4.16,;-1.57,3.03,;2.03,4.94,;1.58,6.41,;2.63,7.53,;4.13,7.19,;5.18,8.31,;4.58,5.71,;3.53,4.59,;-2.74,-2.19,;-4.28,-2.19,;-5.18,-.93,;-4.77,-3.65,;-3.53,-4.56,;-2.28,-3.66,;-.77,-3.99,;-.32,-5.46,;-1.25,-6.68,;-.34,-7.95,;1.14,-7.51,;2.46,-8.29,;3.8,-7.53,;5.13,-8.31,;3.82,-5.99,;2.49,-5.21,;1.15,-5.97,)|
Cn1ccc2c(ccnc12)-c1ncc(Nc2cccc(n2)C2CCNCC2)c2C(=O)NCc12
Cn1ccc2c(ccnc12)-c1ncc(Nc2ccc(cn2)N2CCC(C)(O)CC2)c2C(=O)NCc12
CN1CCC(CC1=O)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)nc1
COC[C@]1(O)CCCN(C1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1 |r|
COC[C@@]1(O)CCCN(C1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1 |r|
OC1CCC2(CC2)N(C1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1
Cn1ncc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)c1C1CCOCC1
CC1(O)CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1
OC1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3ccccn23)nc1
O[C@@H]1CCN(C[C@H]1F)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1 |r|
O[C@H]1CCN(C[C@@H]1F)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1 |r|
CN1CCN(CC2(O)CCN(CC2)c2ccc(Nc3cnc(c4CNC(=O)c34)-c3ccnc4n(C)ccc34)nc2)CC1
CN1CCN(CC2(O)CCN(CC2)c2ccc(Nc3ccc(c4CNC(=O)c34)-c3cnc4c(C)cccn34)nc2)CC1
CN1CCN(CC2(O)CCN(CC2)c2ccc(Nc3ccc(c4CNC(=O)c34)-c3cnc4ccccn34)nc2)CC1
OC1[C@H]2CC[C@@H]1CN(C2)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1 |r|
[H]C12CCC([H])(CN(C1)c1ccc(Nc3ccc(c4CNC(=O)c34)-c3cnc4cc(F)ccn34)nc1)C2O |TLB:9:7:3.2:36|
CN(C)CCN1CCC(CC1=O)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1
CN1CCC(O)(CC1)c1cccc(Nc2cnc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)n1
Cn1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)cc1C1CCOCC1
CN1CC(C1)c1ccn2c(cnc2c1)-c1ccc(Nc2ccc(cn2)N2CCC(O)CC2)c2C(=O)NCc12
CN1CCN(CC2(O)CCN(CC2)c2ccc(Nc3ccc(c4CNC(=O)c34)-c3cnc4cnccn34)nc2)CC1
Cn1ccc2c(ccnc12)-c1ncc(Nc2ccc3CCNCc3n2)c2C(=O)NCc12
COC[C@H]1CN(CC[C@@H]1O)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)nc1 |r|
Cn1ccc2c(ccnc12)-c1ncc(Nc2cccc(n2)C2CNC2)c2C(=O)NCc12
Cn1ccc2c(ccnc12)-c1ncc(Nc2ccc(cn2)N2CC[C@@H](F)[C@H](O)C2)c2C(=O)NCc12 |r|
Cn1ccc2c(ccnc12)-c1ncc(Nc2ccc(cn2)N2CC[C@H](F)[C@@H](O)C2)c2C(=O)NCc12 |r|
CN1CCc2ccc(Nc3cnc(c4CNC(=O)c34)-c3ccnc4n(C)ccc34)nc2C1
CN1CCC[C@@H](C1)c1cccc(Nc2cnc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)n1 |r|
CN1CCC[C@H](C1)c1cccc(Nc2cnc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)n1 |r|
COC[C@H]1CN(CCO1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1 |r|
Cn1cc2c(cnc2cn1)-c1ccc(Nc2ccc(cn2)N2CCC(O)CC2)c2C(=O)NCc12
COC[C@H]1CN(CC[C@H]1O)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)nc1 |r|
Cn1ccc2c(ccnc12)-c1ccc(Nc2ncc(cc2F)N2CCC(O)CC2)c2C(=O)NCc12
Cn1cc(-c2ccc(Nc3ccc(cn3)N3CCC(O)CC3)c3C(=O)NCc23)c2cnncc12
Cn1ccc2c(cnc2n1)-c1ccc(Nc2ccc(cn2)N2CCC(O)CC2)c2C(=O)NCc12
Cn1ccc2c(ccnc12)-c1ncc(Nc2ccc(cn2)C2(O)CCOCC2)c2C(=O)NCc12
Fc1ccn2c(cnc2c1)-c1ccc(Nc2ccc(cn2)N2CCC(CN3CCOCC3)CC2)c2C(=O)NCc12
CC1(CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1)N1CCOCC1
Cn1ccc2c(ccnc12)-c1ncc(Nc2cccc(n2)C2(C)CCNCC2)c2C(=O)NCc12
Cn1ccc2c(ccnc12)-c1ncc(Nc2cccc(n2)N2CC[C@H](C2)N2CCCC2)c2C(=O)NCc12 |r|
CN1CC(C1)c1cccc(Nc2cnc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)n1
CC1(CO)CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1
O[C@@H]1CN(CC[C@H]1F)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cnccn23)nc1 |r|
O[C@H]1CN(CC[C@@H]1F)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cnccn23)nc1 |r|
COC[C@@H]1CN(CC[C@@H]1O)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)nc1 |r|
CN1CCN(CC2(O)CCN(CC2)c2ccc(Nc3ccc(c4CNC(=O)c34)-c3cnc4cc(Cl)ccn34)nc2)CC1
COCC1(O)CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1
Cc1ccn2c(cnc2c1F)-c1ccc(Nc2ccc(cn2)N2CCC(O)(CN3CCOCC3)CC2)c2C(=O)NCc12
Cn1ccc2c(ccnc12)-c1ncc(Nc2cccc(n2)N2CC[C@H]3CNC[C@@H]23)c2C(=O)NCc12 |r|
Cn1ccc2c(ccnc12)-c1ncc(Nc2cccc(n2)N2CC[C@@H]3CNC[C@H]23)c2C(=O)NCc12 |r|
COC[C@@H]1CN(CCO1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1 |r|
Cn1ccc2c(ccnc12)-c1ncc(Nc2cccc(n2)N2CC[C@@H](C2)N2CCCC2)c2C(=O)NCc12 |r|
CN1CCN(CC2(O)CCN(CC2)c2ccc(Nc3ccc(c4CNC(=O)c34)-c3cnc4c(F)c(C)ccn34)nc2)CC1
O=C1NCc2c1c(Nc1ccc(cn1)N1CCC[C@@]3(CCNC3=O)C1)ccc2-c1cnn2CCCCc12 |r|
O=C1NCc2c1c(Nc1ccc(cn1)N1CCC[C@]3(CCNC3=O)C1)ccc2-c1cnn2CCCCc12 |r|
OC1(CN2CCOCC2)CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(Cl)ccn23)nc1
Cn1cc2ncc(-c3ccc(Nc4ccc(cn4)N4CCC(O)CC4)c4C(=O)NCc34)c2cn1
CNC1CN(C1)c1cccc(Nc2cnc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)c1
OC[C@H]1CN(CCO1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1 |r|
CN1CCN(CC1)c1cccc(Nc2cnc(c3CNC(=O)c23)-c2cnc3ccccn23)n1
Cc1ccn2c(cnc2n1)-c1ccc(Nc2ccc(cn2)N2CCO[C@H](CO)C2)c2C(=O)NCc12 |r|
CNC1CCN(CC1(F)F)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)nc1
OC[C@@H]1CN(CCO1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1 |r|
COC1CCN(CC1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2cnc3c(F)cccn23)nc1
CN(C)CCNC(=O)C(C)(C)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3c(F)c(C)ccn23)nc1
CC(C)(O)[C@@H]1CN(CCO1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cnccn23)nc1 |r|
CC(C)(O)[C@H]1CN(CCO1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2cnc3c(F)cccn23)nc1 |r|
Cn1ccc2c(ccnc12)-c1ncc(Nc2ccc(cn2)N2CCO[C@H](C2)C(C)(C)O)c2C(=O)NCc12 |r|
Cc1ccn2c(cnc2c1F)-c1ccc(Nc2ccc(cn2)N2CCO[C@@H](CO)C2)c2C(=O)NCc12 |r|
COc1cccn2c(cnc12)-c1ncc(Nc2ccc(cn2)N2CCC[C@@H](C2)C(C)(C)O)c2C(=O)NCc12 |r|
CC(C)(O)[C@H]1CN(CCO1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2cnc3c(Cl)cccn23)nc1 |r|
Cc1ccn2c(cnc2c1F)-c1ccc(Nc2ccc(cn2)N2CCO[C@@H](C2)C(C)(C)O)c2C(=O)NCc12 |r|
OC1CCN(CC1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2cnn3ccccc23)nc1
Cc1ccn2c(cnc2c1F)-c1ncc(Nc2ccc(cn2)N2CCO[C@H](C2)C(C)(C)O)c2C(=O)NCc12 |r|
Cc1ccn2c(cnc2c1F)-c1ccc(Nc2ccc(CN3CCOCC3)cn2)c2C(=O)NCc12
Cc1ccn2c(cnc2c1)-c1ccc(Nc2ccc(CN3CCOCC3)cn2)c2C(=O)NCc12
CC(C)(O)[C@H]1CN(CCO1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2cnc3ccccn23)nc1 |r|
Cn1ccc2c(ccnc12)-c1ncc(Nc2ccc(cn2)N2CCO[C@@H](C2)C(C)(C)O)c2C(=O)NCc12 |r|
Cn1ccc2c(ccnc12)-c1ncc(Nc2cccc(n2)N2CCC3CNCC23)c2C(=O)NCc12
Cc1ccn2c(cnc2c1F)-c1ncc(Nc2ccc(cn2)N2CCO[C@@H](C2)C(C)(C)O)c2C(=O)NCc12 |r|
CC(C)(O)[C@@H]1CN(CCO1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cccnn23)nc1 |r|
CC(C)(O)[C@@H]1CN(CCO1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3c(cccn23)C(F)F)nc1 |r|
Fc1ccn2c(cnc2c1)-c1ccc(Nc2ccc(cn2)N2CCCC(C2)N2CCOCC2)c2C(=O)NCc12
Fc1ccn2c(cnc2c1)-c1ccc(Nc2ccc(cn2)N2CCO[C@H](CNC3CC3)C2)c2C(=O)NCc12 |r|
CN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1[C@H]1CCOC1 |r|
CN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1[C@@H]1CCOC1 |r|
Cc1ccn2c(cnc2c1F)-c1ncc(Nc2cccc(n2)C2CC[C@@H]3CNC[C@H]23)c2C(=O)NCc12 |r|
Cc1ccn2c(cnc2c1F)-c1ncc(Nc2cccc(n2)C2CCC3CNCC23)c2C(=O)NCc12
FC1CN(C[C@@H]2CN(CCO2)c2ccc(Nc3ccc(c4CNC(=O)c34)-c3cnc4cc(F)ccn34)nc2)C1 |r|
CC(C)(O)[C@@H]1CN(CCO1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2cnc3c(F)cccn23)nc1 |r|
Cn1ccc2c(cccc12)-c1ncc(Nc2ccc(cn2)N2CCO[C@@H](C2)C(C)(C)O)c2C(=O)NCc12 |r|
CC(C)(O)[C@@H]1CN(CCO1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2cnc3ccccn23)nc1 |r|
Cc1ccn2c(cnc2c1F)-c1ccc(Nc2ccc(cn2)N2CCO[C@H](C2)C(C)(C)O)c2C(=O)NCc12 |r|
Cc1ccn2c(cnc2c1F)-c1ccc(Nc2ccc(cn2)N2CCC(CC2)N2CCOCC2)c2C(=O)NCc12
Cc1ccc2c(cnn2c1)-c1ccc(Nc2ccc(cn2)N2CCO[C@@H](C2)C(C)(C)O)c2C(=O)NCc12 |r|
Cc1ccn2c(cnc2c1)-c1ccc(Nc2ccc(cn2)N2CCO[C@@H](C2)C(C)(C)O)c2C(=O)NCc12 |r|
CN(CC1(O)CCCN(C1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1)C1CC1
CC(C)(O)[C@@H]1CN(CCO1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(ccn23)C(F)F)nc1 |r|
Fc1ccn2c(cnc2c1)-c1ccc(Nc2cccc(n2)N2CCC3CNCC23)c2C(=O)NCc12
CN(C[C@@H]1CN(CCO1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1)C1CC1 |r|
Fc1ccn2c(cnc2c1)-c1ccc(Nc2ccc(cn2)N2CCO[C@@H](CNC3CC3)C2)c2C(=O)NCc12 |r|
CN1CCOC2(CCCN(C2)c2ccc(Nc3ccc(c4CNC(=O)c34)-c3cnc4cc(F)ccn34)nc2)C1
Fc1ccn2c(cnc2c1)-c1ccc(Nc2cccc(n2)N2CC[C@H]3CNC[C@@H]23)c2C(=O)NCc12 |r|
Fc1ccn2c(cnc2c1)-c1ccc(Nc2cccc(n2)N2CC[C@@H]3CNC[C@H]23)c2C(=O)NCc12 |r|
CN(C[C@H]1CN(CCO1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1)C1CC1 |r|
Fc1ccn2c(cnc2c1)-c1ccc(Nc2ccc(cn2)N2CCCC3(CNCCO3)C2)c2C(=O)NCc12
Fc1ccn2c(cnc2c1)-c1ccc(Nc2ccc(cn2)N2CCC[C@@H](C2)N2CCOCC2)c2C(=O)NCc12 |r|
Fc1ccn2c(cnc2c1)-c1ccc(Nc2ccc(cn2)N2CCC[C@H](C2)N2CCOCC2)c2C(=O)NCc12 |r|
CN(C)CC1(F)CCCN(C1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1
CCN(CC)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1C1CCOC1
Fc1ccn2c(cnc2c1)-c1ccc(Nc2ccc(C3CCOC3)c(CN3CCCC3)n2)c2C(=O)NCc12
CN1CCO[C@]2(CCCN(C2)c2ccc(Nc3ccc(c4CNC(=O)c34)-c3cnc4cc(F)ccn34)nc2)C1 |r|
CN1CCO[C@@]2(CCCN(C2)c2ccc(Nc3ccc(c4CNC(=O)c34)-c3cnc4cc(F)ccn34)nc2)C1 |r|
Fc1ccn2c(cnc2c1)-c1ccc(Nc2ccc(cn2)N2CCC[C@@]3(CNCCO3)C2)c2C(=O)NCc12 |r|
Fc1ccn2c(cnc2c1)-c1ccc(Nc2ccc(cn2)N2CCC[C@]3(CNCCO3)C2)c2C(=O)NCc12 |r|
CN(C)C1COCCN(C1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1
CCN(CC)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1[C@H]1CCOC1 |r|
CCN(CC)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1[C@@H]1CCOC1 |r|
Fc1ccn2c(cnc2c1)-c1ccc(Nc2ccc(cn2)N2CCO[C@H](Cn3ccnc3)C2)c2C(=O)NCc12 |r|
C[C@H](N1CCC[C@H](O)C1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1 |r|
C[C@@H](N1CCC[C@H](O)C1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1 |r|
Fc1ccn2c(cnc2c1)-c1ccc(Nc2ccc([C@H]3CCOC3)c(CN3CCCC3)n2)c2C(=O)NCc12 |r|
Fc1ccn2c(cnc2c1)-c1ccc(Nc2ccc([C@@H]3CCOC3)c(CN3CCCC3)n2)c2C(=O)NCc12 |r|
CN(C)CC1COCCN1c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1
CN(C)[C@@H]1COCCN(C1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1 |r|
CN(C)[C@H]1COCCN(C1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1 |r|
CC(N(C)C)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1
C[C@H](N1CCO[C@@H](C)C1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1 |r|
C[C@@H](N1CCO[C@@H](C)C1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1 |r|
CN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1N1CCC[C@@H](O)C1 |r|
CN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1N1CCOCC11CC1
C[C@H](N1CCC(O)CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1 |r|
C[C@@H](N1CCC(O)CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1 |r|
C[C@@H]1COCCN1c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1CN(C)C |r|
C[C@H]1CN(CCO1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1CN(C)C |r|
CN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1N1CCOC2(CC2)C1
C[C@H]1COCCN1c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1CN(C)C |r|
CN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1N1CCC[C@H](O)C1 |r|
CN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1O[C@@H]1CCOC1 |r|
CN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1N1CCN(C)C(=O)CC1
CN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1N1CCC(C)(O)CC1
CN(C)C1CCCc2ccc(Nc3ccc(c4CNC(=O)c34)-c3cnc4cc(F)ccn34)nc12
CN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(C)cnn23)ccc1[C@H]1CCOC1 |r|
CN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(C)cnn23)ccc1[C@@H]1CCOC1 |r|
CN(C)Cc1nc(Nc2cnc(c3CNC(=O)c23)-c2cnc3c(C)ccnn23)ccc1C1CCOC1
CN(C)Cc1nc(Nc2cnc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)ccc1[C@@H]1CCOC1 |r|
C[C@@H]1CN(CCO1)c1c(CN(C)C)cc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1CN(C)C |r|
CN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnn3cc(F)ccc23)ccc1[C@H]1CCOC1 |r|
CN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnn3cc(F)ccc23)ccc1[C@@H]1CCOC1 |r|
CN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1O[C@H]1CCOC1 |r|
CN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)ccc1[C@@H]1CCOC1 |r|
CN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)ccc1[C@H]1CCOC1 |r|
CN(C)Cc1nc(Nc2cnc(c3CNC(=O)c23)-c2cccc3n(C)ccc23)ccc1[C@H]1CCOC1 |r|
COC1CN(Cc2nc(Nc3ccc(c4CNC(=O)c34)-c3cnc4cc(F)ccn34)ccc2[C@H]2CCOC2)C1 |r|
COC1CN(Cc2nc(Nc3ccc(c4CNC(=O)c34)-c3cnc4cc(F)ccn34)ccc2[C@@H]2CCOC2)C1 |r|
CN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1[C@H]1CCCOC1 |r|
CN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1[C@@H]1CCCOC1 |r|
Cn1ccc2c(cccc12)-c1ncc(Nc2ccc(C3CCOC3)c(CN3CCCC3)n2)c2C(=O)NCc12
CN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1OC1CCOCC1
CN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1[C@H]1CCCO1 |r|
CN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1N1CC[C@H](O)C1 |r|
CN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1[C@H]1CCN(C)C(=O)C1 |r|
CN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1[C@@H]1CCN(C)C(=O)C1 |r|
CC(C)NCc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1[C@@H]1CCOC1 |r|
CC(C)NCc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1[C@H]1CCOC1 |r|
CN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1[C@@H]1CCCO1 |r|
CN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(C)ccn23)ccc1C1CCOC1
CN1CC[C@H](CC1=O)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)nc1 |r|
CN1CC[C@@H](CC1=O)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)nc1 |r|
CN(C)C(C)(C)C1CN(CCO1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1
OC1CCN(CC1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2ccnn3ccnc23)nc1
Cn1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)cc1C1(O)CCOCC1
CN(C)C[C@]1(O)CCCN(C1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1 |r|
CN(C)C[C@@]1(O)CCCN(C1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1 |r|
COC(C)(C)[C@@H]1CN(CCO1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cnccn23)nc1 |r|
COC(C)(C)[C@H]1CN(CCO1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cnccn23)nc1 |r|
CO[C@H]1CC[C@H](CO)N(C1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnn3CCCCc23)nc1 |r|
CO[C@@H]1CC[C@@H](CO)N(C1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnn3CCCCc23)nc1 |r|
O[C@]1(CCOC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1 |r|
O[C@@]1(CCOC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1 |r|
CN1CCC(C)(CC1)c1cccc(Nc2cnc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)n1
COC1(CO)CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1
CN(C)C[C@]1(O)CCCN(C1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3c(F)c(C)ccn23)nc1 |r|
CN(C)C[C@@]1(O)CCCN(C1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3c(F)c(C)ccn23)nc1 |r|
COC[C@@H]1CN(CCO1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3c(F)c(C)ccn23)nc1 |r|
COC[C@H]1CN(CCO1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3c(F)c(C)ccn23)nc1 |r|
OC1(CCOCC1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2cnc3ccccn23)nc1
CN(C)C(C)(C)C1CCCN(C1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1
Cc1ccn2c(cnc2c1F)-c1ccc(Nc2ccc(cn2)N2CC[C@@H](F)[C@H](O)C2)c2C(=O)NCc12 |r|
Cc1ccn2c(cnc2c1F)-c1ccc(Nc2ccc(cn2)N2CC[C@H](F)[C@@H](O)C2)c2C(=O)NCc12 |r|
CN(C)C[C@@H]1CN(CCO1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)nc1 |r|
CN(C)C[C@H]1CN(CCO1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)nc1 |r|
Cc1ccn2c(cnc2c1F)-c1ccc(Nc2ccc(cn2)C2(O)CCOCC2)c2C(=O)NCc12
OC1CCN(CC1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2ccnn3cccc23)nc1
CN1CCN(CC1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)nc1C
CN(C)C(C)(C)[C@@H]1CN(CCO1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1 |r|
CN(C)C(C)(C)[C@H]1CN(CCO1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1 |r|
OC1CCN(CC1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2ccnc3cnccc23)nc1
CN(C)C[C@@H]1CN(CCO1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(Cl)ccn23)nc1 |r|
CN(C)C[C@H]1CN(CCO1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(Cl)ccn23)nc1 |r|
O[C@H]1COCCN(C1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(Cl)ccn23)nc1 |r|
O[C@@H]1COCCN(C1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(Cl)ccn23)nc1 |r|
C[C@@H]1CC[C@](C)(O)CN1c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnn3CCCCc23)nc1 |r|
C[C@@H]1CC[C@@](C)(O)CN1c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnn3CCCCc23)nc1 |r|
CN1CC(O)(C1)C1CCCN(C1)c1ccc(Nc2ccc(C3=CNC4C=C(F)C=CN34)c3CNC(=O)c23)nc1 |c:30,t:23,27|
O[C@@H]1CN(CC[C@H]1F)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2cnc3ccccn23)nc1 |r|
Cc1ccn2c(cnc2c1F)-c1ccc(Nc2ccc(cn2)[C@]2(O)CCOC2)c2C(=O)NCc12 |r|
Cc1ccn2c(cnc2c1F)-c1ccc(Nc2ccc(cn2)[C@@]2(O)CCOC2)c2C(=O)NCc12 |r|
CN(C)C[C@@H]1CN(CCO1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1 |r|
CN(C)C[C@H]1CN(CCO1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1 |r|
CN1CCN(Cc2ccc(Nc3ccc(c4CNC(=O)c34)-c3cnc4c(F)c(C)ccn34)nc2)CC1
CN(C)C(C)(C)[C@H]1CCCN(C1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1 |r|
CN(C)C(C)(C)[C@@H]1CCCN(C1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1 |r|
OC1(CCOCC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(ccn23)C(F)F)nc1
O[C@]1(CCOC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(ccn23)C(F)F)nc1 |r|
O[C@@]1(CCOC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(ccn23)C(F)F)nc1 |r|
CO[C@@]1(CN(C)C)CCCN(C1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1 |r|
CO[C@]1(CN(C)C)CCCN(C1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1 |r|
CN(C)C[C@@H]1CN(CCO1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3c(F)c(C)ccn23)nc1 |r|
CN(C)C[C@H]1CN(CCO1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3c(F)c(C)ccn23)nc1 |r|
CN1CC[C@]11CCN(C1)c1cccc(Nc2cnc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)n1 |r|
CN1CC[C@@]11CCN(C1)c1cccc(Nc2cnc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)n1 |r|
CN(C)C(C)(C)[C@@H]1CN(CCO1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cnccn23)nc1 |r|
CN(C)C(C)(C)[C@H]1CN(CCO1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cnccn23)nc1 |r|
C[C@H](O)[C@@H]1CN(CCO1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1 |r|
C[C@@H](O)[C@@H]1CN(CCO1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1 |r|
CN1CCN(C[C@H]1C(C)(C)O)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2cnc3c(F)cccn23)nc1 |r|
CN1CCN(C[C@@H]1C(C)(C)O)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2cnc3c(F)cccn23)nc1 |r|
Cn1ccc2c(ncnc12)-c1ccc(Nc2ccc(cn2)N2CCO[C@@H](C2)C(C)(C)O)c2C(=O)NCc12 |r|
Cn1ccc2c(ncnc12)-c1ccc(Nc2ccc(cn2)N2CCO[C@H](C2)C(C)(C)O)c2C(=O)NCc12 |r|
CC(C)(O)[C@H]1COCCN(C1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1 |r|
CC(C)(O)[C@@H]1COCCN(C1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1 |r|
COC[C@@H]1CN(CCO1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3nc(C)ccn23)nc1 |r|
COC[C@H]1CN(CCO1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3nc(C)ccn23)nc1 |r|
CN1C[C@@H]2CCN([C@@H]2C1)c1cccc(Nc2cnc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)n1 |r|
CN1C[C@H]2CCN([C@H]2C1)c1cccc(Nc2cnc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)n1 |r|
OC1CCN(CC1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2cncn3ccnc23)nc1
CN(C)Cc1cc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(Cl)ccn23)ncc1C1(O)CCOCC1
C[C@H](N1CCOCC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1 |r|
C[C@@H](N1CCOCC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1 |r|
Cc1cc(Nc2cnc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)nc(c1)N1CC[C@H]2CNC[C@@H]12 |r|
Cc1cc(Nc2cnc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)nc(c1)N1CC[C@@H]2CNC[C@H]12 |r|
CN1C[C@@H]2CCN([C@@H]2C1)c1cc(C)cc(Nc2cnc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)n1 |r|
CN1C[C@H]2CCN([C@H]2C1)c1cc(C)cc(Nc2cnc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)n1 |r|
Cc1ccn2c(cnc2n1)-c1ccc(Nc2ccc(cn2)N2CCO[C@@H](C2)C(C)(C)O)c2C(=O)NCc12 |r|
Cc1ccn2c(cnc2n1)-c1ccc(Nc2ccc(cn2)N2CCO[C@H](C2)C(C)(C)O)c2C(=O)NCc12 |r|
CN1CCN(CC2(O)CCN(CC2)c2ccc(Nc3cnc(c4CNC(=O)c34)-c3cnc4ccccn34)nc2)CC1
COC[C@@H]1CN(CCO1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2ncnc3n(C)ccc23)nc1 |r|
COC[C@H]1CN(CCO1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2ncnc3n(C)ccc23)nc1 |r|
CN(C)Cc1cc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ncc1C1(O)CCOCC1
O[C@@H]1CN(CC[C@H]1F)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2cnc3c(F)cccn23)nc1 |r|
O[C@H]1CN(CC[C@@H]1F)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2cnc3c(F)cccn23)nc1 |r|
OC1(CN2CCOCC2)CCCN(C1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1
CC1(C)CNCCN1Cc1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3c(F)c(ccn23)C(F)F)nc1
O[C@@]1(CN2CCOCC2)CCCN(C1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1 |r|
O[C@]1(CN2CCOCC2)CCCN(C1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1 |r|
O[C@@H]1CN(CC[C@@H]1F)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2cnc3c(F)cccn23)nc1 |r|
O[C@H]1CN(CC[C@H]1F)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2cnc3c(F)cccn23)nc1 |r|
Cn1ccc2c(ccnc12)-c1ncc(Nc2cncc(n2)N2CC[C@H]3CNC[C@@H]23)c2C(=O)NCc12 |r|
Cn1ccc2c(ccnc12)-c1ncc(Nc2cncc(n2)N2CC[C@@H]3CNC[C@H]23)c2C(=O)NCc12 |r|
OC1(CC1)[C@@H]1CN(CCO1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1 |r|
OC1(CC1)[C@H]1CN(CCO1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1 |r|
CN(C1CNC1)c1nc(Nc2cnc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)ccc1C
CN(C)C(C)(C)C1CN(CCO1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)nc1
CN(C)CCOC1(CCOCC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1
CC(C)(N)[C@@H]1CN(CCO1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1 |r|
CC(C)(N)[C@H]1CN(CCO1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1 |r|
CN1CCN(Cc2ccc(Nc3ccc(c4CNC(=O)c34)-c3cnc4c(F)c(ccn34)C(F)F)nc2)C(C)(C)C1
Cn1ccc2c(ccnc12)-c1ncc(Nc2ccc(cn2)N2CCC[C@@](O)(CN3CCOCC3)C2)c2C(=O)NCc12 |r|
Cn1ccc2c(ccnc12)-c1ncc(Nc2ccc(cn2)N2CCC[C@](O)(CN3CCOCC3)C2)c2C(=O)NCc12 |r|
CNC(C)(C)[C@@H]1CN(CCO1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1 |r|
CNC(C)(C)[C@H]1CN(CCO1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1 |r|
CN1CCCC1C1(O)CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1
CN1CC(O)(C1)[C@H]1CCCN(C1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1 |r|
CN1CC(O)(C1)[C@@H]1CCCN(C1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1 |r|
Cn1ccc2c(ccnc12)-c1ncc(Nc2cccc(n2)N2CC3(CCN3)C2)c2C(=O)NCc12
COc1cc(Nc2cnc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)nc(c1)N1CC[C@H]2CNC[C@@H]12 |r|
COc1cc(Nc2cnc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)nc(c1)N1CC[C@@H]2CNC[C@H]12 |r|
OC1(CCOCC1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2cnc3c(F)cccn23)nc1
Cn1ccc2c(ccnc12)-c1ncc(Nc2ccnc(n2)N2CC[C@H]3CNC[C@@H]23)c2C(=O)NCc12 |r|
Cn1ccc2c(ccnc12)-c1ncc(Nc2ccnc(n2)N2CC[C@@H]3CNC[C@H]23)c2C(=O)NCc12 |r|
CN(C)C1(CC1)[C@@H]1CN(CCO1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1 |r|
CN(C)C1(CC1)[C@H]1CN(CCO1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1 |r|
Cn1ccc2c(ccnc12)-c1ncc(Nc2cccc(n2)N2C[C@H](CN3CCC3)CCC2=O)c2C(=O)NCc12 |r|
Cn1ccc2c(ccnc12)-c1ncc(Nc2cccc(n2)N2C[C@@H](CN3CCC3)CCC2=O)c2C(=O)NCc12 |r|
Fc1ccn2c(cnc2c1)-c1ccc(Nc2ccc(cn2)N2CCO[C@@H]3CNC[C@H]23)c2C(=O)NCc12 |r|
Cn1ccc2c(ccnc12)-c1ncc(Nc2cccc(n2)N2C[C@H](N)CC2=O)c2C(=O)NCc12 |r|
Cn1ccc2c(ccnc12)-c1ncc(Nc2cccc(n2)N2C[C@@H](N)CC2=O)c2C(=O)NCc12 |r|
CN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1N1CCOCC1
Fc1ccn2c(cnc2c1)-c1ccc(Nc2ccc(cn2)N2CCO[C@H]3CNC[C@@H]23)c2C(=O)NCc12 |r|
CN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3c(C)cccn23)ccc1N1CCOC1
CC(C)([C@@H]1CN(CCO1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1)N1CC(O)C1 |r|
CC(C)([C@H]1CN(CCO1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1)N1CC(O)C1 |r|
CN(C)Cc1cccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)n1
CN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1N1CC[C@@H](F)[C@H](O)C1 |r|
CN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1N1CC[C@H](F)[C@@H](O)C1 |r|
NCc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1C1CCOC1
CN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3c(F)c(C)ccn23)ccc1C1CCOC1
CN(C)C1(CCOCC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1
CN(C)Cc1nc(Nc2cnc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)ccc1C1CCOC1
CN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnn3c(C)cccc23)ccc1C1CCOC1
CN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnn3c(C)cccc23)ccc1[C@@H]1CCOC1 |r|
COC[C@@H]1CN(CCO1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1CN(C)C |r|
COC[C@H]1CN(CCO1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1CN(C)C |r|
CN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cnccn23)ccc1[C@H]1CCOC1 |r|
CN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cnccn23)ccc1[C@@H]1CCOC1 |r|
CN(C)C(C)(C)[C@]1(O)CCCN(C1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1 |r|
CN(C)C(C)(C)[C@@]1(O)CCCN(C1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1 |r|
Fc1ccn2c(cnc2c1)-c1ccc(Nc2ccc([C@H]3CCOC3)c(CN3CCC(F)(F)C3)n2)c2C(=O)NCc12 |r|
Fc1ccn2c(cnc2c1)-c1ccc(Nc2ccc([C@@H]3CCOC3)c(CN3CCC(F)(F)C3)n2)c2C(=O)NCc12 |r|
CN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1C1(O)CCOCC1
Fc1ccn2c(cnc2c1)-c1ccc(Nc2ccc([C@H]3CCOC3)c(CN3CCOCC3)n2)c2C(=O)NCc12 |r|
Fc1ccn2c(cnc2c1)-c1ccc(Nc2ccc([C@@H]3CCOC3)c(CN3CCOCC3)n2)c2C(=O)NCc12 |r|
CNCc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1[C@H]1CCOC1 |r|
CNCc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1[C@@H]1CCOC1 |r|
Cn1ccc2c(ccnc12)-c1ncc(Nc2cccc(n2)N2C[C@@H](CC2=O)N2CCC2)c2C(=O)NCc12 |r|
Cn1ccc2c(ccnc12)-c1ncc(Nc2cccc(n2)N2C[C@H](CC2=O)N2CCC2)c2C(=O)NCc12 |r|
CC(C)(NC1CC1)C1CN(CCO1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1
COCCN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1[C@@H]1CCOC1 |r|
COCCN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1[C@H]1CCOC1 |r|
CC(C)N(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1[C@H]1CCOC1 |r|
CC(C)N(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1[C@@H]1CCOC1 |r|
CN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnn3cc(C)ccc23)ccc1[C@H]1CCOC1 |r|
CN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnn3cc(C)ccc23)ccc1[C@@H]1CCOC1 |r|
CN(CCO)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1[C@H]1CCOC1 |r|
CN(CCO)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1[C@@H]1CCOC1 |r|
F[C@H]1CCN(Cc2nc(Nc3ccc(c4CNC(=O)c34)-c3cnc4cc(F)ccn34)ccc2[C@H]2CCOC2)C1 |r|
F[C@H]1CCN(Cc2nc(Nc3ccc(c4CNC(=O)c34)-c3cnc4cc(F)ccn34)ccc2[C@@H]2CCOC2)C1 |r|
CN(Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1[C@H]1CCOC1)C1CC1 |r|
CN(Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1[C@@H]1CCOC1)C1CC1 |r|
FC(F)CNCc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1[C@H]1CCOC1 |r|
FC(F)CNCc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1[C@@H]1CCOC1 |r|
F[C@@H]1CCN(Cc2nc(Nc3ccc(c4CNC(=O)c34)-c3cnc4cc(F)ccn34)ccc2[C@H]2CCOC2)C1 |r|
F[C@@H]1CCN(Cc2nc(Nc3ccc(c4CNC(=O)c34)-c3cnc4cc(F)ccn34)ccc2[C@@H]2CCOC2)C1 |r|
CN(Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1[C@H]1CCOC1)C1COC1 |r|
CN(Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1[C@@H]1CCOC1)C1COC1 |r|
CN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1N1CCC[C@@H](C1)C(C)(C)O |r|
CN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1N1CCC[C@H](C1)C(C)(C)O |r|
CC(C)(N1CCOCC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1
CN(CC(F)F)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1[C@H]1CCOC1 |r|
CN(CC(F)F)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1[C@@H]1CCOC1 |r|
Fc1ccn2c(cnc2c1)-c1ccc(Nc2ccc([C@H]3CCOC3)c(CNCC(F)(F)F)n2)c2C(=O)NCc12 |r|
Fc1ccn2c(cnc2c1)-c1ccc(Nc2ccc([C@@H]3CCOC3)c(CNCC(F)(F)F)n2)c2C(=O)NCc12 |r|
CN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(ccn23)C(F)F)ccc1[C@H]1CCOC1 |r|
CN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(ccn23)C(F)F)ccc1[C@@H]1CCOC1 |r|
CN(Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1[C@H]1CCOC1)CC(F)(F)F |r|
Fc1ccn2c(cnc2c1)-c1ccc(Nc2ccc([C@H]3CCOC3)c(CN3CCC3)n2)c2C(=O)NCc12 |r|
Fc1ccn2c(cnc2c1)-c1ccc(Nc2ccc([C@@H]3CCOC3)c(CN3CCC3)n2)c2C(=O)NCc12 |r|
CCN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1[C@H]1CCOC1 |r|
CCN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1C1CCOC1
CN(C)CCc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1[C@H]1CCOC1 |r|
CN(C)CCc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1[C@@H]1CCOC1 |r|
FC1CN(Cc2nc(Nc3ccc(c4CNC(=O)c34)-c3cnc4cc(F)ccn34)ccc2[C@H]2CCOC2)C1 |r|
FC1CN(Cc2nc(Nc3ccc(c4CNC(=O)c34)-c3cnc4cc(F)ccn34)ccc2[C@@H]2CCOC2)C1 |r|
OC1CN(Cc2nc(Nc3ccc(c4CNC(=O)c34)-c3cnc4cc(F)ccn34)ccc2[C@H]2CCOC2)C1 |r|
OC1CN(Cc2nc(Nc3ccc(c4CNC(=O)c34)-c3cnc4cc(F)ccn34)ccc2[C@@H]2CCOC2)C1 |r|
CN(Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1[C@@H]1CCOC1)CC(F)(F)F |r|
CN(C)Cc1nc(Nc2cnc(c3CNC(=O)c23)-c2ccnc3[nH]ccc23)ccc1[C@@H]1CCOC1 |r|
CN(C)Cc1nc(Nc2cnc(c3CNC(=O)c23)-c2ccnc3[nH]ccc23)ccc1[C@H]1CCOC1 |r|
CN(C)Cc1nc(Nc2cnc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)ccc1N1CCOCC1
CN(C)Cc1nc(Nc2cnc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)ccc1N1CCO[C@@H](C1)C(C)(C)O |r|
CN(C)Cc1nc(Nc2cnc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)ccc1N1CCO[C@H](C1)C(C)(C)O |r|
OCc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1C1CCOC1
Fc1ccn2c(cnc2c1)-c1ccc(Nc2ccc([C@H]3CCOC3)c(n2)N2CCNCC2)c2C(=O)NCc12 |r|
Fc1ccn2c(cnc2c1)-c1ccc(Nc2ccc([C@@H]3CCOC3)c(n2)N2CCNCC2)c2C(=O)NCc12 |r|
CN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1N1CCO[C@@H](C1)C(C)(C)O |r|
CN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1N1CCO[C@H](C1)C(C)(C)O |r|
CN(C)Cc1nc(Nc2cnc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)ccc1N1CCC(O)CC1
CN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1N1CCC(O)CC1
O[C@H]1CCN(Cc2nc(Nc3ccc(c4CNC(=O)c34)-c3cnc4cc(F)ccn34)ccc2[C@H]2CCOC2)C1 |r|
O[C@H]1CCN(Cc2nc(Nc3ccc(c4CNC(=O)c34)-c3cnc4cc(F)ccn34)ccc2[C@@H]2CCOC2)C1 |r|
CO[C@@H]1CCN(Cc2nc(Nc3ccc(c4CNC(=O)c34)-c3cnc4cc(F)ccn34)ccc2[C@H]2CCOC2)C1 |r|
CO[C@@H]1CCN(Cc2nc(Nc3ccc(c4CNC(=O)c34)-c3cnc4cc(F)ccn34)ccc2[C@@H]2CCOC2)C1 |r|
COCC1(O)CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1CN(C)C
O[C@@H]1CCN(Cc2nc(Nc3ccc(c4CNC(=O)c34)-c3cnc4cc(F)ccn34)ccc2[C@H]2CCOC2)C1 |r|
O[C@@H]1CCN(Cc2nc(Nc3ccc(c4CNC(=O)c34)-c3cnc4cc(F)ccn34)ccc2[C@@H]2CCOC2)C1 |r|
CCN(CC)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1N1CCOCC1
CN(C)C1CN(C1)c1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1[C@H]1CCOC1 |r|
CN(C)C1CN(C1)c1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1[C@@H]1CCOC1 |r|
CN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1C1CCC1
CO[C@H]1CCN(Cc2nc(Nc3ccc(c4CNC(=O)c34)-c3cnc4cc(F)ccn34)ccc2C2CCOC2)C1 |r|
CCNC(=O)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1CN(C)C
CN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1C1CCOCC1
CO[C@@H]1CCC(C1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1CN(C)C |r|
CO[C@H]1CCC(C1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1CN(C)C |r|
CN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1N1CCN(C)C(=O)C1
CN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1S(C)(=O)=O
COC[C@@H]1CN(CCO1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)nc1CN(C)C |r|
COC[C@H]1CN(CCO1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)nc1CN(C)C |r|
CN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)cnc1[C@H]1CCOC1 |r|
CN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)cnc1[C@@H]1CCOC1 |r|
CN1CCN(CC1)c1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)cnc1[C@H]1CCOC1 |r|
CN1CCN(CC1)c1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)cnc1[C@@H]1CCOC1 |r|
CN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1[C@@]1(O)CCOC1 |r|
CN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1[C@]1(O)CCOC1 |r|
CN(C)Cc1nc(Nc2cnc(c3CNC(=O)c23)-c2cccc3n(C)ccc23)ccc1O[C@@H]1CCOC1 |r|
CN(C)Cc1nc(Nc2cnc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)ccc1O[C@H]1CCOC1 |r|
CN(C)CCc1nc(Nc2cnc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)ccc1[C@@H]1CCOC1 |r|
CN(C)CCc1nc(Nc2cnc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)ccc1[C@H]1CCOC1 |r|
Cn1ccc2c(ccnc12)-c1ncc(Nc2ccc([C@@H]3CCOC3)c(CN3CC[C@@H](O)C3)n2)c2C(=O)NCc12 |r|
Cn1ccc2c(ccnc12)-c1ncc(Nc2ccc([C@H]3CCOC3)c(CN3CC[C@@H](O)C3)n2)c2C(=O)NCc12 |r|
Cn1ccc2c(ccnc12)-c1ncc(Nc2ccc([C@@H]3CCOC3)c(CN3CC[C@H](O)C3)n2)c2C(=O)NCc12 |r|
Cn1ccc2c(ccnc12)-c1ncc(Nc2ccc([C@H]3CCOC3)c(CN3CC[C@H](O)C3)n2)c2C(=O)NCc12 |r|
CNCc1nc(Nc2cnc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)ccc1[C@@H]1CCOC1 |r|
CNCc1nc(Nc2cnc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)ccc1[C@H]1CCOC1 |r|
CN1CC(C1)Oc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1[C@H]1CCOC1 |r|
CN1CC(C1)Oc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1[C@@H]1CCOC1 |r|
C[C@@H](N(C)C)c1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1[C@H]1CCOC1 |r|
C[C@H](N(C)C)c1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1[C@H]1CCOC1 |r|
CN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1N1CCOC[C@H](O)C1 |r|
CN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1N1CCOC[C@@H](O)C1 |r|
COC1(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1CN(C)C
CN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1C1(CCOCC1)C#N
OC[C@H]1CCCN1Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1[C@H]1CCOC1 |r|
OC[C@H]1CCCN1Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1[C@@H]1CCOC1 |r|
OC[C@@H]1CCCN1Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1[C@H]1CCOC1 |r|
OC[C@@H]1CCCN1Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1[C@@H]1CCOC1 |r|
Cn1ccc2c(ccnc12)-c1ncc(Nc2ccc([C@H]3CCOC3)c(CN)n2)c2C(=O)NCc12 |r|
COC1(CCOCC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1CN(C)C
COCC1(CCOCC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1CN(C)C
CN(C)C(C)(C)c1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1[C@H]1CCOC1 |r|
CN(C)C(C)(C)c1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1[C@@H]1CCOC1 |r|
CN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1C1(F)CCOCC1
CN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1OCC(F)F
Cn1ccc2c(ccnc12)-c1ncc(Nc2ccc([C@@H]3CCOC3)c(CN)n2)c2C(=O)NCc12 |r|
COCC1(CCOC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1CN(C)C
CN(C)CCc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1C1CCOCC1
CN(C)Cc1nc(Nc2cnc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)ccc1N1CCOC2(CC2)C1
CN(C)CCc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1N1CCOCC1
CN(C)[C@H]1CCCc2ccc(Nc3ccc(c4CNC(=O)c34)-c3cnc4cc(F)ccn34)nc12 |r|
CN(C)[C@@H]1CCCc2ccc(Nc3ccc(c4CNC(=O)c34)-c3cnc4cc(F)ccn34)nc12 |r|
CN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1C1(C)CCOC1
CC(C)NCc1nc(Nc2cnc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)ccc1C1CCOCC1
CN(C)Cc1nc(Nc2cnc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)ccc1C1CCOCC1
CN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnn3cc(C)cnc23)ccc1C1CCOC1
CC(C)NCc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1C1CCOCC1
CC(C)(C)NCc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1C1CCOC1
Fc1ccn2c(cnc2c1)-c1ccc(Nc2ccc(C3CCOC3)c(CNCC3CC3)n2)c2C(=O)NCc12
CN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cnccn23)ccc1C1CCOCC1
COCC1(O)CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)nc1CN(C)C
CN(C)Cc1cc(cc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)n1)C1CCCO1
O=C1NCc2c1c(NC1OC=C(C=C1)N1CCOCC1)cnc2-c1c[nH]c2ccccc12 |c:11,13|
Cc1ccc2c(cnn2c1)-c1ccc(Nc2ccc(cn2)N2CCNCC2)c2C(=O)NCc12
CN1CCc2c1nccc2-c1ccc(Nc2ccc(cn2)N2CCNCC2)c2C(=O)NCc12
Cn1ccc2c(ccnc12)-c1ccc(Nc2ccc(cn2)C2CCNCC2)c2C(=O)NCc12
OC1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1
Cn1ccc2c(ncnc12)-c1ccc(Nc2ccc(cn2)N2CCC(O)CC2)c2C(=O)NCc12
OCc1ccn2c(cnc2c1)-c1ccc(Nc2ccc(cn2)N2CCC(O)CC2)c2C(=O)NCc12
CCOc1c(cnn2c(cnc12)-c1ccc(Nc2ccc(cn2)N2CCC(O)CC2)c2C(=O)NCc12)C#N
Cc1cnc2c(cnn2c1)-c1ccc(Nc2ccc(cn2)N2CCC(O)CC2)c2C(=O)NCc12
O=C1NCc2c1c(Nc1ccc(cn1)N1CCOCC1)cnc2-c1cnc2ccccn12
Cn1ccc2c(cccc12)-c1ncc(Nc2ccc(cn2)N2CCNCC2)c2C(=O)NCc12
C[C@H]1NC(=O)c2c1c(ccc2Nc1ccc(cn1)N1CCC(O)CC1)-c1ccnc2n(C)ccc12 |r|
C[C@@H]1NC(=O)c2c1c(ccc2Nc1ccc(cn1)N1CCC(O)CC1)-c1ccnc2n(C)ccc12 |r|
Fc1ccn2c(cnc2c1)-c1ccc(Nc2ccc(cn2)C2CCOCC2)c2C(=O)NCc12
CC(C)(O)C1CCCN(C1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2cnn3CCCCc23)nc1
OC1CCN(CC1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2ccnc3nccn23)nc1
Fc1ccn2c(cnc2c1)-c1ccc(Nc2ccn(n2)C2CCOCC2)c2C(=O)NCc12
OC1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2ncc3cnccn23)nc1
CN(C)CCN1CCC(CC1=O)C1=CB=C(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)C=C1 |c:42,t:13,15|
CN1CC(C1)c1ccn2c(cnc2c1)-c1ccc(Nc2ccc(cc2)N2CCC(O)CC2)c2C(=O)NCc12
COCC1CN(CC[C@@H]1O)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)nc1 |r|
O[C@@H]1CN(CC[C@H]1F)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3ccccn23)nc1 |r|
CNC1CN(C1)c1cccc(Nc2cnc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)n1
Cc1ccc2c(cnn2c1)-c1ccc(Nc2ccc(CN3CCOCC3)cn2)c2C(=O)NCc12
CC(C)(O)[C@@H]1CN(CCO1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2cnc3c(cccn23)C(F)F)nc1 |r|
Cc1ccn2c(cnc2c1F)-c1ncc(Nc2cccc(n2)N2CC[C@@H]3CNC[C@H]23)c2C(=O)NCc12 |r|
Cc1ccn2c(cnc2c1F)-c1ncc(Nc2cccc(n2)N2CCC3CNCC23)c2C(=O)NCc12
CC(C)(O)[C@H]1CN(CCO1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cnccn23)nc1 |r|
Fc1ccn2c(cnc2c1)-c1ccc(Nc2ccc(cn2)N2CCC(CC2)N2CCOCC2)c2C(=O)NCc12
CN(C)Cc1nc(Nc2cnc(c3CNC(=O)c23)-c2cnc3c(C)cccn23)ccc1C1CCOC1
CN(C)Cc1nc(Nc2cnc(c3CNC(=O)c23)-c2cccc3n(C)ccc23)ccc1[C@@H]1CCOC1 |r|
C[C@@H]1CN(CCO1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1CN(C)C |r|
Cn1ccc2c(ccnc12)-c1ncc(Nc2ccc(C3CCOC3)c(CN3CCCC3)n2)c2C(=O)NCc12
CN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3nc(C)ccn23)ccc1[C@H]1CCOC1 |r|
CN1CC(O)(C1)C1CCCN(C1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1
CN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3c(C)cccn23)ccc1[C@H]1CCOC1 |r|
CN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3c(C)cccn23)ccc1[C@@H]1CCOC1 |r|
CN(C)Cc1nc(Nc2cnc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)ccc1[C@H]1CCOC1 |r|
CN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnn3c(C)cccc23)ccc1[C@H]1CCOC1 |r|
CCN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1[C@@H]1CCOC1 |r|
CO[C@@H]1CC[C@H](C1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1CN(C)C |r|
CN1CCN(CC1)c1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1[C@H]1CCOC1 |r|
CN1CCN(CC1)c1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1[C@@H]1CCOC1 |r|
CN(C)Cc1nc(Nc2cnc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)ccc1O[C@@H]1CCOC1 |r|
COCC1(O)CCN(CC1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)nc1CN(C)C
Cc1ccncc1-c1cc2cc(NC(=O)[C@@H]3C[C@@H]3F)ncc2c(N)n1 |r|
Cc1c(cnn1C)-c1cc2cc(NC(=O)[C@H]3C[C@H]3F)ncc2c(N)n1 |r|
Cc1nn(C)c(C)c1-c1cc2cc(NC(=O)[C@H]3C[C@H]3F)ncc2c(N)n1 |r|
Cn1cc(cn1)-c1cc2cc(NC(=O)[C@H]3C[C@H]3F)ncc2c(N)n1 |r|
CCc1ccncc1-c1cc2cc(NC(=O)[C@H]3C[C@@H]3C#N)ncc2c(N)n1 |r|
Cn1cc(cn1)-c1cc2cc(NC(=O)[C@@H]3C[C@@H]3F)ncc2c(N)n1 |r|
Cn1cc(cn1)-c1cc2cc(NC(=O)C3C[C@@H]3F)ncc2c(N)n1 |r|
CNC(=O)Nc1cc2cc(nc(N)c2cn1)-c1cnn(C)c1
COc1ccncc1-c1cc2cc(NC(=O)[C@@H]3C[C@@H]3F)ncc2c(N)n1 |r|
Cc1ccncc1-c1cc2cc(NC(=O)C3CC3(F)F)ncc2c(N)n1
Cc1ncncc1-c1cc2cc(NC(=O)[C@@H]3C[C@@H]3F)ncc2c(N)n1 |r|
CCc1ncncc1-c1cc2cc(NC(=O)[C@@H]3C[C@@H]3F)ncc2c(N)n1 |r|
Nc1nc(cc2cc(NC(=O)[C@@H]3C[C@@H]3F)ncc12)-c1cnccc1C(F)F |r|
Nc1nc(cc2cc(NC(=O)[C@@H]3C[C@@H]3F)ncc12)-c1cnccc1C#N |r|
Cc1cc(N)ncc1-c1cc2cc(NC(=O)[C@H]3C[C@H]3F)ncc2c(N)n1 |r|
Cc1c(F)cncc1-c1cc2cc(NC(=O)[C@@H]3C[C@@H]3F)ncc2c(N)n1 |r|
Cn1nccc1-c1cc2cc(NC(=O)[C@@H]3C[C@@H]3F)ncc2c(N)n1 |r|
Cc1cc2[nH]cnc2cc1-c1cc2cc(NC(=O)[C@@H]3C[C@@H]3F)ncc2c(N)n1 |r|
CCc1ccncc1-c1cc2cc(NC(=O)C3CCC3)ncc2c(N)n1
Nc1nc(cc2cc(NC(=O)[C@@H]3C[C@@H]3C#N)ncc12)-c1cncc2[nH]ccc12 |r|
Cc1cnccc1-c1cc2cc(NC(=O)[C@@H]3C[C@@H]3F)ncc2c(N)n1 |r|
Cc1ccncc1-c1cc2cc(NC(=O)C3CC3)ncc2c(N)n1
Cc1cc(CO)ncc1-c1cc2cc(NC(=O)C3CC3)ncc2c(N)n1
CCc1ccncc1-c1cc2cc(NC(=O)C3CC3)ncc2c(N)n1
Cn1cc(cn1)-c1cc2cc(NC(=O)C3CC3)ncc2c(N)n1
CCc1ccncc1-c1cc2cc(NC(=O)CCC#N)ncc2c(N)n1
CCc1ccncc1-c1cc2cc(NC(=O)CCC(N)=O)ncc2c(N)n1
CCc1ccncc1-c1cc2cc(NC(=O)NCc3cncs3)ncc2c(N)n1
CCc1ccncc1-c1cc2cc(NC(=O)NC(C)C)ncc2c(N)n1
CCc1ccncc1-c1cc2cc(NC(=O)CC#N)ncc2c(N)n1
CCc1ccncc1-c1cc2cc(NC(=O)N(C)C)ncc2c(N)n1
CCc1ccncc1-c1cc2cc(NC(=O)N[C@H](C)C(N)=O)ncc2c(N)n1 |r|
Cc1ccncc1-c1cc2cc(NC(=O)C(C)(C)C#N)ncc2c(N)n1
COC(C)(C)C(=O)Nc1cc2cc(nc(N)c2cn1)-c1cnccc1C
CC(C)C(=O)Nc1cc2cc(nc(N)c2cn1)-c1cnccc1C
C[C@H](C#N)C(=O)Nc1cc2cc(nc(N)c2cn1)-c1cnccc1C |r|
Cc1ccncc1-c1cc2cc(NC(=O)C(C)(C)O)ncc2c(N)n1
Nc1nc(cc2cc(NC(=O)C3CC3)ncc12)N1CCOC1=O
Cc1ccncc1-c1cc2cc(NC(=O)[C@@H]3C[C@H]3C#N)ncc2c(N)n1 |r|
Nc1nc(cc2cc(NC(=O)C3CC3)ncc12)-c1ccc[nH]c1=O
Cc1ccncc1-c1cc2cc(NC(=O)[C@H]3C[C@@H]3C#N)ncc2c(N)n1 |r|
Nc1nc(cc2cc(NC(=O)[C@@H]3C[C@@H]3F)ncc12)-c1cnccc1CO |r|
CCC1CCCN1c1cc2cc(NC(=O)[C@@H]3C[C@@H]3F)ncc2c(N)n1 |r|
Nc1nc(cc2cc(NC(=O)[C@H]3C[C@H]3F)ncc12)-c1cnccc1C1CC1 |r|
CC1CC1C(=O)Nc1cc2cc(nc(N)c2cn1)-c1cnn(C)c1
Cc1cc(ccc1-c1cc2cc(NC(=O)[C@H]3C[C@H]3F)ncc2c(N)n1)C(N)=O |r|
CNC(=O)c1ccc(c(C)c1)-c1cc2cc(NC(=O)[C@H]3C[C@H]3F)ncc2c(N)n1 |r|
CC(C)c1ccncc1-c1cc2cc(NC(=O)[C@@H]3C[C@H]3C#N)ncc2c(N)n1 |r|
Cc1ccncc1-c1cc2cc(NC(=O)[C@H]3C[C@@H]3F)ncc2c(N)n1 |r|
Cc1c(cnc2nc[nH]c12)-c1cc2cc(NC(=O)[C@H]3C[C@H]3F)ncc2c(N)n1 |r|
CCc1ccncc1-c1cc2cc(NC(=O)[C@@H]3C[C@H]3COC)ncc2c(N)n1 |r|
Nc1nc(cc2cc(NC(=O)[C@H]3C[C@H]3F)ncc12)N1CCCC1CCO |r|
COc1cc(c(C)cn1)-c1cc2cc(NC(=O)[C@H]3C[C@H]3F)ncc2c(N)n1 |r|
Cc1c[nH]c(=O)cc1-c1cc2cc(NC(=O)[C@@H]3C[C@@H]3F)ncc2c(N)n1 |r|
CCc1ccncc1-c1cc2cc(NC(=O)OCc3ccccc3)ncc2c(N)n1
Cc1cc2NC(=O)Cc2cc1-c1cc2cc(NC(=O)[C@@H]3C[C@@H]3F)ncc2c(N)n1 |r|
Cc1cc(ncc1-c1cc2cc(NC(=O)[C@@H]3C[C@@H]3F)ncc2c(N)n1)C(C)(C)O |r|
CCc1ccncc1-c1cc2cc(NC(=O)[C@@H]3C[C@@H]3C#N)ncc2c(N)n1 |r|
CCc1ccncc1-c1cc2cc(NC(=O)[C@@H]3C[C@@H]3C(N)=O)ncc2c(N)n1 |r|
Cc1ccnc(C)c1-c1cc2cc(NC(=O)[C@@H]3C[C@@H]3F)ncc2c(N)n1 |r|
Cn1ccc2cncc(-c3cc4cc(NC(=O)[C@@H]5C[C@@H]5F)ncc4c(N)n3)c12 |r|
CCc1cc(=O)n(C)cc1-c1cc2cc(NC(=O)[C@@H]3C[C@@H]3F)ncc2c(N)n1 |r|
CCc1ccncc1-c1cc2cc(NC(=O)N[C@@H]3CCN(C)C3=O)ncc2c(N)n1 |r|
CCc1cc(OC)ncc1-c1cc2cc(NC(=O)[C@@H]3C[C@@H]3F)ncc2c(N)n1 |r|
CCc1cc(N)ncc1-c1cc2cc(NC(=O)[C@@H]3C[C@@H]3F)ncc2c(N)n1 |r|
CCc1ccncc1-c1cc2cc(NC(=O)C3=CC3)ncc2c(N)n1 |t:17|
CCc1ccncc1-c1cc2cc(NC(=O)c3cc(C)[nH]n3)ncc2c(N)n1
CCc1ccncc1-c1cc2cc(NC(=O)c3cc[nH]n3)ncc2c(N)n1
CCc1ccncc1-c1cc2cc(NC(=O)c3ccnn3C)ncc2c(N)n1
CCc1ccncc1-c1cc2cc(NC(=O)c3cnn(C)c3)ncc2c(N)n1
CCc1ccncc1-c1cc2cc(Nc3cnn(C)c3)ncc2c(N)n1
CCc1ccncc1-c1cc2cc(Nc3cn[nH]c3)ncc2c(N)n1
CCc1ccncc1-c1cc2cc(Nc3ccn(C)n3)ncc2c(N)n1
CCc1ccncc1-c1cc2cc(Nc3cc[nH]n3)ncc2c(N)n1
CCc1ccncc1-c1cc2cc(Nc3cnn(c3)C3CCNCC3)ncc2c(N)n1
CCc1ccncc1-c1cc2cc(NS(=O)(=O)C3CC3)ncc2c(N)n1
CCc1ccncc1-c1cc2cc(Nc3cc(C)ncn3)ncc2c(N)n1
CCN(C)C(=O)c1ccnc(Nc2cc3cc(nc(N)c3cn2)-c2cnccc2CC)c1
CC[C@@H](O)c1ccnc(Nc2cc3cc(nc(N)c3cn2)-c2cnccc2CC)c1 |r|
CCc1ccncc1-c1cc2cc(Nc3cccc(CO)n3)ncc2c(N)n1
CCc1ccncc1-c1cc2cc(NC(=O)c3cnn(c3)C3CCNCC3)ncc2c(N)n1
CCc1ccncc1-c1cc2cc(Nc3cnn(CCO)c3)ncc2c(N)n1
CCC1CCCN1c1cc2cc(NC(=O)[C@H]3C[C@H]3F)ncc2c(N)n1 |r|
CCc1ccncc1-c1cc2cc(NC(=O)[C@@H]3C[C@H]3C#N)ncc2c(N)n1 |r|
CCc1ccncc1-c1cc2cc(NC(=O)[C@H]3C[C@H]3C#N)ncc2c(N)n1 |r|
CCc1ccncc1-c1cc2cc(NC(=O)[C@@H]3C[C@H]3C(=O)C3CC(O)C3)ncc2c(N)n1 |r,wU:16.16,wD:18.20,(3.05,6.82,;3.05,8.36,;4.39,9.13,;5.72,8.36,;7.05,9.13,;7.05,10.67,;5.72,11.44,;4.39,10.67,;3.05,11.44,;1.72,10.67,;.39,11.44,;-.95,10.67,;-2.28,11.44,;-3.62,10.67,;-3.62,9.13,;-2.28,8.36,;-4.95,8.36,;-6.49,8.36,;-5.72,7.03,;-5.72,5.49,;-7.05,4.72,;-4.39,4.72,;-3.99,3.23,;-2.5,3.63,;-1.17,2.86,;-2.9,5.12,;-2.28,12.98,;-.95,13.75,;.39,12.98,;1.72,13.75,;1.72,15.29,;3.05,12.98,)|
Nc1nc(cc2cc(NC(=O)[C@H]3C[C@@H]3C#N)ncc12)-c1cncc2C(O)CCCc12 |r|
Cc1cnc(CO)cc1-c1cc2cc(NC(=O)[C@@H]3C[C@@H]3F)ncc2c(N)n1 |r|
Cc1cnc(cc1-c1cc2cc(NC(=O)[C@@H]3C[C@@H]3F)ncc2c(N)n1)C#N |r|
CCc1ccncc1-c1cc2cc(NC(=O)Cc3ccn[nH]3)ncc2c(N)n1
Cc1n[nH]c(C)c1-c1cc2cc(NC(=O)[C@@H]3C[C@@H]3F)ncc2c(N)n1 |r|
Cc1ncc(-c2cc3cc(NC(=O)[C@@H]4C[C@H]4C#N)ncc3c(N)n2)n1C |r|
CCc1ccncc1-c1cc2cc(NCc3ccn[nH]3)ncc2c(N)n1
Nc1nc(cc2cc(NC(=O)[C@@H]3C[C@H]3F)ncc12)-c1cccnc1 |r|
Cc1ccncc1-c1cc2cc(NC(=O)C3CC3F)ncc2c(N)n1
Cc1ccncc1-c1cc2cc(NC(=O)[C@@H]3C[C@H]3F)ncc2c(N)n1 |r|
CCc1ccncc1-c1cc2cc(NC(=O)N[C@@H]3C[C@H](O)C3)ncc2c(N)n1 |r,wU:17.17,19.20,(2.55,-2.38,;2.55,-.84,;3.88,-.07,;5.21,-.84,;6.55,-.07,;6.55,1.47,;5.21,2.24,;3.88,1.47,;2.55,2.24,;1.21,1.47,;-.12,2.24,;-1.46,1.47,;-2.79,2.24,;-4.12,1.47,;-4.12,-.07,;-2.79,-.84,;-5.46,-.84,;-5.46,-2.38,;-6.55,-3.46,;-5.46,-4.55,;-5.46,-6.09,;-4.37,-3.46,;-2.79,3.78,;-1.46,4.55,;-.12,3.78,;1.21,4.55,;1.21,6.09,;2.55,3.78,)|
Nc1nc(cc2cc(NC(=O)[C@@H]3C[C@H]3C#N)ncc12)-c1cnccc1C(F)(F)F |r|
Cc1ccncc1-c1cc2cc(NC(=O)C3C4CNCC34)ncc2c(N)n1
Nc1nc(cc2cc(NC(=O)C3C[C@@H]3C#N)ncc12)-c1cn[nH]c1 |r|
Cc1ccncc1-c1cc2cc(NC(=O)C3CC33CNC3)ncc2c(N)n1
CC(C)c1[nH]ncc1-c1cc2cc(NC(=O)C3C[C@@H]3C#N)ncc2c(N)n1 |r|
Cc1ccncc1-c1cc2cc(NC(=O)C3C4COCC34)ncc2c(N)n1
Cc1ccncc1-c1cc2cc(NC(=O)N[C@H]3CCC[C@@H]3O)ncc2c(N)n1 |r|
C[C@@H](CO)NC(=O)Nc1cc2cc(nc(N)c2cn1)-c1cnccc1C |r|
C[C@H]1CC1C(=O)Nc1cc2cc(nc(N)c2cn1)-c1cnccc1C |r|
Cc1ccncc1-c1cc2cc(NC(=O)C3C[C@@H]3C(F)(F)F)ncc2c(N)n1 |r|
Cc1ccncc1-c1cc2cc(N[C@@H]3CCNC3)ncc2c(N)n1 |r|
Cc1ccncc1-c1cc2cc(NC(=O)[C@@H]3C[C@H]3c3cc[nH]n3)ncc2c(N)n1 |r|
Cc1ccncc1-c1cc2cc(NC(=O)C3C[C@@H]3c3cn[nH]c3)ncc2c(N)n1 |r|
Cc1ccncc1-c1cc2cc(NC(=O)[C@@H]3[C@H]4COC[C@@H]34)ncc2c(N)n1 |r|
COCCN1C[C@H]2[C@@H](C1)[C@@H]2C(=O)Nc1cc2cc(nc(N)c2cn1)-c1cnccc1C |r|
Cc1ccncc1-c1cc2cc(NC(=O)[C@@H]3C[C@]33CCNC3)ncc2c(N)n1 |r|
Cc1ccncc1-c1cc2cc(NC(=O)C3C[C@]33CCNC3)ncc2c(N)n1 |r|
COCCN1CC[C@@]2(C[C@@H]2C(=O)Nc2cc3cc(nc(N)c3cn2)-c2cnccc2C)C1 |r|
COCCN1CC[C@@]2(C[C@H]2C(=O)Nc2cc3cc(nc(N)c3cn2)-c2cnccc2C)C1 |r|
CCOc1ccncc1-c1cc2cc(NC(=O)[C@H]3C[C@@H]3C#N)ncc2c(N)n1 |r|
CNC(=O)Nc1cc2cc(nc(N)c2cn1)-c1cnccc1C
Cc1ccncc1-c1cc2cc(NC(=O)[C@H]3C[C@@H]3c3cccnc3)ncc2c(N)n1 |r|
Nc1nc(cc2cc(NC(=O)[C@@H]3C[C@H]3C#N)ncc12)-c1cn[nH]c1C(F)(F)F |r|
Cc1ccncc1-c1cc2cc(NC(=O)O[C@@H]3CCNC3=O)ncc2c(N)n1 |r|
Cc1cc2[nH]c(=O)oc2cc1-c1cc2cc(NC(=O)C3C[C@@H]3C#N)ncc2c(N)n1 |r|
CN(C)C(=O)[C@@H]1C[C@@H]1C(=O)Nc1cc2cc(nc(N)c2cn1)-c1cnccc1C |r|
CCNC(=O)[C@@H]1C[C@@H]1C(=O)Nc1cc2cc(nc(N)c2cn1)-c1cnccc1C |r|
CN(C)C(=O)[C@@H]1C[C@H]1C(=O)Nc1cc2cc(nc(N)c2cn1)-c1cnccc1C |r|
C[C@@H]1C[C@H]1C(=O)Nc1cc2cc(nc(N)c2cn1)-c1cnccc1C |r|
Cc1ccncc1-c1cc2cc(NC(=O)[C@@H]3C[C@H]3C(F)(F)F)ncc2c(N)n1 |r|
C[C@H]1C[C@H]1C(=O)Nc1cc2cc(nc(N)c2cn1)-c1cnccc1C |r|
Cc1cc2n(C)c(=O)oc2cc1-c1cc2cc(NC(=O)[C@@H]3C[C@H]3C=N)ncc2c(N)n1 |r|
CC(=O)N1C[C@H]2[C@@H](C1)[C@@H]2C(=O)Nc1cc2cc(nc(N)c2cn1)-c1cnccc1C |r|
Cc1cc2[nH]c(=O)oc2cc1-c1cc2cc(NC(=O)[C@H]3C[C@@H]3c3cn[nH]c3)ncc2c(N)n1 |r|
COc1ccc(Cn2cncc2[C@H]2C[C@@H]2C(=O)Nc2cc3cc(nc(N)c3cn2)-c2cnccc2C)cc1 |r|
CCS(=O)(=O)n1cc(cn1)[C@@H]1C[C@H]1C(=O)Nc1cc2cc(nc(N)c2cn1)-c1cnccc1C |r|
Cc1c(cncc1-c1cc2cc(NC(=O)[C@H]3C[C@@H]3C#N)ncc2c(N)n1)C(F)F |r|
Cc1ccncc1-c1cc2cc(NC(=O)[C@H]3C[C@@]33CCN(C3)S(C)(=O)=O)ncc2c(N)n1 |r|
Cc1ccncc1-c1cc2cc(NC(=O)[C@@H]3C[C@@]33CCN(C3)S(C)(=O)=O)ncc2c(N)n1 |r|
Cc1ccncc1-c1cc2cc(NC(=O)C3C[C@]33CN(C3)c3cnccc3C#N)ncc2c(N)n1 |r|
Cc1ccncc1-c1cc2cc(NC(=O)[C@@H]3[C@H]4CN(C[C@@H]34)S(C)(=O)=O)ncc2c(N)n1 |r|
Cc1ccncc1-c1cc2cc(NC(=O)[C@@H]3C[C@H]3c3cnsc3)ncc2c(N)n1 |r|
Cc1ccncc1-c1nc(N)c2cnc(NC(=O)[C@H]3C[C@@H]3C#N)cc2c1F |r|
Cc1ccncc1-c1cc2cc(NC(=O)[C@H]3C[C@@H]3CO)ncc2c(N)n1 |r|
Cc1ccncc1-c1cc2cc(NC(=O)[C@@H]3C[C@H]3CN)ncc2c(N)n1 |r|
CC(=O)Nc1cc2c(F)c(nc(N)c2cn1)-c1cnccc1C
Cc1ccncc1-c1cc2cc(NC(=O)[C@H]3C[C@@H]3CC#N)ncc2c(N)n1 |r|
Cc1ccncc1-c1cc2cc(NC(=O)[C@H]3[C@@H]4CNC(=O)[C@H]34)ncc2c(N)n1 |r|
Cc1ccncc1-c1cc2cc(NC(=O)[C@@H]3C[C@H]3c3cnn(C)c3)ncc2c(N)n1 |r|
Cc1cc2NC(=O)C(O)c2cc1-c1cc2cc(NC(=O)[C@H]3C[C@@H]3C#N)ncc2c(N)n1 |r|
CC(=O)N1CC(C1)n1cc(Nc2cc3cc(nc(N)c3cn2)-c2cnccc2C)cn1
Cc1ccncc1-c1nc(N)c2cnc(NC(=O)Nc3cnn(C)c3)cc2c1F
Cc1ccncc1-c1nc(N)c2cnc(NC(=O)Nc3cnn(C)c3)cc2c1Cl
Cc1cc(ccc1-c1cc2cc(NC(=O)[C@@H]3C[C@H]3C#N)ncc2c(N)n1)C(=O)NCC(F)(F)F |r|
Cc1c(N)cncc1-c1cc2cc(NC(=O)C3C[C@@H]3C#N)ncc2c(N)n1 |r|
CC(=O)N1CCC(CC1)[C@H]1C[C@@H]1C(=O)Nc1cc2cc(nc(N)c2cn1)-c1cnccc1C |r|
Cc1cc(ncc1-c1cc2cc(NC(=O)[C@@H]3C[C@@H]3F)ncc2c(N)n1)-c1ccc[nH]c1=O |r|
Cc1ccncc1-c1cc2cc(Nc3cnn(CCO)c3)ncc2c(N)n1
Cc1ccncc1-c1cc2cc(Nc3ccn(C)c(=O)c3)ncc2c(N)n1
Cc1ccncc1-c1cc2cc(NC(=O)Nc3ccccc3C#N)ncc2c(N)n1
Cc1ccncc1-c1nc(N)c2cnc(NC(=O)[C@@H]3C[C@H]3c3cn[nH]c3)cc2c1F |r|
Cc1ccncc1-c1nc(N)c2cnc(NC(=O)[C@@H]3C[C@H]3c3cn[nH]c3)cc2c1Cl |r|
COCCN1CC(C1)NC(=O)Nc1cc2cc(nc(N)c2cn1)-c1cnccc1C
Cc1ccncc1-c1cc2cc(NC(=O)NC3CNC3)ncc2c(N)n1
C[C@H](C#N)n1cc(NC(=O)Nc2cc3cc(nc(N)c3cn2)-c2cnccc2C)cn1 |r|
Cc1cc(ncc1-c1cc2cc(NC(=O)[C@@H]3C[C@@H]3F)ncc2c(N)n1)N1CC[C@H](N)C1 |r|
CNC(=O)c1c(C)c(c(C)n1C)-c1cc2cc(NC(=O)C3C[C@H]3C#N)ncc2c(N)n1 |r|
C[C@@H]1C[C@H]1C(=O)Nc1cc2cc(nc(N)c2cn1)-c1c(C)ncc(N)c1C |r|
CNC(=O)C(C)(C)n1cc(Nc2cc3cc(nc(N)c3cn2)-c2cnccc2C)cn1
CN(C)C(=O)C(C)(C)n1cc(Nc2cc3cc(nc(N)c3cn2)-c2cnccc2C)cn1
CNC(=O)Cn1cc(Cc2cc3cc(nc(N)c3cn2)-c2cnccc2C)cn1
Cc1cc(C)c(cc1C(N)=O)-c1cc2cc(NC(=O)[C@@H]3C[C@H]3C#N)ncc2c(N)n1 |r|
C[C@H]1COC(=O)N1c1cc2cc(NC(=O)[C@@H]3C[C@H]3C#N)ncc2c(N)n1 |r|
Cc1[nH]ncc1-c1cc2cc(NC(=O)[C@@H]3C[C@H]3C(F)(F)F)ncc2c(N)n1 |r|
Cc1nn(C)c(C)c1-c1cc2cc(NC(=O)[C@H]3C[C@@H]3C(F)(F)F)ncc2c(N)n1 |r|
Cc1ccncc1-c1cc2cc(NC(=O)[C@H]3C[C@@H]3c3ncccn3)ncc2c(N)n1 |r|
Cc1c(N)cncc1-c1cc2cc(NC(=O)[C@H]3C[C@@H]3C(F)(F)F)ncc2c(N)n1 |r|
Nc1nc(cc2cc(NC(=O)C3C[C@H]3C#N)ncc12)-c1cnccc1CCO |r|
Nc1nc(cc2cc(NC(=O)[C@H]3C[C@@H]3CC#N)ncc12)-c1cnccc1CCO |r|
Cc1ccncc1-c1cc2cc(NC(=O)[C@@H]3C[C@H]3CC#N)ncc2c(N)n1 |r|
Cc1ccncc1-c1nc(N)c2cnc(NC(=O)[C@H]3C[C@@H]3c3cn[nH]c3)cc2c1F |r|
Cc1ccncc1-c1cc2cc(NC(=O)[C@H]3C[C@@H]3c3cnn(C)c3)ncc2c(N)n1 |r|
Cc1c(N)cncc1-c1cc2cc(NC(=O)[C@@H]3C[C@H]3C#N)ncc2c(N)n1 |r|
Cc1c(N)cncc1-c1cc2cc(NC(=O)[C@H]3C[C@@H]3C#N)ncc2c(N)n1 |r|
Cc1ccncc1-c1nc(N)c2cnc(NC(=O)C3CC3)cc2c1C1=C[C@@H](O)CC1 |r,t:28|
Cc1ccncc1-c1nc(N)c2cnc(NC(=O)[C@H]3C[C@@H]3CC#N)cc2c1C |r|
Cc1ccnc(-c2ccccc2)c1-c1cc2cc(NC(=O)[C@H]3C[C@@H]3CC#N)ncc2c(N)n1 |r|
CC(=O)OC[C@@]1(C)C[C@@H]1C(=O)Nc1cc2cc(nc(N)c2cn1)-c1cnccc1C |r|
CC(=O)OC[C@]1(C)C[C@@H]1C(=O)Nc1cc2cc(nc(N)c2cn1)-c1cnccc1C |r|
Cc1ccncc1-c1cc2cc(NC(=O)C3CC3(C)CO)ncc2c(N)n1
Cc1ccncc1-c1nc(N)c2cnc(NC(=O)[C@@H]3C[C@H]3CC#N)cc2c1Br |r|
Nc1nc(cc2cc(NC(=O)[C@@H]3C[C@@H]3F)ncc12)-c1cncc2NCCc12 |r|
C[C@@H](CO)n1cc(Nc2cc3cc(nc(N)c3cn2)-c2cnccc2C)cn1 |r|
Cn1cc(cn1)[C@@H]1C[C@H]1C(=O)Nc1cc2cc(nc(N)c2cn1)-c1cnccc1CCO |r|
Cn1cc(cn1)[C@H]1C[C@@H]1C(=O)Nc1cc2cc(nc(N)c2cn1)-c1cnccc1CCO |r|
CNc1cncc(c1C)-c1cc2cc(NC(=O)[C@H]3C[C@H]3F)ncc2c(N)n1 |r|
CC(C#N)n1cc(Nc2cc3cc(nc(N)c3cn2)-c2cnccc2C)cn1
CC(=O)N1CC[C@@H](C1)n1cc(Nc2cc3cc(nc(N)c3cn2)-c2cnccc2C)cn1 |r|
Cc1ccncc1-c1cc2cc(Nc3cnn(c3)[C@H]3CN(CC[C@@H]3O)C3COC3)ncc2c(N)n1 |r|
Cc1ccncc1-c1cc2cc(Nc3cnn(c3)[C@@H]3CCN(C[C@H]3O)C3COC3)ncc2c(N)n1 |r|
C[C@@H](O)c1cc(Nc2cc3cc(nc(N)c3cn2)-c2cnccc2C)nn1C |r|
Nc1nc(cc2cc(NC(=O)[C@@H]3C[C@@H]3F)ncc12)-c1cncc2NC(=O)COc12 |r|
Nc1nc(cc2cc(NC(=O)[C@@H]3C[C@@H]3F)ncc12)-c1cncc2NCCOc12 |r|
Nc1nc(cc2cc(NC(=O)[C@@H]3C[C@H]3C#N)ncc12)-c1ccccc1C#N |r|
CC(C)(O)Cc1ccncc1-c1cc2cc(NC(=O)[C@@H]3C[C@H]3C#N)ncc2c(N)n1 |r|
CNC(=O)c1cncc(c1C)-c1cc2cc(NC(=O)[C@H]3C[C@H]3F)ncc2c(N)n1 |r|
Nc1nc(cc2cc(NC(=O)[C@@H]3C[C@H]3C#N)ncc12)-c1cnccc1CC#N |r|
COCc1ccncc1-c1cc2cc(NC(=O)[C@@H]3C[C@H]3C#N)ncc2c(N)n1 |r|
COCCc1ccncc1-c1cc2cc(NC(=O)[C@H]3C[C@@H]3C#N)ncc2c(N)n1 |r|
COCc1ccncc1-c1cc2cc(NC(=O)C3[C@@H]4CC[C@H](C#N)[C@H]34)ncc2c(N)n1 |r|
Cc1ccncc1-c1cc2cc(NC(=O)[C@H]3C[C@@H]3C3CNC(=O)O3)ncc2c(N)n1 |r|
CC(O)Cc1ccncc1-c1cc2cc(NC(=O)[C@H]3C[C@@H]3C#N)ncc2c(N)n1 |r|
Cc1ccncc1-c1nc(N)c2cnc(NC(=O)[C@H]3C[C@@H]3c3cnn(C)c3)cc2c1Cl |r|
Cc1ccncc1-c1nc(N)c2cnc(NC(=O)[C@@H]3C[C@H]3c3cnn(C)c3)cc2c1Cl |r|
Nc1nc(cc2cc(NC(=O)C3C[C@H]3C#N)ncc12)-c1cnccc1-c1cn[nH]c1 |r|
Nc1nc(cc2cc(NC(=O)[C@H]3C[C@@H]3C#N)ncc12)-c1cnccc1-c1cn[nH]c1 |r|
Cc1cc(ncc1-c1cc2cc(NC(=O)[C@@H]3C[C@H]3CC#N)ncc2c(N)n1)-c1cnn(C)c1 |r|
Cc1cc(ncc1-c1cc2cc(NC(=O)[C@H]3C[C@@H]3CC#N)ncc2c(N)n1)-c1cnn(C)c1 |r|
COC(C)(C)[C@@H]1C[C@H]1C(=O)Nc1cc2cc(nc(N)c2cn1)-c1cnccc1C |r|
COC(C)(C)[C@H]1C[C@@H]1C(=O)Nc1cc2cc(nc(N)c2cn1)-c1cnccc1C |r|
Cc1ccncc1-c1cc2cc(NC(=O)[C@@H]3C[C@H]3C(C)(C)O)ncc2c(N)n1 |r|
Cc1ccncc1-c1cc2cc(NC(=O)[C@H]3C[C@@H]3C(C)(C)O)ncc2c(N)n1 |r|
Nc1nc(cc2cc(NC(=O)[C@@H]3C[C@H]3C#N)ncc12)-c1cnccc1-c1cc[nH]n1 |r|
Nc1nc(cc2cc(NC(=O)[C@H]3C[C@@H]3C#N)ncc12)-c1cnccc1-c1cc[nH]n1 |r|
Nc1nc(cc2cc(NC(=O)[C@H]3C[C@@H]3c3cnsc3)ncc12)-c1cnccc1CCO |r|
Nc1nc(cc2cc(NC(=O)[C@@H]3C[C@H]3c3cnsc3)ncc12)-c1cnccc1CCO |r|
Cc1c(N)cncc1-c1cc2cc(NC(=O)[C@H]3C[C@@H]3CC#N)ncc2c(N)n1 |r|
Cc1c(N)cncc1-c1cc2cc(NC(=O)[C@@H]3C[C@H]3CC#N)ncc2c(N)n1 |r|
CN1CC[C@H](C1=O)n1cc(Nc2cc3cc(nc(N)c3cn2)-c2cnccc2C)cn1 |r|
CN1CC[C@@H](C1=O)n1cc(Nc2cc3cc(nc(N)c3cn2)-c2cnccc2C)cn1 |r|
CN1CCC[C@H](C1=O)n1cc(Nc2cc3cc(nc(N)c3cn2)-c2cnccc2C)cn1 |r|
CN1CCC[C@@H](C1=O)n1cc(Nc2cc3cc(nc(N)c3cn2)-c2cnccc2C)cn1 |r|
Nc1nc(cc2cc(NC(=O)[C@@H]3C[C@H]3c3cccnc3)ncc12)-c1cnccc1CCO |r|
Nc1nc(cc2cc(NC(=O)[C@H]3C[C@@H]3c3cccnc3)ncc12)-c1cnccc1CCO |r|
Cc1ccncc1-c1cc2cc(NC(=O)[C@@H]3[C@H]4CN(C[C@@H]34)C3COC3)ncc2c(N)n1 |r|
CN1CCc2cc(Nc3cc4cc(nc(N)c4cn3)-c3cnccc3C)nn2CC1=O
Cc1ccncc1-c1cc2cc(Nc3cnn(CC(F)F)c3)ncc2c(N)n1
Cc1ccncc1-c1nc(N)c2cnc(NC(=O)C3CC3)cc2c1-c1cn[nH]c1
Cc1ccncc1-c1cc2cc(Nc3cc(C4CC4)n(CCO)n3)ncc2c(N)n1
Cc1ccncc1-c1cc2cc(Nc3cnn(CC(C)(C)O)c3)ncc2c(N)n1
Cc1cc(Nc2cc3cc(nc(N)c3cn2)-c2cnccc2C)n(CCO)n1
Cc1cc(Nc2cc3cc(nc(N)c3cn2)-c2cnccc2C)cn1CCO
CNC(=O)c1cc(Nc2cc3cc(nc(N)c3cn2)-c2cnccc2C)nn1C
Cc1ccncc1-c1cc2cc(Nc3ccc(CS(N)(=O)=O)cc3)ncc2c(N)n1
Cc1ccncc1-c1cc2cc(Nc3ccc(cc3)N3CCNCC3=O)ncc2c(N)n1
Cc1ccncc1-c1cc2cc(Nc3cnn(c3)C(C)(C)CO)ncc2c(N)n1
Cc1ccc(F)cc1-c1cc2cc(NC(=O)[C@H]3C[C@@H]3c3cnn(C)c3)ncc2c(N)n1 |r|
Cc1ccc(O)cc1-c1cc2cc(NC(=O)C3CC3c3cnn(C)c3)ncc2c(N)n1
Cc1ccncc1-c1nc(N)c2cnc(NC(=O)[C@@H]3C[C@H]3CC#N)cc2c1Cl |r|
Cc1ccncc1-c1nc(N)c2cnc(NC(=O)[C@H]3C[C@@H]3CC#N)cc2c1Cl |r|
CCc1c(nc(N)c2cnc(NC(=O)[C@H]3C[C@@H]3CC#N)cc12)-c1cnccc1C |r|
CCc1c(nc(N)c2cnc(NC(=O)[C@@H]3C[C@H]3CC#N)cc12)-c1cnccc1C |r|
C[C@H](C#N)n1cc(Nc2cc3cc(nc(N)c3cn2)-c2cnccc2C)cn1 |r|
C[C@@H](C#N)n1cc(Nc2cc3cc(nc(N)c3cn2)-c2cnccc2C)cn1 |r|
Cc1ccncc1-c1nc(N)c2cnc(NC(=O)[C@H]3C[C@@H]3CC#N)cc2c1C=C |r|
C[C@@H]1[C@H](CC#N)[C@H]1C(=O)Nc1cc2cc(nc(N)c2cn1)-c1cnccc1C |r|
C[C@H]1[C@@H](CC#N)[C@@H]1C(=O)Nc1cc2cc(nc(N)c2cn1)-c1cnccc1C |r|
C[C@H]1[C@H](CC#N)[C@H]1C(=O)Nc1cc2cc(nc(N)c2cn1)-c1cnccc1C |r|
C[C@@H]1[C@@H](CC#N)[C@@H]1C(=O)Nc1cc2cc(nc(N)c2cn1)-c1cnccc1C |r|
Cc1ccc(O)cc1-c1cc2cc(NC(=O)[C@H]3C[C@@H]3c3cnn(C)c3)ncc2c(N)n1 |r|
Cc1ccc(O)cc1-c1cc2cc(NC(=O)[C@@H]3C[C@H]3c3cnn(C)c3)ncc2c(N)n1 |r|
COc1ccc(C)c(c1)-c1cc2cc(NC(=O)[C@H]3C[C@@H]3c3cnn(C)c3)ncc2c(N)n1 |r|
COc1ccc(C)c(c1)-c1cc2cc(NC(=O)C3C[C@H]3c3cnn(C)c3)ncc2c(N)n1 |r|
CN(C)C(=O)c1ccc(C)c(c1)-c1cc2cc(NC(=O)[C@H]3C[C@@H]3c3cnn(C)c3)ncc2c(N)n1 |r|
CN(C)C(=O)c1ccc(C)c(c1)-c1cc2cc(NC(=O)[C@@H]3C[C@H]3c3cnn(C)c3)ncc2c(N)n1 |r|
Cc1ccncc1-c1cc2cc(NC(=O)[C@H]3C[C@@H]3c3cnn(CCOCCN)c3)ncc2c(N)n1 |r|
Cc1ccncc1-c1cc2cc(NC(=O)[C@@H]3C[C@H]3c3cnn(CCOCCN)c3)ncc2c(N)n1 |r|
COC1CN(C1)[C@@H]1C[C@H]2[C@@H](C1)[C@@H]2C(=O)Nc1cc2cc(nc(N)c2cn1)-c1cnccc1C |r|
NCCOCCn1cc(cn1)[C@H]1C[C@@H]1C(=O)Nc1cc2cc(nc(N)c2cn1)-c1c(Cl)cccc1Cl |r|
NCCOCCn1cc(cn1)[C@@H]1C[C@H]1C(=O)Nc1cc2cc(nc(N)c2cn1)-c1c(Cl)cccc1Cl |r|
Cc1ccncc1-c1cc2cc(NC(=O)[C@@H]3[C@H]4CC(C[C@@H]34)N3CCOCC3)ncc2c(N)n1 |r|
Cc1ccccc1-c1cc2cc(NC(=O)[C@@H]3C[C@H]3c3cnn(C)c3)ncc2c(N)n1 |r|
Cc1ccccc1-c1cc2cc(NC(=O)[C@H]3C[C@@H]3c3cnn(C)c3)ncc2c(N)n1 |r|
Cc1ccc(cc1-c1cc2cc(NC(=O)[C@@H]3CC3c3cnn(C)c3)ncc2c(N)n1)C#N |r|
Cc1ccc(cc1-c1cc2cc(NC(=O)[C@H]3C[C@@H]3c3cnn(C)c3)ncc2c(N)n1)C#N |r|
Cn1cc(cn1)[C@@H]1C[C@H]1C(=O)Nc1cc2cc(nc(N)c2cn1)-c1c(F)cccc1Cl |r|
Cn1cc(cn1)[C@H]1C[C@@H]1C(=O)Nc1cc2cc(nc(N)c2cn1)-c1c(F)cccc1Cl |r|
Cn1cc(cn1)[C@@H]1C[C@H]1C(=O)Nc1cc2cc(nc(N)c2cn1)-c1ccccc1Cl |r|
Cn1cc(cn1)[C@H]1C[C@@H]1C(=O)Nc1cc2cc(nc(N)c2cn1)-c1ccccc1Cl |r|
Cn1cc(cn1)[C@@H]1C[C@H]1C(=O)Nc1cc2cc(nc(N)c2cn1)-c1c(F)cccc1F |r|
Cn1cc(cn1)[C@H]1C[C@@H]1C(=O)Nc1cc2cc(nc(N)c2cn1)-c1c(F)cccc1F |r|
Cc1cc(ncc1-c1cc2cc(NC(=O)[C@H]3C[C@@H]3c3cnn(C)c3)ncc2c(N)n1)-c1ncco1 |r|
Cc1cc(ncc1-c1cc2cc(NC(=O)[C@@H]3C[C@H]3c3cnn(C)c3)ncc2c(N)n1)-c1ncco1 |r|
Nc1nc(cc2cc(NC(=O)[C@H]3C[C@@H]3CC#N)ncc12)-c1c(Cl)cccc1Cl |r|
Nc1nc(cc2cc(NC(=O)C3C[C@H]3CC#N)ncc12)-c1c(Cl)cccc1Cl |r|
Cc1ccncc1-c1cc2cc(NC(=O)[C@@H]3C[C@@]33CCNC(=O)C3)ncc2c(N)n1 |r|
Cc1ccncc1-c1cc2cc(NC(=O)[C@H]3C[C@]33CCNC(=O)C3)ncc2c(N)n1 |r|
Cc1ccncc1-c1cc2cc(NC(=O)C3C[C@@]33CCNC(=O)C3)ncc2c(N)n1 |r|
Cc1ccncc1-c1cc2cc(NC(=O)[C@@H]3C[C@]33CCNC(=O)C3)ncc2c(N)n1 |r|
Cc1ccncc1-c1nc(N)c2cnc(NC(=O)[C@@H]3C[C@H]3CC#N)cc2c1C1CC1 |r|
Cc1ccncc1-c1nc(N)c2cnc(NC(=O)[C@H]3C[C@@H]3CC#N)cc2c1C1CC1 |r|
Cc1ccnc(-c2ccccc2)c1-c1cc2cc(NC(=O)[C@H]3C[C@@H]3c3cnn(C)c3)ncc2c(N)n1 |r|
Cc1ccnc(-c2ccccc2)c1-c1cc2cc(NC(=O)[C@@H]3C[C@H]3c3cnn(C)c3)ncc2c(N)n1 |r|
C[C@H]1CC[C@@H]1C(=O)Nc1cc2cc(nc(N)c2cn1)-c1cnccc1C |r|
C[C@@H]1CC[C@@H]1C(=O)Nc1cc2cc(nc(N)c2cn1)-c1cnccc1C |r|
C[C@@H]1CC[C@H]1C(=O)Nc1cc2cc(nc(N)c2cn1)-c1cnccc1C |r|
C[C@H]1CC[C@H]1C(=O)Nc1cc2cc(nc(N)c2cn1)-c1cnccc1C |r|
Cc1ccncc1-c1cc2cc(NC(=O)[C@H]3C[C@@H]3C3CCOCC3)ncc2c(N)n1 |r|
Cc1ccncc1-c1cc2cc(NC(=O)[C@@H]3C[C@H]3C3CCOCC3)ncc2c(N)n1 |r|
C[C@@H]1[C@H]([C@@H]1c1cnn(C)c1)C(=O)Nc1cc2cc(nc(N)c2cn1)-c1cnccc1C |r|
C[C@H]1[C@@H]([C@H]1c1cnn(C)c1)C(=O)Nc1cc2cc(nc(N)c2cn1)-c1cnccc1C |r|
C[C@@H]1[C@@H]([C@H]1c1cnn(C)c1)C(=O)Nc1cc2cc(nc(N)c2cn1)-c1cnccc1C |r|
C[C@H]1[C@H]([C@@H]1c1cnn(C)c1)C(=O)Nc1cc2cc(nc(N)c2cn1)-c1cnccc1C |r|
COCCn1cc(cn1)[C@@H]1C[C@H]1C(=O)Nc1cc2cc(nc(N)c2cn1)-c1cnccc1C |r|
COCCn1cc(cn1)[C@H]1C[C@@H]1C(=O)Nc1cc2cc(nc(N)c2cn1)-c1cnccc1C |r|
Cn1cc(cn1)[C@H]1CC1C(=O)Nc1cc2c(Cl)c(nc(N)c2cn1)-c1cnccc1CCO |r|
Cn1cc(cn1)[C@@H]1C[C@H]1C(=O)Nc1cc2c(Cl)c(nc(N)c2cn1)-c1cnccc1CCO |r|
Cc1cc(ncc1-c1cc2cc(NC(=O)[C@@H]3C[C@H]3CC#N)ncc2c(N)n1)-c1ccccc1 |r|
Cc1cc(ncc1-c1cc2cc(NC(=O)[C@H]3C[C@@H]3CC#N)ncc2c(N)n1)-c1ccccc1 |r|
Cc1ccncc1-c1cc2cc(NC(=O)C3CC33CC3)ncc2c(N)n1
Cc1ccncc1-c1cc2cc(NCC3CC3(F)F)ncc2c(N)n1
Cc1ccncc1-c1cc2cc(NCC(F)F)ncc2c(N)n1
Cn1cc(cn1)[C@H]1C[C@@H]1C(=O)Nc1cc2cc(nc(N)c2cn1)-c1cnc2c(cnn(C)c2=O)c1 |r|
CN(C)C(=O)c1cc(C)c(cn1)-c1cc2cc(NC(=O)[C@H]3C[C@@H]3c3cnn(C)c3)ncc2c(N)n1 |r|
COC(=O)c1cc(C)c(cn1)-c1cc2cc(NC(=O)[C@H]3C[C@@H]3c3cnn(C)c3)ncc2c(N)n1 |r|
Cc1cc(ncc1-c1cc2cc(NC(=O)[C@@H]3C[C@H]3c3cnn(C)c3)ncc2c(N)n1)C(O)=O |r|
Cc1cc(ncc1-c1cc2cc(NC(=O)[C@H]3C[C@@H]3c3cnn(C)c3)ncc2c(N)n1)N1CCC1=O |r|
Cc1cc(ncc1-c1cc2cc(NC(=O)[C@H]3C[C@@H]3c3cnn(C)c3)ncc2c(N)n1)-c1ccn(C)n1 |r|
Cc1cc(ncc1-c1cc2cc(NC(=O)[C@H]3C[C@@H]3c3cnn(C)c3)ncc2c(N)n1)-n1cccn1 |r|
CNC(=O)c1cc(C)c(cn1)-c1cc2cc(NC(=O)[C@@H]3C[C@H]3c3cnn(C)c3)ncc2c(N)n1 |r|
Cn1cc(cn1)[C@H]1C[C@@H]1C(=O)Nc1cc2cc(nc(N)c2cn1)-c1cnc(N)c(c1)C(F)(F)F |r|
Cc1cc(ncc1-c1cc2cc(NC(=O)[C@H]3C[C@@H]3c3cnn(C)c3)ncc2c(N)n1)C(=O)OCc1ccccc1 |r|
C[C@H]1[C@@H]([C@H]1c1cnn(C)c1)C(=O)Nc1cc2cc(nc(N)c2cn1)-c1c(C)cc(cc1F)-c1ncco1 |r|
C[C@@H]1[C@@H]([C@H]1c1cnn(C)c1)C(=O)Nc1cc2cc(nc(N)c2cn1)-c1c(C)cc(cc1F)-c1ncco1 |r|
Cc1cc(cc(F)c1-c1cc2cc(NC(=O)[C@H]3C[C@@H]3c3cnn(C)c3)ncc2c(N)n1)C(N)=O |r|
Cc1cc(cc(F)c1-c1cc2cc(NC(=O)[C@@H]3C[C@H]3c3cnn(C)c3)ncc2c(N)n1)C(N)=O |r|
Cc1ccc2c(CC[C@@]2(C)O)c1-c1cc2cc(NC(=O)[C@H]3C[C@@H]3CC#N)ncc2c(N)n1 |r|
C[C@@H]1[C@H]([C@@H]1c1cnn(C)c1)C(=O)Nc1cc2cc(nc(N)c2cn1)-c1c(C)cccc1F |r|
C[C@@H]1[C@@H]([C@H]1c1cnn(C)c1)C(=O)Nc1cc2cc(nc(N)c2cn1)-c1c(C)cccc1F |r|
C[C@H]1[C@H]([C@@H]1c1cnn(C)c1)C(=O)Nc1cc2cc(nc(N)c2cn1)-c1c(C)cccc1F |r|
C[C@H]1[C@@H]([C@H]1c1cnn(C)c1)C(=O)Nc1cc2cc(nc(N)c2cn1)-c1c(C)cccc1F |r|
C[C@H]1[C@@H]([C@H]1c1cnn(C)c1)C(=O)Nc1cc2cc(nc(N)c2cn1)-c1cccc(N)c1C |r|
Cc1cccc(F)c1-c1cc2cc(NC(=O)[C@@H]3C[C@H]3CC#N)ncc2c(N)n1 |r|
Cc1cccc(F)c1-c1cc2cc(NC(=O)[C@H]3C[C@@H]3CC#N)ncc2c(N)n1 |r|
Cc1cccc(Cl)c1-c1cc2cc(NC(=O)[C@@H]3C[C@H]3CC#N)ncc2c(N)n1 |r|
Cc1cccc(Cl)c1-c1cc2cc(NC(=O)[C@H]3C[C@@H]3CC#N)ncc2c(N)n1 |r|
Cc1c(N)ccc(Cl)c1-c1cc2cc(NC(=O)[C@H]3C[C@@H]3CC#N)ncc2c(N)n1 |r|
Cc1c(N)ccc(Cl)c1-c1cc2cc(NC(=O)[C@@H]3C[C@H]3CC#N)ncc2c(N)n1 |r|
Cc1c(N)cccc1-c1cc2cc(NC(=O)[C@@H]3C[C@H]3CC#N)ncc2c(N)n1 |r|
Cc1c(N)cccc1-c1cc2cc(NC(=O)[C@H]3C[C@@H]3CC#N)ncc2c(N)n1 |r|
Cn1cc(cn1)[C@H]1C[C@@H]1C(=O)Nc1cc2cc(nc(N)c2cn1)-c1cc(ccc1Cl)C#N |r|
Cc1ccccc1-c1cc2cc(NC(=O)[C@@H]3C[C@H]3CC#N)ncc2c(N)n1 |r|
Cc1ccccc1-c1cc2cc(NC(=O)[C@H]3C[C@@H]3CC#N)ncc2c(N)n1 |r|
Cc1ccc(cc1-c1cc2cc(NC(=O)[C@@H]3C[C@H]3CC#N)ncc2c(N)n1)C#N |r|
Cc1ccc(cc1-c1cc2cc(NC(=O)[C@H]3C[C@@H]3CC#N)ncc2c(N)n1)C#N |r|
Cc1cc(ccc1-c1cc2cc(NC(=O)[C@H]3C[C@@H]3c3cnn(C)c3)ncc2c(N)n1)-c1nc(co1)-c1ccccc1 |r|
Cc1cc(ccc1-c1cc2cc(NC(=O)[C@@H]3C[C@H]3c3cnn(C)c3)ncc2c(N)n1)-c1nc(co1)-c1ccccc1 |r|
CC(C)c1coc(n1)-c1ccc(c(C)c1)-c1cc2cc(NC(=O)[C@H]3C[C@@H]3c3cnn(C)c3)ncc2c(N)n1 |r|
CC(C)c1coc(n1)-c1ccc(c(C)c1)-c1cc2cc(NC(=O)[C@@H]3C[C@H]3c3cnn(C)c3)ncc2c(N)n1 |r|
Cn1cc(cn1)[C@@H]1C[C@H]1C(=O)Nc1cc2cc(nc(N)c2cn1)-c1c(Cl)cccc1Cl |r|
Cn1cc(cn1)[C@H]1C[C@@H]1C(=O)Nc1cc2cc(nc(N)c2cn1)-c1c(Cl)cccc1Cl |r|
Cc1cc(ccc1-c1cc2cc(NC(=O)[C@H]3C[C@@H]3c3cnn(C)c3)ncc2c(N)n1)-c1ncco1 |r|
Cc1cc(ccc1-c1cc2cc(NC(=O)[C@@H]3C[C@H]3c3cnn(C)c3)ncc2c(N)n1)-c1ncco1 |r|
Cc1cccc(CC#N)c1-c1cc2cc(NC(=O)[C@@H]3C[C@H]3c3cnn(C)c3)ncc2c(N)n1 |r|
Cc1cccc(F)c1-c1cc2cc(NC(=O)[C@@H]3C[C@H]3c3cnn(C)c3)ncc2c(N)n1 |r|
CC(C)[C@H]1COC(=N1)c1cc(C)c(cn1)-c1cc2cc(NC(=O)[C@H]3C[C@@H]3c3cnn(C)c3)ncc2c(N)n1 |r,c:6|
COC(=O)[C@@H]1COC(=N1)c1cc(C)c(cn1)-c1cc2cc(NC(=O)[C@H]3C[C@@H]3c3cnn(C)c3)ncc2c(N)n1 |r,c:7|
COC(=O)[C@@H]1COC(=N1)c1cc(C)c(cn1)-c1cc2cc(NC(=O)[C@@H]3C[C@H]3c3cnn(C)c3)ncc2c(N)n1 |r,c:7|
COCc1cc(C)c(cn1)-c1cc2cc(NC(=O)[C@H]3C[C@@H]3c3cnn(C)c3)ncc2c(N)n1 |r|
COCc1cc(C)c(cn1)-c1cc2cc(NC(=O)[C@@H]3C[C@H]3c3cnn(C)c3)ncc2c(N)n1 |r|
Cc1ccncc1-c1cc2cc(Nc3ccc(CC#N)cn3)ncc2c(N)n1
Cc1ccncc1C#Cc1cc2cc(NC(=O)[C@H]3C[C@@H]3c3cnn(C)c3)ncc2c(N)n1 |r|
Cc1ccncc1C#Cc1cc2cc(NC(=O)[C@@H]3C[C@H]3c3cnn(C)c3)ncc2c(N)n1 |r|
COc1cncc(c1C)-c1cc2cc(NC(=O)[C@H]3C[C@@H]3c3cnn(C)c3)ncc2c(N)n1 |r|
COc1cncc(c1C)-c1cc2cc(NC(=O)[C@@H]3C[C@H]3c3cnn(C)c3)ncc2c(N)n1 |r|
COc1cc(C)c(cn1)-c1cc2cc(NC(=O)[C@H]3C[C@@H]3c3cnn(C)c3)ncc2c(N)n1 |r|
COc1cc(C)c(cn1)-c1cc2cc(NC(=O)[C@@H]3C[C@H]3c3cnn(C)c3)ncc2c(N)n1 |r|
Cc1ccnc(Cc2ccccc2)c1-c1cc2cc(NC(=O)[C@@H]3C[C@H]3c3cnn(C)c3)ncc2c(N)n1 |r|
Cc1cc(ncc1-c1cc2cc(NC(=O)[C@@H]3C[C@H]3c3cnn(C)c3)ncc2c(N)n1)-n1cccn1 |r|
Cc1cc(ncc1-c1cc2cc(NC(=O)[C@@H]3C[C@H]3c3cnn(C)c3)ncc2c(N)n1)N1CCC1=O |r|
COC(=O)c1cc(C)c(cn1)-c1cc2cc(NC(=O)[C@@H]3C[C@H]3c3cnn(C)c3)ncc2c(N)n1 |r|
Cc1cc(ncc1-c1cc2cc(NC(=O)[C@@H]3C[C@H]3c3cnn(C)c3)ncc2c(N)n1)-c1ccn(C)n1 |r|
Cc1nc2c(cnn(C)c2=O)cc1-c1cc2cc(NC(=O)[C@H]3C[C@@H]3c3cnn(C)c3)ncc2c(N)n1 |r|
Cc1nc2c(cnn(C)c2=O)cc1-c1cc2cc(NC(=O)[C@@H]3C[C@H]3c3cnn(C)c3)ncc2c(N)n1 |r|
Cc1c(cnc2c1cnn(C)c2=O)-c1cc2cc(NC(=O)[C@H]3C[C@@H]3c3cnn(C)c3)ncc2c(N)n1 |r|
Cc1c(cnc2c1cnn(C)c2=O)-c1cc2cc(NC(=O)[C@@H]3C[C@H]3c3cnn(C)c3)ncc2c(N)n1 |r|
Cc1nc2c(cnn(C)c2=O)c(C)c1-c1cc2cc(NC(=O)[C@H]3C[C@@H]3c3cnn(C)c3)ncc2c(N)n1 |r|
Cc1nc2c(cnn(C)c2=O)c(C)c1-c1cc2cc(NC(=O)[C@@H]3C[C@H]3c3cnn(C)c3)ncc2c(N)n1 |r|
Cc1ccncc1-c1cc2cc(NC(=O)[C@@H]3[C@H]4CC(C[C@@H]34)NS(C)(=O)=O)ncc2c(N)n1 |r|
CN1CC2(CC2)c2cc(Nc3cc4cc(nc(N)c4cn3)-c3cncc(N)c3C)nn2CC1=O
CN1CCc2cc(Nc3cc4cc(nc(N)c4cn3)-c3cncc(N)c3C)nn2CC1=O
Cc1ccncc1-c1cc2cc(Nc3cc4COC[C@H](C#N)n4n3)ncc2c(N)n1 |r|
Cc1ccncc1-c1cc2cc(Nc3cc4COC[C@@H](C#N)n4n3)ncc2c(N)n1 |r|
CN1C=C(C)c2ccc(Nc3cc4cc(nc(N)c4cn3)-c3cnccc3C)nc2CC1=O |t:2|
CC(C)N1CCc2cc(Nc3cc4cc(nc(N)c4cn3)[C@@H](C)Oc3ccccn3)nn2CC1=O |r|
CC(C)N1CCc2cc(Nc3cc4cc(nc(N)c4cn3)[C@@H](C)n3ccccc3=O)nn2CC1=O |r|
Cc1ccc2c(CC[C@]2(C)O)c1-c1cc2cc(NC(=O)[C@H]3C[C@@H]3CC#N)ncc2c(N)n1 |r|
C[C@@H]1[C@@H]([C@H]1c1cnn(C)c1)C(=O)Nc1cc2cc(nc(N)c2cn1)-c1cccc(N)c1C |r|
C[C@@H]1[C@H]([C@@H]1c1cnn(C)c1)C(=O)Nc1cc2cc(nc(N)c2cn1)-c1cccc(N)c1C |r|
C[C@H]1[C@H]([C@@H]1c1cnn(C)c1)C(=O)Nc1cc2cc(nc(N)c2cn1)-c1cccc(N)c1C |r|
CN1CCc2cc(Nc3cc4cc(nc(N)c4cn3)-c3c(C)cccc3F)nn2CC1=O
COCc1cccc(C)c1-c1cc2cc(NC(=O)[C@@H]3C[C@H]3c3cnn(C)c3)ncc2c(N)n1 |r|
COCc1cccc(C)c1-c1cc2cc(NC(=O)[C@H]3C[C@@H]3c3cnn(C)c3)ncc2c(N)n1 |r|
O[C@@H]1C[C@@H]2CC[C@H](C1)N2c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cnccn23)nc1 |r,TLB:9:8:5.4:7.2.1|
Cn1ccc2c(ccnc12)-c1ncc(Nc2ccc(cn2)N2C[C@@H]3C[C@H]2COC3)c2C(=O)NCc12 |r|
O[C@H]1C[C@@H]2CC[C@H](C1)N2c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cnccn23)nc1 |r,TLB:9:8:5.4:2.1.7|
CNC1CN(C1)c1cccc(Cc2cnc(c3CNC(=O)c23)-c2ccnc3n(C)ccc23)n1
Cc1ccn2c(cnc2c1F)-c1ccc(Nc2ccc(cn2)N2CCO[C@@H](CP)C2)c2C(=O)NCc12 |r|
COc1cccn2c(cnc12)-c1ncc(Nc2ccc(cn2)N2CCO[C@@H](C2)C(C)(C)O)c2C(=O)NCc12 |r|
CN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3nc(C)ccn23)ccc1C1CCOC1
CO[C@H]1CCN(Cc2nc(Nc3ccc(c4CNC(=O)c34)-c3cnc4cc(F)ccn34)ccc2[C@H]2CCOC2)C1 |r|
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2cccc(N3CCN(C)CC3)c2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc3c(c2)NC(=O)CC3)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(-c3cn[nH]c3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(CCO)CC3)c(F)c2)cnc2c1NCC(C)O2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CC4CCC(C3)N4C)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C4CCCC4)CC3)c(F)c2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(-c3cc[nH]n3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C4CCCC4)CC3)cc2)cnc2c1NCC(C)O2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(S(C)(=O)=O)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc3c(c2)C(=O)NCC3)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(-c3cnco3)cc2)cnc2c1NCCO2
CCC1CNc2c(ncc(Nc3cc[nH]c(=O)c3C(=O)Nc3ccc(N4CCN(C)CC4)cc3)c2C)O1
Cc1nc2cc(NC(=O)c3c(Nc4cnc5c(c4C)NCCO5)cc[nH]c3=O)ccc2[nH]1
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(CCO)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C4CCCC4)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C)CC3)cc2)cnc2c1NCC(C(C)C)O2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(CCCS(C)(=O)=O)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C(C)C)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(CC(C)(C)O)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C)CC3)cc2)cnc2c1NCC1(CC1)O2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc3c(c2)CN(C)CC3)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C)CC3)c(Cl)c2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C(=O)C4CCCC4)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C)CC3)c(C#N)c2)cnc2c1NCC(C)O2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(CCN4CCOCC4)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(S(C)(=O)=O)CC3)cc2)cnc2c1NCCO2
COCC(=O)N1CCN(c2ccc(NC(=O)c3c(Nc4cnc5c(c4C)NCCO5)cc[nH]c3=O)cc2)CC1
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2cnn(C3CCN(C)CC3)c2)cnc2c1NCC(C)O2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C)CC3)c(CN(C)C)c2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C)CC3)c(N)c2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(-c3cccnc3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(Cc4ccn[nH]4)CC3)cc2)cnc2c1NCC(C)O2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(C[C@H]3COC(=O)N3)cc2)cnc2c1NCCO2
CCn1nccc1-c1ccc(NC(=O)c2c(Nc3cnc4c(c3C)NCCO4)cc[nH]c2=O)cc1
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(-c3ccncc3)cc2)cnc2c1NCCO2
COCCN1CCN(c2ccc(NC(=O)c3c(Nc4cnc5c(c4C)NCCO5)cc[nH]c3=O)cc2F)CC1
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2cnc(-n3nccn3)c(Cl)c2)cnc2c1NCCO2
CCn1nc(C(F)(F)F)cc1-c1ccc(NC(=O)c2c(Nc3cnc4c(c3C)NCCO4)cc[nH]c2=O)cc1
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCCC(N)C3)cc2)cnc2c1NCCO2
Cc1cc(N2CCN(C)CC2)ccc1NC(=O)c1c(Nc2cnc3c(c2C)NCCO3)cc[nH]c1=O
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc3c(c2)OCCO3)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C)C[C@@H]3C)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCC(N)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C)CC3)c(C(F)(F)F)c2)cnc2c1NCC(C)O2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(S(=O)(=O)NC3CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C)CC3=O)cc2)cnc2c1NCCO2
COCCC(=O)N1CCN(c2ccc(NC(=O)c3c(Nc4cnc5c(c4C)NCCO5)cc[nH]c3=O)cc2)CC1
COCC1CN(C)CCN1c1ccc(NC(=O)c2c(Nc3cnc4c(c3C)NCC(C)O4)cc[nH]c2=O)cc1
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(CN3CCS(=O)(=O)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCNC(=O)C3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(CCO)CC3)cc2)cnc2c1NCC(C)O2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C)CC3)cc2)cnc2c1NCC(C)O2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(Cc3ccncc3)cc2)cnc2c1NCCO2
CN1CCN(c2ccc(NC(=O)c3c(Nc4cnc5c(c4)NCCO5)cc[nH]c3=O)cc2)CC1
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(c4cccnc4)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C)CC3)cc2)cnc2c1NCC(F)O2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc3[nH]ncc3c2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc3c(c2)OCC(=O)N3)cnc2c1NCCO2
CNC(=O)N1CCN(c2ccc(NC(=O)c3c(Nc4cnc5c(c4C)NCCO5)cc[nH]c3=O)cc2)CC1
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C)CC3)nc2)cnc2c1NCC(C)O2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CC4CCC3CN4C)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C)CC3)c(Br)c2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(c4ccncc4)CC3)cc2)cnc2c1NCCO2
Cc1cc(NC(=O)c2c(Nc3cnc4c(c3C)NCC(C)O4)cc[nH]c2=O)ccc1N1CCN(C)CC1
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3C[C@@H]4C[C@H]3CN4C)cc2)cnc2c1NCCO2
CN1CCN(c2ccc(NC(=O)c3c(Nc4cnc5c(c4)N(C)CCO5)cc[nH]c3=O)cc2)CC1
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(c4ccccn4)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN4CCCC4C3)cc2)cnc2c1NCC(C)O2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc3cn[nH]c3c2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(-c3ccnn3C(C)C)cc2)cnc2c1NCCO2
COCCN(C)C(=O)N1CCN(c2ccc(NC(=O)c3c(Nc4cnc5c(c4C)NCCO5)cc[nH]c3=O)cc2)CC1
COCCN1CCC(c2ccc(NC(=O)c3c(Nc4cnc5c(c4C)NCCO5)cc[nH]c3=O)cc2)CC1
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(CCC4CNC4)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C)CC3)cc2)cnc2c1NCC(C)O2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C)CC3)c(N(C)C)c2)cnc2c1NCCO2
COc1cc(NC(=O)c2c(Nc3cnc4c(c3C)NCC(C)O4)cc[nH]c2=O)ccc1N1CCN(C)CC1
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc3c(c2)N(C)C(=O)CO3)cnc2c1NCCO2
Cc1c(Nc2nc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C4CCN(C)CC4)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C)CC3)c(CO)c2)cnc2c1NCC(C)O2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc3c(c2)NCCO3)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C)C(=O)C3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C(=O)[C@@H]4C[C@@H]4F)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCOCC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C)C[C@H]3C)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc3ncc(O)nc3c2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C)CC3)cc2)cnc2c1NCC(C)O2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(CN3CCN(C)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(C(N)=O)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCC(N4CCN(C)CC4)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C)CC3)cc2)cnc2c1NC(=O)CO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C4CC4)CC3)cc2)cnc2c1NCCO2
CC(=O)Nc1ccc(NC(=O)c2c(Nc3cnc4c(c3C)NCCO4)cc[nH]c2=O)cn1
COCCN1CCN(c2ccc(NC(=O)c3c(Nc4cnc5c(c4C)NCCO5)cc[nH]c3=O)cc2C)CC1
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C)CC3)c(N)c2)cnc2c1NCC(C)O2
CNc1cc(NC(=O)c2c(Nc3cnc4c(c3C)NCCO4)cc[nH]c2=O)ccc1N1CCN(C)CC1
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3c2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc3sc(NC(=O)[C@@H]4C[C@@H]4F)nc3c2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(CC(=O)N(C)C)CC3)cc2)cnc2c1NCCO2
CN1CCN(c2ccc(NC(=O)c3c(Nc4cnc5c(c4C#N)NCCO5)cc[nH]c3=O)cc2)CC1
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCC(C(C)(C)O)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCC(C)(CO)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCC(C(C)O)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C(=O)c4ccn[nH]4)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C(=O)C4CC(C)(C)C4)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C(=O)C4CC4C)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C(=O)C4(C)CCC4)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C(=O)C4CC(C)C4)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(Cc4ccnn4C)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C(=O)C4CC4(C)C)CC3)cc2)cnc2c1NCCO2
COC(C)(C)CN1CCN(c2ccc(NC(=O)c3c(Nc4cnc5c(c4C)NCCO5)cc[nH]c3=O)cc2)CC1
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C4CCCC4)CC3)c(N)c2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C(=O)CC4CC4)CC3)cc2)cnc2c1NCCO2
CCC(=O)N1CCN(c2ccc(NC(=O)c3c(Nc4cnc5c(c4C)NCC(C)O5)cc[nH]c3=O)cc2Cl)CC1
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C(=O)C4CCC4)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C(=O)C(C)C)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C(=O)c4ccnn4C)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C(=O)N4CC(C)(C)C4)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C(=O)C4CC(F)(F)C4)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C(=O)N4CC(F)(F)C4)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C(=O)N4CC5(CCC5)C4)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C(=O)N4CC5(COC5)C4)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C(=O)c4ccn(C)n4)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN4CCOC[C@H]4C3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C(=O)N4CCCC4)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C(=O)N4CCC4)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCC(N4CCN(C(C)C)CC4)CC3)c(F)c2)cnc2c1NCC(C)O2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN4CCOC[C@@H]4C3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN4CCC[C@H]4C3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN4CCC[C@@H]4C3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(C3CCCCC3)cc2)cnc2c1NCCO2
Cc1c(NC2C=CNC(=O)C2C(=O)Nc2ccc(-c3ccccc3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C(=O)C4CC4)CC3)cc2)cnc2c1NCCO2
CCC(C)C(=O)N1CCN(c2ccc(NC(=O)c3c(Nc4cnc5c(c4C)NCCO5)cc[nH]c3=O)cc2)CC1
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C(=O)C4C(C)(C)C4(C)C)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C(=O)C(C)C)CC3)cc2)cnc2c1NCC(C)O2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(c4ccn(C)n4)CC3)cc2)cnc2c1NCCO2
Cc1ncccc1N1CCN(c2ccc(NC(=O)c3c(Nc4cnc5c(c4C)NCCO5)cc[nH]c3=O)cc2)CC1
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(c4cncnc4)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(c4ncn(C)n4)CC3)cc2)cnc2c1NCCO2
Cc1cc(N2CCN(c3ccc(NC(=O)c4c(Nc5cnc6c(c5C)NCCO6)cc[nH]c4=O)cc3)CC2)ccn1
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C(=O)C(C)(C)C)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C(=O)C(C)(C)F)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C(=O)C(C)C)[C@@H](C)C3)cc2)cnc2c1NCCO2
COC(C)(C)C(=O)N1CCN(c2ccc(NC(=O)c3c(Nc4cnc5c(c4C)NCCO5)cc[nH]c3=O)cc2)CC1
CCC(=O)N1CCN(c2ccc(NC(=O)c3c(Nc4cnc5c(c4C)NCCO5)cc[nH]c3=O)cc2)C[C@@H]1C
COCCN1CCN(c2ccc(NC(=O)c3c(Nc4cnc5c(c4C)NCCO5)cc[nH]c3=O)cc2)C[C@@H]1C
CCC(=O)N1CCN(c2ccc(NC(=O)c3c(Nc4cnc5c(c4C)NCCO5)cc[nH]c3=O)cc2)C[C@H]1C
COCCN1CCN(c2ccc(NC(=O)c3c(Nc4cnc5c(c4C)NCCO5)cc[nH]c3=O)cc2)C[C@H]1C
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C(=O)C(C)C)[C@H](C)C3)cc2)cnc2c1NCCO2
CO[C@@H](C)C(=O)N1CCN(c2ccc(NC(=O)c3c(Nc4cnc5c(c4C)NCCO5)cc[nH]c3=O)cc2)CC1
COCC(C)N1CCN(c2ccc(NC(=O)c3c(Nc4cnc5c(c4C)NCCO5)cc[nH]c3=O)cc2)CC1
Cc1c(Nc2nc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C#N)CC3)cc2)cnc2c1NCCO2
CO[C@H](C)C(=O)N1CCN(c2ccc(NC(=O)c3c(Nc4cnc5c(c4C)NCCO5)cc[nH]c3=O)cc2)CC1
CNC(C)C(=O)N1CCN(c2ccc(NC(=O)c3c(Nc4cnc5c(c4C)NCCO5)cc[nH]c3=O)cc2)CC1
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C(=O)C4(C)CC4)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C(=O)C4CCN(C)C4)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C(=O)C(C)(C)O)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C(=O)C(C)N(C)C)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN4C(=O)CCC4C3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C)CC3)c(F)c2)cnc2c1NCC(C)O2
CCN1CCN(c2ccc(NC(=O)c3c(Nc4cnc5c(c4C)NCC(C)O5)cc[nH]c3=O)cc2F)CC1
CCC(=O)N1CCN(c2ccc(NC(=O)c3c(Nc4cnc5c(c4C)NCC(C)O5)cc[nH]c3=O)cc2)CC1
Cc1ccc(N2CCN(c3ccc(NC(=O)c4c(Nc5cnc6c(c5C)NCCO6)cc[nH]c4=O)cc3)CC2)cn1
COCc1cc(N2CCN(c3ccc(NC(=O)c4c(Nc5cnc6c(c5C)NCCO6)cc[nH]c4=O)cc3)CC2)ccn1
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(c4ccnc(C(=O)N(C)C)c4)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(c4nccn4C)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(c4cscn4)CC3)cc2)cnc2c1NCCO2
CCOCCN1CCN(c2ccc(NC(=O)c3c(Nc4cnc5c(c4C)NCCO5)cc[nH]c3=O)cc2)CC1
COC(C)CN1CCN(c2ccc(NC(=O)c3c(Nc4cnc5c(c4C)NCCO5)cc[nH]c3=O)cc2)CC1
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(CC(C)C)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(c4nccs4)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C(=O)C4CC4)CC3)cc2)cnc2c1NCC(C)O2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C(=O)C4CN(C)C4)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN4C(=O)CCCC4C3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCC(O)(CN(C)C)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C4CC4)CC3)c(F)c2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN4C(=O)N(C)CC4C3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C(C)c4ccn[nH]4)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C4COC4)CC3)c(F)c2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C4(C)COC4)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCC(N(C)C(=O)C(C)C)C3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCC4(CC3)CC4)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C(C)(C)C)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(C3CCN(C(C)C)CC3)cc2)cnc2c1NCC(C)O2
CCN1CCN(c2ccc(NC(=O)c3c(Nc4cnc5c(c4C)NCC(C)O5)cc[nH]c3=O)cc2F)CC1
CCN1CCN(c2ccc(NC(=O)c3c(Nc4cnc5c(c4C)NCC(C)O5)cc[nH]c3=O)cc2F)CC1
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(CCF)CC3)c(F)c2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCC(O)(CN(C)C)CC3)c(F)c2)cnc2c1NCC(C)O2
CCN1CCN(c2c(F)cc(NC(=O)c3c(Nc4cnc5c(c4C)NCCO5)cc[nH]c3=O)cc2Cl)CC1
CCN1CCN(c2c(F)cc(NC(=O)c3c(Nc4cnc5c(c4C)NCCO5)cc[nH]c3=O)cc2F)CC1
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C4CC4)CC3)c(Cl)c2)cnc2c1NCCO2
COC1(CN(C)C)CCN(c2ccc(NC(=O)c3c(Nc4cnc5c(c4C)NCCO5)cc[nH]c3=O)cc2)CC1
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C)CC3)c(CN)c2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C)CC3)c(CCO)c2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCC(N)C3)cc2)cnc2c1NCCO2
COc1ncc(C(C)(C)O)c2cc(NC(=O)c3c(Nc4cnc5c(c4C)NCCO5)cc[nH]c3=O)ccc12
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCCC3CO)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCC(O)C3)cc2)cnc2c1NCCO2
CCCN1CCN(c2ccc(NC(=O)c3c(Nc4cnc5c(c4C)NCCO5)cc[nH]c3=O)cc2)CC1
Cc1cc(NC(=O)c2c(Nc3cnc4c(c3C)NCCO4)cc[nH]c2=O)ccc1N1CCN(C2CC2)CC1
CCOc1cc(NC(=O)c2c(Nc3cnc4c(c3C)NCCO4)cc[nH]c2=O)ccc1N1CCN(C2CC2)CC1
CC(=O)N1CCN(c2ccc(NC(=O)c3c(Nc4cnc5c(c4C)NCCO5)cc[nH]c3=O)cc2)CC1
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C(=O)CCO)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C(C)C)CC3)cc2)cnc2c1NCC(C)O2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C(C)C)CC3)cc2)cnc2c1NCC(C)O2
COCCCN1CCN(c2ccc(NC(=O)c3c(Nc4cnc5c(c4C)NCC(C)O5)cc[nH]c3=O)cc2)CC1
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(c4ccn(C)n4)CC3)cc2)cnc2c1NCC(C)O2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C)CC3CO)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2cnn(CC(F)(F)F)c2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(c4cnn(C)c4)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2cc[nH]c(=O)c2C(=O)Nc2ccc(N3CCC(C4CC4)CC3)cc2)cnc2c1NCCO2
Cc1c(Nc2nc[nH]c(=O)c2C(=O)Nc2ccc(N3CCN(C(C)C)CC3)cc2)cnc2c1NCCO2
COCCN1CCN(c2ccc(NC(=O)c3c(Nc4cnc5c(c4C)NCCO5)nc[nH]c3=O)cc2)CC1
CN(C)Cc1cc(Nc2ncc(-c3cnc4cc(F)ccn34)c3c2C(=O)NC3)ccc1N1CCOCC1
Cn1ccc2c(-c3ccc(Nc4ccc5c(n4)OC[C@H]4CNCCN54)c4c3CNC4=O)ccnc21
CCN1CCN2c3ccc(Nc4ccc(-c5ccnc6c5ccn6C)c5c4C(=O)NC5)nc3OC[C@H]2C1
Cn1ccc2c(-c3ncc(Nc4ccc5c(n4)OC[C@@H]4COCCN54)c4c3CNC4=O)ccnc21
O=C1NCc2c(-c3cnc4cc(F)ccn34)ccc(Nc3ccc4c(n3)OC[C@@H]3COCCN43)c21
O=C1NCc2c(-c3cnc4cc(F)ccn34)ccc(Nc3ccc4c(n3)OC[C@H]3COCCN43)c21
O=C1NCc2c(-c3cnc4cc(F)ccn34)ccc(Nc3ccc4c(n3)OC[C@@H]3COCC[C@H]43)c21
O=C1NCc2c(-c3cnc4cc(F)ccn34)ccc(Nc3ccc4c(n3)OC[C@H]3COCC[C@@H]43)c21
O=C1NCc2c(-c3cnc4cc(F)ccn34)ccc(Nc3ccc4c(n3)OC[C@@H]3COC[C@H]43)c21
O=C1NCc2c(-c3cnc4cc(F)ccn34)ccc(Nc3ccc4c(n3)OC[C@H]3COC[C@@H]43)c21
COc1cccc(F)c1-c1ccc(Nc2ccc(N3CCOCC3)c(CN(C)C)n2)c2c1CNC2=O
CN1Cc2nc(Nc3ccc(-c4cnc5cc(F)ccn45)c4c3C(=O)NC4)ccc2N2CCOCC2C1
CN1Cc2nc(Nc3ccc(-c4cnc5cc(F)ccn45)c4c3C(=O)NC4)ccc2C2COCC2C1
O=C1NCc2c(-c3cnc4cc(F)ccn34)ccc(Nc3ccc4c(n3)CNC(=O)C3COCC43)c21
Cn1ccc2c(-c3ncc(Nc4ccc5c(n4)OC[C@H]4COCCN54)c4c3CNC4=O)ccnc21
O=C1NCc2c(-c3cnc4cc(F)ccn34)ccc(Nc3ccc4c(n3)CNC(=O)[C@H]3COC[C@@H]43)c21
O=C1NCc2c(-c3cnc4cc(F)ccn34)ccc(Nc3ccc4c(n3)CNC(=O)[C@@H]3COC[C@H]43)c21
Cn1ccc2c(-c3ccc(Nc4ccc5c(n4)CNC(=O)C4COCC54)c4c3CNC4=O)ccnc21
CN1Cc2nc(Nc3cnc(-c4ccnc5c4ccn5C)c4c3C(=O)NC4)ccc2N2CCOCC2C1
CN1Cc2nc(Nc3ccc(-c4ccnc5c4ccn5C)c4c3C(=O)NC4)ccc2N2CCOCC2C1
Cn1ccc2c(-c3ccc(Nc4ccc5c(n4)NC(=O)[C@@H]4CCCN4C5)c4c3CNC4=O)ccnc21
Cn1ccc2c(-c3ccc(Nc4ccc5c(n4)CNCC4COCCN54)c4c3CNC4=O)ccnc21
CCN7Cc5nc(Nc3cnc(c1ccnc2c1ccn2C)c4CNC(=O)c34)ccc5N6CCOCC6C7
CN7Cc5nc(Nc3cnc(c1ccnc2c1ccn2C)c4CNC(=O)c34)ccc5N6CCOC[C@@H]6C7
CN1Cc2nc(Nc3cnc(-c4ccnc5c4ccn5C)c4c3C(=O)NC4)ccc2N2CCOC[C@H]2C1
[2H]C([2H])([2H])n1ccc2c(-c3ncc(Nc4ccc5c(n4)CN(C)CC4COCCN54)c4c3CNC4=O)ccnc21
[2H]C([2H])([2H])n1ccc2c(-c3ncc(Nc4ccc5c(n4)CN(C)C[C@H]4COCCN54)c4c3CNC4=O)ccnc21
[2H]C([2H])([2H])n1ccc2c(-c3ncc(Nc4ccc5c(n4)CN(C)C[C@@H]4COCCN54)c4c3CNC4=O)ccnc21
[2H]C([2H])([2H])n1ccc2c(-c3ncc(Nc4ccc5c(n4)OC[C@@H]4COCCN54)c4c3CNC4=O)ccnc21
CN1Cc2nc(Nc3cnc(-c4ccnc5c4ccn5C)c4cc[nH]c(=O)c34)ccc2N2CCOCC2C1
CN1Cc2nc(Nc3cnc(-c4cnc5cc(F)ccn45)c4c3C(=O)NC4)ccc2N2CCOCC2C1
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CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N([C@@H]1C[C@@H](C1)N1CCC(C)(C)C1)C(=O)C21CCN(CC1)C(=O)C(C)(C)O |r,wU:27.30,29.35,(5.83,-5.18,;6.6,-3.85,;8.14,-3.85,;5.83,-2.52,;6.73,-1.27,;5.83,-.02,;4.36,-.5,;3.03,.27,;1.69,-.5,;1.69,-2.04,;3.03,-2.81,;3.03,-4.35,;1.69,-5.12,;1.69,-6.66,;.36,-7.43,;-.97,-6.66,;-.97,-5.12,;.36,-4.35,;.36,-2.81,;4.36,-2.04,;.36,.27,;.36,1.81,;-.97,2.58,;-2.31,1.81,;-2.31,.27,;-.97,-.5,;-3.77,-.21,;-4.17,-1.69,;-5.5,-2.46,;-4.73,-3.8,;-3.4,-3.03,;-5.13,-5.28,;-4.23,-6.53,;-5.13,-7.78,;-6.6,-7.3,;-8.14,-7.3,;-7.37,-8.63,;-6.6,-5.76,;-4.68,1.04,;-6.22,1.04,;-3.77,2.29,;-2.68,3.37,;-3.08,4.86,;-4.57,5.26,;-5.66,4.17,;-5.26,2.68,;-4.97,6.75,;-3.88,7.84,;-6.45,7.15,;-6.85,5.66,;-7.94,6.75,;-6.85,8.63,)|
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CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N([C@@H]1C[C@@H](C1)N1C3CCC1COC3)C(=O)C21CCN(CC1)C(=O)C1(C)COC1 |r,wU:27.30,29.35,(5.76,-5.37,;6.53,-4.04,;8.07,-4.04,;5.76,-2.7,;6.66,-1.46,;5.76,-.21,;4.29,-.69,;2.96,.08,;1.62,-.69,;1.62,-2.23,;2.96,-3,;2.96,-4.54,;1.62,-5.31,;1.62,-6.85,;.29,-7.62,;-1.04,-6.85,;-1.04,-5.31,;.29,-4.54,;.29,-3,;4.29,-2.23,;.29,.08,;.29,1.62,;-1.04,2.39,;-2.38,1.62,;-2.38,.08,;-1.04,-.69,;-3.84,-.39,;-4.24,-1.88,;-5.57,-2.65,;-4.8,-3.98,;-3.47,-3.21,;-5.2,-5.47,;-6.69,-5.87,;-6.29,-7.36,;-5.2,-7.65,;-4.11,-6.56,;-4.51,-8.05,;-6,-8.45,;-7.09,-7.36,;-4.75,.85,;-6.29,.85,;-3.84,2.1,;-2.75,3.19,;-3.15,4.67,;-4.64,5.07,;-5.73,3.98,;-5.33,2.5,;-5.04,6.56,;-3.95,7.65,;-6.53,6.96,;-6.92,8.45,;-8.07,6.96,;-8.07,5.42,;-6.53,5.42,)|
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CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N([C@@H]1C[C@@H](C1)N1C[C@H](C)[C@H](C)C1)C(=O)C21CCN(CC1)C(=O)C1(C)COC1 |r,wU:27.30,29.35,33.38,35.40,(5.76,-4.95,;6.53,-3.61,;8.07,-3.61,;5.76,-2.28,;6.66,-1.03,;5.76,.21,;4.29,-.26,;2.96,.51,;1.62,-.26,;1.62,-1.8,;2.96,-2.57,;2.96,-4.11,;1.62,-4.88,;1.62,-6.42,;.29,-7.19,;-1.04,-6.42,;-1.04,-4.88,;.29,-4.11,;.29,-2.57,;4.29,-1.8,;.29,.51,;.29,2.05,;-1.04,2.82,;-2.38,2.05,;-2.38,.51,;-1.04,-.26,;-3.84,.03,;-4.24,-1.46,;-5.57,-2.23,;-4.8,-3.56,;-3.47,-2.79,;-5.2,-5.05,;-6.67,-5.52,;-6.67,-7.06,;-8,-7.83,;-5.2,-7.54,;-4.43,-8.87,;-4.3,-6.29,;-4.75,1.28,;-6.29,1.28,;-3.84,2.52,;-2.75,3.61,;-3.15,5.1,;-4.64,5.5,;-5.73,4.41,;-5.33,2.92,;-5.04,6.99,;-3.95,8.08,;-6.53,7.38,;-6.92,8.87,;-8.07,7.38,;-8.07,5.84,;-6.53,5.84,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N([C@@H]1C[C@@H](C1)N1C[C@H](C)[C@H](C)C1)C(=O)C21CCN(CC1)C(=O)[C@@H]1CCCO1 |r,wU:27.30,29.35,33.38,35.40,wD:48.55,(6.23,-4.93,;7,-3.6,;8.54,-3.6,;6.23,-2.27,;7.14,-1.02,;6.23,.23,;4.77,-.25,;3.43,.52,;2.1,-.25,;2.1,-1.79,;3.43,-2.56,;3.43,-4.1,;2.1,-4.87,;2.1,-6.41,;.77,-7.18,;-.57,-6.41,;-.57,-4.87,;.77,-4.1,;.77,-2.56,;4.77,-1.79,;.77,.52,;.77,2.06,;-.57,2.83,;-1.9,2.06,;-1.9,.52,;-.57,-.25,;-3.37,.04,;-3.76,-1.44,;-5.1,-2.21,;-4.33,-3.55,;-2.99,-2.78,;-4.73,-5.04,;-6.19,-5.51,;-6.19,-7.05,;-7.53,-7.82,;-4.73,-7.53,;-3.96,-8.86,;-3.82,-6.28,;-4.27,1.29,;-5.81,1.29,;-3.37,2.54,;-2.28,3.62,;-2.68,5.11,;-4.16,5.51,;-5.25,4.42,;-4.85,2.93,;-4.56,7,;-3.47,8.09,;-6.05,7.4,;-7.3,6.49,;-8.54,7.4,;-8.07,8.86,;-6.53,8.86,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N([C@@H]1C[C@@H](C1)N1C[C@H](C)[C@H](C)C1)C(=O)C21CCN(CC1)C(=O)C(C)(C)CO |r,wU:27.30,29.35,33.38,35.40,(5.73,-5.49,;6.5,-4.16,;8.04,-4.16,;5.73,-2.82,;6.63,-1.58,;5.73,-.33,;4.26,-.81,;2.93,-.04,;1.6,-.81,;1.6,-2.35,;2.93,-3.12,;2.93,-4.66,;1.6,-5.43,;1.6,-6.97,;.26,-7.74,;-1.07,-6.97,;-1.07,-5.43,;.26,-4.66,;.26,-3.12,;4.26,-2.35,;.26,-.04,;.26,1.5,;-1.07,2.27,;-2.4,1.5,;-2.4,-.04,;-1.07,-.81,;-3.87,-.51,;-4.27,-2,;-5.6,-2.77,;-4.83,-4.1,;-3.5,-3.33,;-5.23,-5.59,;-6.69,-6.07,;-6.69,-7.61,;-8.03,-8.38,;-5.23,-8.08,;-4.46,-9.42,;-4.32,-6.84,;-4.77,.73,;-6.31,.73,;-3.87,1.98,;-2.78,3.07,;-3.18,4.56,;-4.67,4.95,;-5.75,3.87,;-5.36,2.38,;-5.06,6.44,;-3.98,7.53,;-6.55,6.84,;-6.95,5.35,;-8.04,6.44,;-6.95,8.33,;-5.86,9.42,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N([C@H]1C[C@H](C1)N1CCCCC1)C(=O)C21CCN(CC1)C(=O)C1(C)CCO1 |r,wU:27.30,29.35,(6.04,-5.29,;6.81,-3.96,;8.35,-3.96,;6.04,-2.63,;6.94,-1.38,;6.04,-.13,;4.57,-.61,;3.24,.16,;1.91,-.61,;1.91,-2.15,;3.24,-2.92,;3.24,-4.46,;1.91,-5.23,;1.91,-6.77,;.57,-7.54,;-.76,-6.77,;-.76,-5.23,;.57,-4.46,;.57,-2.92,;4.57,-2.15,;.57,.16,;.57,1.7,;-.76,2.47,;-2.1,1.7,;-2.1,.16,;-.76,-.61,;-3.56,-.32,;-3.96,-1.8,;-3.19,-3.14,;-4.52,-3.91,;-5.29,-2.57,;-4.92,-5.4,;-6.41,-5.79,;-6.81,-7.28,;-5.72,-8.37,;-4.23,-7.97,;-3.83,-6.48,;-4.47,.93,;-6.01,.93,;-3.56,2.18,;-2.47,3.26,;-2.87,4.75,;-4.36,5.15,;-5.45,4.06,;-5.05,2.57,;-4.76,6.64,;-3.67,7.73,;-6.24,7.04,;-5.47,8.37,;-7.58,6.27,;-8.35,7.6,;-7.01,8.37,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N([C@@H]1C[C@@H](C1)N1CCC(C)(C)C1)C(=O)C21CCN(CC1)C(=O)C1(C)CCO1 |r,wU:27.30,29.35,(6.04,-5.39,;6.81,-4.05,;8.35,-4.05,;6.04,-2.72,;6.94,-1.48,;6.04,-.23,;4.57,-.71,;3.24,.06,;1.91,-.71,;1.91,-2.25,;3.24,-3.02,;3.24,-4.56,;1.91,-5.33,;1.91,-6.87,;.57,-7.64,;-.76,-6.87,;-.76,-5.33,;.57,-4.56,;.57,-3.02,;4.57,-2.25,;.57,.06,;.57,1.6,;-.76,2.37,;-2.1,1.6,;-2.1,.06,;-.76,-.71,;-3.56,-.41,;-3.96,-1.9,;-5.29,-2.67,;-4.52,-4,;-3.19,-3.23,;-4.92,-5.49,;-4.02,-6.74,;-4.92,-7.98,;-6.39,-7.51,;-7.72,-8.28,;-7.72,-6.74,;-6.39,-5.97,;-4.47,.83,;-6.01,.83,;-3.56,2.08,;-2.47,3.17,;-2.87,4.66,;-4.36,5.06,;-5.45,3.97,;-5.05,2.48,;-4.76,6.54,;-3.67,7.63,;-6.24,6.94,;-5.47,8.28,;-7.58,6.17,;-8.35,7.51,;-7.01,8.28,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N([C@@H]1C[C@@H](C1)N1CCC(C)(C)C1)C(=O)C21CCN(CC1)C(=O)[C@@H]1CCCO1 |r,wU:27.30,29.35,wD:48.55,(6.23,-5.17,;7,-3.84,;8.54,-3.84,;6.23,-2.5,;7.14,-1.26,;6.23,-.01,;4.77,-.49,;3.43,.28,;2.1,-.49,;2.1,-2.03,;3.43,-2.8,;3.43,-4.34,;2.1,-5.11,;2.1,-6.65,;.77,-7.42,;-.57,-6.65,;-.57,-5.11,;.77,-4.34,;.77,-2.8,;4.77,-2.03,;.77,.28,;.77,1.82,;-.57,2.59,;-1.9,1.82,;-1.9,.28,;-.57,-.49,;-3.37,-.19,;-3.76,-1.68,;-5.1,-2.45,;-4.33,-3.79,;-2.99,-3.02,;-4.73,-5.27,;-3.82,-6.52,;-4.73,-7.77,;-6.19,-7.29,;-6.96,-8.62,;-7.73,-7.29,;-6.19,-5.75,;-4.27,1.05,;-5.81,1.05,;-3.37,2.3,;-2.28,3.39,;-2.68,4.87,;-4.16,5.27,;-5.25,4.18,;-4.85,2.7,;-4.56,6.76,;-3.47,7.85,;-6.05,7.16,;-7.3,6.25,;-8.54,7.16,;-8.07,8.62,;-6.53,8.62,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N([C@@H]1C[C@@H](C1)N1CCC(C)(C)C1)C(=O)C21CCN(CC1)C(=O)[C@H]1CCCO1 |r,wU:48.55,27.30,29.35,(6.23,-5.17,;7,-3.84,;8.54,-3.84,;6.23,-2.5,;7.14,-1.26,;6.23,-.01,;4.77,-.49,;3.43,.28,;2.1,-.49,;2.1,-2.03,;3.43,-2.8,;3.43,-4.34,;2.1,-5.11,;2.1,-6.65,;.77,-7.42,;-.57,-6.65,;-.57,-5.11,;.77,-4.34,;.77,-2.8,;4.77,-2.03,;.77,.28,;.77,1.82,;-.57,2.59,;-1.9,1.82,;-1.9,.28,;-.57,-.49,;-3.37,-.19,;-3.76,-1.68,;-5.1,-2.45,;-4.33,-3.79,;-2.99,-3.02,;-4.73,-5.27,;-3.82,-6.52,;-4.73,-7.77,;-6.19,-7.29,;-6.96,-8.62,;-7.73,-7.29,;-6.19,-5.75,;-4.27,1.05,;-5.81,1.05,;-3.37,2.3,;-2.28,3.39,;-2.68,4.87,;-4.16,5.27,;-5.25,4.18,;-4.85,2.7,;-4.56,6.76,;-3.47,7.85,;-6.05,7.16,;-7.3,6.25,;-8.54,7.16,;-8.07,8.62,;-6.53,8.62,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N([C@@H]1C[C@@H](C1)N1CCC(C)(C)C1)C(=O)C21CCN(CC1)C(=O)[C@@]1(C)CCCO1 |r,wU:27.30,29.35,48.55,wD:48.56,(-.39,-4.19,;-1.9,-3.87,;-2.93,-5.01,;-2.37,-2.4,;-1.47,-1.16,;-2.37,.09,;-3.84,-.39,;-5.17,.38,;-6.5,-.39,;-6.5,-1.93,;-5.17,-2.7,;-5.17,-4.24,;-6.5,-5.01,;-6.5,-6.55,;-7.84,-7.32,;-9.17,-6.55,;-9.17,-5.01,;-7.84,-4.24,;-7.84,-2.7,;-3.84,-1.93,;-7.84,.38,;-7.84,1.92,;-9.17,2.69,;-10.51,1.92,;-10.51,.38,;-9.17,-.39,;-11.97,-.09,;-12.45,-1.56,;-13.82,-2.26,;-13.12,-3.63,;-11.75,-2.93,;-13.6,-5.1,;-12.69,-6.34,;-13.6,-7.59,;-15.06,-7.11,;-16.6,-7.11,;-15.46,-8.6,;-15.06,-5.57,;-12.88,1.15,;-14.42,1.15,;-11.97,2.4,;-10.94,3.54,;-11.42,5.01,;-12.92,5.33,;-13.95,4.18,;-13.48,2.72,;-13.4,6.79,;-12.37,7.94,;-14.9,7.11,;-15.3,8.6,;-14.82,5.57,;-16.26,5.02,;-17.23,6.22,;-16.39,7.51,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N([C@@H]1C[C@@H](C1)N1CCC(C)(C)C1)C(=O)C21CCN(CC1)C(=O)[C@]1(C)CCCO1 |r,wU:27.30,29.35,48.56,wD:48.55,(17.23,-4.19,;15.72,-3.87,;14.69,-5.01,;15.25,-2.4,;16.15,-1.16,;15.25,.09,;13.78,-.39,;12.45,.38,;11.12,-.39,;11.12,-1.93,;12.45,-2.7,;12.45,-4.24,;11.12,-5.01,;11.12,-6.55,;9.78,-7.32,;8.45,-6.55,;8.45,-5.01,;9.78,-4.24,;9.78,-2.7,;13.78,-1.93,;9.78,.38,;9.78,1.92,;8.45,2.69,;7.12,1.92,;7.12,.38,;8.45,-.39,;5.65,-.09,;5.17,-1.56,;3.8,-2.26,;4.5,-3.63,;5.87,-2.93,;4.03,-5.1,;4.93,-6.34,;4.03,-7.59,;2.56,-7.11,;1.02,-7.11,;2.16,-8.6,;2.56,-5.57,;4.75,1.15,;3.21,1.15,;5.65,2.4,;6.68,3.54,;6.21,5.01,;4.7,5.33,;3.67,4.18,;4.14,2.72,;4.22,6.79,;5.25,7.94,;2.72,7.11,;2.32,8.6,;2.8,5.57,;1.36,5.02,;.39,6.22,;1.23,7.51,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N([C@@H]1C[C@@H](C1)N1CCC(C)(C)C1)C(=O)C21CCN(CC1)C(=O)C1(C)CCCO1 |r,wU:27.30,29.35,(5.99,-5.18,;6.76,-3.85,;8.3,-3.85,;5.99,-2.52,;6.9,-1.27,;5.99,-.02,;4.53,-.5,;3.2,.27,;1.86,-.5,;1.86,-2.04,;3.2,-2.81,;3.2,-4.35,;1.86,-5.12,;1.86,-6.66,;.53,-7.43,;-.81,-6.66,;-.81,-5.12,;.53,-4.35,;.53,-2.81,;4.53,-2.04,;.53,.27,;.53,1.81,;-.81,2.58,;-2.14,1.81,;-2.14,.27,;-.81,-.5,;-3.6,-.21,;-4,-1.69,;-5.34,-2.46,;-4.57,-3.8,;-3.23,-3.03,;-4.97,-5.28,;-4.06,-6.53,;-4.97,-7.78,;-6.43,-7.3,;-7.2,-8.63,;-7.97,-7.3,;-6.43,-5.76,;-4.51,1.04,;-6.05,1.04,;-3.6,2.29,;-2.52,3.37,;-2.91,4.86,;-4.4,5.26,;-5.49,4.17,;-5.09,2.68,;-4.8,6.75,;-3.71,7.84,;-6.29,7.15,;-6.69,8.63,;-5.81,5.68,;-7.06,4.78,;-8.3,5.68,;-7.83,7.15,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N([C@@H]1C[C@@H](C1)N1CCC(C)(C)C1)C(=O)C21CCN(CC1)C(=O)[C@H]1CCOC1 |r,wU:48.55,27.30,29.35,(6.23,-5.17,;7,-3.84,;8.54,-3.84,;6.23,-2.5,;7.14,-1.26,;6.23,-.01,;4.77,-.49,;3.43,.28,;2.1,-.49,;2.1,-2.03,;3.43,-2.8,;3.43,-4.34,;2.1,-5.11,;2.1,-6.65,;.77,-7.42,;-.57,-6.65,;-.57,-5.11,;.77,-4.34,;.77,-2.8,;4.77,-2.03,;.77,.28,;.77,1.82,;-.57,2.59,;-1.9,1.82,;-1.9,.28,;-.57,-.49,;-3.37,-.19,;-3.76,-1.68,;-5.1,-2.45,;-4.33,-3.79,;-2.99,-3.02,;-4.73,-5.27,;-3.82,-6.52,;-4.73,-7.77,;-6.19,-7.29,;-6.96,-8.62,;-7.73,-7.29,;-6.19,-5.75,;-4.27,1.05,;-5.81,1.05,;-3.37,2.3,;-2.28,3.39,;-2.68,4.87,;-4.16,5.27,;-5.25,4.18,;-4.85,2.7,;-4.56,6.76,;-3.47,7.85,;-6.05,7.16,;-7.3,6.25,;-8.54,7.16,;-8.07,8.62,;-6.53,8.62,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N([C@@H]1C[C@@H](C1)N1CCC(C)(C)C1)C(=O)C21CCN(CC1)C(=O)[C@@H]1CCOC1 |r,wU:27.30,29.35,wD:48.55,(6.23,-5.17,;7,-3.84,;8.54,-3.84,;6.23,-2.5,;7.14,-1.26,;6.23,-.01,;4.77,-.49,;3.43,.28,;2.1,-.49,;2.1,-2.03,;3.43,-2.8,;3.43,-4.34,;2.1,-5.11,;2.1,-6.65,;.77,-7.42,;-.57,-6.65,;-.57,-5.11,;.77,-4.34,;.77,-2.8,;4.77,-2.03,;.77,.28,;.77,1.82,;-.57,2.59,;-1.9,1.82,;-1.9,.28,;-.57,-.49,;-3.37,-.19,;-3.76,-1.68,;-5.1,-2.45,;-4.33,-3.79,;-2.99,-3.02,;-4.73,-5.27,;-3.82,-6.52,;-4.73,-7.77,;-6.19,-7.29,;-6.96,-8.62,;-7.73,-7.29,;-6.19,-5.75,;-4.27,1.05,;-5.81,1.05,;-3.37,2.3,;-2.28,3.39,;-2.68,4.87,;-4.16,5.27,;-5.25,4.18,;-4.85,2.7,;-4.56,6.76,;-3.47,7.85,;-6.05,7.16,;-7.3,6.25,;-8.54,7.16,;-8.07,8.62,;-6.53,8.62,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N([C@@H]1C[C@@H](C1)N1CCC(C)(C)C1)C(=O)C21CCN(CC1)C(=O)C1(C)CCOC1 |r,wU:27.30,29.35,(5.99,-5.18,;6.76,-3.85,;8.3,-3.85,;5.99,-2.52,;6.9,-1.27,;5.99,-.02,;4.53,-.5,;3.2,.27,;1.86,-.5,;1.86,-2.04,;3.2,-2.81,;3.2,-4.35,;1.86,-5.12,;1.86,-6.66,;.53,-7.43,;-.81,-6.66,;-.81,-5.12,;.53,-4.35,;.53,-2.81,;4.53,-2.04,;.53,.27,;.53,1.81,;-.81,2.58,;-2.14,1.81,;-2.14,.27,;-.81,-.5,;-3.6,-.21,;-4,-1.69,;-5.34,-2.46,;-4.57,-3.8,;-3.23,-3.03,;-4.97,-5.28,;-4.06,-6.53,;-4.97,-7.78,;-6.43,-7.3,;-7.2,-8.63,;-7.97,-7.3,;-6.43,-5.76,;-4.51,1.04,;-6.05,1.04,;-3.6,2.29,;-2.52,3.37,;-2.91,4.86,;-4.4,5.26,;-5.49,4.17,;-5.09,2.68,;-4.8,6.75,;-3.71,7.84,;-6.29,7.15,;-6.69,8.63,;-5.81,5.68,;-7.06,4.78,;-8.3,5.68,;-7.83,7.15,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N([C@@H]1C[C@@H](C1)N1CCC(C)(C)C1)C(=O)C21CCN(CC1)C(=O)[C@@H]1OCC[C@@H]1C |r,wU:27.30,29.35,48.55,52.61,(5.94,5.06,;6.97,6.2,;8.48,5.88,;6.49,7.67,;7.4,8.92,;6.49,10.16,;5.03,9.69,;3.7,10.46,;2.36,9.69,;2.36,8.15,;3.7,7.38,;3.7,5.84,;2.36,5.07,;2.36,3.53,;1.03,2.76,;-.31,3.53,;-.31,5.07,;1.03,5.84,;1.03,7.38,;5.03,8.15,;1.03,10.46,;1.03,12,;-.31,12.77,;-1.64,12,;-1.64,10.46,;-.31,9.69,;-3.1,9.98,;-3.58,8.51,;-4.95,7.82,;-4.25,6.44,;-2.88,7.14,;-4.73,4.98,;-3.82,3.73,;-4.73,2.49,;-6.19,2.96,;-7.73,2.8,;-6.82,1.56,;-6.19,4.5,;-4.01,11.23,;-5.55,11.23,;-3.1,12.47,;-2.07,13.62,;-2.55,15.08,;-4.06,15.4,;-5.09,14.26,;-4.61,12.79,;-4.53,16.86,;-3.5,18.01,;-6.04,17.19,;-6.81,18.52,;-8.31,18.2,;-8.48,16.67,;-7.07,16.04,;-6.75,14.53,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N([C@@H]1C[C@@H](C1)N1CCC(C)(C)C1)C(=O)C21CCN(CC1)C(=O)[C@H]1OCC[C@H]1C |r,wU:27.30,29.35,wD:48.55,52.61,(5.94,-15.01,;6.97,-13.87,;8.48,-14.19,;6.49,-12.41,;7.4,-11.16,;6.49,-9.91,;5.03,-10.39,;3.7,-9.62,;2.36,-10.39,;2.36,-11.93,;3.7,-12.7,;3.7,-14.24,;2.36,-15.01,;2.36,-16.55,;1.03,-17.32,;-.31,-16.55,;-.31,-15.01,;1.03,-14.24,;1.03,-12.7,;5.03,-11.93,;1.03,-9.62,;1.03,-8.08,;-.31,-7.31,;-1.64,-8.08,;-1.64,-9.62,;-.31,-10.39,;-3.1,-10.1,;-3.58,-11.56,;-4.95,-12.26,;-4.25,-13.63,;-2.88,-12.93,;-4.73,-15.1,;-3.82,-16.34,;-4.73,-17.59,;-6.19,-17.11,;-7.73,-17.27,;-6.82,-18.52,;-6.19,-15.57,;-4.01,-8.85,;-5.55,-8.85,;-3.1,-7.6,;-2.07,-6.46,;-2.55,-4.99,;-4.06,-4.67,;-5.09,-5.82,;-4.61,-7.28,;-4.53,-3.21,;-3.5,-2.07,;-6.04,-2.89,;-6.81,-1.56,;-8.31,-1.88,;-8.48,-3.41,;-7.07,-4.03,;-6.75,-5.54,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N([C@@H]1C[C@@H](C1)N1CCC(C)(C)C1)C(=O)C21CCN(CC1)C(=O)[C@H]1CC[C@@H](C)O1 |r,wU:27.30,29.35,48.55,51.59,(6.43,5.84,;7.46,6.98,;8.97,6.66,;6.99,8.45,;7.89,9.7,;6.99,10.94,;5.52,10.47,;4.19,11.24,;2.85,10.47,;2.85,8.93,;4.19,8.16,;4.19,6.62,;2.85,5.85,;2.85,4.31,;1.52,3.54,;.19,4.31,;.19,5.85,;1.52,6.62,;1.52,8.16,;5.52,8.93,;1.52,11.24,;1.52,12.78,;.19,13.55,;-1.15,12.78,;-1.15,11.24,;.19,10.47,;-2.61,10.76,;-3.09,9.29,;-4.46,8.6,;-3.76,7.22,;-2.39,7.92,;-4.24,5.76,;-3.33,4.51,;-4.24,3.27,;-5.7,3.74,;-7.23,3.58,;-6.33,2.34,;-5.7,5.28,;-3.52,12.01,;-5.06,12.01,;-2.61,13.25,;-1.58,14.4,;-2.06,15.86,;-3.56,16.18,;-4.59,15.04,;-4.12,13.57,;-4.04,17.65,;-3.01,18.79,;-5.55,17.97,;-6.58,16.82,;-7.98,17.45,;-7.82,18.98,;-8.97,20.01,;-6.32,19.3,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N([C@@H]1C[C@@H](C1)N1CCC(C)(C)C1)C(=O)C21CCN(CC1)C(=O)[C@@H]1CC[C@H](C)O1 |r,wU:27.30,29.35,wD:48.55,51.59,(6.43,-16.51,;7.46,-15.36,;8.97,-15.68,;6.99,-13.9,;7.89,-12.65,;6.99,-11.4,;5.52,-11.88,;4.19,-11.11,;2.85,-11.88,;2.85,-13.42,;4.19,-14.19,;4.19,-15.73,;2.85,-16.5,;2.85,-18.04,;1.52,-18.81,;.19,-18.04,;.19,-16.5,;1.52,-15.73,;1.52,-14.19,;5.52,-13.42,;1.52,-11.11,;1.52,-9.57,;.19,-8.8,;-1.15,-9.57,;-1.15,-11.11,;.19,-11.88,;-2.61,-11.59,;-3.09,-13.05,;-4.46,-13.75,;-3.76,-15.12,;-2.39,-14.42,;-4.24,-16.59,;-3.33,-17.83,;-4.24,-19.08,;-5.7,-18.6,;-7.23,-18.76,;-6.33,-20.01,;-5.7,-17.06,;-3.52,-10.34,;-5.06,-10.34,;-2.61,-9.09,;-1.58,-7.95,;-2.06,-6.49,;-3.56,-6.17,;-4.59,-7.31,;-4.12,-8.77,;-4.04,-4.7,;-3.01,-3.56,;-5.55,-4.38,;-6.58,-5.52,;-7.98,-4.9,;-7.82,-3.37,;-8.97,-2.34,;-6.32,-3.05,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N([C@@H]1C[C@@H](C1)N1CCC(C)(C)C1)C(=O)C21CCN(CC1)C(=O)CC1COC1 |r,wU:27.30,29.35,(5.85,-6.13,;6.62,-4.8,;8.16,-4.8,;5.85,-3.46,;6.76,-2.22,;5.85,-.97,;4.39,-1.45,;3.05,-.68,;1.72,-1.45,;1.72,-2.99,;3.05,-3.76,;3.05,-5.3,;1.72,-6.07,;1.72,-7.61,;.39,-8.38,;-.95,-7.61,;-.95,-6.07,;.39,-5.3,;.39,-3.76,;4.39,-2.99,;.39,-.68,;.39,.86,;-.95,1.63,;-2.28,.86,;-2.28,-.68,;-.95,-1.45,;-3.75,-1.15,;-4.14,-2.64,;-5.48,-3.41,;-4.71,-4.75,;-3.37,-3.98,;-5.11,-6.23,;-4.2,-7.48,;-5.11,-8.73,;-6.57,-8.25,;-6.57,-9.79,;-8.11,-8.25,;-6.57,-6.71,;-4.65,.09,;-6.19,.09,;-3.75,1.34,;-2.66,2.43,;-3.06,3.91,;-4.54,4.31,;-5.63,3.22,;-5.23,1.74,;-4.94,5.8,;-3.85,6.89,;-6.43,6.2,;-6.83,7.69,;-6.06,9.02,;-7.39,9.79,;-8.16,8.46,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N([C@H]1C[C@H](C1)N1CCCCC1)C(=O)C21CCN(CC1)C(=O)C1CCO1 |r,wU:27.30,29.35,(6.04,-5.29,;6.81,-3.96,;8.35,-3.96,;6.04,-2.63,;6.94,-1.38,;6.04,-.13,;4.57,-.61,;3.24,.16,;1.91,-.61,;1.91,-2.15,;3.24,-2.92,;3.24,-4.46,;1.91,-5.23,;1.91,-6.77,;.57,-7.54,;-.76,-6.77,;-.76,-5.23,;.57,-4.46,;.57,-2.92,;4.57,-2.15,;.57,.16,;.57,1.7,;-.76,2.47,;-2.1,1.7,;-2.1,.16,;-.76,-.61,;-3.56,-.32,;-3.96,-1.8,;-3.19,-3.14,;-4.52,-3.91,;-5.29,-2.57,;-4.92,-5.4,;-6.41,-5.79,;-6.81,-7.28,;-5.72,-8.37,;-4.23,-7.97,;-3.83,-6.48,;-4.47,.93,;-6.01,.93,;-3.56,2.18,;-2.47,3.26,;-2.87,4.75,;-4.36,5.15,;-5.45,4.06,;-5.05,2.57,;-4.76,6.64,;-3.67,7.73,;-6.24,7.04,;-7.58,6.27,;-8.35,7.6,;-7.01,8.37,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N([C@@H]1C[C@@H](C1)N1CCC(C)(C)C1)C(=O)C21CCN(CC1)C(=O)C1CCOCC1 |r,wU:27.30,29.35,(6.47,-5.38,;7.24,-4.05,;8.78,-4.05,;6.47,-2.72,;7.38,-1.47,;6.47,-.22,;5.01,-.7,;3.67,.07,;2.34,-.7,;2.34,-2.24,;3.67,-3.01,;3.67,-4.55,;2.34,-5.32,;2.34,-6.86,;1.01,-7.63,;-.33,-6.86,;-.33,-5.32,;1.01,-4.55,;1.01,-3.01,;5.01,-2.24,;1.01,.07,;1.01,1.61,;-.33,2.38,;-1.66,1.61,;-1.66,.07,;-.33,-.7,;-3.12,-.41,;-3.52,-1.89,;-4.86,-2.66,;-4.09,-4,;-2.75,-3.23,;-4.49,-5.48,;-3.58,-6.73,;-4.49,-7.98,;-5.95,-7.5,;-6.72,-8.83,;-7.49,-7.5,;-5.95,-5.96,;-4.03,.84,;-5.57,.84,;-3.12,2.09,;-2.04,3.18,;-2.43,4.66,;-3.92,5.06,;-5.01,3.97,;-4.61,2.48,;-4.32,6.55,;-3.23,7.64,;-5.81,6.95,;-6.21,8.44,;-7.69,8.83,;-8.78,7.74,;-8.38,6.26,;-6.9,5.86,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N([C@@H]1C[C@@H](C1)N1CCC(C)(C)C1)C(=O)C21CCN(CC1)C(=O)C1CCCCO1 |r,wU:27.30,29.35,(6.47,-5.38,;7.24,-4.05,;8.78,-4.05,;6.47,-2.72,;7.38,-1.47,;6.47,-.22,;5.01,-.7,;3.67,.07,;2.34,-.7,;2.34,-2.24,;3.67,-3.01,;3.67,-4.55,;2.34,-5.32,;2.34,-6.86,;1.01,-7.63,;-.33,-6.86,;-.33,-5.32,;1.01,-4.55,;1.01,-3.01,;5.01,-2.24,;1.01,.07,;1.01,1.61,;-.33,2.38,;-1.66,1.61,;-1.66,.07,;-.33,-.7,;-3.12,-.41,;-3.52,-1.89,;-4.86,-2.66,;-4.09,-4,;-2.75,-3.23,;-4.49,-5.48,;-3.58,-6.73,;-4.49,-7.98,;-5.95,-7.5,;-6.72,-8.83,;-7.49,-7.5,;-5.95,-5.96,;-4.03,.84,;-5.57,.84,;-3.12,2.09,;-2.04,3.18,;-2.43,4.66,;-3.92,5.06,;-5.01,3.97,;-4.61,2.48,;-4.32,6.55,;-3.23,7.64,;-5.81,6.95,;-6.9,5.86,;-8.38,6.26,;-8.78,7.74,;-7.69,8.83,;-6.21,8.44,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N([C@@H]1C[C@@H](C1)N1CCC(C)(C)C1)C(=O)C21CCN(CC1)C(=O)C1CCCOC1 |r,wU:27.30,29.35,(6.47,-5.38,;7.24,-4.05,;8.78,-4.05,;6.47,-2.72,;7.38,-1.47,;6.47,-.22,;5.01,-.7,;3.67,.07,;2.34,-.7,;2.34,-2.24,;3.67,-3.01,;3.67,-4.55,;2.34,-5.32,;2.34,-6.86,;1.01,-7.63,;-.33,-6.86,;-.33,-5.32,;1.01,-4.55,;1.01,-3.01,;5.01,-2.24,;1.01,.07,;1.01,1.61,;-.33,2.38,;-1.66,1.61,;-1.66,.07,;-.33,-.7,;-3.12,-.41,;-3.52,-1.89,;-4.86,-2.66,;-4.09,-4,;-2.75,-3.23,;-4.49,-5.48,;-3.58,-6.73,;-4.49,-7.98,;-5.95,-7.5,;-6.72,-8.83,;-7.49,-7.5,;-5.95,-5.96,;-4.03,.84,;-5.57,.84,;-3.12,2.09,;-2.04,3.18,;-2.43,4.66,;-3.92,5.06,;-5.01,3.97,;-4.61,2.48,;-4.32,6.55,;-3.23,7.64,;-5.81,6.95,;-6.9,5.86,;-8.38,6.26,;-8.78,7.74,;-7.69,8.83,;-6.21,8.44,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N([C@@H]1C[C@@H](C1)N1CCC(C)(C)C1)C(=O)C21CCN(CC1)C(=O)C1(C)CCOCC1 |r,wU:27.30,29.35,(6.47,-5.38,;7.24,-4.05,;8.78,-4.05,;6.47,-2.72,;7.38,-1.47,;6.47,-.22,;5.01,-.7,;3.67,.07,;2.34,-.7,;2.34,-2.24,;3.67,-3.01,;3.67,-4.55,;2.34,-5.32,;2.34,-6.86,;1.01,-7.63,;-.33,-6.86,;-.33,-5.32,;1.01,-4.55,;1.01,-3.01,;5.01,-2.24,;1.01,.07,;1.01,1.61,;-.33,2.38,;-1.66,1.61,;-1.66,.07,;-.33,-.7,;-3.12,-.41,;-3.52,-1.89,;-4.86,-2.66,;-4.09,-4,;-2.75,-3.23,;-4.49,-5.48,;-3.58,-6.73,;-4.49,-7.98,;-5.95,-7.5,;-6.72,-8.83,;-7.49,-7.5,;-5.95,-5.96,;-4.03,.84,;-5.57,.84,;-3.12,2.09,;-2.04,3.18,;-2.43,4.66,;-3.92,5.06,;-5.01,3.97,;-4.61,2.48,;-4.32,6.55,;-3.23,7.64,;-5.81,6.95,;-4.72,8.04,;-6.21,8.44,;-7.69,8.83,;-8.78,7.74,;-8.38,6.26,;-6.9,5.86,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N([C@H]1C[C@H](C1)N1CCCCC1)C(=O)C21CCN(CC1)C(=O)C1(C)CC1 |r,wU:27.30,29.35,(5.27,-5.72,;6.04,-4.38,;7.58,-4.38,;5.27,-3.05,;6.17,-1.8,;5.27,-.56,;3.8,-1.03,;2.47,-.26,;1.14,-1.03,;1.14,-2.57,;2.47,-3.34,;2.47,-4.88,;1.14,-5.65,;1.14,-7.19,;-.2,-7.96,;-1.53,-7.19,;-1.53,-5.65,;-.2,-4.88,;-.2,-3.34,;3.8,-2.57,;-.2,-.26,;-.2,1.28,;-1.53,2.05,;-2.87,1.28,;-2.87,-.26,;-1.53,-1.03,;-4.33,-.74,;-4.73,-2.23,;-3.96,-3.56,;-5.29,-4.33,;-6.06,-3,;-5.69,-5.82,;-7.18,-6.22,;-7.58,-7.7,;-6.49,-8.79,;-5,-8.39,;-4.6,-6.91,;-5.24,.51,;-6.78,.51,;-4.33,1.75,;-3.24,2.84,;-3.64,4.33,;-5.13,4.73,;-6.22,3.64,;-5.82,2.15,;-5.53,6.22,;-7.01,6.61,;-4.44,7.3,;-5.77,8.07,;-2.95,7.7,;-4.04,8.79,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N([C@H]1C[C@H](C1)N1CCCCC1)C(=O)C21CCN(CC1)C(=O)C12CC(F)(C1)C2 |r,wU:27.30,29.35,(5.27,-6.29,;6.04,-4.95,;7.58,-4.95,;5.27,-3.62,;6.17,-2.37,;5.27,-1.13,;3.8,-1.6,;2.47,-.83,;1.14,-1.6,;1.14,-3.14,;2.47,-3.91,;2.47,-5.45,;1.14,-6.22,;1.14,-7.76,;-.2,-8.53,;-1.53,-7.76,;-1.53,-6.22,;-.2,-5.45,;-.2,-3.91,;3.8,-3.14,;-.2,-.83,;-.2,.71,;-1.53,1.48,;-2.87,.71,;-2.87,-.83,;-1.53,-1.6,;-4.33,-1.31,;-4.73,-2.8,;-3.96,-4.13,;-5.29,-4.9,;-6.06,-3.57,;-5.69,-6.39,;-7.18,-6.79,;-7.58,-8.27,;-6.49,-9.36,;-5,-8.96,;-4.6,-7.48,;-5.24,-.06,;-6.78,-.06,;-4.33,1.18,;-3.24,2.27,;-3.64,3.76,;-5.13,4.16,;-6.22,3.07,;-5.82,1.58,;-5.53,5.65,;-7.01,6.04,;-4.44,6.73,;-2.9,6.73,;-2.9,8.27,;-1.81,9.36,;-4.44,8.27,;-4.15,7.85,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N([C@@H]1C[C@@H](C1)N1CCC(C)(C)C1)C(=O)C21CCN(CC1)C(C)=O |r,wU:27.30,29.35,(5.72,-5.07,;6.49,-3.73,;8.03,-3.73,;5.72,-2.4,;6.63,-1.15,;5.72,.09,;4.26,-.38,;2.93,.39,;1.59,-.38,;1.59,-1.92,;2.93,-2.69,;2.93,-4.23,;1.59,-5,;1.59,-6.54,;.26,-7.31,;-1.08,-6.54,;-1.08,-5,;.26,-4.23,;.26,-2.69,;4.26,-1.92,;.26,.39,;.26,1.93,;-1.08,2.7,;-2.41,1.93,;-2.41,.39,;-1.08,-.38,;-3.87,-.09,;-4.27,-1.58,;-5.61,-2.35,;-4.84,-3.68,;-3.5,-2.91,;-5.24,-5.17,;-4.33,-6.41,;-5.24,-7.66,;-6.7,-7.18,;-8.03,-6.41,;-8.03,-7.95,;-6.7,-5.64,;-4.78,1.16,;-6.32,1.16,;-3.87,2.4,;-2.79,3.49,;-3.18,4.98,;-4.67,5.38,;-5.76,4.29,;-5.36,2.8,;-5.07,6.87,;-6.56,7.26,;-3.98,7.95,)|
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CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N([C@H]1C[C@H](C1)N1CCC[C@@H](C)C1)C(=O)C21CCN(CC1)C(C)=O |r,wU:27.30,29.35,35.40,(6.01,-4.97,;6.78,-3.64,;8.32,-3.64,;6.01,-2.3,;6.92,-1.06,;6.01,.19,;4.55,-.29,;3.21,.48,;1.88,-.29,;1.88,-1.83,;3.21,-2.6,;3.21,-4.14,;1.88,-4.91,;1.88,-6.45,;.55,-7.22,;-.79,-6.45,;-.79,-4.91,;.55,-4.14,;.55,-2.6,;4.55,-1.83,;.55,.48,;.55,2.02,;-.79,2.79,;-2.12,2.02,;-2.12,.48,;-.79,-.29,;-3.59,.01,;-3.99,-1.48,;-3.22,-2.82,;-4.55,-3.59,;-5.32,-2.25,;-4.95,-5.07,;-3.86,-6.16,;-4.26,-7.65,;-5.74,-8.05,;-6.83,-6.96,;-8.32,-7.36,;-6.43,-5.47,;-4.49,1.25,;-6.03,1.25,;-3.59,2.5,;-2.5,3.59,;-2.9,5.07,;-4.38,5.47,;-5.47,4.38,;-5.07,2.9,;-4.78,6.96,;-6.27,7.36,;-3.69,8.05,)|
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CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N([C@H]1C[C@H](C1)N1CC3CCC(C1)O3)C(=O)C21CCN(CC1)C(C)=O |r,wU:27.30,29.35,(5.27,-4.97,;6.04,-3.64,;7.58,-3.64,;5.27,-2.3,;6.17,-1.06,;5.27,.19,;3.8,-.29,;2.47,.48,;1.14,-.29,;1.14,-1.83,;2.47,-2.6,;2.47,-4.14,;1.14,-4.91,;1.14,-6.45,;-.2,-7.22,;-1.53,-6.45,;-1.53,-4.91,;-.2,-4.14,;-.2,-2.6,;3.8,-1.83,;-.2,.48,;-.2,2.02,;-1.53,2.79,;-2.87,2.02,;-2.87,.48,;-1.53,-.29,;-4.33,.01,;-4.73,-1.48,;-3.96,-2.82,;-5.29,-3.59,;-6.06,-2.25,;-5.69,-5.07,;-7.18,-5.47,;-7.58,-6.96,;-6.53,-6.18,;-5.44,-6.47,;-5,-7.65,;-4.6,-6.16,;-6.49,-8.05,;-5.24,1.25,;-6.78,1.25,;-4.33,2.5,;-3.24,3.59,;-3.64,5.07,;-5.13,5.47,;-6.22,4.38,;-5.82,2.9,;-5.53,6.96,;-7.01,7.36,;-4.44,8.05,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N([C@H]1C[C@H](C1)N1CCCC3(CC3)C1)C(=O)C21CCN(CC1)C(=O)C1(C)COC1 |r,wU:27.30,29.35,(6.04,-5.29,;6.81,-3.96,;8.35,-3.96,;6.04,-2.63,;6.94,-1.38,;6.04,-.13,;4.57,-.61,;3.24,.16,;1.91,-.61,;1.91,-2.15,;3.24,-2.92,;3.24,-4.46,;1.91,-5.23,;1.91,-6.77,;.57,-7.54,;-.76,-6.77,;-.76,-5.23,;.57,-4.46,;.57,-2.92,;4.57,-2.15,;.57,.16,;.57,1.7,;-.76,2.47,;-2.1,1.7,;-2.1,.16,;-.76,-.61,;-3.56,-.32,;-3.96,-1.8,;-3.19,-3.14,;-4.52,-3.91,;-5.29,-2.57,;-4.92,-5.4,;-3.83,-6.48,;-4.23,-7.97,;-5.72,-8.37,;-6.81,-7.28,;-8.29,-6.88,;-7.9,-8.37,;-6.41,-5.79,;-4.47,.93,;-6.01,.93,;-3.56,2.18,;-2.47,3.26,;-2.87,4.75,;-4.36,5.15,;-5.45,4.06,;-5.05,2.57,;-4.76,6.64,;-3.67,7.73,;-6.24,7.04,;-5.47,8.37,;-7.01,8.37,;-8.35,7.6,;-7.58,6.27,)|
C[C@@H](O)C(=O)N1CCC2(CC1)C(=O)N([C@H]1C[C@H](C1)N1CCCC3(CC3)C1)c1cc(ccc21)-c1cc2ncn(C(C)C)c2c(Nc2ccncc2F)n1 |r,wU:14.14,16.19,1.1,(-7.36,5.87,;-6.27,6.96,;-6.67,8.45,;-4.78,6.56,;-3.69,7.65,;-4.38,5.07,;-2.9,4.67,;-2.5,3.19,;-3.59,2.1,;-5.07,2.5,;-5.47,3.98,;-4.49,.85,;-6.03,.85,;-3.59,-.39,;-3.99,-1.88,;-3.22,-3.21,;-4.55,-3.98,;-5.32,-2.65,;-4.95,-5.47,;-3.86,-6.56,;-4.26,-8.05,;-5.74,-8.45,;-6.83,-7.36,;-8.32,-6.96,;-7.92,-8.45,;-6.43,-5.87,;-2.12,.08,;-.79,-.69,;.55,.08,;.55,1.62,;-.79,2.39,;-2.12,1.62,;1.88,-.69,;3.21,.08,;4.55,-.69,;6.01,-.21,;6.92,-1.46,;6.01,-2.7,;6.78,-4.04,;6.01,-5.37,;8.32,-4.04,;4.55,-2.23,;3.21,-3,;3.21,-4.54,;1.88,-5.31,;1.88,-6.85,;.55,-7.62,;-.79,-6.85,;-.79,-5.31,;.55,-4.54,;.55,-3,;1.88,-2.23,)|
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CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N([C@@H]1C[C@@H](C1)N1CC(C)(C)C[C@H]1CO)C(=O)C21CCN(CC1)C1COC1 |r,wU:27.30,29.35,37.43,(6.12,-4.91,;7.15,-3.76,;8.66,-4.08,;6.68,-2.3,;7.58,-1.05,;6.68,.19,;5.21,-.28,;3.88,.49,;2.55,-.28,;2.55,-1.82,;3.88,-2.59,;3.88,-4.13,;2.55,-4.9,;2.55,-6.44,;1.21,-7.21,;-.12,-6.44,;-.12,-4.9,;1.21,-4.13,;1.21,-2.59,;5.21,-1.82,;1.21,.49,;1.21,2.03,;-.12,2.8,;-1.45,2.03,;-1.45,.49,;-.12,-.28,;-2.92,.01,;-3.39,-1.45,;-4.77,-2.15,;-4.07,-3.52,;-2.7,-2.83,;-4.54,-4.99,;-3.64,-6.24,;-4.54,-7.48,;-4.94,-8.97,;-3.45,-8.57,;-6.01,-7.01,;-6.01,-5.47,;-7.25,-4.56,;-8.66,-5.19,;-3.82,1.26,;-5.36,1.26,;-2.92,2.5,;-1.89,3.65,;-2.36,5.11,;-3.87,5.43,;-4.9,4.29,;-4.43,2.82,;-4.35,6.9,;-3.65,8.27,;-5.02,8.97,;-5.72,7.6,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N([C@@H]1C[C@@H](C1)N1CC(C)(C)C[C@@H]1CO)C(=O)C21CCN(CC1)C1COC1 |r,wU:27.30,29.35,wD:37.43,(6.12,-4.91,;7.15,-3.76,;8.66,-4.08,;6.68,-2.3,;7.58,-1.05,;6.68,.19,;5.21,-.28,;3.88,.49,;2.55,-.28,;2.55,-1.82,;3.88,-2.59,;3.88,-4.13,;2.55,-4.9,;2.55,-6.44,;1.21,-7.21,;-.12,-6.44,;-.12,-4.9,;1.21,-4.13,;1.21,-2.59,;5.21,-1.82,;1.21,.49,;1.21,2.03,;-.12,2.8,;-1.45,2.03,;-1.45,.49,;-.12,-.28,;-2.92,.01,;-3.39,-1.45,;-4.77,-2.15,;-4.07,-3.52,;-2.7,-2.83,;-4.54,-4.99,;-3.64,-6.24,;-4.54,-7.48,;-4.94,-8.97,;-3.45,-8.57,;-6.01,-7.01,;-6.01,-5.47,;-7.25,-4.56,;-8.66,-5.19,;-3.82,1.26,;-5.36,1.26,;-2.92,2.5,;-1.89,3.65,;-2.36,5.11,;-3.87,5.43,;-4.9,4.29,;-4.43,2.82,;-4.35,6.9,;-3.65,8.27,;-5.02,8.97,;-5.72,7.6,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N(C1CC(C1)N1CCC[C@H](C)C1)C(=O)C21CCN(CC1)C1COC1 |r,wU:35.40,(14.97,3.01,;13.44,2.79,;12.87,1.36,;12.49,4,;12.9,5.48,;11.62,6.33,;10.41,5.38,;8.89,5.63,;7.91,4.45,;8.45,3,;9.97,2.75,;10.5,1.3,;9.52,.12,;8,.37,;7.02,-.81,;7.56,-2.26,;9.07,-2.51,;10.06,-1.33,;11.57,-1.59,;10.95,3.93,;6.39,4.7,;5.41,3.52,;3.89,3.77,;3.36,5.22,;4.34,6.4,;5.86,6.15,;3.51,7.7,;4.08,9.14,;3.47,10.55,;4.88,11.16,;5.49,9.75,;5.45,12.59,;6.98,12.75,;7.61,14.16,;6.7,15.41,;5.17,15.25,;4.27,16.49,;4.54,13.84,;2.02,7.32,;.83,8.3,;1.92,5.79,;1.99,4.25,;.69,3.42,;-.68,4.14,;-.74,5.67,;.56,6.5,;-1.98,3.31,;-2.31,1.81,;-3.82,2.14,;-3.48,3.65,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N(C1CC(C1)N1CC[C@H](F)C1)C(=O)C21CCN(CC1)C1COC1 |r,wU:34.39,(14.97,3.01,;13.44,2.79,;12.87,1.36,;12.49,4,;12.9,5.48,;11.62,6.33,;10.41,5.38,;8.89,5.63,;7.91,4.45,;8.45,3,;9.97,2.75,;10.5,1.3,;9.52,.12,;8,.37,;7.02,-.81,;7.56,-2.26,;9.07,-2.51,;10.06,-1.33,;11.57,-1.59,;10.95,3.93,;6.39,4.7,;5.41,3.52,;3.89,3.77,;3.36,5.22,;4.34,6.4,;5.86,6.15,;3.51,7.7,;4.08,9.14,;3.47,10.55,;4.88,11.16,;5.49,9.75,;5.45,12.59,;6.96,12.91,;7.12,14.44,;5.71,15.07,;5.39,16.58,;4.68,13.93,;2.02,7.32,;.83,8.3,;1.92,5.79,;1.99,4.25,;.69,3.42,;-.68,4.14,;-.74,5.67,;.56,6.5,;-1.98,3.31,;-2.31,1.81,;-3.82,2.14,;-3.48,3.65,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N(C1CC(C1)N1CCC(F)CC1)C(=O)C21CCN(CC1)C1COC1 |(14.97,3.01,;13.44,2.79,;12.87,1.36,;12.49,4,;12.9,5.48,;11.62,6.33,;10.41,5.38,;8.89,5.63,;7.91,4.45,;8.45,3,;9.97,2.75,;10.5,1.3,;9.52,.12,;8,.37,;7.02,-.81,;7.56,-2.26,;9.07,-2.51,;10.06,-1.33,;11.57,-1.59,;10.95,3.93,;6.39,4.7,;5.41,3.52,;3.89,3.77,;3.36,5.22,;4.34,6.4,;5.86,6.15,;3.51,7.7,;4.08,9.14,;3.47,10.55,;4.88,11.16,;5.49,9.75,;5.45,12.59,;6.98,12.75,;7.61,14.16,;6.7,15.41,;7.33,16.81,;5.17,15.25,;4.54,13.84,;2.02,7.32,;.83,8.3,;1.92,5.79,;1.99,4.25,;.69,3.42,;-.68,4.14,;-.74,5.67,;.56,6.5,;-1.98,3.31,;-2.31,1.81,;-3.82,2.14,;-3.48,3.65,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N(C1CC(C1)N1CC[C@H](C)C1)C(=O)C21CCN(CC1)C1COC1 |r,wU:34.39,(14.97,3.01,;13.44,2.79,;12.87,1.36,;12.49,4,;12.9,5.48,;11.62,6.33,;10.41,5.38,;8.89,5.63,;7.91,4.45,;8.45,3,;9.97,2.75,;10.5,1.3,;9.52,.12,;8,.37,;7.02,-.81,;7.56,-2.26,;9.07,-2.51,;10.06,-1.33,;11.57,-1.59,;10.95,3.93,;6.39,4.7,;5.41,3.52,;3.89,3.77,;3.36,5.22,;4.34,6.4,;5.86,6.15,;3.51,7.7,;4.08,9.14,;3.47,10.55,;4.88,11.16,;5.49,9.75,;5.45,12.59,;6.96,12.91,;7.12,14.44,;5.71,15.07,;5.39,16.58,;4.68,13.93,;2.02,7.32,;.83,8.3,;1.92,5.79,;1.99,4.25,;.69,3.42,;-.68,4.14,;-.74,5.67,;.56,6.5,;-1.98,3.31,;-2.31,1.81,;-3.82,2.14,;-3.48,3.65,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N(C1CC(C1)N1CCCC(C)(C)C1)C(=O)C21CCN(CC1)C1COC1 |(14.97,3.01,;13.44,2.79,;12.87,1.36,;12.49,4,;12.9,5.48,;11.62,6.33,;10.41,5.38,;8.89,5.63,;7.91,4.45,;8.45,3,;9.97,2.75,;10.5,1.3,;9.52,.12,;8,.37,;7.02,-.81,;7.56,-2.26,;9.07,-2.51,;10.06,-1.33,;11.57,-1.59,;10.95,3.93,;6.39,4.7,;5.41,3.52,;3.89,3.77,;3.36,5.22,;4.34,6.4,;5.86,6.15,;3.51,7.7,;4.08,9.14,;3.47,10.55,;4.88,11.16,;5.49,9.75,;5.45,12.59,;6.98,12.75,;7.61,14.16,;6.7,15.41,;5.17,15.25,;4.27,16.49,;5.8,16.65,;4.54,13.84,;2.02,7.32,;.83,8.3,;1.92,5.79,;1.99,4.25,;.69,3.42,;-.68,4.14,;-.74,5.67,;.56,6.5,;-1.98,3.31,;-2.31,1.81,;-3.82,2.14,;-3.48,3.65,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N(C1CC(C1)N1CC[C@@H](F)C1)C(=O)C21CCN(CC1)C1COC1 |r,wD:34.39,(14.97,3.01,;13.44,2.79,;12.87,1.36,;12.49,4,;12.9,5.48,;11.62,6.33,;10.41,5.38,;8.89,5.63,;7.91,4.45,;8.45,3,;9.97,2.75,;10.5,1.3,;9.52,.12,;8,.37,;7.02,-.81,;7.56,-2.26,;9.07,-2.51,;10.06,-1.33,;11.57,-1.59,;10.95,3.93,;6.39,4.7,;5.41,3.52,;3.89,3.77,;3.36,5.22,;4.34,6.4,;5.86,6.15,;3.51,7.7,;4.08,9.14,;3.47,10.55,;4.88,11.16,;5.49,9.75,;5.45,12.59,;6.96,12.91,;7.12,14.44,;5.71,15.07,;5.39,16.58,;4.68,13.93,;2.02,7.32,;.83,8.3,;1.92,5.79,;1.99,4.25,;.69,3.42,;-.68,4.14,;-.74,5.67,;.56,6.5,;-1.98,3.31,;-2.31,1.81,;-3.82,2.14,;-3.48,3.65,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N(C1CC(C1)N1CC[C@@H](C)C1)C(=O)C21CCN(CC1)C1COC1 |r,wD:34.39,(14.97,3.01,;13.44,2.79,;12.87,1.36,;12.49,4,;12.9,5.48,;11.62,6.33,;10.41,5.38,;8.89,5.63,;7.91,4.45,;8.45,3,;9.97,2.75,;10.5,1.3,;9.52,.12,;8,.37,;7.02,-.81,;7.56,-2.26,;9.07,-2.51,;10.06,-1.33,;11.57,-1.59,;10.95,3.93,;6.39,4.7,;5.41,3.52,;3.89,3.77,;3.36,5.22,;4.34,6.4,;5.86,6.15,;3.51,7.7,;4.08,9.14,;3.47,10.55,;4.88,11.16,;5.49,9.75,;5.45,12.59,;6.96,12.91,;7.12,14.44,;5.71,15.07,;5.39,16.58,;4.68,13.93,;2.02,7.32,;.83,8.3,;1.92,5.79,;1.99,4.25,;.69,3.42,;-.68,4.14,;-.74,5.67,;.56,6.5,;-1.98,3.31,;-2.31,1.81,;-3.82,2.14,;-3.48,3.65,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N(C1CC(C1)N1CCC(C1)C(F)F)C(=O)C21CCN(CC1)C1COC1 |(14.97,3.01,;13.44,2.79,;12.87,1.36,;12.49,4,;12.9,5.48,;11.62,6.33,;10.41,5.38,;8.89,5.63,;7.91,4.45,;8.45,3,;9.97,2.75,;10.5,1.3,;9.52,.12,;8,.37,;7.02,-.81,;7.56,-2.26,;9.07,-2.51,;10.06,-1.33,;11.57,-1.59,;10.95,3.93,;6.39,4.7,;5.41,3.52,;3.89,3.77,;3.36,5.22,;4.34,6.4,;5.86,6.15,;3.51,7.7,;4.08,9.14,;3.47,10.55,;4.88,11.16,;5.49,9.75,;5.45,12.59,;6.96,12.91,;7.12,14.44,;5.71,15.07,;4.68,13.93,;5.39,16.58,;3.93,17.05,;6.53,17.61,;2.02,7.32,;.83,8.3,;1.92,5.79,;1.99,4.25,;.69,3.42,;-.68,4.14,;-.74,5.67,;.56,6.5,;-1.98,3.31,;-2.31,1.81,;-3.82,2.14,;-3.48,3.65,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N(C1CC(C1)N1CC(F)C3(CC3)C1)C(=O)C21CCN(CC1)C1COC1 |(14.97,3.01,;13.44,2.79,;12.87,1.36,;12.49,4,;12.9,5.48,;11.62,6.33,;10.41,5.38,;8.89,5.63,;7.91,4.45,;8.45,3,;9.97,2.75,;10.5,1.3,;9.52,.12,;8,.37,;7.02,-.81,;7.56,-2.26,;9.07,-2.51,;10.06,-1.33,;11.57,-1.59,;10.95,3.93,;6.39,4.7,;5.41,3.52,;3.89,3.77,;3.36,5.22,;4.34,6.4,;5.86,6.15,;3.51,7.7,;4.08,9.14,;3.47,10.55,;4.88,11.16,;5.49,9.75,;5.45,12.59,;4.68,13.93,;5.71,15.07,;5.39,16.58,;7.12,14.44,;8.02,15.69,;8.65,14.28,;6.96,12.91,;2.02,7.32,;.83,8.3,;1.92,5.79,;1.99,4.25,;.69,3.42,;-.68,4.14,;-.74,5.67,;.56,6.5,;-1.98,3.31,;-2.31,1.81,;-3.82,2.14,;-3.48,3.65,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N(C1CC(C1)N1C3CCC1COC3)C(=O)C21CCN(CC1)C1COC1 |(14.97,3.01,;13.44,2.79,;12.87,1.36,;12.49,4,;12.9,5.48,;11.62,6.33,;10.41,5.38,;8.89,5.63,;7.91,4.45,;8.45,3,;9.97,2.75,;10.5,1.3,;9.52,.12,;8,.37,;7.02,-.81,;7.56,-2.26,;9.07,-2.51,;10.06,-1.33,;11.57,-1.59,;10.95,3.93,;6.39,4.7,;5.41,3.52,;3.89,3.77,;3.36,5.22,;4.34,6.4,;5.86,6.15,;3.51,7.7,;4.08,9.14,;3.47,10.55,;4.88,11.16,;5.49,9.75,;5.45,12.59,;4.54,13.84,;5.95,14.55,;6.82,14.29,;6.98,12.75,;7.61,14.16,;6.7,15.41,;5.17,15.25,;2.02,7.32,;.83,8.3,;1.92,5.79,;1.99,4.25,;.69,3.42,;-.68,4.14,;-.74,5.67,;.56,6.5,;-1.98,3.31,;-2.31,1.81,;-3.82,2.14,;-3.48,3.65,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N(C1CC(C1)N1CCCCC1)C(=O)C21CCN(CC1)C1COC1 |(14.97,3.01,;13.44,2.79,;12.87,1.36,;12.49,4,;12.9,5.48,;11.62,6.33,;10.41,5.38,;8.89,5.63,;7.91,4.45,;8.45,3,;9.97,2.75,;10.5,1.3,;9.52,.12,;8,.37,;7.02,-.81,;7.56,-2.26,;9.07,-2.51,;10.06,-1.33,;11.57,-1.59,;10.95,3.93,;6.39,4.7,;5.41,3.52,;3.89,3.77,;3.36,5.22,;4.34,6.4,;5.86,6.15,;3.51,7.7,;4.08,9.14,;3.47,10.55,;4.88,11.16,;5.49,9.75,;5.45,12.59,;6.98,12.75,;7.61,14.16,;6.7,15.41,;5.17,15.25,;4.54,13.84,;2.02,7.32,;.83,8.3,;1.92,5.79,;1.99,4.25,;.69,3.42,;-.68,4.14,;-.74,5.67,;.56,6.5,;-1.98,3.31,;-2.31,1.81,;-3.82,2.14,;-3.48,3.65,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N(C1CC(C1)NCC(C)(C)O)C(=O)C2(C)C |(13.94,7.78,;12.91,6.63,;13.39,5.17,;11.4,6.95,;10.78,8.36,;9.25,8.2,;8.93,6.69,;7.59,5.92,;7.59,4.38,;8.93,3.61,;10.26,4.38,;11.59,3.61,;11.59,2.07,;10.26,1.3,;10.26,-.24,;11.59,-1.01,;12.93,-.24,;12.93,1.3,;14.26,2.07,;10.26,5.92,;6.26,3.61,;6.26,2.07,;4.92,1.3,;3.59,2.07,;3.59,3.61,;4.92,4.38,;2.13,4.09,;1.65,5.55,;.28,6.25,;.98,7.62,;2.35,6.93,;.5,9.09,;1.53,10.23,;3.04,9.91,;3.36,11.42,;4.54,9.59,;2.72,8.41,;1.22,2.84,;-.32,2.84,;2.13,1.6,;2.43,.09,;.99,.55,)|
CC(C)n1cnc2cc(nc(Nc3cc(C)ncc3F)c12)-c1ccc2c(c1)N([C@@H]1C[C@@H](C1)NCC(C)(C)O)C(=O)C2(C)C |r,wU:28.31,30.36,(5.79,-2.53,;6.82,-1.39,;8.33,-1.71,;6.34,.08,;7.25,1.32,;6.34,2.57,;4.88,2.09,;3.55,2.86,;2.21,2.09,;2.21,.55,;3.55,-.22,;3.55,-1.76,;2.21,-2.53,;2.21,-4.07,;.88,-4.84,;.88,-6.38,;-.46,-4.07,;-.46,-2.53,;.88,-1.76,;.88,-.22,;4.88,.55,;.88,2.86,;.88,4.4,;-.46,5.17,;-1.79,4.4,;-1.79,2.86,;-.46,2.09,;-3.25,2.39,;-3.73,.92,;-5.1,.22,;-4.4,-1.15,;-3.03,-.45,;-4.88,-2.61,;-6.39,-2.93,;-6.86,-4.4,;-8.33,-3.92,;-8.01,-5.43,;-5.83,-5.54,;-4.16,3.63,;-5.7,3.63,;-3.25,4.88,;-4.43,5.88,;-2.89,6.38,)|
CC(C)n1cnc2cc(nc(Nc3cc(C)ncc3F)c12)-c1ccc2c(c1)N([C@H]1C[C@H](C1)N1CCCCC1)C(=O)C2(C)C |r,wU:28.31,30.36,(5.67,-2.9,;6.07,-1.41,;7.61,-1.41,;5.59,.06,;6.5,1.3,;5.59,2.55,;4.13,2.07,;2.8,2.84,;1.46,2.07,;1.46,.53,;2.8,-.24,;2.8,-1.78,;1.46,-2.55,;1.46,-4.09,;.13,-4.86,;.13,-6.4,;-1.2,-4.09,;-1.2,-2.55,;.13,-1.78,;.13,-.24,;4.13,.53,;.13,2.84,;.13,4.38,;-1.2,5.15,;-2.54,4.38,;-2.54,2.84,;-1.2,2.07,;-4,2.37,;-4.48,.9,;-3.78,-.47,;-5.15,-1.17,;-5.85,.2,;-5.63,-2.63,;-7.13,-2.95,;-7.61,-4.42,;-6.58,-5.56,;-5.07,-5.24,;-4.6,-3.78,;-4.91,3.61,;-6.45,3.61,;-4,4.86,;-5.34,5.63,;-4,6.4,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N([C@H]1C[C@H](C1)N1CCCCC1)C(=O)C2(C)O |r,wU:27.30,29.35,(5.06,-2.95,;6.09,-1.8,;7.59,-2.12,;5.61,-.34,;6.52,.91,;5.61,2.15,;4.15,1.68,;2.81,2.45,;1.48,1.68,;1.48,.14,;2.81,-.63,;2.81,-2.17,;1.48,-2.94,;1.48,-4.48,;.15,-5.25,;-1.19,-4.48,;-1.19,-2.94,;.15,-2.17,;.15,-.63,;4.15,.14,;.15,2.45,;.15,3.99,;-1.19,4.76,;-2.52,3.99,;-2.52,2.45,;-1.19,1.68,;-3.99,1.97,;-4.46,.51,;-3.76,-.87,;-5.14,-1.57,;-5.83,-.19,;-5.61,-3.03,;-7.12,-3.35,;-7.59,-4.82,;-6.56,-5.96,;-5.06,-5.64,;-4.58,-4.17,;-4.89,3.22,;-6.43,3.22,;-3.99,4.46,;-3.63,5.96,;-5.16,5.46,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N([C@H]1C[C@H](C1)N1CCCCC1)C(=O)[C@@]2(C)O |r,wU:27.30,29.35,39.47,wD:39.46,(-.37,-2.12,;-1.88,-1.8,;-2.91,-2.94,;-2.36,-.33,;-1.45,.91,;-2.36,2.16,;-3.82,1.68,;-5.16,2.45,;-6.49,1.68,;-6.49,.14,;-5.16,-.63,;-5.16,-2.17,;-6.49,-2.94,;-6.49,-4.48,;-7.82,-5.25,;-9.16,-4.48,;-9.16,-2.94,;-7.82,-2.17,;-7.82,-.63,;-3.82,.14,;-7.82,2.45,;-7.82,3.99,;-9.16,4.76,;-10.49,3.99,;-10.49,2.45,;-9.16,1.68,;-11.95,1.98,;-12.43,.51,;-11.73,-.86,;-13.1,-1.56,;-13.8,-.19,;-13.58,-3.03,;-15.09,-3.35,;-15.56,-4.81,;-14.53,-5.95,;-13.02,-5.63,;-12.55,-4.17,;-12.86,3.22,;-14.4,3.22,;-11.95,4.47,;-11.56,5.95,;-13.04,5.56,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N([C@H]1C[C@H](C1)N1CCCCC1)C(=O)[C@]2(C)O |r,wU:27.30,29.35,39.46,wD:39.47,(15.56,-2.12,;14.06,-1.8,;13.02,-2.94,;13.58,-.33,;14.48,.91,;13.58,2.16,;12.11,1.68,;10.78,2.45,;9.45,1.68,;9.45,.14,;10.78,-.63,;10.78,-2.17,;9.45,-2.94,;9.45,-4.48,;8.11,-5.25,;6.78,-4.48,;6.78,-2.94,;8.11,-2.17,;8.11,-.63,;12.11,.14,;8.11,2.45,;8.11,3.99,;6.78,4.76,;5.45,3.99,;5.45,2.45,;6.78,1.68,;3.98,1.98,;3.51,.51,;4.21,-.86,;2.83,-1.56,;2.13,-.19,;2.36,-3.03,;.85,-3.35,;.37,-4.81,;1.41,-5.95,;2.91,-5.63,;3.39,-4.17,;3.08,3.22,;1.54,3.22,;3.98,4.47,;4.38,5.95,;2.89,5.56,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N([C@@H]1C[C@@H](C1)N1CCC3(CC3)C1)C(=O)C2(C)C |r,wU:27.30,29.35,(5.56,-2.7,;6.59,-1.56,;8.1,-1.88,;6.12,-.09,;7.02,1.15,;6.12,2.4,;4.65,1.92,;3.32,2.69,;1.99,1.92,;1.99,.38,;3.32,-.39,;3.32,-1.93,;1.99,-2.7,;1.99,-4.24,;.65,-5.01,;-.68,-4.24,;-.68,-2.7,;.65,-1.93,;.65,-.39,;4.65,.38,;.65,2.69,;.65,4.23,;-.68,5,;-2.01,4.23,;-2.01,2.69,;-.68,1.92,;-3.48,2.22,;-3.96,.75,;-5.33,.05,;-4.63,-1.32,;-3.26,-.62,;-5.1,-2.78,;-4.2,-4.03,;-5.1,-5.28,;-6.57,-4.8,;-8.1,-4.96,;-7.2,-6.21,;-6.57,-3.26,;-4.38,3.46,;-5.92,3.46,;-3.48,4.71,;-4.65,5.71,;-3.12,6.21,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N([C@@H]1C[C@@H](C1)N1C[C@H](C)[C@H](C)C1)C(=O)C2(C)C |r,wU:27.30,29.35,33.38,35.40,(5.42,-2.44,;6.45,-1.29,;7.96,-1.61,;5.98,.17,;6.88,1.42,;5.98,2.67,;4.51,2.19,;3.18,2.96,;1.84,2.19,;1.84,.65,;3.18,-.12,;3.18,-1.66,;1.84,-2.43,;1.84,-3.97,;.51,-4.74,;-.82,-3.97,;-.82,-2.43,;.51,-1.66,;.51,-.12,;4.51,.65,;.51,2.96,;.51,4.5,;-.82,5.27,;-2.16,4.5,;-2.16,2.96,;-.82,2.19,;-3.62,2.48,;-4.1,1.02,;-5.47,.32,;-4.77,-1.05,;-3.4,-.35,;-5.25,-2.52,;-6.71,-2.99,;-6.71,-4.53,;-7.96,-5.44,;-5.25,-5.01,;-4.77,-6.47,;-4.34,-3.76,;-4.53,3.73,;-6.07,3.73,;-3.62,4.98,;-4.79,5.98,;-3.26,6.47,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N([C@H]1C[C@H](C1)N1CC3CCC1CC3)C(=O)C2(C)C |r,wU:27.30,29.35,(5.06,-2.95,;6.09,-1.8,;7.59,-2.12,;5.61,-.34,;6.52,.91,;5.61,2.15,;4.15,1.68,;2.81,2.45,;1.48,1.68,;1.48,.14,;2.81,-.63,;2.81,-2.17,;1.48,-2.94,;1.48,-4.48,;.15,-5.25,;-1.19,-4.48,;-1.19,-2.94,;.15,-2.17,;.15,-.63,;4.15,.14,;.15,2.45,;.15,3.99,;-1.19,4.76,;-2.52,3.99,;-2.52,2.45,;-1.19,1.68,;-3.99,1.97,;-4.46,.51,;-3.76,-.87,;-5.14,-1.57,;-5.83,-.19,;-5.61,-3.03,;-4.58,-4.17,;-5.06,-5.64,;-6.56,-5.96,;-7.59,-4.82,;-7.12,-3.35,;-6.75,-4.83,;-5.38,-4.13,;-4.89,3.22,;-6.43,3.22,;-3.99,4.46,;-5.16,5.46,;-3.63,5.96,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N([C@H]1C[C@H](C1)N1CCCCCC1)C(=O)C2(C)C |r,wU:27.30,29.35,(5.22,-2.49,;6.25,-1.34,;7.76,-1.66,;5.78,.12,;6.68,1.37,;5.78,2.61,;4.31,2.14,;2.98,2.91,;1.65,2.14,;1.65,.6,;2.98,-.17,;2.98,-1.71,;1.65,-2.48,;1.65,-4.02,;.31,-4.79,;-1.02,-4.02,;-1.02,-2.48,;.31,-1.71,;.31,-.17,;4.31,.6,;.31,2.91,;.31,4.45,;-1.02,5.22,;-2.35,4.45,;-2.35,2.91,;-1.02,2.14,;-3.82,2.43,;-4.3,.97,;-3.6,-.4,;-4.97,-1.1,;-5.67,.27,;-5.44,-2.57,;-6.97,-2.77,;-7.76,-4.1,;-7.22,-5.54,;-5.75,-6.01,;-4.47,-5.17,;-4.33,-3.63,;-4.72,3.68,;-6.26,3.68,;-3.82,4.92,;-5.31,5.32,;-2.73,6.01,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N([C@@H]1C[C@@H](C1)N1CC3C(C1)C3(C)C)C(=O)C2(C)C |r,wU:27.30,29.35,(5.18,-1.7,;6.21,-.56,;7.72,-.88,;5.74,.9,;6.64,2.15,;5.74,3.4,;4.27,2.92,;2.94,3.69,;1.6,2.92,;1.6,1.38,;2.94,.61,;2.94,-.93,;1.6,-1.7,;1.6,-3.24,;.27,-4.01,;-1.06,-3.24,;-1.06,-1.7,;.27,-.93,;.27,.61,;4.27,1.38,;.27,3.69,;.27,5.23,;-1.06,6,;-2.4,5.23,;-2.4,3.69,;-1.06,2.92,;-3.86,3.21,;-4.34,1.75,;-5.71,1.05,;-5.01,-.32,;-3.64,.38,;-5.49,-1.79,;-6.95,-2.26,;-6.95,-3.8,;-5.49,-4.28,;-4.58,-3.03,;-6.63,-5.31,;-6.23,-6.8,;-7.72,-6.4,;-4.77,4.46,;-6.31,4.46,;-3.86,5.71,;-5.35,6.11,;-2.77,6.8,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N([C@@H]1C[C@@H](C1)N1CC3CC3C1)C(=O)C2(C)C |r,wU:27.30,29.35,(4.8,-2.65,;5.83,-1.51,;7.33,-1.83,;5.35,-.04,;6.26,1.2,;5.35,2.45,;3.89,1.97,;2.55,2.74,;1.22,1.97,;1.22,.43,;2.55,-.34,;2.55,-1.88,;1.22,-2.65,;1.22,-4.19,;-.11,-4.96,;-1.45,-4.19,;-1.45,-2.65,;-.11,-1.88,;-.11,-.34,;3.89,.43,;-.11,2.74,;-.11,4.28,;-1.45,5.05,;-2.78,4.28,;-2.78,2.74,;-1.45,1.97,;-4.25,2.27,;-4.72,.8,;-6.09,.1,;-5.39,-1.27,;-4.02,-.57,;-5.87,-2.73,;-7.33,-3.21,;-7.33,-4.75,;-7.01,-6.26,;-5.87,-5.23,;-4.96,-3.98,;-5.15,3.51,;-6.69,3.51,;-4.25,4.76,;-5.42,5.76,;-3.89,6.26,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N([C@H]1C[C@H](C1)N1CC3CCC(C3)C1)C(=O)C2(C)C |r,wU:27.30,29.35,(5.06,-2.95,;6.09,-1.8,;7.59,-2.12,;5.61,-.34,;6.52,.91,;5.61,2.15,;4.15,1.68,;2.81,2.45,;1.48,1.68,;1.48,.14,;2.81,-.63,;2.81,-2.17,;1.48,-2.94,;1.48,-4.48,;.15,-5.25,;-1.19,-4.48,;-1.19,-2.94,;.15,-2.17,;.15,-.63,;4.15,.14,;.15,2.45,;.15,3.99,;-1.19,4.76,;-2.52,3.99,;-2.52,2.45,;-1.19,1.68,;-3.99,1.97,;-4.46,.51,;-3.76,-.87,;-5.14,-1.57,;-5.83,-.19,;-5.61,-3.03,;-7.12,-3.35,;-7.59,-4.82,;-6.7,-4.01,;-5.36,-4.43,;-5.06,-5.64,;-6.56,-5.96,;-4.58,-4.17,;-4.89,3.22,;-6.43,3.22,;-3.99,4.46,;-5.16,5.46,;-3.63,5.96,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N([C@H]1C[C@H](C1)N1CCCCC1)C(=O)C2(C)C |r,wU:27.30,29.35,(5.79,-2.2,;6.82,-1.05,;8.33,-1.37,;6.34,.41,;7.25,1.66,;6.34,2.91,;4.88,2.43,;3.55,3.2,;2.21,2.43,;2.21,.89,;3.55,.12,;3.55,-1.42,;2.21,-2.19,;2.21,-3.73,;.88,-4.5,;-.46,-3.73,;-.46,-2.19,;.88,-1.42,;.88,.12,;4.88,.89,;.88,3.2,;.88,4.74,;-.46,5.51,;-1.79,4.74,;-1.79,3.2,;-.46,2.43,;-3.25,2.72,;-3.73,1.26,;-3.03,-.11,;-4.4,-.81,;-5.1,.56,;-4.88,-2.28,;-6.39,-2.6,;-6.86,-4.06,;-5.83,-5.21,;-4.32,-4.89,;-3.85,-3.42,;-4.16,3.97,;-5.7,3.97,;-3.25,5.22,;-4.43,6.22,;-2.89,6.71,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N([C@@H]1C[C@@H](C1)NCC(C)(C)F)C(=O)C2(C)C |r,wU:27.30,29.35,(5.79,-2.95,;6.82,-1.8,;8.33,-2.12,;6.34,-.34,;7.25,.91,;6.34,2.15,;4.88,1.68,;3.55,2.45,;2.21,1.68,;2.21,.14,;3.55,-.63,;3.55,-2.17,;2.21,-2.94,;2.21,-4.48,;.88,-5.25,;-.46,-4.48,;-.46,-2.94,;.88,-2.17,;.88,-.63,;4.88,.14,;.88,2.45,;.88,3.99,;-.46,4.76,;-1.79,3.99,;-1.79,2.45,;-.46,1.68,;-3.25,1.97,;-3.73,.51,;-5.1,-.19,;-4.4,-1.57,;-3.03,-.87,;-4.88,-3.03,;-6.39,-3.35,;-6.86,-4.82,;-8.33,-4.34,;-8.01,-5.85,;-5.83,-5.96,;-4.16,3.22,;-5.7,3.22,;-3.25,4.46,;-4.43,5.46,;-2.89,5.96,)|
CC(C)n1cnc2cc(nc(Nc3c(F)cncc3F)c12)-c1ccc2c(c1)N([C@H]1C[C@H](C1)N1CCCCC1)C(=O)C2(C)C |r,wU:28.31,30.36,(5.06,-2.95,;6.09,-1.8,;7.59,-2.12,;5.61,-.34,;6.52,.91,;5.61,2.15,;4.15,1.68,;2.81,2.45,;1.48,1.68,;1.48,.14,;2.81,-.63,;2.81,-2.17,;1.48,-2.94,;.15,-2.17,;.15,-.63,;-1.19,-2.94,;-1.19,-4.48,;.15,-5.25,;1.48,-4.48,;2.81,-5.25,;4.15,.14,;.15,2.45,;.15,3.99,;-1.19,4.76,;-2.52,3.99,;-2.52,2.45,;-1.19,1.68,;-3.99,1.97,;-4.46,.51,;-3.76,-.87,;-5.14,-1.57,;-5.83,-.19,;-5.61,-3.03,;-7.12,-3.35,;-7.59,-4.82,;-6.56,-5.96,;-5.06,-5.64,;-4.58,-4.17,;-4.89,3.22,;-6.43,3.22,;-3.99,4.46,;-5.16,5.46,;-3.63,5.96,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N([C@@H]1C[C@@H](C1)N1C[C@H]3CC[C@@H]1C3)C(=O)C2(C)C |r,wU:27.30,29.35,wD:36.42,33.43,(5.06,-2.95,;6.09,-1.8,;7.59,-2.12,;5.61,-.34,;6.52,.91,;5.61,2.15,;4.15,1.68,;2.81,2.45,;1.48,1.68,;1.48,.14,;2.81,-.63,;2.81,-2.17,;1.48,-2.94,;1.48,-4.48,;.15,-5.25,;-1.19,-4.48,;-1.19,-2.94,;.15,-2.17,;.15,-.63,;4.15,.14,;.15,2.45,;.15,3.99,;-1.19,4.76,;-2.52,3.99,;-2.52,2.45,;-1.19,1.68,;-3.99,1.97,;-4.46,.51,;-5.83,-.19,;-5.14,-1.57,;-3.76,-.87,;-5.61,-3.03,;-4.58,-4.17,;-5.06,-5.64,;-6.56,-5.96,;-7.59,-4.82,;-7.12,-3.35,;-6.35,-4.68,;-4.89,3.22,;-6.43,3.22,;-3.99,4.46,;-5.16,5.46,;-3.63,5.96,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N(C1CC(C1)N1CCCCC1)C(=O)C21CCN(CC1)C(C)=O |(-7.45,6.11,;-5.94,5.79,;-4.91,6.94,;-5.47,4.33,;-6.37,3.08,;-5.47,1.83,;-4,2.31,;-2.67,1.54,;-1.33,2.31,;-1.33,3.85,;-2.67,4.62,;-2.67,6.16,;-1.33,6.93,;-1.33,8.47,;,9.24,;1.33,8.47,;1.33,6.93,;,6.16,;,4.62,;-4,3.85,;,1.54,;1.33,2.31,;2.67,1.54,;2.67,,;1.33,-.77,;;1.65,-2.28,;.62,-3.42,;.7,-4.96,;-.83,-5.04,;-.91,-3.5,;-1.86,-6.18,;-1.39,-7.65,;-2.42,-8.79,;-3.93,-8.47,;-4.4,-7.01,;-3.37,-5.86,;3.19,-2.44,;3.96,-3.77,;3.81,-1.03,;4.84,-2.17,;6.35,-1.85,;6.82,-.39,;5.79,.75,;4.29,.43,;8.33,-.07,;8.81,1.39,;9.36,-1.21,)|
CC(C)n1cnc2cc(nc(Nc3ccc(F)nc3F)c12)-c1ccc2c(c1)N([C@H]1C[C@H](C1)N1CCCCC1)C(=O)C21CCN(CC1)C(=O)[C@@H](C)O |r,wU:28.31,30.36,48.57,(5.24,-5.29,;6.27,-4.14,;7.77,-4.47,;5.79,-2.68,;6.7,-1.43,;5.79,-.19,;4.33,-.66,;2.99,.11,;1.66,-.66,;1.66,-2.2,;2.99,-2.97,;2.99,-4.51,;1.66,-5.28,;1.66,-6.82,;.32,-7.59,;-1.01,-6.82,;-2.34,-7.59,;-1.01,-5.28,;.32,-4.51,;.32,-2.97,;4.33,-2.2,;.32,.11,;.32,1.65,;-1.01,2.42,;-2.34,1.65,;-2.34,.11,;-1.01,-.66,;-3.81,-.37,;-4.28,-1.83,;-3.58,-3.21,;-4.96,-3.91,;-5.66,-2.53,;-5.43,-5.37,;-6.94,-5.69,;-7.41,-7.16,;-6.38,-8.3,;-4.88,-7.98,;-4.4,-6.52,;-4.71,.88,;-6.25,.88,;-3.81,2.12,;-2.78,3.27,;-3.25,4.73,;-4.76,5.05,;-5.79,3.91,;-5.31,2.44,;-5.24,6.52,;-4.2,7.66,;-6.74,6.84,;-7.77,5.69,;-7.22,8.3,)|
CC(C)n1cnc2cc(nc(Nc3ncc(F)cc3F)c12)-c1ccc2c(c1)N([C@H]1C[C@H](C1)N1CCCCC1)C(=O)C21CCN(CC1)C(C)=O |r,wU:28.31,30.36,(5.06,-4.97,;6.09,-3.82,;7.59,-4.14,;5.61,-2.36,;6.52,-1.11,;5.61,.13,;4.15,-.34,;2.81,.43,;1.48,-.34,;1.48,-1.88,;2.81,-2.65,;2.81,-4.19,;1.48,-4.96,;1.48,-6.5,;.15,-7.27,;-1.19,-6.5,;-2.52,-7.27,;-1.19,-4.96,;.15,-4.19,;.15,-2.65,;4.15,-1.88,;.15,.43,;.15,1.97,;-1.19,2.74,;-2.52,1.97,;-2.52,.43,;-1.19,-.34,;-3.99,-.05,;-4.46,-1.51,;-3.76,-2.89,;-5.14,-3.59,;-5.83,-2.21,;-5.61,-5.05,;-7.12,-5.37,;-7.59,-6.84,;-6.56,-7.98,;-5.06,-7.66,;-4.58,-6.2,;-4.89,1.2,;-6.43,1.2,;-3.99,2.44,;-2.96,3.59,;-3.43,5.05,;-4.94,5.37,;-5.97,4.23,;-5.49,2.76,;-5.41,6.84,;-6.92,7.16,;-4.38,7.98,)|
CC(C)n1cnc2cc(nc(Nc3ccc(F)nc3F)c12)-c1ccc2c(c1)N([C@H]1C[C@H](C1)N1CCCCC1)C(=O)C21CCN(CC1)C(C)=O |r,wU:28.31,30.36,(5.06,-4.97,;6.09,-3.82,;7.59,-4.14,;5.61,-2.36,;6.52,-1.11,;5.61,.13,;4.15,-.34,;2.81,.43,;1.48,-.34,;1.48,-1.88,;2.81,-2.65,;2.81,-4.19,;1.48,-4.96,;1.48,-6.5,;.15,-7.27,;-1.19,-6.5,;-2.52,-7.27,;-1.19,-4.96,;.15,-4.19,;.15,-2.65,;4.15,-1.88,;.15,.43,;.15,1.97,;-1.19,2.74,;-2.52,1.97,;-2.52,.43,;-1.19,-.34,;-3.99,-.05,;-4.46,-1.51,;-3.76,-2.89,;-5.14,-3.59,;-5.83,-2.21,;-5.61,-5.05,;-7.12,-5.37,;-7.59,-6.84,;-6.56,-7.98,;-5.06,-7.66,;-4.58,-6.2,;-4.89,1.2,;-6.43,1.2,;-3.99,2.44,;-2.96,3.59,;-3.43,5.05,;-4.94,5.37,;-5.97,4.23,;-5.49,2.76,;-5.41,6.84,;-6.92,7.16,;-4.38,7.98,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N([C@@H]1C[C@@H](C1)N1CCC(C)(C)C1)C(=O)C21CCOCC1 |r,wU:27.30,29.35,(5.57,-3.38,;6.6,-2.23,;8.1,-2.55,;6.12,-.77,;7.03,.48,;6.12,1.72,;4.66,1.25,;3.32,2.02,;1.99,1.25,;1.99,-.29,;3.32,-1.06,;3.32,-2.6,;1.99,-3.37,;1.99,-4.91,;.66,-5.68,;-.68,-4.91,;-.68,-3.37,;.66,-2.6,;.66,-1.06,;4.66,-.29,;.66,2.02,;.66,3.56,;-.68,4.33,;-2.01,3.56,;-2.01,2.02,;-.68,1.25,;-3.48,1.54,;-3.95,.08,;-5.32,-.62,;-4.62,-1.99,;-3.25,-1.3,;-5.1,-3.46,;-4.19,-4.7,;-5.1,-5.95,;-6.56,-5.47,;-8.1,-5.47,;-6.96,-6.96,;-6.56,-3.93,;-4.38,2.79,;-5.92,2.79,;-3.48,4.03,;-2.44,5.18,;-2.92,6.64,;-4.43,6.96,;-5.46,5.82,;-4.98,4.35,)|
CC[C@H](C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N([C@H]1C[C@H](C1)N1CCCCC1)C(=O)C21CCN(CC1)C(C)=O |r,wU:28.31,30.36,wD:2.2,(8.11,-3,;7.08,-4.14,;5.57,-3.82,;4.54,-4.97,;5.1,-2.36,;6,-1.11,;5.1,.13,;3.63,-.34,;2.3,.43,;.96,-.34,;.96,-1.88,;2.3,-2.65,;2.3,-4.19,;.96,-4.96,;.96,-6.5,;-.37,-7.27,;-1.7,-6.5,;-1.7,-4.96,;-.37,-4.19,;-.37,-2.65,;3.63,-1.88,;-.37,.43,;-.37,1.97,;-1.7,2.74,;-3.04,1.97,;-3.04,.43,;-1.7,-.34,;-4.5,-.05,;-4.98,-1.51,;-4.28,-2.89,;-5.65,-3.59,;-6.35,-2.21,;-6.13,-5.05,;-7.63,-5.37,;-8.11,-6.84,;-7.08,-7.98,;-5.57,-7.66,;-5.1,-6.2,;-5.41,1.2,;-6.95,1.2,;-4.5,2.44,;-3.47,3.59,;-3.95,5.05,;-5.45,5.37,;-6.48,4.23,;-6.01,2.76,;-5.93,6.84,;-7.44,7.16,;-4.9,7.98,)|
CCn1cnc2cc(nc(Nc3ccc(F)nc3F)c12)-c1ccc2c(c1)N([C@H]1C[C@H](C1)N1CCCCC1)C(=O)C21CCN(CC1)C(=O)[C@@H](C)O |r,wU:27.30,29.35,47.56,(7.77,-4.47,;6.27,-4.14,;5.79,-2.68,;6.7,-1.43,;5.79,-.19,;4.33,-.66,;2.99,.11,;1.66,-.66,;1.66,-2.2,;2.99,-2.97,;2.99,-4.51,;1.66,-5.28,;1.66,-6.82,;.32,-7.59,;-1.01,-6.82,;-2.34,-7.59,;-1.01,-5.28,;.32,-4.51,;.32,-2.97,;4.33,-2.2,;.32,.11,;.32,1.65,;-1.01,2.42,;-2.34,1.65,;-2.34,.11,;-1.01,-.66,;-3.81,-.37,;-4.28,-1.83,;-3.58,-3.21,;-4.96,-3.91,;-5.66,-2.53,;-5.43,-5.37,;-6.94,-5.69,;-7.41,-7.16,;-6.38,-8.3,;-4.88,-7.98,;-4.4,-6.52,;-4.71,.88,;-6.25,.88,;-3.81,2.12,;-2.78,3.27,;-3.25,4.73,;-4.76,5.05,;-5.79,3.91,;-5.31,2.44,;-5.24,6.52,;-4.2,7.66,;-6.74,6.84,;-7.77,5.69,;-7.22,8.3,)|
CC(C)NC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C32CCN(CC2)C(C)=O)c(F)cn1 |r,wU:29.31,31.36,(-2.52,-9.94,;-1.19,-9.17,;.15,-9.94,;-1.19,-7.63,;.15,-6.86,;1.48,-7.63,;.15,-5.32,;1.48,-4.55,;1.48,-3.01,;2.81,-2.24,;2.81,-.7,;1.48,.07,;1.48,1.61,;2.81,2.38,;4.15,1.61,;5.61,2.09,;6.52,.84,;5.61,-.4,;6.09,-1.87,;5.06,-3.01,;7.59,-2.19,;4.15,.07,;.15,2.38,;.15,3.92,;-1.19,4.69,;-2.52,3.92,;-2.52,2.38,;-1.19,1.61,;-3.99,1.91,;-4.46,.44,;-3.76,-.93,;-5.14,-1.63,;-5.83,-.26,;-5.61,-3.09,;-7.12,-3.41,;-7.59,-4.88,;-6.56,-6.02,;-5.06,-5.7,;-4.58,-4.24,;-4.89,3.15,;-6.43,3.15,;-3.99,4.4,;-2.96,5.54,;-3.43,7.01,;-4.94,7.33,;-5.97,6.18,;-5.49,4.72,;-5.41,8.79,;-6.92,9.11,;-4.38,9.94,;.15,-2.24,;.15,-.7,;-1.19,-3.01,;-1.19,-4.55,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N([C@@H]1C[C@@H](C1)N1CCC(C)(C)C1)C(=O)C21CCN(CC1)C1COC1 |r,wU:27.30,29.35,(5.46,-5.15,;6.5,-4,;8,-4.32,;6.02,-2.54,;6.92,-1.29,;6.02,-.04,;4.55,-.52,;3.22,.25,;1.89,-.52,;1.89,-2.06,;3.22,-2.83,;3.22,-4.37,;1.89,-5.14,;1.89,-6.68,;.55,-7.45,;-.78,-6.68,;-.78,-5.14,;.55,-4.37,;.55,-2.83,;4.55,-2.06,;.55,.25,;.55,1.79,;-.78,2.56,;-2.11,1.79,;-2.11,.25,;-.78,-.52,;-3.58,-.23,;-4.05,-1.69,;-5.43,-2.39,;-4.73,-3.76,;-3.36,-3.06,;-5.2,-5.23,;-4.3,-6.47,;-5.2,-7.72,;-6.67,-7.24,;-8,-8.01,;-6.27,-8.73,;-6.67,-5.7,;-4.48,1.02,;-6.02,1.02,;-3.58,2.27,;-2.55,3.41,;-3.02,4.87,;-4.53,5.19,;-5.56,4.05,;-5.08,2.59,;-5.01,6.66,;-4.31,8.03,;-5.68,8.73,;-6.38,7.36,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N([C@@H]1C[C@@H](C1)N1CCC(C)(C)C1)C(=O)C21CCN(CC1)C(=O)C1COC1 |r,wU:27.30,29.35,(5.79,-4.89,;6.82,-3.75,;8.32,-4.07,;6.34,-2.28,;7.25,-1.03,;6.34,.21,;4.88,-.26,;3.54,.51,;2.21,-.26,;2.21,-1.8,;3.54,-2.57,;3.54,-4.11,;2.21,-4.88,;2.21,-6.42,;.87,-7.19,;-.46,-6.42,;-.46,-4.88,;.87,-4.11,;.87,-2.57,;4.88,-1.8,;.87,.51,;.87,2.05,;-.46,2.82,;-1.79,2.05,;-1.79,.51,;-.46,-.26,;-3.26,.03,;-3.73,-1.44,;-5.11,-2.13,;-4.41,-3.51,;-3.03,-2.81,;-4.88,-4.97,;-3.98,-6.22,;-4.88,-7.46,;-6.35,-6.99,;-7.83,-7.39,;-6.35,-8.53,;-6.35,-5.45,;-4.16,1.28,;-5.7,1.28,;-3.26,2.52,;-2.23,3.67,;-2.7,5.13,;-4.21,5.45,;-5.24,4.31,;-4.76,2.84,;-4.69,6.92,;-3.65,8.06,;-6.19,7.24,;-7.03,8.53,;-8.32,7.69,;-7.48,6.4,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N([C@@H]1C[C@@H](C1)N1CCC(C)(C)C1)C(=O)C21CCN(CC1)C(=O)C1(C)COC1 |r,wU:27.30,29.35,(5.79,-4.89,;6.82,-3.75,;8.32,-4.07,;6.34,-2.28,;7.25,-1.03,;6.34,.21,;4.88,-.26,;3.54,.51,;2.21,-.26,;2.21,-1.8,;3.54,-2.57,;3.54,-4.11,;2.21,-4.88,;2.21,-6.42,;.87,-7.19,;-.46,-6.42,;-.46,-4.88,;.87,-4.11,;.87,-2.57,;4.88,-1.8,;.87,.51,;.87,2.05,;-.46,2.82,;-1.79,2.05,;-1.79,.51,;-.46,-.26,;-3.26,.03,;-3.73,-1.44,;-5.11,-2.13,;-4.41,-3.51,;-3.03,-2.81,;-4.88,-4.97,;-3.98,-6.22,;-4.88,-7.46,;-6.35,-6.99,;-6.35,-8.53,;-7.83,-7.39,;-6.35,-5.45,;-4.16,1.28,;-5.7,1.28,;-3.26,2.52,;-2.23,3.67,;-2.7,5.13,;-4.21,5.45,;-5.24,4.31,;-4.76,2.84,;-4.69,6.92,;-3.65,8.06,;-6.19,7.24,;-5.32,8.5,;-7.03,8.53,;-8.32,7.69,;-7.48,6.4,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N([C@@H]1C[C@@H](C1)N1CCC(C)(C)C1)C(=O)C21CCN(CC1)C(=O)C1COC1 |r,wU:27.30,29.35,(5.79,-4.89,;6.82,-3.75,;8.32,-4.07,;6.34,-2.28,;7.25,-1.03,;6.34,.21,;4.88,-.26,;3.54,.51,;2.21,-.26,;2.21,-1.8,;3.54,-2.57,;3.54,-4.11,;2.21,-4.88,;2.21,-6.42,;.87,-7.19,;-.46,-6.42,;-.46,-4.88,;.87,-4.11,;.87,-2.57,;4.88,-1.8,;.87,.51,;.87,2.05,;-.46,2.82,;-1.79,2.05,;-1.79,.51,;-.46,-.26,;-3.26,.03,;-3.73,-1.44,;-5.11,-2.13,;-4.41,-3.51,;-3.03,-2.81,;-4.88,-4.97,;-3.98,-6.22,;-4.88,-7.46,;-6.35,-6.99,;-6.35,-8.53,;-7.83,-7.39,;-6.35,-5.45,;-4.16,1.28,;-5.7,1.28,;-3.26,2.52,;-2.23,3.67,;-2.7,5.13,;-4.21,5.45,;-5.24,4.31,;-4.76,2.84,;-4.69,6.92,;-3.65,8.06,;-6.19,7.24,;-7.03,8.53,;-8.32,7.69,;-7.48,6.4,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N([C@@H]1C[C@@H](C1)N1CCC(C)(C)C1)C(=O)C21CCN(CC1)C(=O)[C@@H]1CCO1 |r,wU:27.30,29.35,wD:48.55,(-.37,-4.07,;-1.88,-3.75,;-2.91,-4.89,;-2.36,-2.28,;-1.45,-1.03,;-2.36,.21,;-3.82,-.26,;-5.15,.51,;-6.49,-.26,;-6.49,-1.8,;-5.15,-2.57,;-5.15,-4.11,;-6.49,-4.88,;-6.49,-6.42,;-7.82,-7.19,;-9.15,-6.42,;-9.15,-4.88,;-7.82,-4.11,;-7.82,-2.57,;-3.82,-1.8,;-7.82,.51,;-7.82,2.05,;-9.15,2.82,;-10.49,2.05,;-10.49,.51,;-9.15,-.26,;-11.95,.03,;-12.43,-1.44,;-13.8,-2.13,;-13.1,-3.51,;-11.73,-2.81,;-13.58,-4.97,;-12.67,-6.22,;-13.58,-7.46,;-15.04,-6.99,;-16.58,-6.99,;-15.04,-8.53,;-15.04,-5.45,;-12.86,1.28,;-14.4,1.28,;-11.95,2.52,;-10.92,3.67,;-11.4,5.13,;-12.9,5.45,;-13.94,4.31,;-13.46,2.84,;-13.38,6.92,;-12.35,8.06,;-14.89,7.24,;-16.18,6.4,;-17.02,7.69,;-15.73,8.53,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N([C@@H]1C[C@@H](C1)N1CCC(C)(C)C1)C(=O)C21CCN(CC1)C(=O)[C@H]1CCO1 |r,wU:27.30,29.35,48.55,(17.02,-4.07,;15.51,-3.75,;14.48,-4.89,;15.04,-2.28,;15.94,-1.03,;15.04,.21,;13.57,-.26,;12.24,.51,;10.9,-.26,;10.9,-1.8,;12.24,-2.57,;12.24,-4.11,;10.9,-4.88,;10.9,-6.42,;9.57,-7.19,;8.24,-6.42,;8.24,-4.88,;9.57,-4.11,;9.57,-2.57,;13.57,-1.8,;9.57,.51,;9.57,2.05,;8.24,2.82,;6.9,2.05,;6.9,.51,;8.24,-.26,;5.44,.03,;4.96,-1.44,;3.59,-2.13,;4.29,-3.51,;5.66,-2.81,;3.81,-4.97,;4.72,-6.22,;3.81,-7.46,;2.35,-6.99,;.81,-6.99,;2.35,-8.53,;2.35,-5.45,;4.53,1.28,;2.99,1.28,;5.44,2.52,;6.47,3.67,;5.99,5.13,;4.49,5.45,;3.46,4.31,;3.93,2.84,;4.01,6.92,;5.04,8.06,;2.5,7.24,;1.21,6.4,;.37,7.69,;1.66,8.53,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N([C@H]1C[C@H](C1)N1CCC[C@@H](F)C1)C(=O)C21CCN(CC1)C1COC1 |r,wU:27.30,29.35,35.40,(5.81,-5.43,;6.84,-4.29,;8.35,-4.61,;6.36,-2.82,;7.27,-1.58,;6.36,-.33,;4.9,-.81,;3.57,-.04,;2.23,-.81,;2.23,-2.35,;3.57,-3.12,;3.57,-4.66,;2.23,-5.43,;2.23,-6.97,;.9,-7.74,;-.43,-6.97,;-.43,-5.43,;.9,-4.66,;.9,-3.12,;4.9,-2.35,;.9,-.04,;.9,1.5,;-.43,2.27,;-1.77,1.5,;-1.77,-.04,;-.43,-.81,;-3.23,-.51,;-3.71,-1.98,;-3.01,-3.35,;-4.38,-4.05,;-5.08,-2.68,;-4.86,-5.51,;-3.83,-6.66,;-4.3,-8.12,;-5.81,-8.44,;-6.84,-7.3,;-8.35,-7.62,;-6.36,-5.83,;-4.14,.73,;-5.68,.73,;-3.23,1.98,;-2.2,3.12,;-2.68,4.59,;-4.19,4.91,;-5.22,3.76,;-4.74,2.3,;-4.66,6.37,;-3.96,7.74,;-5.33,8.44,;-6.03,7.07,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N([C@H]1C[C@H](C1)N1CCCC(C)(F)C1)C(=O)C21CCN(CC1)C1COC1 |r,wU:27.30,29.35,(5.79,-5.43,;6.82,-4.29,;8.33,-4.61,;6.34,-2.82,;7.25,-1.58,;6.34,-.33,;4.88,-.81,;3.55,-.04,;2.21,-.81,;2.21,-2.35,;3.55,-3.12,;3.55,-4.66,;2.21,-5.43,;2.21,-6.97,;.88,-7.74,;-.46,-6.97,;-.46,-5.43,;.88,-4.66,;.88,-3.12,;4.88,-2.35,;.88,-.04,;.88,1.5,;-.46,2.27,;-1.79,1.5,;-1.79,-.04,;-.46,-.81,;-3.25,-.51,;-3.73,-1.98,;-3.03,-3.35,;-4.4,-4.05,;-5.1,-2.68,;-4.88,-5.51,;-3.85,-6.66,;-4.32,-8.12,;-5.83,-8.44,;-6.86,-7.3,;-8.33,-6.82,;-8.01,-8.33,;-6.39,-5.83,;-4.16,.73,;-5.7,.73,;-3.25,1.98,;-2.22,3.12,;-2.7,4.59,;-4.21,4.91,;-5.24,3.76,;-4.76,2.3,;-4.68,6.37,;-3.98,7.74,;-5.35,8.44,;-6.05,7.07,)|
CC(C)n1cnc2cc(nc(Nc3ccc(=O)n(C)c3)c12)-c1ccc2c(c1)N([C@H]1C[C@H](C1)N1CCCC(C)(C)C1)C(=O)C2(C)C |r,wU:28.31,30.36,(5.79,-2.53,;6.82,-1.39,;8.33,-1.71,;6.34,.08,;7.25,1.32,;6.34,2.57,;4.88,2.09,;3.55,2.86,;2.21,2.09,;2.21,.55,;3.55,-.22,;3.55,-1.76,;2.21,-2.53,;.88,-1.76,;-.46,-2.53,;-.46,-4.07,;-1.79,-4.84,;.88,-4.84,;.88,-6.38,;2.21,-4.07,;4.88,.55,;.88,2.86,;.88,4.4,;-.46,5.17,;-1.79,4.4,;-1.79,2.86,;-.46,2.09,;-3.25,2.39,;-3.73,.92,;-3.03,-.45,;-4.4,-1.15,;-5.1,.22,;-4.88,-2.61,;-3.85,-3.76,;-4.32,-5.22,;-5.83,-5.54,;-6.86,-4.4,;-8.33,-3.92,;-8.01,-5.43,;-6.39,-2.93,;-4.16,3.63,;-5.7,3.63,;-3.25,4.88,;-4.43,5.88,;-2.89,6.38,)|
CC(C)n1cnc2cc(nc(Nc3ccc(=O)[nH]c3)c12)-c1ccc2c(c1)N([C@H]1C[C@H](C1)N1CCCC(C)(C)C1)C(=O)C2(C)C |r,wU:27.30,29.35,(5.79,-2.95,;6.82,-1.8,;8.33,-2.12,;6.34,-.34,;7.25,.91,;6.34,2.15,;4.88,1.68,;3.55,2.45,;2.21,1.68,;2.21,.14,;3.55,-.63,;3.55,-2.17,;2.21,-2.94,;.88,-2.17,;-.46,-2.94,;-.46,-4.48,;-1.79,-5.25,;.88,-5.25,;2.21,-4.48,;4.88,.14,;.88,2.45,;.88,3.99,;-.46,4.76,;-1.79,3.99,;-1.79,2.45,;-.46,1.68,;-3.25,1.97,;-3.73,.51,;-3.03,-.87,;-4.4,-1.57,;-5.1,-.19,;-4.88,-3.03,;-3.85,-4.17,;-4.32,-5.64,;-5.83,-5.96,;-6.86,-4.82,;-8.33,-4.34,;-8.01,-5.85,;-6.39,-3.35,;-4.16,3.22,;-5.7,3.22,;-3.25,4.46,;-4.43,5.46,;-2.89,5.96,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N([C@H]1C[C@H](C1)N1CCCCC1)C(=O)C2(C)C |r,wU:27.30,29.35,(5.06,-2.95,;6.09,-1.8,;7.59,-2.12,;5.61,-.34,;6.52,.91,;5.61,2.15,;4.15,1.68,;2.81,2.45,;1.48,1.68,;1.48,.14,;2.81,-.63,;2.81,-2.17,;1.48,-2.94,;1.48,-4.48,;.15,-5.25,;-1.19,-4.48,;-1.19,-2.94,;.15,-2.17,;.15,-.63,;4.15,.14,;.15,2.45,;.15,3.99,;-1.19,4.76,;-2.52,3.99,;-2.52,2.45,;-1.19,1.68,;-3.99,1.97,;-4.46,.51,;-3.76,-.87,;-5.14,-1.57,;-5.83,-.19,;-5.61,-3.03,;-7.12,-3.35,;-7.59,-4.82,;-6.56,-5.96,;-5.06,-5.64,;-4.58,-4.17,;-4.89,3.22,;-6.43,3.22,;-3.99,4.46,;-5.16,5.46,;-3.63,5.96,)|
CC(C)CN[C@H]1C[C@H](C1)N1C(=O)C(C)(C)c2ccc(cc12)-c1cc2ncn(C(C)C)c2c(Nc2ccncc2F)n1 |r,wU:7.9,5.4,(-5.81,-5.96,;-6.84,-4.82,;-8.35,-5.14,;-6.36,-3.35,;-4.86,-3.03,;-4.38,-1.57,;-5.08,-.19,;-3.71,.51,;-3.01,-.87,;-3.23,1.97,;-4.14,3.22,;-5.68,3.22,;-3.23,4.46,;-4.4,5.46,;-2.87,5.96,;-1.77,3.99,;-.43,4.76,;.9,3.99,;.9,2.45,;-.43,1.68,;-1.77,2.45,;2.23,1.68,;3.57,2.45,;4.9,1.68,;6.36,2.15,;7.27,.91,;6.36,-.34,;6.84,-1.8,;5.81,-2.95,;8.35,-2.12,;4.9,.14,;3.57,-.63,;3.57,-2.17,;2.23,-2.94,;2.23,-4.48,;.9,-5.25,;-.43,-4.48,;-.43,-2.94,;.9,-2.17,;.9,-.63,;2.23,.14,)|
CCn1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N([C@@H]1C[C@@H](C1)N1CC(C)(C)C1)C(=O)C2(C)C |r,wU:26.29,28.34,(7.54,-1.81,;6.04,-1.49,;5.56,-.03,;6.47,1.22,;5.56,2.46,;4.1,1.99,;2.76,2.76,;1.43,1.99,;1.43,.45,;2.76,-.32,;2.76,-1.86,;1.43,-2.63,;1.43,-4.17,;.1,-4.94,;-1.24,-4.17,;-1.24,-2.63,;.1,-1.86,;.1,-.32,;4.1,.45,;.1,2.76,;.1,4.3,;-1.24,5.07,;-2.57,4.3,;-2.57,2.76,;-1.24,1.99,;-4.04,2.28,;-4.51,.82,;-5.88,.12,;-5.19,-1.25,;-3.81,-.55,;-5.66,-2.72,;-7.03,-3.42,;-6.33,-4.79,;-5.92,-6.27,;-7.54,-5.74,;-4.96,-4.09,;-4.94,3.53,;-6.48,3.53,;-4.04,4.77,;-5.21,5.77,;-3.68,6.27,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N([C@@H]1C[C@@H](C1)N1CC[C@](C)(F)C1)C(=O)C21CCN(CC1)C1COC1 |r,wU:27.30,29.35,34.39,wD:34.40,(5.54,-5.12,;6.57,-3.97,;8.08,-4.3,;6.1,-2.51,;7,-1.26,;6.1,-.02,;4.63,-.49,;3.3,.28,;1.96,-.49,;1.96,-2.03,;3.3,-2.8,;3.3,-4.34,;1.96,-5.11,;1.96,-6.65,;.63,-7.42,;-.7,-6.65,;-.7,-5.11,;.63,-4.34,;.63,-2.8,;4.63,-2.03,;.63,.28,;.63,1.82,;-.7,2.59,;-2.04,1.82,;-2.04,.28,;-.7,-.49,;-3.5,-.2,;-3.98,-1.66,;-5.35,-2.36,;-4.65,-3.74,;-3.28,-3.04,;-5.13,-5.2,;-4.22,-6.45,;-5.13,-7.69,;-6.59,-7.22,;-6.59,-8.76,;-8.08,-7.62,;-6.59,-5.68,;-4.41,1.05,;-5.95,1.05,;-3.5,2.29,;-2.47,3.44,;-2.95,4.9,;-4.45,5.22,;-5.48,4.08,;-5.01,2.61,;-4.93,6.69,;-4.23,8.06,;-5.6,8.76,;-6.3,7.38,)|
CCn1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N([C@@H]1C[C@@H](C1)N1CCC(C)(C)C1)C(=O)C21CCN(CC1)C1COC1 |r,wU:26.29,28.34,(8.08,-4.32,;6.57,-4,;6.1,-2.54,;7,-1.29,;6.1,-.04,;4.63,-.52,;3.3,.25,;1.96,-.52,;1.96,-2.06,;3.3,-2.83,;3.3,-4.37,;1.96,-5.14,;1.96,-6.68,;.63,-7.45,;-.7,-6.68,;-.7,-5.14,;.63,-4.37,;.63,-2.83,;4.63,-2.06,;.63,.25,;.63,1.79,;-.7,2.56,;-2.04,1.79,;-2.04,.25,;-.7,-.52,;-3.5,-.23,;-3.98,-1.69,;-5.35,-2.39,;-4.65,-3.76,;-3.28,-3.06,;-5.13,-5.23,;-4.22,-6.47,;-5.13,-7.72,;-6.59,-7.24,;-8.08,-7.64,;-6.19,-8.73,;-6.59,-5.7,;-4.41,1.02,;-5.95,1.02,;-3.5,2.27,;-2.47,3.41,;-2.95,4.87,;-4.45,5.19,;-5.48,4.05,;-5.01,2.59,;-4.93,6.66,;-4.23,8.03,;-5.6,8.73,;-6.3,7.36,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C3(C)C)c(F)cn1 |r,wU:27.29,29.34,(-1.19,-7.53,;-1.19,-5.99,;.15,-5.22,;1.48,-5.99,;.15,-3.68,;1.48,-2.91,;1.48,-1.37,;2.81,-.6,;2.81,.94,;1.48,1.71,;1.48,3.25,;2.81,4.02,;4.15,3.25,;5.61,3.72,;6.52,2.48,;5.61,1.23,;6.09,-.23,;5.06,-1.38,;7.59,-.55,;4.15,1.71,;.15,4.02,;.15,5.56,;-1.19,6.33,;-2.52,5.56,;-2.52,4.02,;-1.19,3.25,;-3.99,3.54,;-4.46,2.08,;-3.76,.71,;-5.14,.01,;-5.83,1.38,;-5.61,-1.46,;-7.12,-1.78,;-7.59,-3.24,;-6.56,-4.39,;-5.06,-4.07,;-4.58,-2.6,;-4.89,4.79,;-6.43,4.79,;-3.99,6.03,;-5.16,7.03,;-3.63,7.53,;.15,-.6,;.15,.94,;-1.19,-1.37,;-1.19,-2.91,)|
CC[C@H](C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N([C@H]1C[C@H](C1)N1CCCCC1)C(=O)C21CCN(CC1)C1COC1 |r,wU:28.31,30.36,wD:2.2,(8.11,-3.46,;7.08,-4.61,;5.57,-4.29,;4.54,-5.43,;5.1,-2.82,;6,-1.58,;5.1,-.33,;3.63,-.81,;2.3,-.04,;.96,-.81,;.96,-2.35,;2.3,-3.12,;2.3,-4.66,;.96,-5.43,;.96,-6.97,;-.37,-7.74,;-1.7,-6.97,;-1.7,-5.43,;-.37,-4.66,;-.37,-3.12,;3.63,-2.35,;-.37,-.04,;-.37,1.5,;-1.7,2.27,;-3.04,1.5,;-3.04,-.04,;-1.7,-.81,;-4.5,-.51,;-4.98,-1.98,;-4.28,-3.35,;-5.65,-4.05,;-6.35,-2.68,;-6.13,-5.51,;-7.63,-5.83,;-8.11,-7.3,;-7.08,-8.44,;-5.57,-8.12,;-5.1,-6.66,;-5.41,.73,;-6.95,.73,;-4.5,1.98,;-3.47,3.12,;-3.95,4.59,;-5.45,4.91,;-6.48,3.76,;-6.01,2.3,;-5.93,6.37,;-5.23,7.74,;-6.6,8.44,;-7.3,7.07,)|
CC[C@H](C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N([C@@H]1C[C@@H](C1)N1CCC(C)(C)C1)C(=O)C21CCN(CC1)C1COC1 |r,wU:28.31,30.36,wD:2.2,(8.62,-3.18,;7.59,-4.32,;6.08,-4,;5.05,-5.15,;5.61,-2.54,;6.51,-1.29,;5.61,-.04,;4.14,-.52,;2.81,.25,;1.48,-.52,;1.48,-2.06,;2.81,-2.83,;2.81,-4.37,;1.48,-5.14,;1.48,-6.68,;.14,-7.45,;-1.19,-6.68,;-1.19,-5.14,;.14,-4.37,;.14,-2.83,;4.14,-2.06,;.14,.25,;.14,1.79,;-1.19,2.56,;-2.53,1.79,;-2.53,.25,;-1.19,-.52,;-3.99,-.23,;-4.47,-1.69,;-5.84,-2.39,;-5.14,-3.76,;-3.77,-3.06,;-5.62,-5.23,;-4.71,-6.47,;-5.62,-7.72,;-7.08,-7.24,;-8.62,-7.24,;-7.48,-8.73,;-7.08,-5.7,;-4.9,1.02,;-6.44,1.02,;-3.99,2.27,;-2.96,3.41,;-3.44,4.87,;-4.94,5.19,;-5.97,4.05,;-5.5,2.59,;-5.42,6.66,;-4.72,8.03,;-6.09,8.73,;-6.79,7.36,)|
CC(C)n1cnc2cc(nc(Nc3ccnc(F)c3F)c12)-c1ccc2c(c1)N(C1CC(C1)N1CCCCC1)C(=O)C21CCN(CC1)C1COC1 |(14.97,3.01,;13.44,2.79,;12.87,1.36,;12.49,4,;12.9,5.48,;11.62,6.33,;10.41,5.38,;8.89,5.63,;7.91,4.45,;8.45,3,;9.97,2.75,;10.5,1.3,;9.52,.12,;10.06,-1.33,;9.07,-2.51,;7.56,-2.26,;7.02,-.81,;5.5,-.56,;8,.37,;7.46,1.82,;10.95,3.93,;6.39,4.7,;5.41,3.52,;3.89,3.77,;3.36,5.22,;4.34,6.4,;5.86,6.15,;3.51,7.7,;4.08,9.14,;3.47,10.55,;4.88,11.16,;5.49,9.75,;5.45,12.59,;4.49,13.8,;5.06,15.23,;6.58,15.46,;7.54,14.25,;6.97,12.82,;2.02,7.32,;.83,8.3,;1.92,5.79,;1.99,4.25,;.69,3.42,;-.68,4.14,;-.74,5.67,;.56,6.5,;-1.98,3.31,;-2.31,1.81,;-3.82,2.14,;-3.48,3.65,)|
CC(C)n1cnc2cc(nc(Nc3cc(F)ncc3F)c12)-c1ccc2c(c1)N([C@H]1C[C@H](C1)N1CCCCC1)C(=O)C21CCN(CC1)C1COC1 |r,wU:28.31,30.36,(5.06,-5.02,;6.09,-3.87,;7.59,-4.19,;5.61,-2.41,;6.52,-1.16,;5.61,.09,;4.15,-.39,;2.81,.38,;1.48,-.39,;1.48,-1.93,;2.81,-2.7,;2.81,-4.24,;1.48,-5.01,;1.48,-6.55,;.15,-7.32,;.15,-8.86,;-1.19,-6.55,;-1.19,-5.01,;.15,-4.24,;.15,-2.7,;4.15,-1.93,;.15,.38,;.15,1.92,;-1.19,2.69,;-2.52,1.92,;-2.52,.38,;-1.19,-.39,;-3.99,-.1,;-4.46,-1.56,;-3.76,-2.93,;-5.14,-3.63,;-5.83,-2.26,;-5.61,-5.1,;-7.12,-5.42,;-7.59,-6.88,;-6.56,-8.03,;-5.06,-7.71,;-4.58,-6.24,;-4.89,1.15,;-6.43,1.15,;-3.99,2.4,;-2.96,3.54,;-3.43,5,;-4.94,5.32,;-5.97,4.18,;-5.49,2.72,;-5.41,6.79,;-4.72,8.16,;-6.09,8.86,;-6.79,7.49,)|
CC(C)n1cnc2cc(nc(Nc3ccnc(F)c3F)c12)-c1ccc2c(c1)N([C@@H]1C[C@@H](C1)N1CCC(C)(C)C1)C(=O)C21CCN(CC1)C1COC1 |r,wU:28.31,30.36,(5.54,-5.15,;6.57,-4,;8.08,-4.32,;6.1,-2.54,;7,-1.29,;6.1,-.04,;4.63,-.52,;3.3,.25,;1.96,-.52,;1.96,-2.06,;3.3,-2.83,;3.3,-4.37,;1.96,-5.14,;1.96,-6.68,;.63,-7.45,;-.7,-6.68,;-.7,-5.14,;-2.04,-4.37,;.63,-4.37,;.63,-2.83,;4.63,-2.06,;.63,.25,;.63,1.79,;-.7,2.56,;-2.04,1.79,;-2.04,.25,;-.7,-.52,;-3.5,-.23,;-3.98,-1.69,;-5.35,-2.39,;-4.65,-3.76,;-3.28,-3.06,;-5.13,-5.23,;-4.22,-6.47,;-5.13,-7.72,;-6.59,-7.24,;-8.08,-7.64,;-6.99,-8.73,;-6.59,-5.7,;-4.41,1.02,;-5.95,1.02,;-3.5,2.27,;-2.47,3.41,;-2.95,4.87,;-4.45,5.19,;-5.48,4.05,;-5.01,2.59,;-4.93,6.66,;-4.23,8.03,;-5.6,8.73,;-6.3,7.36,)|
CC(C)n1cnc2cc(nc(Nc3ccnc(F)c3F)c12)-c1ccc2c(c1)N([C@H]1C[C@H](C1)N1CCCCC1)C(=O)C2(C)C |r,wU:28.31,30.36,(5.06,-2.95,;6.09,-1.8,;7.59,-2.12,;5.61,-.34,;6.52,.91,;5.61,2.15,;4.15,1.68,;2.81,2.45,;1.48,1.68,;1.48,.14,;2.81,-.63,;2.81,-2.17,;1.48,-2.94,;1.48,-4.48,;.15,-5.25,;-1.19,-4.48,;-1.19,-2.94,;-2.52,-2.17,;.15,-2.17,;.15,-.63,;4.15,.14,;.15,2.45,;.15,3.99,;-1.19,4.76,;-2.52,3.99,;-2.52,2.45,;-1.19,1.68,;-3.99,1.97,;-4.46,.51,;-3.76,-.87,;-5.14,-1.57,;-5.83,-.19,;-5.61,-3.03,;-7.12,-3.35,;-7.59,-4.82,;-6.56,-5.96,;-5.06,-5.64,;-4.58,-4.17,;-4.89,3.22,;-6.43,3.22,;-3.99,4.46,;-5.16,5.46,;-3.63,5.96,)|
CC(C)n1cnc2cc(nc(Nc3ccnc(F)c3F)c12)-c1cnc2c(c1)N([C@H]1C[C@H](C1)N1CCCCC1)C(=O)C2(C)C |r,wU:28.31,30.36,(5.06,-2.95,;6.09,-1.8,;7.59,-2.12,;5.61,-.34,;6.52,.91,;5.61,2.15,;4.15,1.68,;2.81,2.45,;1.48,1.68,;1.48,.14,;2.81,-.63,;2.81,-2.17,;1.48,-2.94,;1.48,-4.48,;.15,-5.25,;-1.19,-4.48,;-1.19,-2.94,;-2.52,-2.17,;.15,-2.17,;.15,-.63,;4.15,.14,;.15,2.45,;.15,3.99,;-1.19,4.76,;-2.52,3.99,;-2.52,2.45,;-1.19,1.68,;-3.99,1.97,;-4.46,.51,;-3.76,-.87,;-5.14,-1.57,;-5.83,-.19,;-5.61,-3.03,;-7.12,-3.35,;-7.59,-4.82,;-6.56,-5.96,;-5.06,-5.64,;-4.58,-4.17,;-4.89,3.22,;-6.43,3.22,;-3.99,4.46,;-5.16,5.46,;-3.63,5.96,)|
CC(C)n1cnc2cc(nc(Nc3ccc(F)nc3F)c12)-c1ccc2c(c1)N([C@H]1C[C@H](C1)N1CCCCC1)C(=O)C21CCN(CC1)C(=O)C1(C)COC1 |r,wU:28.31,30.36,(5.79,-5.2,;6.82,-4.06,;8.32,-4.38,;6.34,-2.59,;7.25,-1.35,;6.34,-.1,;4.88,-.58,;3.54,.19,;2.21,-.58,;2.21,-2.12,;3.54,-2.89,;3.54,-4.43,;2.21,-5.2,;2.21,-6.74,;.87,-7.51,;-.46,-6.74,;-1.79,-7.51,;-.46,-5.2,;.87,-4.43,;.87,-2.89,;4.88,-2.12,;.87,.19,;.87,1.73,;-.46,2.5,;-1.79,1.73,;-1.79,.19,;-.46,-.58,;-3.26,-.28,;-3.73,-1.75,;-3.03,-3.12,;-4.41,-3.82,;-5.11,-2.45,;-4.88,-5.28,;-6.39,-5.6,;-6.86,-7.07,;-5.83,-8.21,;-4.33,-7.89,;-3.85,-6.43,;-4.16,.96,;-5.7,.96,;-3.26,2.21,;-2.23,3.35,;-2.7,4.82,;-4.21,5.14,;-5.24,3.99,;-4.76,2.53,;-4.69,6.6,;-3.65,7.75,;-6.19,6.92,;-5.32,8.19,;-7.03,8.21,;-8.32,7.37,;-7.48,6.08,)|
COc1cc(F)c(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C32CCN(CC2)C(C)=O)cn1 |r,wU:27.29,29.34,(-2.52,-8.4,;-2.52,-6.86,;-1.19,-6.09,;-1.19,-4.55,;.15,-3.78,;.15,-2.24,;1.48,-4.55,;2.81,-3.78,;2.81,-2.24,;1.48,-1.47,;1.48,.07,;2.81,.84,;4.15,.07,;5.61,.55,;6.52,-.7,;5.61,-1.94,;6.09,-3.41,;5.06,-4.55,;7.59,-3.73,;4.15,-1.47,;.15,.84,;.15,2.38,;-1.19,3.15,;-2.52,2.38,;-2.52,.84,;-1.19,.07,;-3.99,.37,;-4.46,-1.1,;-3.76,-2.47,;-5.14,-3.17,;-5.83,-1.8,;-5.61,-4.63,;-7.12,-4.95,;-7.59,-6.42,;-6.56,-7.56,;-5.06,-7.24,;-4.58,-5.78,;-4.89,1.61,;-6.43,1.61,;-3.99,2.86,;-2.96,4,;-3.43,5.47,;-4.94,5.79,;-5.97,4.64,;-5.49,3.18,;-5.41,7.25,;-6.92,7.57,;-4.38,8.4,;1.48,-6.09,;.15,-6.86,)|
CC(C)n1cnc2cc(nc(Nc3cc(CO)ncc3F)c12)-c1ccc2c(c1)N([C@H]1C[C@H](C1)N1CCCCC1)C(=O)C21CCN(CC1)C(C)=O |r,wU:29.32,31.37,(5.06,-4.17,;6.09,-3.02,;7.59,-3.34,;5.61,-1.56,;6.52,-.31,;5.61,.93,;4.15,.46,;2.81,1.23,;1.48,.46,;1.48,-1.08,;2.81,-1.85,;2.81,-3.39,;1.48,-4.16,;1.48,-5.7,;.15,-6.47,;.15,-8.01,;-1.19,-8.78,;-1.19,-5.7,;-1.19,-4.16,;.15,-3.39,;.15,-1.85,;4.15,-1.08,;.15,1.23,;.15,2.77,;-1.19,3.54,;-2.52,2.77,;-2.52,1.23,;-1.19,.46,;-3.99,.75,;-4.46,-.71,;-3.76,-2.08,;-5.14,-2.78,;-5.83,-1.41,;-5.61,-4.25,;-7.12,-4.57,;-7.59,-6.03,;-6.56,-7.18,;-5.06,-6.86,;-4.58,-5.39,;-4.89,2,;-6.43,2,;-3.99,3.24,;-2.96,4.39,;-3.43,5.85,;-4.94,6.17,;-5.97,5.03,;-5.49,3.56,;-5.41,7.64,;-6.92,7.96,;-4.38,8.78,)|
CC(C)n1cnc2cc(nc(Nc3cc(ncc3F)N(C)C)c12)-c1ccc2c(c1)N([C@H]1C[C@H](C1)N1CCCCC1)C(=O)C21CCN(CC1)C(C)=O |r,wU:30.33,32.38,(5.06,-4.17,;6.09,-3.02,;7.59,-3.34,;5.61,-1.56,;6.52,-.31,;5.61,.93,;4.15,.46,;2.81,1.23,;1.48,.46,;1.48,-1.08,;2.81,-1.85,;2.81,-3.39,;1.48,-4.16,;1.48,-5.7,;.15,-6.47,;-1.19,-5.7,;-1.19,-4.16,;.15,-3.39,;.15,-1.85,;.15,-8.01,;1.48,-8.78,;-1.19,-8.78,;4.15,-1.08,;.15,1.23,;.15,2.77,;-1.19,3.54,;-2.52,2.77,;-2.52,1.23,;-1.19,.46,;-3.99,.75,;-4.46,-.71,;-3.76,-2.08,;-5.14,-2.78,;-5.83,-1.41,;-5.61,-4.25,;-7.12,-4.57,;-7.59,-6.03,;-6.56,-7.18,;-5.06,-6.86,;-4.58,-5.39,;-4.89,2,;-6.43,2,;-3.99,3.24,;-2.96,4.39,;-3.43,5.85,;-4.94,6.17,;-5.97,5.03,;-5.49,3.56,;-5.41,7.64,;-6.92,7.96,;-4.38,8.78,)|
CC(C)n1cnc2cc(nc(Nc3cc(CO)ncc3F)c12)-c1ccc2c(c1)N([C@@H]1C[C@@H](C1)N1CC(C)(C)C1)C(=O)C2(C)C |r,wU:29.32,31.37,(5.01,-2.15,;6.04,-1,;7.54,-1.32,;5.56,.46,;6.47,1.71,;5.56,2.95,;4.1,2.48,;2.76,3.25,;1.43,2.48,;1.43,.94,;2.76,.17,;2.76,-1.37,;1.43,-2.14,;1.43,-3.68,;.1,-4.45,;.1,-5.99,;-1.24,-6.76,;-1.24,-3.68,;-1.24,-2.14,;.1,-1.37,;.1,.17,;4.1,.94,;.1,3.25,;.1,4.79,;-1.24,5.56,;-2.57,4.79,;-2.57,3.25,;-1.24,2.48,;-4.04,2.77,;-4.51,1.31,;-5.88,.61,;-5.19,-.76,;-3.81,-.06,;-5.66,-2.23,;-7.03,-2.93,;-6.33,-4.3,;-5.92,-5.78,;-7.54,-5.25,;-4.96,-3.6,;-4.94,4.02,;-6.48,4.02,;-4.04,5.26,;-5.21,6.26,;-3.68,6.76,)|
CC(C)n1cnc2cc(nc(Nc3ccnc(F)c3F)c12)-c1ccc2c(c1)N([C@H]1C[C@H](C1)N1CCCCC1)C(=O)C2(C)O |r,wU:28.31,30.36,(5.06,-2.95,;6.09,-1.8,;7.59,-2.12,;5.61,-.34,;6.52,.91,;5.61,2.15,;4.15,1.68,;2.81,2.45,;1.48,1.68,;1.48,.14,;2.81,-.63,;2.81,-2.17,;1.48,-2.94,;1.48,-4.48,;.15,-5.25,;-1.19,-4.48,;-1.19,-2.94,;-2.52,-2.17,;.15,-2.17,;.15,-.63,;4.15,.14,;.15,2.45,;.15,3.99,;-1.19,4.76,;-2.52,3.99,;-2.52,2.45,;-1.19,1.68,;-3.99,1.97,;-4.46,.51,;-3.76,-.87,;-5.14,-1.57,;-5.83,-.19,;-5.61,-3.03,;-7.12,-3.35,;-7.59,-4.82,;-6.56,-5.96,;-5.06,-5.64,;-4.58,-4.17,;-4.89,3.22,;-6.43,3.22,;-3.99,4.46,;-3.63,5.96,;-5.16,5.46,)|
CC(C)n1cnc2cc(nc(Nc3ccnc(F)c3F)c12)-c1ccc2c(c1)N([C@H]1C[C@H](C1)N1CCCCC1)C(=O)C21CCN(CC1)C(=O)[C@@H](C)O |r,wU:28.31,30.36,48.57,(5.24,-5.29,;6.27,-4.14,;7.77,-4.47,;5.79,-2.68,;6.7,-1.43,;5.79,-.19,;4.33,-.66,;2.99,.11,;1.66,-.66,;1.66,-2.2,;2.99,-2.97,;2.99,-4.51,;1.66,-5.28,;1.66,-6.82,;.32,-7.59,;-1.01,-6.82,;-1.01,-5.28,;-2.34,-4.51,;.32,-4.51,;.32,-2.97,;4.33,-2.2,;.32,.11,;.32,1.65,;-1.01,2.42,;-2.34,1.65,;-2.34,.11,;-1.01,-.66,;-3.81,-.37,;-4.28,-1.83,;-3.58,-3.21,;-4.96,-3.91,;-5.66,-2.53,;-5.43,-5.37,;-6.94,-5.69,;-7.41,-7.16,;-6.38,-8.3,;-4.88,-7.98,;-4.4,-6.52,;-4.71,.88,;-6.25,.88,;-3.81,2.12,;-2.78,3.27,;-3.25,4.73,;-4.76,5.05,;-5.79,3.91,;-5.31,2.44,;-5.24,6.52,;-4.2,7.66,;-6.74,6.84,;-7.77,5.69,;-7.22,8.3,)|
CC(C)n1cnc2cc(nc(Nc3ccnc(F)c3F)c12)-c1ccc2c(c1)N([C@H]1C[C@H](C1)N1CCCCC1)C(=O)C21CCN(CC1)C(=O)C(C)(C)CO |r,wU:28.31,30.36,(5.71,-5.45,;6.74,-4.31,;8.25,-4.63,;6.27,-2.84,;7.17,-1.59,;6.27,-.35,;4.8,-.82,;3.47,-.05,;2.13,-.82,;2.13,-2.36,;3.47,-3.13,;3.47,-4.67,;2.13,-5.44,;2.13,-6.98,;.8,-7.75,;-.53,-6.98,;-.53,-5.44,;-1.87,-4.67,;.8,-4.67,;.8,-3.13,;4.8,-2.36,;.8,-.05,;.8,1.49,;-.53,2.26,;-1.87,1.49,;-1.87,-.05,;-.53,-.82,;-3.33,-.53,;-3.81,-2,;-3.11,-3.37,;-4.48,-4.07,;-5.18,-2.69,;-4.96,-5.53,;-6.46,-5.85,;-6.94,-7.32,;-5.91,-8.46,;-4.4,-8.14,;-3.93,-6.68,;-4.24,.72,;-5.78,.72,;-3.33,1.96,;-2.3,3.11,;-2.78,4.57,;-4.28,4.89,;-5.31,3.75,;-4.84,2.28,;-4.76,6.36,;-3.73,7.5,;-6.27,6.68,;-6.59,5.17,;-7.73,6.2,;-6.74,8.14,;-8.25,8.46,)|
CNC(=O)c1ccc(F)c(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C3(C)C)n1 |r,wU:30.32,32.37,(1.48,-7.53,;1.48,-5.99,;.15,-5.22,;-1.19,-5.99,;.15,-3.68,;-1.19,-2.91,;-1.19,-1.37,;.15,-.6,;.15,.94,;1.48,-1.37,;2.81,-.6,;2.81,.94,;1.48,1.71,;1.48,3.25,;2.81,4.02,;4.15,3.25,;5.61,3.72,;6.52,2.48,;5.61,1.23,;6.09,-.23,;5.06,-1.38,;7.59,-.55,;4.15,1.71,;.15,4.02,;.15,5.56,;-1.19,6.33,;-2.52,5.56,;-2.52,4.02,;-1.19,3.25,;-3.99,3.54,;-4.46,2.08,;-3.76,.71,;-5.14,.01,;-5.83,1.38,;-5.61,-1.46,;-7.12,-1.78,;-7.59,-3.24,;-6.56,-4.39,;-5.06,-4.07,;-4.58,-2.6,;-4.89,4.79,;-6.43,4.79,;-3.99,6.03,;-5.16,7.03,;-3.63,7.53,;1.48,-2.91,)|
CC(C)n1cnc2cc(nc(Nc3cc4ccncc4cc3F)c12)-c1ccc2c(c1)N(C1CC(C1)N1CCCCC1)C(=O)C21CCN(CC1)C(C)=O |(-7.45,6.11,;-5.94,5.79,;-4.91,6.94,;-5.47,4.33,;-6.37,3.08,;-5.47,1.83,;-4,2.31,;-2.67,1.54,;-1.33,2.31,;-1.33,3.85,;-2.67,4.62,;-2.67,6.16,;-1.33,6.93,;,6.16,;1.33,6.93,;2.67,6.16,;4,6.93,;4,8.47,;2.67,9.24,;1.33,8.47,;,9.24,;-1.33,8.47,;-2.67,9.24,;-4,3.85,;,1.54,;1.33,2.31,;2.67,1.54,;2.67,,;1.33,-.77,;;1.65,-2.28,;.62,-3.42,;.7,-4.96,;-.83,-5.04,;-.91,-3.5,;-1.86,-6.18,;-1.39,-7.65,;-2.42,-8.79,;-3.93,-8.47,;-4.4,-7.01,;-3.37,-5.86,;3.19,-2.44,;3.96,-3.77,;3.81,-1.03,;4.84,-2.17,;6.35,-1.85,;6.82,-.39,;5.79,.75,;4.29,.43,;8.33,-.07,;8.81,1.39,;9.36,-1.21,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N(C1CC(C1)N1CCCCC1)C(=O)C21CCN(CC1)C(=O)C(C)(C)CO |(14.97,3.01,;13.44,2.79,;12.87,1.36,;12.49,4,;12.9,5.48,;11.62,6.33,;10.41,5.38,;8.89,5.63,;7.91,4.45,;8.45,3,;9.97,2.75,;10.5,1.3,;9.52,.12,;10.06,-1.33,;9.07,-2.51,;7.56,-2.26,;7.02,-.81,;8,.37,;7.46,1.82,;10.95,3.93,;6.39,4.7,;5.41,3.52,;3.89,3.77,;3.36,5.22,;4.34,6.4,;5.86,6.15,;3.51,7.7,;4.08,9.14,;3.47,10.55,;4.88,11.16,;5.49,9.75,;5.45,12.59,;4.49,13.8,;5.06,15.23,;6.58,15.46,;7.54,14.25,;6.97,12.82,;2.02,7.32,;.83,8.3,;1.92,5.79,;1.99,4.25,;.69,3.42,;-.68,4.14,;-.74,5.67,;.56,6.5,;-1.98,3.31,;-1.91,1.77,;-3.34,4.03,;-2.63,5.39,;-4.06,2.66,;-4.71,4.74,;-6.01,3.91,)|
COC1(CCC1)C(=O)N1CCC2(CC1)C(=O)N(C1CC(C1)N1CCCCC1)c1cc(ccc21)-c1cc2ncn(C(C)C)c2c(Nc2ccncc2F)n1 |(-6.01,3.91,;-4.64,3.2,;-3.34,4.03,;-4.11,5.36,;-3.31,6.28,;-2.28,5.14,;-1.98,3.31,;-1.91,1.77,;-.68,4.14,;.69,3.42,;1.99,4.25,;1.92,5.79,;.56,6.5,;-.74,5.67,;2.02,7.32,;.83,8.3,;3.51,7.7,;4.08,9.14,;3.47,10.55,;4.88,11.16,;5.49,9.75,;5.45,12.59,;4.49,13.8,;5.06,15.23,;6.58,15.46,;7.54,14.25,;6.97,12.82,;4.34,6.4,;5.86,6.15,;6.39,4.7,;5.41,3.52,;3.89,3.77,;3.36,5.22,;7.91,4.45,;8.89,5.63,;10.41,5.38,;11.62,6.33,;12.9,5.48,;12.49,4,;13.44,2.79,;14.97,3.01,;12.87,1.36,;10.95,3.93,;9.97,2.75,;10.5,1.3,;9.52,.12,;10.06,-1.33,;9.07,-2.51,;7.56,-2.26,;7.02,-.81,;8,.37,;7.46,1.82,;8.45,3,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N(C1CC(C1)N1CCCC(C)(C)C1)C(=O)C21CCN(CC1)C(=O)C1CCO1 |(14.97,3.01,;13.44,2.79,;12.87,1.36,;12.49,4,;12.9,5.48,;11.62,6.33,;10.41,5.38,;8.89,5.63,;7.91,4.45,;8.45,3,;9.97,2.75,;10.5,1.3,;9.52,.12,;10.06,-1.33,;9.07,-2.51,;7.56,-2.26,;7.02,-.81,;8,.37,;7.46,1.82,;10.95,3.93,;6.39,4.7,;5.41,3.52,;3.89,3.77,;3.36,5.22,;4.34,6.4,;5.86,6.15,;3.51,7.7,;4.08,9.14,;3.47,10.55,;4.88,11.16,;5.49,9.75,;5.45,12.59,;6.97,12.82,;7.54,14.25,;6.58,15.46,;5.06,15.23,;4.11,16.44,;5.22,16.76,;4.49,13.8,;2.02,7.32,;.83,8.3,;1.92,5.79,;1.99,4.25,;.69,3.42,;-.68,4.14,;-.74,5.67,;.56,6.5,;-1.98,3.31,;-1.91,1.77,;-3.34,4.03,;-2.28,5.14,;-3.31,6.28,;-4.11,5.36,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N(C1CC(C1)N1CCCCC1)C(=O)C21CCN(CC1)C(=O)C1CCC[C@@H]1O |r,wD:51.60,(14.97,3.01,;13.44,2.79,;12.87,1.36,;12.49,4,;12.9,5.48,;11.62,6.33,;10.41,5.38,;8.89,5.63,;7.91,4.45,;8.45,3,;9.97,2.75,;10.5,1.3,;9.52,.12,;10.06,-1.33,;9.07,-2.51,;7.56,-2.26,;7.02,-.81,;8,.37,;7.46,1.82,;10.95,3.93,;6.39,4.7,;5.41,3.52,;3.89,3.77,;3.36,5.22,;4.34,6.4,;5.86,6.15,;3.51,7.7,;4.08,9.14,;3.47,10.55,;4.88,11.16,;5.49,9.75,;5.45,12.59,;4.49,13.8,;5.06,15.23,;6.58,15.46,;7.54,14.25,;6.97,12.82,;2.02,7.32,;.83,8.3,;1.92,5.79,;1.99,4.25,;.69,3.42,;-.68,4.14,;-.74,5.67,;.56,6.5,;-1.98,3.31,;-1.91,1.77,;-3.34,4.03,;-4.75,3.4,;-5.78,4.54,;-5.01,5.88,;-3.5,5.56,;-2.36,6.59,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N(C1CC(C1)N1C[C@@H]3CC[C@@H]3C1)C(=O)C21CCN(CC1)C(=O)C1(C)COC1 |r,wU:36.40,33.38,(14.97,3.01,;13.44,2.79,;12.87,1.36,;12.49,4,;12.9,5.48,;11.62,6.33,;10.41,5.38,;8.89,5.63,;7.91,4.45,;8.45,3,;9.97,2.75,;10.5,1.3,;9.52,.12,;10.06,-1.33,;9.07,-2.51,;7.56,-2.26,;7.02,-.81,;8,.37,;7.46,1.82,;10.95,3.93,;6.39,4.7,;5.41,3.52,;3.89,3.77,;3.36,5.22,;4.34,6.4,;5.86,6.15,;3.51,7.7,;4.08,9.14,;3.47,10.55,;4.88,11.16,;5.49,9.75,;5.45,12.59,;6.96,12.91,;7.12,14.44,;7.74,15.85,;6.34,16.48,;5.71,15.07,;4.68,13.93,;2.02,7.32,;.83,8.3,;1.92,5.79,;1.99,4.25,;.69,3.42,;-.68,4.14,;-.74,5.67,;.56,6.5,;-1.98,3.31,;-1.91,1.77,;-3.34,4.03,;-4.64,3.2,;-4.11,5.36,;-3.21,6.6,;-2.44,5.27,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N(C1CC(C1)N1C[C@@H]3CC[C@@H]3C1)C(=O)C21CCN(CC1)C(=O)C1CCCO1 |r,wU:36.40,33.38,(14.97,3.01,;13.44,2.79,;12.87,1.36,;12.49,4,;12.9,5.48,;11.62,6.33,;10.41,5.38,;8.89,5.63,;7.91,4.45,;8.45,3,;9.97,2.75,;10.5,1.3,;9.52,.12,;10.06,-1.33,;9.07,-2.51,;7.56,-2.26,;7.02,-.81,;8,.37,;7.46,1.82,;10.95,3.93,;6.39,4.7,;5.41,3.52,;3.89,3.77,;3.36,5.22,;4.34,6.4,;5.86,6.15,;3.51,7.7,;4.08,9.14,;3.47,10.55,;4.88,11.16,;5.49,9.75,;5.45,12.59,;6.96,12.91,;7.12,14.44,;7.74,15.85,;6.34,16.48,;5.71,15.07,;4.68,13.93,;2.02,7.32,;.83,8.3,;1.92,5.79,;1.99,4.25,;.69,3.42,;-.68,4.14,;-.74,5.67,;.56,6.5,;-1.98,3.31,;-1.91,1.77,;-3.34,4.03,;-4.75,3.4,;-5.78,4.54,;-5.01,5.88,;-3.5,5.56,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N(C1CC(C1)N1C[C@@H]3CC[C@@H]3C1)C(=O)C21CCN(CC1)C(=O)C(C)(C)CO |r,wU:36.40,33.38,(14.97,3.01,;13.44,2.79,;12.87,1.36,;12.49,4,;12.9,5.48,;11.62,6.33,;10.41,5.38,;8.89,5.63,;7.91,4.45,;8.45,3,;9.97,2.75,;10.5,1.3,;9.52,.12,;10.06,-1.33,;9.07,-2.51,;7.56,-2.26,;7.02,-.81,;8,.37,;7.46,1.82,;10.95,3.93,;6.39,4.7,;5.41,3.52,;3.89,3.77,;3.36,5.22,;4.34,6.4,;5.86,6.15,;3.51,7.7,;4.08,9.14,;3.47,10.55,;4.88,11.16,;5.49,9.75,;5.45,12.59,;6.96,12.91,;7.12,14.44,;7.74,15.85,;6.34,16.48,;5.71,15.07,;4.68,13.93,;2.02,7.32,;.83,8.3,;1.92,5.79,;1.99,4.25,;.69,3.42,;-.68,4.14,;-.74,5.67,;.56,6.5,;-1.98,3.31,;-1.91,1.77,;-3.34,4.03,;-3.5,5.56,;-3.39,2.49,;-4.75,3.4,;-5.78,4.54,)|
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CC(C)n1cnc2cc(nc(Nc3cc(F)ncc3F)c12)-c1ccc2c(c1)N(C1CC(C1)N1CCC(C)(C)C1)C(=O)C21CCN(CC1)C(=O)C1(C)COC1 |(11.59,-4.02,;10.07,-4.24,;9.5,-5.67,;9.11,-3.04,;9.53,-1.55,;8.24,-.7,;7.04,-1.66,;5.52,-1.4,;4.54,-2.59,;5.07,-4.03,;6.59,-4.29,;7.13,-5.73,;6.14,-6.92,;4.63,-6.66,;3.64,-7.85,;2.13,-7.59,;4.18,-9.29,;5.7,-9.55,;6.68,-8.36,;8.2,-8.62,;7.57,-3.1,;3.02,-2.33,;2.03,-3.51,;.52,-3.26,;-.02,-1.81,;.96,-.63,;2.48,-.88,;.14,.67,;.71,2.11,;.09,3.52,;1.51,4.13,;2.12,2.72,;2.07,5.56,;3.58,5.88,;3.74,7.41,;2.34,8.04,;2.01,9.55,;3.53,9.01,;1.3,6.9,;-1.35,.29,;-2.54,1.27,;-1.45,-1.25,;-1.39,-2.78,;-2.69,-3.61,;-4.05,-2.9,;-4.12,-1.36,;-2.82,-.53,;-5.35,-3.72,;-5.29,-5.26,;-6.72,-3.01,;-5.65,-1.89,;-8.02,-3.83,;-8.95,-2.15,;-7.49,-1.67,)|
CC(C)n1cnc2cc(nc(Nc3cc(C)ncc3F)c12)-c1ccc2c(c1)N(C1CC(C1)N1CC3CCC(C3)C1)C(=O)C21CCN(CC1)C(C)=O |(11.59,-4.02,;10.07,-4.24,;9.5,-5.67,;9.11,-3.04,;9.53,-1.55,;8.24,-.7,;7.04,-1.66,;5.52,-1.4,;4.54,-2.59,;5.07,-4.03,;6.59,-4.29,;7.13,-5.73,;6.14,-6.92,;4.63,-6.66,;3.64,-7.85,;2.13,-7.59,;4.18,-9.29,;5.7,-9.55,;6.68,-8.36,;8.2,-8.62,;7.57,-3.1,;3.02,-2.33,;2.03,-3.51,;.52,-3.26,;-.02,-1.81,;.96,-.63,;2.48,-.88,;.14,.67,;.71,2.11,;.09,3.52,;1.51,4.13,;2.12,2.72,;2.07,5.56,;1.17,6.81,;1.8,8.21,;1.8,6.67,;3.24,6.09,;4.23,7.13,;3.33,8.37,;3.61,5.72,;-1.35,.29,;-2.54,1.27,;-1.45,-1.25,;-1.39,-2.78,;-2.69,-3.61,;-4.05,-2.9,;-4.12,-1.36,;-2.82,-.53,;-5.35,-3.72,;-6.72,-3.01,;-5.29,-5.26,)|
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CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N([C@H]1C[C@H](C1)N1CCCCC1)C(=O)C21CCN(CC1)C(=O)C(C)(C)C |r,wU:27.30,29.35,(7.77,-4.47,;6.27,-4.14,;5.24,-5.29,;5.79,-2.68,;6.7,-1.43,;5.79,-.19,;4.33,-.66,;2.99,.11,;1.66,-.66,;1.66,-2.2,;2.99,-2.97,;2.99,-4.51,;1.66,-5.28,;1.66,-6.82,;.32,-7.59,;-1.01,-6.82,;-1.01,-5.28,;.32,-4.51,;.32,-2.97,;4.33,-2.2,;.32,.11,;.32,1.65,;-1.01,2.42,;-2.34,1.65,;-2.34,.11,;-1.01,-.66,;-3.81,-.37,;-4.28,-1.83,;-3.58,-3.21,;-4.96,-3.91,;-5.66,-2.53,;-5.43,-5.37,;-6.94,-5.69,;-7.41,-7.16,;-6.38,-8.3,;-4.88,-7.98,;-4.4,-6.52,;-4.71,.88,;-6.25,.88,;-3.81,2.12,;-2.78,3.27,;-3.25,4.73,;-4.76,5.05,;-5.79,3.91,;-5.31,2.44,;-5.24,6.52,;-4.2,7.66,;-6.74,6.84,;-7.22,8.3,;-7.77,5.69,;-5.71,7.98,)|
CC(C)C(=O)N1CCC2(CC1)C(=O)N([C@H]1C[C@H](C1)N1CCCCC1)c1cc(ccc21)-c1cc2ncn(C(C)C)c2c(Nc2ccncc2F)n1 |r,wU:14.14,16.19,(-7.22,8.3,;-6.74,6.84,;-7.77,5.69,;-5.24,6.52,;-4.2,7.66,;-4.76,5.05,;-3.25,4.73,;-2.78,3.27,;-3.81,2.12,;-5.31,2.44,;-5.79,3.91,;-4.71,.88,;-6.25,.88,;-3.81,-.37,;-4.28,-1.83,;-3.58,-3.21,;-4.96,-3.91,;-5.66,-2.53,;-5.43,-5.37,;-6.94,-5.69,;-7.41,-7.16,;-6.38,-8.3,;-4.88,-7.98,;-4.4,-6.52,;-2.34,.11,;-1.01,-.66,;.32,.11,;.32,1.65,;-1.01,2.42,;-2.34,1.65,;1.66,-.66,;2.99,.11,;4.33,-.66,;5.79,-.19,;6.7,-1.43,;5.79,-2.68,;6.27,-4.14,;7.77,-4.47,;5.24,-5.29,;4.33,-2.2,;2.99,-2.97,;2.99,-4.51,;1.66,-5.28,;1.66,-6.82,;.32,-7.59,;-1.01,-6.82,;-1.01,-5.28,;.32,-4.51,;.32,-2.97,;1.66,-2.2,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N([C@@H]1C[C@@H](C1)N1C[C@@H]3CC[C@@H]3C1)C(=O)C21CCN(CC1)C(C)=O |r,wU:27.30,29.35,33.38,36.40,(7.57,-3.63,;6.07,-3.31,;5.3,-4.64,;5.59,-1.85,;6.5,-.6,;5.59,.65,;4.13,.17,;2.79,.94,;1.46,.17,;1.46,-1.37,;2.79,-2.14,;2.79,-3.68,;1.46,-4.45,;1.46,-5.99,;.12,-6.76,;-1.21,-5.99,;-1.21,-4.45,;.12,-3.68,;.12,-2.14,;4.13,-1.37,;.12,.94,;.12,2.48,;-1.21,3.25,;-2.54,2.48,;-2.54,.94,;-1.21,.17,;-4.01,.46,;-4.48,-1,;-5.86,-1.7,;-5.16,-3.07,;-3.78,-2.37,;-5.63,-4.54,;-7.1,-5.01,;-7.1,-6.55,;-7.57,-8.02,;-6.11,-8.49,;-5.63,-7.03,;-4.73,-5.78,;-4.91,1.71,;-6.45,1.71,;-4.01,2.96,;-2.98,4.1,;-3.45,5.56,;-4.96,5.88,;-5.99,4.74,;-5.51,3.28,;-5.43,7.35,;-6.94,7.67,;-4.4,8.49,)|
CC(C)n1cnc2cc(nc(Nc3cc(C)ncc3F)c12)-c1ccc2c(c1)N([C@@H]1C[C@@H](C1)N1CCC(C)(C)C1)C(=O)C21CCN(CC1)C(C)=O |r,wU:28.31,30.36,(8.08,-3.73,;6.57,-3.41,;5.54,-4.55,;6.1,-1.94,;7,-.7,;6.1,.55,;4.63,.07,;3.3,.84,;1.96,.07,;1.96,-1.47,;3.3,-2.24,;3.3,-3.78,;1.96,-4.55,;1.96,-6.09,;.63,-6.86,;.63,-8.4,;-.7,-6.09,;-.7,-4.55,;.63,-3.78,;.63,-2.24,;4.63,-1.47,;.63,.84,;.63,2.38,;-.7,3.15,;-2.04,2.38,;-2.04,.84,;-.7,.07,;-3.5,.37,;-3.98,-1.1,;-5.35,-1.8,;-4.65,-3.17,;-3.28,-2.47,;-5.13,-4.63,;-4.22,-5.88,;-5.13,-7.13,;-6.59,-6.65,;-8.08,-7.05,;-6.99,-8.14,;-6.59,-5.11,;-4.41,1.61,;-5.95,1.61,;-3.5,2.86,;-2.47,4,;-2.95,5.47,;-4.45,5.79,;-5.48,4.64,;-5.01,3.18,;-4.93,7.25,;-6.44,7.57,;-3.9,8.4,)|
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CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N([C@@H]1C[C@@H](C1)N1CC(C)(C)C1)C(=O)C21CCN(CC1)C1COC1 |r,wU:27.30,29.35,(7.61,-4.37,;6.1,-4.05,;5.07,-5.19,;5.62,-2.59,;6.53,-1.34,;5.62,-.09,;4.16,-.57,;2.83,.2,;1.49,-.57,;1.49,-2.11,;2.83,-2.88,;2.83,-4.42,;1.49,-5.19,;1.49,-6.73,;.16,-7.5,;-1.18,-6.73,;-1.18,-5.19,;.16,-4.42,;.16,-2.88,;4.16,-2.11,;.16,.2,;.16,1.74,;-1.18,2.51,;-2.51,1.74,;-2.51,.2,;-1.18,-.57,;-3.97,-.28,;-4.45,-1.74,;-5.82,-2.44,;-5.12,-3.81,;-3.75,-3.11,;-5.6,-5.28,;-6.97,-5.98,;-6.27,-7.35,;-7.61,-8.12,;-5.5,-8.68,;-4.9,-6.65,;-4.88,.97,;-6.42,.97,;-3.97,2.22,;-2.94,3.36,;-3.42,4.83,;-4.93,5.15,;-5.96,4,;-5.48,2.54,;-5.4,6.61,;-4.7,7.98,;-6.07,8.68,;-6.77,7.31,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N(C1CC(C1)N1CCCC3(CC3)C1)C(=O)C21CCN(CC1)C(C)=O |(-2.25,10.49,;-.74,10.17,;.29,11.32,;-.27,8.71,;-1.17,7.46,;-.27,6.22,;1.2,6.69,;2.53,5.92,;3.86,6.69,;3.86,8.23,;2.53,9,;2.53,10.54,;3.86,11.31,;5.2,10.54,;6.53,11.31,;6.53,12.85,;5.2,13.62,;3.86,12.85,;2.53,13.62,;1.2,8.23,;5.2,5.92,;5.2,4.38,;6.53,3.61,;7.87,4.38,;7.87,5.92,;6.53,6.69,;9.33,6.4,;9.81,7.86,;11.18,8.56,;10.48,9.93,;9.11,9.24,;10.95,11.4,;9.92,12.54,;10.4,14.01,;11.91,14.33,;12.94,13.18,;14.08,14.21,;14.4,12.71,;12.46,11.72,;10.23,5.15,;11.77,5.15,;9.33,3.91,;10.84,3.59,;11.31,2.12,;10.28,.98,;8.78,1.3,;8.3,2.76,;10.76,-.49,;9.73,-1.63,;12.26,-.81,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N([C@@H]1C[C@@H](C1)N1CCC3(CC3)C1)C(=O)C21CCN(CC1)C(C)=O |r,wU:27.30,29.35,(8.1,-3.9,;6.59,-3.58,;5.56,-4.72,;6.12,-2.11,;7.02,-.87,;6.12,.38,;4.65,-.1,;3.32,.67,;1.99,-.1,;1.99,-1.64,;3.32,-2.41,;3.32,-3.95,;1.99,-4.72,;1.99,-6.26,;.65,-7.03,;-.68,-6.26,;-.68,-4.72,;.65,-3.95,;.65,-2.41,;4.65,-1.64,;.65,.67,;.65,2.21,;-.68,2.98,;-2.01,2.21,;-2.01,.67,;-.68,-.1,;-3.48,.2,;-3.96,-1.27,;-5.33,-1.97,;-4.63,-3.34,;-3.26,-2.64,;-5.1,-4.8,;-4.2,-6.05,;-5.1,-7.3,;-6.57,-6.82,;-8.1,-6.98,;-7.2,-8.23,;-6.57,-5.28,;-4.38,1.44,;-5.92,1.44,;-3.48,2.69,;-2.45,3.83,;-2.92,5.3,;-4.43,5.62,;-5.46,4.47,;-4.99,3.01,;-4.91,7.08,;-3.88,8.23,;-6.41,7.4,)|
COC(C)(C)CN(C)C1CC(C1)N1C(=O)C2(CCN(CC2)C(C)=O)c2ccc(cc12)-c1cc2ncn(C(C)C)c2c(Nc2ccncc2F)n1 |(6.86,6.84,;5.83,7.98,;4.32,7.66,;3.29,8.8,;5.35,6.52,;3.85,6.2,;4.88,5.05,;6.39,5.37,;4.4,3.59,;5.1,2.21,;3.73,1.51,;3.03,2.89,;3.25,.05,;4.16,-1.2,;5.7,-1.2,;3.25,-2.44,;4.76,-2.76,;5.24,-4.23,;4.21,-5.37,;2.7,-5.05,;2.22,-3.59,;4.68,-6.84,;3.65,-7.98,;6.19,-7.16,;1.79,-1.97,;.46,-2.74,;-.88,-1.97,;-.88,-.43,;.46,.34,;1.79,-.43,;-2.21,.34,;-3.55,-.43,;-4.88,.34,;-6.34,-.13,;-7.25,1.11,;-6.34,2.36,;-6.82,3.82,;-8.33,4.14,;-5.79,4.97,;-4.88,1.88,;-3.55,2.65,;-3.55,4.19,;-2.21,4.96,;-.88,4.19,;.46,4.96,;.46,6.5,;-.88,7.27,;-2.21,6.5,;-3.55,7.27,;-2.21,1.88,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N(C1CC(C1)N1CC3CC3C1)C(=O)C21CCN(CC1)C(C)=O |(-8.33,4.14,;-6.82,3.82,;-5.79,4.97,;-6.34,2.36,;-7.25,1.11,;-6.34,-.13,;-4.88,.34,;-3.55,-.43,;-2.21,.34,;-2.21,1.88,;-3.55,2.65,;-3.55,4.19,;-2.21,4.96,;-.88,4.19,;.46,4.96,;.46,6.5,;-.88,7.27,;-2.21,6.5,;-3.55,7.27,;-4.88,1.88,;-.88,-.43,;-.88,-1.97,;.46,-2.74,;1.79,-1.97,;1.79,-.43,;.46,.34,;3.25,.05,;3.73,1.51,;5.1,2.21,;4.4,3.59,;3.03,2.89,;4.88,5.05,;6.34,5.53,;6.34,7.07,;5.78,8.79,;4.88,7.54,;3.97,6.3,;4.16,-1.2,;5.7,-1.2,;3.25,-2.44,;4.76,-2.76,;5.24,-4.23,;4.21,-5.37,;2.7,-5.05,;2.22,-3.59,;4.68,-6.84,;3.65,-7.98,;6.19,-7.16,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N(C1CC(C1)N1CC3CCC(C3)C1)C(=O)C21CCN(CC1)C(C)=O |(-8.33,4.14,;-6.82,3.82,;-5.79,4.97,;-6.34,2.36,;-7.25,1.11,;-6.34,-.13,;-4.88,.34,;-3.55,-.43,;-2.21,.34,;-2.21,1.88,;-3.55,2.65,;-3.55,4.19,;-2.21,4.96,;-.88,4.19,;.46,4.96,;.46,6.5,;-.88,7.27,;-2.21,6.5,;-3.55,7.27,;-4.88,1.88,;-.88,-.43,;-.88,-1.97,;.46,-2.74,;1.79,-1.97,;1.79,-.43,;.46,.34,;3.25,.05,;3.73,1.51,;5.1,2.21,;4.4,3.59,;3.03,2.89,;4.88,5.05,;3.85,6.2,;4.32,7.66,;4.64,6.15,;5.72,5.81,;6.86,6.84,;5.83,7.98,;6.39,5.37,;4.16,-1.2,;5.7,-1.2,;3.25,-2.44,;4.76,-2.76,;5.24,-4.23,;4.21,-5.37,;2.7,-5.05,;2.22,-3.59,;4.68,-6.84,;3.65,-7.98,;6.19,-7.16,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N(C1CC(C1)N1CCCC3(CCC3)C1)C(=O)C21CCN(CC1)C(C)=O |(-8.33,4.14,;-6.82,3.82,;-5.79,4.97,;-6.34,2.36,;-7.25,1.11,;-6.34,-.13,;-4.88,.34,;-3.55,-.43,;-2.21,.34,;-2.21,1.88,;-3.55,2.65,;-3.55,4.19,;-2.21,4.96,;-.88,4.19,;.46,4.96,;.46,6.5,;-.88,7.27,;-2.21,6.5,;-3.55,7.27,;-4.88,1.88,;-.88,-.43,;-.88,-1.97,;.46,-2.74,;1.79,-1.97,;1.79,-.43,;.46,.34,;3.25,.05,;3.73,1.51,;5.1,2.21,;4.4,3.59,;3.03,2.89,;4.88,5.05,;3.85,6.2,;4.32,7.66,;5.83,7.98,;6.86,6.84,;8.01,7.87,;9.27,7.3,;8.33,6.36,;6.39,5.37,;4.16,-1.2,;5.7,-1.2,;3.25,-2.44,;4.76,-2.76,;5.24,-4.23,;4.21,-5.37,;2.7,-5.05,;2.22,-3.59,;4.68,-6.84,;3.65,-7.98,;6.19,-7.16,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N(C1CC(C1)N1CCC3CC3C1)C(=O)C21CCN(CC1)C(C)=O |(-8.33,4.14,;-6.82,3.82,;-5.79,4.97,;-6.34,2.36,;-7.25,1.11,;-6.34,-.13,;-4.88,.34,;-3.55,-.43,;-2.21,.34,;-2.21,1.88,;-3.55,2.65,;-3.55,4.19,;-2.21,4.96,;-.88,4.19,;.46,4.96,;.46,6.5,;-.88,7.27,;-2.21,6.5,;-3.55,7.27,;-4.88,1.88,;-.88,-.43,;-.88,-1.97,;.46,-2.74,;1.79,-1.97,;1.79,-.43,;.46,.34,;3.25,.05,;3.73,1.51,;5.1,2.21,;4.4,3.59,;3.03,2.89,;4.88,5.05,;3.85,6.2,;4.32,7.66,;5.83,7.98,;7.34,8.3,;6.86,6.84,;6.39,5.37,;4.16,-1.2,;5.7,-1.2,;3.25,-2.44,;4.76,-2.76,;5.24,-4.23,;4.21,-5.37,;2.7,-5.05,;2.22,-3.59,;4.68,-6.84,;3.65,-7.98,;6.19,-7.16,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N(C1CC(C1)N1CCCC[C@@H]1C)C(=O)C21CCN(CC1)C(C)=O |r,wD:36.42,(-8.33,4.14,;-6.82,3.82,;-5.79,4.97,;-6.34,2.36,;-7.25,1.11,;-6.34,-.13,;-4.88,.34,;-3.55,-.43,;-2.21,.34,;-2.21,1.88,;-3.55,2.65,;-3.55,4.19,;-2.21,4.96,;-.88,4.19,;.46,4.96,;.46,6.5,;-.88,7.27,;-2.21,6.5,;-3.55,7.27,;-4.88,1.88,;-.88,-.43,;-.88,-1.97,;.46,-2.74,;1.79,-1.97,;1.79,-.43,;.46,.34,;3.25,.05,;3.73,1.51,;5.1,2.21,;4.4,3.59,;3.03,2.89,;4.88,5.05,;3.85,6.2,;4.32,7.66,;5.83,7.98,;6.86,6.84,;6.39,5.37,;7.42,4.23,;4.16,-1.2,;5.7,-1.2,;3.25,-2.44,;4.76,-2.76,;5.24,-4.23,;4.21,-5.37,;2.7,-5.05,;2.22,-3.59,;4.68,-6.84,;3.65,-7.98,;6.19,-7.16,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N(C1CC(C1)N1CCCCCC1)C(=O)C21CCN(CC1)C(C)=O |(-8.33,4.14,;-6.82,3.82,;-5.79,4.97,;-6.34,2.36,;-7.25,1.11,;-6.34,-.13,;-4.88,.34,;-3.55,-.43,;-2.21,.34,;-2.21,1.88,;-3.55,2.65,;-3.55,4.19,;-2.21,4.96,;-.88,4.19,;.46,4.96,;.46,6.5,;-.88,7.27,;-2.21,6.5,;-3.55,7.27,;-4.88,1.88,;-.88,-.43,;-.88,-1.97,;.46,-2.74,;1.79,-1.97,;1.79,-.43,;.46,.34,;3.25,.05,;3.73,1.51,;5.1,2.21,;4.4,3.59,;3.03,2.89,;4.88,5.05,;3.85,6.2,;4.01,7.73,;5.34,8.5,;6.87,8.34,;7.75,6.71,;6.97,5.33,;4.16,-1.2,;5.7,-1.2,;3.25,-2.44,;4.76,-2.76,;5.24,-4.23,;4.21,-5.37,;2.7,-5.05,;2.22,-3.59,;4.68,-6.84,;3.65,-7.98,;6.19,-7.16,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N(C1CC(C1)N1CC3CCC(C3)C1)C(=O)C21CCN(CC1)C(C)=O |(-8.33,4.14,;-6.82,3.82,;-5.79,4.97,;-6.34,2.36,;-7.25,1.11,;-6.34,-.13,;-4.88,.34,;-3.55,-.43,;-2.21,.34,;-2.21,1.88,;-3.55,2.65,;-3.55,4.19,;-2.21,4.96,;-.88,4.19,;.46,4.96,;.46,6.5,;-.88,7.27,;-2.21,6.5,;-3.55,7.27,;-4.88,1.88,;-.88,-.43,;-.88,-1.97,;.46,-2.74,;1.79,-1.97,;1.79,-.43,;.46,.34,;3.25,.05,;3.73,1.51,;5.1,2.21,;4.4,3.59,;3.03,2.89,;4.88,5.05,;3.85,6.2,;4.32,7.66,;4.64,6.15,;5.62,5.93,;6.86,6.84,;5.83,7.98,;6.39,5.37,;4.16,-1.2,;5.7,-1.2,;3.25,-2.44,;4.76,-2.76,;5.24,-4.23,;4.21,-5.37,;2.7,-5.05,;2.22,-3.59,;4.68,-6.84,;3.65,-7.98,;6.19,-7.16,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N(C1CC(C1)N1CC3CC3(C)C1)C(=O)C21CCN(CC1)C(C)=O |(-7.59,4.14,;-6.09,3.82,;-5.06,4.97,;-5.61,2.36,;-6.52,1.11,;-5.61,-.13,;-4.15,.34,;-2.81,-.43,;-1.48,.34,;-1.48,1.88,;-2.81,2.65,;-2.81,4.19,;-1.48,4.96,;-.15,4.19,;1.19,4.96,;1.19,6.5,;-.15,7.27,;-1.48,6.5,;-2.81,7.27,;-4.15,1.88,;-.15,-.43,;-.15,-1.97,;1.19,-2.74,;2.52,-1.97,;2.52,-.43,;1.19,.34,;3.99,.05,;4.46,1.51,;5.83,2.21,;5.14,3.59,;3.76,2.89,;5.61,5.05,;4.71,6.3,;5.61,7.54,;6.64,8.69,;7.08,7.07,;8.6,7.27,;7.08,5.53,;4.89,-1.2,;6.43,-1.2,;3.99,-2.44,;5.49,-2.76,;5.97,-4.23,;4.94,-5.37,;3.43,-5.05,;2.96,-3.59,;5.41,-6.84,;4.38,-7.98,;6.92,-7.16,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N(C1CC(C1)N1CCCC1)C(=O)C2(C)C |(-7.59,4.14,;-6.09,3.82,;-5.06,4.97,;-5.61,2.36,;-6.52,1.11,;-5.61,-.13,;-4.15,.34,;-2.81,-.43,;-1.48,.34,;-1.48,1.88,;-2.81,2.65,;-2.81,4.19,;-1.48,4.96,;-.15,4.19,;1.19,4.96,;1.19,6.5,;-.15,7.27,;-1.48,6.5,;-2.81,7.27,;-4.15,1.88,;-.15,-.43,;-.15,-1.97,;1.19,-2.74,;2.52,-1.97,;2.52,-.43,;1.19,.34,;3.99,.05,;4.46,1.51,;5.83,2.21,;5.14,3.59,;3.76,2.89,;5.61,5.05,;7.08,5.53,;7.08,7.07,;5.61,7.54,;4.71,6.3,;4.89,-1.2,;6.43,-1.2,;3.99,-2.44,;5.49,-2.76,;2.96,-3.59,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N(C1CC(C1)N1CCC(C)(C)C1)C(=O)C2(C)C |(-7.33,2.17,;-5.83,1.85,;-4.8,2.99,;-5.35,.38,;-6.26,-.86,;-5.35,-2.11,;-3.89,-1.63,;-2.55,-2.4,;-1.22,-1.63,;-1.22,-.09,;-2.55,.68,;-2.55,2.22,;-1.22,2.99,;.11,2.22,;1.45,2.99,;1.45,4.53,;.11,5.3,;-1.22,4.53,;-2.55,5.3,;-3.89,-.09,;.11,-2.4,;.11,-3.94,;1.45,-4.71,;2.78,-3.94,;2.78,-2.4,;1.45,-1.63,;4.25,-1.93,;4.72,-.46,;6.09,.24,;5.39,1.61,;4.02,.91,;5.87,3.07,;7.33,3.55,;7.33,5.09,;5.87,5.56,;5.39,7.03,;6.96,6.65,;4.96,4.32,;5.15,-3.17,;6.69,-3.17,;4.25,-4.42,;5.75,-4.74,;3.21,-5.56,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N(C1CC(C1)N1C3CC1COC3)C(=O)C2(C)C |(-7.33,2.17,;-5.83,1.85,;-4.8,2.99,;-5.35,.38,;-6.26,-.86,;-5.35,-2.11,;-3.89,-1.63,;-2.55,-2.4,;-1.22,-1.63,;-1.22,-.09,;-2.55,.68,;-2.55,2.22,;-1.22,2.99,;.11,2.22,;1.45,2.99,;1.45,4.53,;.11,5.3,;-1.22,4.53,;-2.55,5.3,;-3.89,-.09,;.11,-2.4,;.11,-3.94,;1.45,-4.71,;2.78,-3.94,;2.78,-2.4,;1.45,-1.63,;4.25,-1.93,;4.72,-.46,;6.09,.24,;5.39,1.61,;4.02,.91,;5.87,3.07,;7.38,3.39,;6.35,4.54,;4.84,4.22,;5.32,5.68,;6.82,6,;7.85,4.86,;5.15,-3.17,;6.69,-3.17,;4.25,-4.42,;5.75,-4.74,;3.21,-5.56,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N(C1CC(C1)N1CCC[C@@H](C)C1)C(=O)C2(C)C |r,wU:35.40,(-7.33,2.17,;-5.83,1.85,;-4.8,2.99,;-5.35,.38,;-6.26,-.86,;-5.35,-2.11,;-3.89,-1.63,;-2.55,-2.4,;-1.22,-1.63,;-1.22,-.09,;-2.55,.68,;-2.55,2.22,;-1.22,2.99,;.11,2.22,;1.45,2.99,;1.45,4.53,;.11,5.3,;-1.22,4.53,;-2.55,5.3,;-3.89,-.09,;.11,-2.4,;.11,-3.94,;1.45,-4.71,;2.78,-3.94,;2.78,-2.4,;1.45,-1.63,;4.25,-1.93,;4.72,-.46,;6.09,.24,;5.39,1.61,;4.02,.91,;5.87,3.07,;4.84,4.22,;5.32,5.68,;6.82,6,;7.85,4.86,;9.36,5.18,;7.38,3.39,;5.15,-3.17,;6.69,-3.17,;4.25,-4.42,;5.75,-4.74,;3.21,-5.56,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N(C1CC(C1)N1CC[C@H](C)C1)C(=O)C2(C)C |r,wU:34.39,(-7.33,2.17,;-5.83,1.85,;-4.8,2.99,;-5.35,.38,;-6.26,-.86,;-5.35,-2.11,;-3.89,-1.63,;-2.55,-2.4,;-1.22,-1.63,;-1.22,-.09,;-2.55,.68,;-2.55,2.22,;-1.22,2.99,;.11,2.22,;1.45,2.99,;1.45,4.53,;.11,5.3,;-1.22,4.53,;-2.55,5.3,;-3.89,-.09,;.11,-2.4,;.11,-3.94,;1.45,-4.71,;2.78,-3.94,;2.78,-2.4,;1.45,-1.63,;4.25,-1.93,;4.72,-.46,;6.09,.24,;5.39,1.61,;4.02,.91,;5.87,3.07,;7.33,3.55,;7.33,5.09,;5.87,5.56,;5.39,7.03,;4.96,4.32,;5.15,-3.17,;6.69,-3.17,;4.25,-4.42,;5.75,-4.74,;3.21,-5.56,)|
CC(C)n1cnc2cc(nc(Nc3ccncc3F)c12)-c1ccc2c(c1)N(C1CC(C1)N1CC3CCC1CC3)C(=O)C21CCN(CC1)C(C)=O |(-7.33,2.17,;-5.83,1.85,;-4.8,2.99,;-5.35,.38,;-6.26,-.86,;-5.35,-2.11,;-3.89,-1.63,;-2.55,-2.4,;-1.22,-1.63,;-1.22,-.09,;-2.55,.68,;-2.55,2.22,;-1.22,2.99,;.11,2.22,;1.45,2.99,;1.45,4.53,;.11,5.3,;-1.22,4.53,;-2.55,5.3,;-3.89,-.09,;.11,-2.4,;.11,-3.94,;1.45,-4.71,;2.78,-3.94,;2.78,-2.4,;1.45,-1.63,;4.25,-1.93,;4.72,-.46,;6.09,.24,;5.39,1.61,;4.02,.91,;5.87,3.07,;7.38,3.39,;7.85,4.86,;6.82,6,;5.32,5.68,;4.84,4.22,;6.17,4.99,;6.8,3.58,;5.15,-3.17,;6.69,-3.17,;4.25,-4.42,;3.21,-5.56,;3.69,-7.03,;5.2,-7.35,;6.23,-6.2,;5.75,-4.74,;5.67,-8.81,;4.64,-9.96,;7.18,-9.13,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N(C2CC(C2)N2CCCCC2)C(=O)C3(C)C)ncc1C |(6.53,12.85,;6.53,11.31,;5.2,10.54,;3.86,11.31,;5.2,9,;3.86,8.23,;3.86,6.69,;2.53,5.92,;2.53,4.38,;3.86,3.61,;3.86,2.07,;2.53,1.3,;1.2,2.07,;-.27,1.6,;-1.17,2.84,;-.27,4.09,;-.74,5.55,;-2.25,5.87,;.29,6.7,;1.2,3.61,;5.2,1.3,;5.2,-.24,;6.53,-1.01,;7.87,-.24,;7.87,1.3,;6.53,2.07,;9.33,1.78,;9.81,3.24,;9.11,4.62,;10.48,5.31,;11.18,3.94,;10.95,6.78,;9.92,7.92,;10.4,9.39,;11.91,9.71,;12.94,8.56,;12.46,7.1,;10.23,.53,;11.77,.53,;9.33,-.71,;8.7,-2.12,;10.66,-1.48,;5.2,5.92,;6.53,6.69,;6.53,8.23,;7.87,9,)|
CC(C)n1cnc2cc(nc(Nc3cc(C(=O)NC4(CF)CC4)c(C)cn3)c12)-c1ccc2c(c1)N([C@H]1C[C@H](C1)N1CCCCC1)C(=O)C2(C)C |r,wU:35.39,37.44,(7.59,-1.32,;6.09,-1,;5.06,-2.14,;5.61,.47,;6.52,1.71,;5.61,2.96,;4.15,2.48,;2.81,3.25,;1.48,2.48,;1.48,.94,;2.81,.17,;2.81,-1.37,;1.48,-2.14,;1.48,-3.68,;.15,-4.45,;.15,-5.99,;-1.19,-6.76,;1.48,-6.76,;2.81,-5.99,;4.15,-6.76,;5.48,-5.99,;3.58,-4.65,;2.04,-4.65,;-1.19,-3.68,;-2.52,-4.45,;-1.19,-2.14,;.15,-1.37,;4.15,.94,;.15,3.25,;.15,4.79,;-1.19,5.56,;-2.52,4.79,;-2.52,3.25,;-1.19,2.48,;-3.99,2.78,;-4.46,1.31,;-3.76,-.06,;-5.14,-.76,;-5.83,.61,;-5.61,-2.22,;-7.12,-2.54,;-7.59,-4.01,;-6.56,-5.15,;-5.06,-4.83,;-4.58,-3.37,;-4.89,4.02,;-6.43,4.02,;-3.99,5.27,;-3.59,6.76,;-5.08,6.36,)|
CN[C@@H]1CCCN(C1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2ccnc3n(C)cc(C)c23)nc1 |r|
Cn1cnc2c(ccnc12)-c1ccc(Nc2ccc(cn2)N2CCNCC2)c2C(=O)NCc12
CN1CCN(CC1)C1=CNC(Nc2cnc(c3CNC(=O)c23)-c2c([nH]c3ccccc23)-c2ccccc2)C=C1 |c:43,t:8,(-7.49,7.53,;-6.15,6.76,;-4.82,7.53,;-3.49,6.76,;-3.49,5.22,;-4.82,4.45,;-6.15,5.22,;-2.15,4.45,;-.82,5.22,;.51,4.45,;.51,2.91,;1.85,2.14,;1.85,.6,;.51,-.17,;.51,-1.71,;1.85,-2.48,;3.18,-1.71,;4.65,-2.18,;5.55,-.94,;4.65,.31,;5.12,1.77,;3.18,-.17,;1.85,-4.02,;3.09,-4.92,;2.62,-6.39,;1.08,-6.39,;.05,-7.53,;-1.46,-7.21,;-1.93,-5.75,;-.9,-4.6,;.6,-4.92,;4.56,-4.45,;5.7,-5.48,;7.17,-5,;7.49,-3.5,;6.34,-2.46,;4.88,-2.94,;-.82,2.14,;-2.15,2.91,)|
Cc1ccc2c(cnn2c1)-c1ccc(Nc2ccc(cn2)N2CCOCC2)c2C(=O)NCc12
OC1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnn3nccnc23)nc1
Fc1ccn2c(cnc2c1)-c1ccc(Nc2ccc(cn2)N2C[C@H]3CC[C@H](C3)C2)c2C(=O)NCc12 |r|
[H]C12CCC([H])(C1)CN(C2)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1
CN1C=CC2=C(C=CNC12)c1ncc(Nc2cccc(n2)N2CC[C@H]3CNC[C@@H]23)c2C(=O)NCc12 |r,c:2,6,t:4|
Cc1ccn2c(cnc2c1F)-c1ncc(Nc2ccc(CN3CCOCC3)cn2)c2C(=O)NCc12
Cn1ccc2c(ccnc12)-c1ncc(NC2NC(CN3CCCC3)=C(C=C2)C2CCOC2)c2C(=O)NCc12 |c:26,28|
CO[C@@H]1CN([C@@H](CO)CO1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnn3CCCCc23)nc1 |r|
CO[C@H]1CN([C@H](CO)CO1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnn3CCCCc23)nc1 |r|
CN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1C1CC[C@@H](F)[C@H](O)C1 |r|
CN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1C1CC[C@H](F)[C@@H](O)C1 |r|
CNCc1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nncn1C(C)C)N(C)C
CNCc1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nncn1C(C)C)N1CCC1
CNCc1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nncn1C(C)C)N1[C@H](C)C[C@H]1C |r|
CCN(CC)c1cc2C(=O)N(Cc2c(CNC)n1)c1cccc(n1)-c1nncn1C(C)C
CNCc1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nncn1C(C)C)C1CC1
CNCc1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nncn1C(C)C)N(C)C(C)C
CNCc1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nncn1C(C)C)C1(C)CC1
CNCc1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nncn1C(C)C)N1[C@H](C)CC[C@H]1C |r|
CCN(CC)c1cc2C(=O)N(Cc2c(CNC)n1)c1cccc(n1)-c1nncn1CC
CNCc1nc(cc2C(=O)N(Cc12)c1cccc(n1)N1[C@@H](C)COC1=O)N(C)C |r|
CC(C)c1[nH]ncc1-c1cccc(n1)N1Cc2c(cc(nc2CN)N(C)C)C1=O
CC(C)n1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2CN)N(C)C)C1=O
C[C@@H](CC(F)(F)F)n1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2CN)N(C)C)C1=O |r|
CC[C@H](C)n1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2CNC)N(C)C)C1=O |r|
CNCc1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nncn1[C@@H](C)CC(F)(F)F)N1CCCC1 |r|
CN(C)c1cc2C(=O)N(Cc2c(CN)n1)c1cccc(n1)-c1nncn1CC1CC1
CNCc1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nncn1[C@@H](C)CC(F)(F)F)N(C)C |r|
CC[C@@H](CC(F)(F)F)n1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2CNC)N(C)C)C1=O |r|
CC[C@H](CC(F)(F)F)n1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2CNC)N(C)C)C1=O |r|
CCn1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2CNC)N(C)C)C1=O
CNCc1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nncn1CC1CC1)N(C)C
CNCc1nc(cc2C(=O)N(Cc12)c1ccc(F)c(n1)-c1cn[nH]c1C(C)C)N(C)C
CNCc1nccc2C(=O)N(Cc12)c1cccc(n1)-c1nncn1C(C)C
CNCc1nc(NC)cc2C(=O)N(Cc12)c1cccc(n1)-c1nncn1C(C)C
CNCc1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nncn1C(C)C)N1[C@H]2CC[C@@H]1CC2 |r,THB:5:27:32.33:30.29|
C[C@H]1COC(=O)N1c1cccc(n1)N1Cc2c(cc(nc2CN)C2CC2)C1=O |r|
CNCc1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nncn1C(C)C)N1[C@@H](C)CC[C@H]1C |r|
CNCc1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nncn1C(C)C)C(C)(C)C
CNCc1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nncn1C(C)C)C(C)C
CC(C)n1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2CN)C2CC2)C1=O
C[C@H]1COC(=O)N1c1cccc(n1)N1Cc2c(cc(nc2CN)N(C)C)C1=O |r|
CNCc1nc(cc2C(=O)N(Cc12)c1cccc(n1)N1[C@@H](C)COC1=O)N1CCC1 |r|
CC(C)n1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2CN)N2[C@@H](C)C[C@H]2C)C1=O |r|
CC(C)c1cnnn1-c1cccc(n1)N1Cc2c(cc(nc2CN)N(C)C)C1=O
C[C@H]1COC(=O)N1c1cccc(n1)N1Cc2c(cc(nc2CN)C(C)(C)C)C1=O |r|
CNCc1nc(cc2C(=O)N(Cc12)c1cccc(n1)N1[C@H](COC1=O)C(F)F)N(C)C |r|
CCN(CC)c1cc2C(=O)N(Cc2c(CN)n1)c1cccc(n1)-c1nncn1C(C)C
CNCc1nc(cc2C(=O)N(Cc12)c1cccc(n1)N1[C@@H](C)COC1=O)C(C)(C)C |r|
CNCc1nc(cc2C(=O)N(Cc12)c1cccc(n1)N1[C@@H](C)COC1=O)C1CC1 |r|
CC(C)c1cc2C(=O)N(Cc2c(CN)n1)c1cccc(n1)N1[C@@H](C)COC1=O |r|
C[C@H]1COC(=O)N1c1cccc(n1)N1Cc2c(cc(nc2CN)C2(C)CC2)C1=O |r|
C[C@@H]1C[C@@H](C)N1c1cc2C(=O)N(Cc2c(CN)n1)c1cccc(n1)N1[C@@H](C)COC1=O |r|
C[C@H]1COC(=O)N1c1cccc(n1)N1Cc2c(cc(nc2CN)N2CCC2)C1=O |r|
CNCc1nc(cc2C(=O)N(Cc12)c1cccc(n1)N1[C@@H](CF)COC1=O)N(C)C |r|
CCCn1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2CNC)N(C)C)C1=O
CNCc1nc(C)cc2C(=O)N(Cc12)c1cccc(n1)-c1nncn1C(C)C
CCN(C)c1cc2C(=O)N(Cc2c(CNC)n1)c1cccc(n1)-c1nncn1C(C)C
CNCc1nc(cc2C(=O)N(Cc12)c1cccc(n1)N1[C@@H](C)COC1=O)C1(C)CC1 |r|
CNCc1nc(N)cc2C(=O)N(Cc12)c1cccc(n1)-c1nncn1C(C)C
CC[C@H](CC(F)(F)F)n1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2CNC)C(C)(C)C)C1=O |r|
CNCc1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nncn1C(C)C)C(F)(F)F
CNCc1cc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nncn1C(C)C)N1[C@@H](C)C[C@H]1C |r|
CCCn1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2CNC)N2CCC[C@H]2C)C1=O |r|
CCCn1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2CN)N(C)CC)C1=O
CCC(CC)n1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2CNC)C2(C)CC2)C1=O
CC[C@H](C)n1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2CNC)C2(C)CC2)C1=O |r|
CCCn1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2CNC)N(C)CC)C1=O
CCN(C)c1cc2C(=O)N(Cc2c(CN)n1)c1cccc(n1)-c1nncn1CC
CCn1c(C)nnc1-c1cccc(n1)N1Cc2c(cc(nc2CN)N2CCC[C@H]2C)C1=O |r|
CCCn1c(C)nnc1-c1cccc(n1)N1Cc2c(cc(nc2CNC)N2CCC[C@H]2C)C1=O |r|
CCCn1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2CNC)N(C)C(C)C)C1=O
CCCn1c(C)nnc1-c1cccc(n1)N1Cc2c(cc(nc2CNC)N(C)C(C)C)C1=O
CNCc1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nncn1C1CCC1)C1(C)CC1
CCc1nnc(-c2cccc(n2)N2Cc3c(cc(nc3CNC)N3CCC[C@H]3C)C2=O)n1CC |r|
CCc1nnc(-c2cccc(n2)N2Cc3c(cc(nc3CNC)N(C)C(C)C)C2=O)n1CC
C[C@@H]1CCCN1c1cc2C(=O)N(Cc2c(CN)n1)c1cccc(n1)N1[C@@H](CF)COC1=O |r|
CNCc1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nncn1C(C)C)C1CCC1
CCN(C(C)C)c1cc2C(=O)N(Cc2c(CNC)n1)c1cccc(n1)-c1nncn1C(C)C
CCn1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2CNC)N(C)C(C)C)C1=O
CC[C@@H](CC(F)(F)F)n1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2CNC)N(C)C(C)C)C1=O |r|
CC[C@H](CC(F)(F)F)n1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2CNC)N(C)C(C)C)C1=O |r|
CNCc1nc(cc2C(=O)N(Cc12)c1cccc(n1)N1[C@@H](C)COC1=O)N(C)C(C)C |r|
CCN(CC)c1cc2C(=O)N(Cc2c(CN)n1)c1cccc(n1)-c1nncn1CC
CCNc1cc2C(=O)N(Cc2c(CNC)n1)c1cccc(n1)-c1nncn1CC
CCNc1cc2C(=O)N(Cc2c(CNC)n1)c1cccc(n1)-c1nncn1C(C)C
CNCc1nc(NC(C)C)cc2C(=O)N(Cc12)c1cccc(n1)-c1nncn1C(C)C
CCCn1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2CNC)N(CC)CC)C1=O
CNCc1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nncn1C)N(C)C(C)C
CCCn1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2CN)N(C)C(C)C)C1=O
CNCc1nc(cc2C(=O)N(Cc12)c1ccc(F)c(n1)-c1nncn1C(C)C)C1(C)CC1
CCN(C(C)C)c1cc2C(=O)N(Cc2c(CNC)n1)c1cccc(n1)-c1nncn1CC
CC1(CC1)c1cc2C(=O)N(Cc2c(CN)n1)c1cccc(n1)N1[C@@H](CF)COC1=O |r|
NCc1nc(cc2C(=O)N(Cc12)c1cccc(n1)N1[C@@H](CF)COC1=O)C1CC1 |r|
CNCc1nc(cc2C(=O)N(Cc12)c1cccc(n1)N1[C@@H](CF)COC1=O)C1CC1 |r|
CCN(CC)c1cc2C(=O)N(Cc2c(CN(C)C)n1)c1cccc(n1)-c1nncn1CC
CCn1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2CN)N(C)C(C)C)C1=O
CCCn1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2CN)C2(C)CC2)C1=O
CNCc1nc(cc2C(=O)N(Cc12)c1cccc(n1)N1[C@@H](CF)COC1=O)C1(C)CC1 |r|
CCn1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2CNC)N2CCC2)C1=O
CCCn1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2CNC)N2CCC2)C1=O
CCCn1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2CNC)C2(C)CC2)C1=O
CCn1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2CNC)C2(C)CC2)C1=O
CCN(CC)c1cc2C(=O)N(Cc2c(CNC)n1)c1cccc(n1)-c1cnc(C)n1CC
CCN(CC)c1cc2C(=O)N(Cc2c(CNC)n1)c1cccc(n1)-c1nnc(C)n1CC
CCN(C(C)C)c1cc2C(=O)N(Cc2c(CNC)n1)c1cccc(n1)N1[C@@H](CF)COC1=O |r|
CCCn1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2CNC)N(CC)C(C)C)C1=O
CC(C)N(C)c1cc2C(=O)N(Cc2c(CN)n1)c1cccc(n1)N1[C@@H](C)COC1=O |r|
CCn1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2CNC)C2CCC2)C1=O
CCCn1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2CNC)C2CCC2)C1=O
CNCc1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nncn1C(C)C)N1CCC[C@H]1C |r|
CCCn1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2CNC)N2[C@H](C)CC[C@H]2C)C1=O |r|
CCn1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2CNC)N2[C@H](C)CC[C@H]2C)C1=O |r|
CC(C)n1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2CN)N2CCC[C@H]2C)C1=O |r|
CCN(C(C)C)c1cc2C(=O)N(Cc2c(CNC)n1)c1cccc(n1)-c1nncn1C
CNCc1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nncn1C(C)C)N1CCCC1(C)C
CCn1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2CN)N2[C@H](C)CC[C@H]2C)C1=O |r|
CCn1c(C)nnc1-c1cccc(n1)N1Cc2c(cc(nc2CNC)N2[C@H](C)CC[C@H]2C)C1=O |r|
CNCc1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nncn1C(C)C)N1C[C@H](C)O[C@H](C)C1 |r|
CCCn1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2CNC)N2CCC[C@H]2C(F)(F)F)C1=O |r|
CCn1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2CNC)N2CCC[C@@H]2C)C1=O |r|
CCn1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2CNC)N2CCC[C@H]2C)C1=O |r|
CNCc1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nnc(C)n1C(C)C)N1[C@H](C)CC[C@H]1C |r|
CCC(CC)n1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2CN)N(C)C)C1=O
CNCc1nc(cc2C(=O)N(Cc12)c1cccc(n1)N1[C@@H](CF)COC1=O)N1[C@H](C)CC[C@H]1C |r|
CCC(CC)n1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2CN)N2[C@H](C)CC[C@H]2C)C1=O |r|
CCCn1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2CNC)N2CCC[C@@H]2C(F)(F)F)C1=O |r|
CCn1c(C)nnc1-c1cccc(n1)N1Cc2c(cc(nc2CNC)N2CCC[C@H]2C)C1=O |r|
CCC(CC)n1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2CN)N(CC)CC)C1=O
CCN(C(C)C)c1cc2C(=O)N(Cc2c(CN)n1)c1cccc(n1)N1[C@@H](CF)COC1=O |r|
C[C@@H]1CC[C@@H](C)N1c1cc2C(=O)N(Cc2c(CN)n1)c1cccc(n1)N1[C@@H](CF)COC1=O |r|
C[C@@H]1CCCN1c1cc2C(=O)N(Cc2c(CN)n1)c1cccc(n1)N1[C@@H](C)COC1=O |r|
CCC(CC)n1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2CN)C2(C)CC2)C1=O
CCn1c(C)nnc1-c1cccc(n1)N1Cc2c(cc(nc2CN)C2(C)CC2)C1=O
CCCn1c(C)nnc1-c1cccc(n1)N1Cc2c(cc(nc2CN)C2(C)CC2)C1=O
CCC(CC)n1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2CN)C2CC2)C1=O
CCCn1c(C)nnc1-c1cccc(n1)N1Cc2c(cc(nc2CNC)N(C)CC)C1=O
CCN(C)c1cc2C(=O)N(Cc2c(CNC)n1)c1cccc(n1)-c1nncn1CC
C[C@H]1CCCN1c1cc2C(=O)N(Cc2c(CN)n1)c1cccc(n1)N1[C@@H](C)COC1=O |r|
CCCn1c(C)nnc1-c1cccc(n1)N1Cc2c(cc(nc2CN)N2CCC[C@H]2C)C1=O |r|
CCCn1c(C)nnc1-c1cccc(n1)N1Cc2c(cc(nc2CN)N2CCC[C@@H]2C)C1=O |r|
CCC(CC)n1c(C)nnc1-c1cccc(n1)N1Cc2c(cc(nc2CNC)N2CCC[C@@H]2C)C1=O |r|
CCCn1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2CN)N2[C@H](C)CC[C@H]2C)C1=O |r|
C[C@@H]1CC[C@@H](C)N1c1cc2C(=O)N(Cc2c(CN)n1)c1cccc(n1)N1[C@@H](C)COC1=O |r|
CCC(CC)n1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2CNC)N2CCC[C@@H]2C)C1=O |r|
CC[C@@H](C)n1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2CNC)C2(C)CC2)C1=O |r|
CCN(C(C)C)c1cc2C(=O)N(Cc2c(CN)n1)c1cccc(n1)-c1nncs1
CCN(C(C)C)c1cc2C(=O)N(Cc2c(CN)n1)c1cccc(n1)-c1nncn1CC
CCC(CC)n1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2CNC)C2CC2)C1=O
CCC(CC)n1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2CN)N2CCC[C@H]2C)C1=O |r|
CCC(CC)n1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2CNC)N2CCC[C@H]2C)C1=O |r|
CCN(C(C)C)c1cc2C(=O)N(Cc2c(CN)n1)c1cccc(n1)-c1nncn1C(C)C
CCCn1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2CN)N(CC)C(C)C)C1=O
CCC(CC)n1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2CN)N(C)C(C)C)C1=O
CCC(CC)n1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2CN)N2CCCC2(C)C)C1=O
CCC(CC)n1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2CN)N2CCC[C@@H]2C)C1=O |r|
CCC(CC)n1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2CN)N(C)CC)C1=O
CCn1c(C)nnc1-c1cccc(n1)N1Cc2c(cc(nc2CN)N2CCCC2(C)C)C1=O
CCCn1c(C)nnc1-c1cccc(n1)N1Cc2c(cc(nc2CN)N2CCCC2(C)C)C1=O
CC(C)n1c(C)nnc1-c1cccc(n1)N1Cc2c(cc(nc2CN)N2CCC[C@H]2C)C1=O |r|
CCn1c(C)nnc1-c1cccc(n1)N1Cc2c(cc(nc2CN)N2CCC[C@@H]2C)C1=O |r|
CCn1c(C)nnc1-c1cccc(n1)N1Cc2c(cc(nc2CN)N(C)C(C)C)C1=O
CCN(C)c1cc2C(=O)N(Cc2c(CN)n1)c1cccc(n1)-c1nnc(C)n1C(C)C
CCCn1c(C)nnc1-c1cccc(n1)N1Cc2c(cc(nc2CN)N(C)CC)C1=O
CC(C)n1c(C)nnc1-c1cccc(n1)N1Cc2c(cc(nc2CN)N2CCC[C@@H]2C)C1=O |r|
CCN(CC)c1cc2C(=O)N(Cc2c(CN)n1)c1cccc(n1)-c1nnc(C)n1CC
CC(C)n1c(C)nnc1-c1cccc(n1)N1Cc2c(cc(nc2CN)N2CCCC2(C)C)C1=O
CC(C)N(C)c1cc2C(=O)N(Cc2c(CN)n1)c1cccc(n1)-c1nnc(C)n1C(C)C
CCC(CC)n1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2CN)N(CC)C(C)C)C1=O
CCN(C(C)C)c1cc2C(=O)N(Cc2c(CN)n1)c1cccc(n1)-c1nnc(C)n1CC
CCn1c(C)nnc1-c1cccc(n1)N1Cc2c(cc(nc2CN)N2[C@H](C)CC[C@H]2C)C1=O |r|
CC(C)n1c(C)nnc1-c1cccc(n1)N1Cc2c(cc(nc2CN)N2[C@H](C)CC[C@H]2C)C1=O |r|
CCCn1c(C)nnc1-c1cccc(n1)N1Cc2c(cc(nc2CN)N(CC)CC)C1=O
CCN(C)c1cc2C(=O)N(Cc2c(CN)n1)c1cccc(n1)-c1nnc(C)n1CC
CCCn1c(C)nnc1-c1cccc(n1)N1Cc2c(cc(nc2CN)N(C)C(C)C)C1=O
CC[C@H](C)n1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2CNC)N(C)CC)C1=O |r|
CN(C)c1cc2C(=O)N(Cc2c(CN)n1)c1cccc(n1)N1[C@@H](CF)COC1=O |r|
CCCn1c(CC)nnc1-c1cccc(n1)N1Cc2c(cc(nc2CNC)N2CCC[C@H]2C)C1=O |r|
CCc1nnc(-c2cccc(n2)N2Cc3c(cc(nc3CNC)N3CCC[C@H]3C)C2=O)n1CC(C)C |r|
CNCc1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nncn1CC(C)C)N(C)C
CNCc1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nncn1[C@@H](C)C(C)C)N(C)C |r|
CNCc1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nncn1C1CCCC1)C1(C)CC1
CCC(CC(F)(F)F)n1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2CNC)C2(C)CC2)C1=O
CNCc1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nncn1[C@H](C)C(C)C)N(C)C |r|
CC[C@H](CO)n1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2CNC)C2(C)CC2)C1=O |r|
CC[C@@H](CO)n1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2CNC)C2(C)CC2)C1=O |r|
CCc1nnc(-c2cccc(n2)N2Cc3c(cc(nc3CN)N3CCC[C@H]3C)C2=O)n1CC |r|
CCCn1c(CC)nnc1-c1cccc(n1)N1Cc2c(cc(nc2CN)N2CCC[C@H]2C)C1=O |r|
CNCc1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nnc(C)n1C1CCC1)C1(C)CC1
Cc1nnc(-c2cccc(n2)N2Cc3c(cc(nc3CN)C3(C)CC3)C2=O)n1C1CCC1
COc1cc2CN(C)Cc2cc1Nc1ncc(Cl)c(Nc2ccccc2P(C)(C)=O)n1
COc1cc2CCN(C)Cc2cc1Nc1ncc(Cl)c(Nc2ccccc2P(C)(C)=O)n1
COc1cc2CCN(C)CCc2cc1Nc1ncc(Cl)c(Nc2ccccc2P(C)(C)=O)n1
COc1cc2CN(C)CCCc2cc1Nc1ncc(Cl)c(Nc2ccccc2P(C)(C)=O)n1
CN1CCc2cc(F)c(Nc3ncc(Cl)c(Nc4ccccc4P(C)(C)=O)n3)cc2C1
CN1CCc2cc(Cl)c(Nc3ncc(Cl)c(Nc4ccccc4P(C)(C)=O)n3)cc2C1
CCc1cc2CCN(C)Cc2cc1Nc1ncc(Cl)c(Nc2ccccc2P(C)(C)=O)n1
CN1CCc2cc(C=C)c(Nc3ncc(Cl)c(Nc4ccccc4P(C)(C)=O)n3)cc2C1
COc1c(Nc2ncc(Cl)c(Nc3ccccc3P(C)(C)=O)n2)cc2CN3CCCCC3Cc2c1N
COc1cc2CC3CCCCN3Cc2cc1Nc1ncc(Cl)c(Nc2ccccc2P(C)(C)=O)n1
COc1cc2CCN(Cc2cc1Nc1ncc(Cl)c(Nc2ccccc2P(C)(C)=O)n1)C(C)C
CCN1CCc2cc(OC)c(Nc3ncc(Cl)c(Nc4ccccc4P(C)(C)=O)n3)cc2C1
COc1cc2CCC[C@@H](N(C)C)c2cc1Nc1ncc(Cl)c(Nc2ccccc2P(C)(C)=O)n1
COc1cc2CC[C@@H](N(C)C)c2cc1Nc1ncc(Cl)c(Nc2ccccc2P(C)(C)=O)n1
COc1cc2CCC[C@H](N(C)C)c2cc1Nc1ncc(Cl)c(Nc2ccccc2P(C)(C)=O)n1
COc1cc2CC[C@H](N(C)C)c2cc1Nc1ncc(Cl)c(Nc2ccccc2P(C)(C)=O)n1
COc1cc2CC(Cc2cc1Nc1ncc(Cl)c(Nc2ccccc2P(C)(C)=O)n1)N(C)C
COc1cc2CN(C)CCc2cc1Nc1ncc(Cl)c(Nc2ccccc2P(C)(C)=O)n1
CCP(=O)(CC)c1ccccc1Nc1nc(Nc2cc3CN(C)CCc3cc2OC)ncc1Cl
CCP(=O)(CC)c1ccccc1Nc1nc(Nc2cc3CN(C)CCc3cc2Cl)ncc1Cl
CN1CCc2cc(Nc3ncc(Cl)c(Nc4ccccc4P(C)(C)=O)n3)c(Cl)cc2C1
COc1cc2CCN(C)Cc2cc1Nc1ncc(Br)c(Nc2ccccc2P(C)(C)=O)n1
COc1cc2CCN(C)Cc2cc1Nc1ncc(OC)c(Nc2ccccc2P(C)(C)=O)n1
CN1CCc2c(Br)cc(Nc3ncc(Cl)c(Nc4ccccc4P(C)(C)=O)n3)cc2C1
COc1cc2CCN(C)Cc2cc1Nc1nccc(Nc2ccccc2P(C)(C)=O)n1
COc1cc2CCN(C)Cc2cc1Nc1ncc(F)c(Nc2ccccc2P(C)(C)=O)n1
COc1cc2CCN(C)Cc2cc1Nc1ncc(c(Nc2ccccc2P(C)(C)=O)n1)C(F)(F)F
COc1cc2CCN(C)C(C)(C)c2cc1Nc1ncc(Cl)c(Nc2ccccc2P(C)(C)=O)n1
COc1cc2CCN(C)C(C)c2cc1Nc1ncc(Cl)c(Nc2ccccc2P(C)(C)=O)n1
COc1cc2CCN(C)Cc2cc1Nc1ncc(Cl)c(Nc2ccccc2S(=O)(=O)C(C)C)n1
COc1cc2CCN(C)Cc2cc1Nc1ncc(Cl)c(Nc2ccccc2C(=O)N(C)C)n1
CNC(=O)c1ccccc1Nc1nc(Nc2cc3CN(C)CCc3cc2OC)ncc1Cl
COc1cc2CCNC(=O)c2cc1Nc1ncc(Cl)c(Nc2ccccc2P(C)(C)=O)n1
COc1cc2CCCN(C)C(=O)c2cc1Nc1ncc(Cl)c(Nc2ccccc2P(C)(C)=O)n1
COc1cc2CCCN(C)Cc2cc1Nc1ncc(Cl)c(Nc2ccccc2P(C)(C)=O)n1
CCOc1cc2CCN(C)Cc2cc1Nc1ncc(Cl)c(Nc2ccccc2P(C)(C)=O)n1
CP(C)(=O)c1ccccc1Nc1nc(Nc2cc3CNCCc3cc2C(F)(F)F)ncc1Cl
COc1cc2CNCCc2cc1Nc1ncc(Cl)c(Nc2ccccc2P(C)(C)=O)n1
COc1cc2CCNCc2cc1Nc1ncc(Cl)c(Nc2ccccc2P(C)(C)=O)n1
COc1cc2c(CNCC2(C)C)cc1Nc1ncc(Cl)c(Nc2ccccc2P(C)(C)=O)n1
COc1cc2CCN(Cc2cc1Nc1ncc(Cl)c(Nc2ccccc2P(C)(C)=O)n1)C1COC1
COc1cc2c(CN(C)CC2(C)C)cc1Nc1ncc(Cl)c(Nc2ccccc2P(C)(C)=O)n1
CN1CCc2cc(c(Nc3ncc(Cl)c(Nc4ccccc4P(C)(C)=O)n3)cc2C1)C(F)(F)F
COc1cc2CCN(C)Cc2cc1Nc1ncc(C=C)c(Nc2ccccc2P(C)(C)=O)n1
COc1cc2CCN(C)Cc2cc1Nc1ncc(-c2cnn(C)c2)c(Nc2ccccc2P(C)(C)=O)n1
CCc1cnc(Nc2cc3CN(C)CCc3cc2OC)nc1Nc1ccccc1P(C)(C)=O
CNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N(C2CC(C2)N2CCCCC2)C(=O)C3(C)C)ccc1C |(9.2,8.23,;9.2,6.69,;7.87,5.92,;7.87,4.38,;6.53,6.69,;5.2,5.92,;3.86,6.69,;2.53,5.92,;2.53,4.38,;3.86,3.61,;3.86,2.07,;2.53,1.3,;1.2,2.07,;-.27,1.6,;-1.17,2.84,;-.27,4.09,;-.74,5.55,;-2.25,5.87,;.29,6.7,;1.2,3.61,;5.2,1.3,;5.2,-.24,;6.53,-1.01,;7.87,-.24,;7.87,1.3,;6.53,2.07,;9.33,1.78,;9.81,3.24,;9.11,4.62,;10.48,5.31,;11.18,3.94,;10.95,6.78,;9.92,7.92,;10.4,9.39,;11.91,9.71,;12.94,8.56,;12.46,7.1,;10.23,.53,;11.77,.53,;9.33,-.71,;8.7,-2.12,;10.66,-1.48,;3.86,8.23,;5.2,9,;6.53,8.23,;7.87,9,)|
CC(C)n1cnc2cc(nc(Nc3ccc(C)c(c3)C(=O)NC3CCC3)c12)-c1ccc2c(c1)N([C@H]1C[C@H](C1)N1CCCCC1)C(=O)C2(C)C |r,wU:34.38,36.43,(4.79,-2.11,;5.88,-1.02,;7.37,-1.42,;5.48,.47,;6.38,1.71,;5.48,2.96,;4.01,2.48,;2.68,3.25,;1.35,2.48,;1.35,.94,;2.68,.17,;2.68,-1.37,;1.35,-2.14,;.01,-1.37,;-1.32,-2.14,;-1.32,-3.68,;-2.65,-4.45,;.01,-4.45,;1.35,-3.68,;.01,-5.99,;-1.32,-6.76,;1.35,-6.76,;2.68,-5.99,;4.17,-6.39,;4.57,-4.9,;3.08,-4.5,;4.01,.94,;.01,3.25,;.01,4.79,;-1.32,5.56,;-2.65,4.79,;-2.65,3.25,;-1.32,2.48,;-4.12,2.78,;-4.52,1.29,;-3.75,-.04,;-5.08,-.81,;-5.85,.52,;-5.48,-2.3,;-6.97,-2.7,;-7.37,-4.19,;-6.28,-5.28,;-4.79,-4.88,;-4.39,-3.39,;-5.02,4.02,;-6.56,4.02,;-4.12,5.27,;-5.45,6.04,;-3.72,6.76,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@@H]2C[C@@H](C2)N2CCC(C)(C)C2)C(=O)C3(C)C)ccc1C |r,wU:27.29,29.34,(3.24,-5.99,;1.91,-6.76,;.57,-5.99,;-.76,-6.76,;.57,-4.45,;1.91,-3.68,;1.91,-2.14,;3.24,-1.37,;3.24,.17,;1.91,.94,;1.91,2.48,;3.24,3.25,;4.57,2.48,;6.04,2.96,;6.94,1.71,;6.04,.47,;6.44,-1.02,;5.35,-2.11,;7.92,-1.42,;4.57,.94,;.57,3.25,;.57,4.79,;-.76,5.56,;-2.09,4.79,;-2.09,3.25,;-.76,2.48,;-3.56,2.78,;-3.96,1.29,;-5.29,.52,;-4.52,-.81,;-3.19,-.04,;-4.92,-2.3,;-4.01,-3.55,;-4.92,-4.79,;-6.38,-4.32,;-7.92,-4.32,;-6.78,-5.8,;-6.38,-2.78,;-4.46,4.02,;-6,4.02,;-3.56,5.27,;-4.89,6.04,;-3.16,6.76,;.57,-1.37,;-.76,-2.14,;-.76,-3.68,;-2.09,-4.45,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@@H]2C[C@@H](C2)N2CC[C@@H](F)C2)C(=O)C3(C)C)ccc1C |r,wU:27.29,29.34,34.38,(3.14,-5.99,;1.8,-6.76,;.47,-5.99,;-.86,-6.76,;.47,-4.45,;1.8,-3.68,;1.8,-2.14,;3.14,-1.37,;3.14,.17,;1.8,.94,;1.8,2.48,;3.14,3.25,;4.47,2.48,;5.94,2.96,;6.84,1.71,;5.94,.47,;6.33,-1.02,;5.24,-2.11,;7.82,-1.42,;4.47,.94,;.47,3.25,;.47,4.79,;-.86,5.56,;-2.2,4.79,;-2.2,3.25,;-.86,2.48,;-3.66,2.78,;-4.06,1.29,;-5.39,.52,;-4.62,-.81,;-3.29,-.04,;-5.02,-2.3,;-4.12,-3.55,;-5.02,-4.79,;-6.49,-4.32,;-7.82,-5.09,;-6.49,-2.78,;-4.57,4.02,;-6.11,4.02,;-3.66,5.27,;-5,6.04,;-3.26,6.76,;.47,-1.37,;-.86,-2.14,;-.86,-3.68,;-2.2,-4.45,)|
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CNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@@H]2C[C@@H](C2)N2CC4C(C2)C4(F)F)C(=O)C3(C)C)ccc1C |r,wU:27.29,29.34,(3.05,-5.91,;1.72,-6.68,;.39,-5.91,;-.95,-6.68,;.39,-4.37,;1.72,-3.6,;1.72,-2.06,;3.05,-1.29,;3.05,.25,;1.72,1.02,;1.72,2.56,;3.05,3.33,;4.39,2.56,;5.85,3.04,;6.76,1.79,;5.85,.55,;6.25,-.94,;5.16,-2.03,;7.74,-1.34,;4.39,1.02,;.39,3.33,;.39,4.87,;-.95,5.64,;-2.28,4.87,;-2.28,3.33,;-.95,2.56,;-3.75,2.86,;-4.14,1.37,;-5.48,.6,;-4.71,-.74,;-3.37,.03,;-5.11,-2.22,;-6.57,-2.7,;-6.57,-4.24,;-5.11,-4.72,;-4.2,-3.47,;-6.25,-5.75,;-7.74,-6.14,;-5.16,-6.83,;-4.65,4.1,;-6.19,4.1,;-3.75,5.35,;-4.83,6.44,;-3.35,6.83,;.39,-1.29,;-.95,-2.06,;-.95,-3.6,;-2.28,-4.37,)|
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CNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@@H]2C[C@@H](C2)N[C@@H]2CCOC[C@H]2C)C(=O)C3(C)C)ccc1C |r,wU:27.29,29.34,32.35,wD:37.42,(3.97,-5.91,;2.64,-6.68,;1.3,-5.91,;-.03,-6.68,;1.3,-4.37,;2.64,-3.6,;2.64,-2.06,;3.97,-1.29,;3.97,.25,;2.64,1.02,;2.64,2.56,;3.97,3.33,;5.3,2.56,;6.77,3.04,;7.67,1.79,;6.77,.54,;7.17,-.94,;6.08,-2.03,;8.65,-1.34,;5.3,1.02,;1.3,3.33,;1.3,4.87,;-.03,5.64,;-1.36,4.87,;-1.36,3.33,;-.03,2.56,;-2.83,2.85,;-3.23,1.37,;-4.56,.6,;-3.79,-.74,;-2.46,.03,;-4.19,-2.22,;-5.68,-2.62,;-6.77,-1.53,;-8.25,-1.93,;-8.65,-3.42,;-7.57,-4.51,;-6.08,-4.11,;-4.99,-5.2,;-3.73,4.1,;-5.27,4.1,;-2.83,5.35,;-3.92,6.43,;-2.06,6.68,;1.3,-1.29,;-.03,-2.06,;-.03,-3.6,;-1.36,-4.37,)|
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Cc1ccc(Nc2nc(cc3ncn(C4CC4)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCC[C@@H](F)C2)C(=O)C3(C)C)cc1C(N)=O |r,wU:25.28,27.33,33.38,(-1.71,-4.45,;-.37,-3.68,;-.37,-2.14,;.96,-1.37,;2.29,-2.14,;3.63,-1.37,;3.63,.17,;2.29,.94,;2.29,2.48,;3.63,3.25,;4.96,2.48,;6.43,2.96,;7.33,1.71,;6.43,.47,;6.83,-1.02,;6.43,-2.51,;7.91,-2.11,;4.96,.94,;.96,3.25,;.96,4.79,;-.37,5.56,;-1.71,4.79,;-1.71,3.25,;-.37,2.48,;-3.17,2.78,;-3.57,1.29,;-2.8,-.04,;-4.13,-.81,;-4.9,.52,;-4.53,-2.3,;-3.42,-3.4,;-3.82,-4.91,;-5.33,-5.31,;-6.43,-4.2,;-7.91,-4.6,;-6.02,-2.7,;-4.08,4.02,;-5.62,4.02,;-3.17,5.27,;-4.26,6.36,;-2.77,6.76,;2.29,-3.68,;.96,-4.45,;.96,-5.99,;2.29,-6.76,;-.37,-6.76,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2cnc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C3(C)C)ccc1C |r,wU:27.29,29.34,(2.69,-5.99,;1.35,-6.76,;.02,-5.99,;-1.32,-6.76,;.02,-4.45,;1.35,-3.68,;1.35,-2.14,;2.69,-1.37,;2.69,.17,;1.35,.94,;1.35,2.48,;2.69,3.25,;4.02,2.48,;5.48,2.96,;6.39,1.71,;5.48,.47,;5.88,-1.02,;4.79,-2.11,;7.37,-1.42,;4.02,.94,;.02,3.25,;.02,4.79,;-1.32,5.56,;-2.65,4.79,;-2.65,3.25,;-1.32,2.48,;-4.11,2.78,;-4.51,1.29,;-3.74,-.04,;-5.08,-.81,;-5.85,.52,;-5.48,-2.3,;-6.96,-2.7,;-7.37,-4.2,;-6.27,-5.31,;-4.77,-4.91,;-4.36,-3.4,;-5.02,4.02,;-6.56,4.02,;-4.11,5.27,;-5.2,6.36,;-3.72,6.76,;.02,-1.37,;-1.32,-2.14,;-1.32,-3.68,;-2.65,-4.45,)|
CC(C)n1cnc2cc(nc(Nc3ccc(C)c(c3)C(=O)NC3(CC3)C(F)F)c12)-c1cnc2c(c1)N([C@H]1C[C@H](C1)N1CCCCC1)C(=O)C2(C)C |r,wU:36.40,38.45,(4.79,-1.16,;5.88,-.07,;7.37,-.47,;5.48,1.42,;6.39,2.66,;5.48,3.91,;4.02,3.43,;2.69,4.2,;1.35,3.43,;1.35,1.89,;2.69,1.12,;2.69,-.42,;1.35,-1.19,;.02,-.42,;-1.32,-1.19,;-1.32,-2.73,;-2.65,-3.5,;.02,-3.5,;1.35,-2.73,;.02,-5.04,;-1.32,-5.81,;1.35,-5.81,;2.69,-5.04,;4.23,-5.04,;3.46,-3.7,;3.46,-6.37,;5,-6.37,;2.69,-7.71,;4.02,1.89,;.02,4.2,;.02,5.74,;-1.32,6.51,;-2.65,5.74,;-2.65,4.2,;-1.32,3.43,;-4.11,3.73,;-4.51,2.24,;-3.74,.9,;-5.08,.13,;-5.85,1.47,;-5.48,-1.35,;-6.96,-1.75,;-7.37,-3.25,;-6.27,-4.36,;-4.77,-3.96,;-4.36,-2.46,;-5.02,4.97,;-6.56,4.97,;-4.11,6.22,;-5.2,7.31,;-3.72,7.71,)|
CC(C)n1cnc2cc(nc(Nc3ccc(C)c(c3)C(=O)NCC(F)F)c12)-c1ccc2c(c1)N([C@H]1C[C@H](C1)N1CCCCC1)C(=O)C2(C)C |r,wU:34.37,36.42,(4.79,-.18,;5.88,.9,;7.37,.51,;5.48,2.39,;6.39,3.64,;5.48,4.88,;4.02,4.41,;2.69,5.18,;1.35,4.41,;1.35,2.87,;2.69,2.1,;2.69,.56,;1.35,-.21,;.02,.56,;-1.32,-.21,;-1.32,-1.75,;-2.65,-2.52,;.02,-2.52,;1.35,-1.75,;.02,-4.06,;1.35,-4.83,;-1.32,-4.83,;-1.32,-6.37,;-2.65,-7.14,;-3.98,-6.37,;-2.65,-8.68,;4.02,2.87,;.02,5.18,;.02,6.72,;-1.32,7.49,;-2.65,6.72,;-2.65,5.18,;-1.32,4.41,;-4.11,4.7,;-4.51,3.21,;-3.74,1.88,;-5.08,1.11,;-5.85,2.44,;-5.48,-.38,;-6.96,-.77,;-7.37,-2.28,;-6.27,-3.38,;-4.77,-2.98,;-4.36,-1.48,;-5.02,5.95,;-6.56,5.95,;-4.11,7.19,;-5.45,7.96,;-3.72,8.68,)|
CC(C)n1cnc2cc(nc(Nc3ccc(C)c(c3)C(=O)NC(C)C(F)F)c12)-c1ccc2c(c1)N([C@H]1C[C@H](C1)N1CCCCC1)C(=O)C2(C)C |r,wU:35.38,37.43,(4.79,-.18,;5.88,.9,;7.37,.51,;5.48,2.39,;6.39,3.64,;5.48,4.88,;4.02,4.41,;2.69,5.18,;1.35,4.41,;1.35,2.87,;2.69,2.1,;2.69,.56,;1.35,-.21,;.02,.56,;-1.32,-.21,;-1.32,-1.75,;-2.65,-2.52,;.02,-2.52,;1.35,-1.75,;.02,-4.06,;1.35,-4.83,;-1.32,-4.83,;-1.32,-6.37,;.02,-7.14,;-2.65,-7.14,;-3.98,-6.37,;-2.65,-8.68,;4.02,2.87,;.02,5.18,;.02,6.72,;-1.32,7.49,;-2.65,6.72,;-2.65,5.18,;-1.32,4.41,;-4.11,4.7,;-4.51,3.21,;-3.74,1.88,;-5.08,1.11,;-5.85,2.44,;-5.48,-.38,;-6.96,-.77,;-7.37,-2.28,;-6.27,-3.38,;-4.77,-2.98,;-4.36,-1.48,;-5.02,5.95,;-6.56,5.95,;-4.11,7.19,;-5.45,7.96,;-3.72,8.68,)|
CC(C)n1cnc2cc(nc(Nc3ccc(C)c(c3)C(=O)N[C@@H](C)C(F)F)c12)-c1ccc2c(c1)N([C@H]1C[C@H](C1)N1CCCCC1)C(=O)C2(C)C |r,wU:35.38,37.43,22.23,(4.79,-.18,;5.88,.9,;7.37,.51,;5.48,2.39,;6.39,3.64,;5.48,4.88,;4.02,4.41,;2.69,5.18,;1.35,4.41,;1.35,2.87,;2.69,2.1,;2.69,.56,;1.35,-.21,;.02,.56,;-1.32,-.21,;-1.32,-1.75,;-2.65,-2.52,;.02,-2.52,;1.35,-1.75,;.02,-4.06,;1.35,-4.83,;-1.32,-4.83,;-1.32,-6.37,;.02,-7.14,;-2.65,-7.14,;-3.98,-6.37,;-2.65,-8.68,;4.02,2.87,;.02,5.18,;.02,6.72,;-1.32,7.49,;-2.65,6.72,;-2.65,5.18,;-1.32,4.41,;-4.11,4.7,;-4.51,3.21,;-3.74,1.88,;-5.08,1.11,;-5.85,2.44,;-5.47,-.38,;-6.96,-.77,;-7.37,-2.28,;-6.27,-3.38,;-4.77,-2.98,;-4.36,-1.48,;-5.02,5.95,;-6.56,5.95,;-4.11,7.19,;-5.45,7.96,;-3.72,8.68,)|
CC(C)n1cnc2cc(nc(Nc3ccc(C)c(c3)C(=O)N[C@H](C)C(F)F)c12)-c1ccc2c(c1)N([C@H]1C[C@H](C1)N1CCCCC1)C(=O)C2(C)C |r,wU:35.38,37.43,wD:22.23,(4.79,-.18,;5.88,.9,;7.37,.51,;5.48,2.39,;6.39,3.64,;5.48,4.88,;4.02,4.41,;2.69,5.18,;1.35,4.41,;1.35,2.87,;2.69,2.1,;2.69,.56,;1.35,-.21,;.02,.56,;-1.32,-.21,;-1.32,-1.75,;-2.65,-2.52,;.02,-2.52,;1.35,-1.75,;.02,-4.06,;1.35,-4.83,;-1.32,-4.83,;-1.32,-6.37,;.02,-7.14,;-2.65,-7.14,;-3.98,-6.37,;-2.65,-8.68,;4.02,2.87,;.02,5.18,;.02,6.72,;-1.32,7.49,;-2.65,6.72,;-2.65,5.18,;-1.32,4.41,;-4.11,4.7,;-4.51,3.21,;-3.74,1.88,;-5.08,1.11,;-5.85,2.44,;-5.47,-.38,;-6.96,-.77,;-7.37,-2.28,;-6.27,-3.38,;-4.77,-2.98,;-4.36,-1.48,;-5.02,5.95,;-6.56,5.95,;-4.11,7.19,;-5.45,7.96,;-3.72,8.68,)|
CCNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C32CCOCC2)ccc1C |r,wU:28.30,30.35,(.02,-8.66,;-1.32,-7.89,;-1.32,-6.35,;.02,-5.58,;1.35,-6.35,;.02,-4.04,;1.35,-3.27,;1.35,-1.73,;2.69,-.96,;2.69,.58,;1.35,1.35,;1.35,2.89,;2.69,3.66,;4.02,2.89,;5.48,3.37,;6.39,2.12,;5.48,.88,;5.88,-.61,;4.79,-1.7,;7.37,-1.01,;4.02,1.35,;.02,3.66,;.02,5.2,;-1.32,5.97,;-2.65,5.2,;-2.65,3.66,;-1.32,2.89,;-4.11,3.19,;-4.51,1.7,;-3.74,.37,;-5.08,-.4,;-5.85,.93,;-5.48,-1.89,;-6.96,-2.29,;-7.37,-3.79,;-6.27,-4.89,;-4.77,-4.5,;-4.36,-2.99,;-5.02,4.43,;-6.56,4.43,;-4.11,5.68,;-3.03,6.77,;-3.42,8.26,;-4.91,8.66,;-6,7.57,;-5.6,6.08,;.02,-.96,;-1.32,-1.73,;-1.32,-3.27,;-2.65,-4.04,)|
CC(C)n1cnc2cc(nc(Nc3ccc(C)c(c3)C(=O)NC3CCC3)c12)-c1ccc2c(c1)N([C@H]1C[C@H](C1)N1CCCCC1)C(=O)C21CCOCC1 |r,wU:34.38,36.43,(4.79,-.99,;5.88,.1,;7.37,-.3,;5.48,1.58,;6.39,2.83,;5.48,4.07,;4.02,3.6,;2.69,4.37,;1.35,3.6,;1.35,2.06,;2.69,1.29,;2.69,-.25,;1.35,-1.02,;.02,-.25,;-1.32,-1.02,;-1.32,-2.56,;-2.65,-3.33,;.02,-3.33,;1.35,-2.56,;.02,-4.87,;1.35,-5.64,;-1.32,-5.64,;-1.32,-7.18,;-2.4,-8.27,;-1.32,-9.36,;-.23,-8.27,;4.02,2.06,;.02,4.37,;.02,5.91,;-1.32,6.68,;-2.65,5.91,;-2.65,4.37,;-1.32,3.6,;-4.11,3.89,;-4.51,2.41,;-3.74,1.07,;-5.08,.3,;-5.85,1.64,;-5.48,-1.19,;-6.96,-1.58,;-7.37,-3.09,;-6.27,-4.19,;-4.77,-3.79,;-4.36,-2.29,;-5.02,5.14,;-6.56,5.14,;-4.11,6.38,;-3.03,7.47,;-3.42,8.96,;-4.91,9.36,;-6,8.27,;-5.6,6.78,)|
CCCNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C3(C)C)ccc1C |r,wU:29.31,31.36,(5.35,-5.99,;4.02,-6.76,;2.69,-5.99,;1.35,-6.76,;.02,-5.99,;-1.32,-6.76,;.02,-4.45,;1.35,-3.68,;1.35,-2.14,;2.69,-1.37,;2.69,.17,;1.35,.94,;1.35,2.48,;2.69,3.25,;4.02,2.48,;5.48,2.96,;6.39,1.71,;5.48,.47,;5.88,-1.02,;4.79,-2.11,;7.37,-1.42,;4.02,.94,;.02,3.25,;.02,4.79,;-1.32,5.56,;-2.65,4.79,;-2.65,3.25,;-1.32,2.48,;-4.11,2.78,;-4.51,1.29,;-3.74,-.04,;-5.08,-.81,;-5.85,.52,;-5.48,-2.3,;-6.96,-2.7,;-7.37,-4.2,;-6.27,-5.31,;-4.77,-4.91,;-4.36,-3.4,;-5.02,4.02,;-6.56,4.02,;-4.11,5.27,;-3.72,6.76,;-5.45,6.04,;.02,-1.37,;-1.32,-2.14,;-1.32,-3.68,;-2.65,-4.45,)|
CC(C)n1cnc2cc(nc(Nc3ccc(C)c(c3)C(=O)NCCC(F)F)c12)-c1ccc2c(c1)N([C@H]1C[C@H](C1)N1CCCCC1)C(=O)C2(C)C |r,wU:35.38,37.43,(4.79,-2.11,;5.88,-1.02,;7.37,-1.42,;5.48,.47,;6.39,1.71,;5.48,2.96,;4.02,2.48,;2.69,3.25,;1.35,2.48,;1.35,.94,;2.69,.17,;2.69,-1.37,;1.35,-2.14,;.02,-1.37,;-1.32,-2.14,;-1.32,-3.68,;-2.65,-4.45,;.02,-4.45,;1.35,-3.68,;.02,-5.99,;-1.32,-6.76,;1.35,-6.76,;2.69,-5.99,;4.02,-6.76,;5.35,-5.99,;6.69,-6.76,;5.35,-4.45,;4.02,.94,;.02,3.25,;.02,4.79,;-1.32,5.56,;-2.65,4.79,;-2.65,3.25,;-1.32,2.48,;-4.11,2.78,;-4.51,1.29,;-3.74,-.04,;-5.08,-.81,;-5.85,.52,;-5.48,-2.3,;-6.96,-2.7,;-7.37,-4.2,;-6.27,-5.31,;-4.77,-4.91,;-4.36,-3.4,;-5.02,4.02,;-6.56,4.02,;-4.11,5.27,;-3.72,6.76,;-5.45,6.04,)|
CC(C)n1cnc2cc(nc(Nc3ccc(C)c(c3)C(=O)NC3CC3)c12)-c1ccc2c(c1)N([C@H]1C[C@H](C1)N1CCCCC1)C(=O)C2(C)C |r,wU:33.37,35.42,(4.79,-2.11,;5.88,-1.02,;7.37,-1.42,;5.48,.47,;6.39,1.71,;5.48,2.96,;4.02,2.48,;2.69,3.25,;1.35,2.48,;1.35,.94,;2.69,.17,;2.69,-1.37,;1.35,-2.14,;.02,-1.37,;-1.32,-2.14,;-1.32,-3.68,;-2.65,-4.45,;.02,-4.45,;1.35,-3.68,;.02,-5.99,;-1.32,-6.76,;1.35,-6.76,;2.69,-5.99,;4.23,-5.99,;3.46,-4.65,;4.02,.94,;.02,3.25,;.02,4.79,;-1.32,5.56,;-2.65,4.79,;-2.65,3.25,;-1.32,2.48,;-4.11,2.78,;-4.51,1.29,;-3.74,-.04,;-5.08,-.81,;-5.85,.52,;-5.48,-2.3,;-6.96,-2.7,;-7.37,-4.2,;-6.27,-5.31,;-4.77,-4.91,;-4.36,-3.4,;-5.02,4.02,;-6.56,4.02,;-4.11,5.27,;-3.72,6.76,;-5.45,6.04,)|
CC(C)n1cnc2cc(nc(Nc3ccc(C)c(c3)C(=O)NC3(CC3)C(F)F)c12)-c1ccc2c(c1)N([C@H]1C[C@H](C1)N1CCCCC1)C(=O)C2(C)C |r,wU:36.40,38.45,(4.79,-1.34,;5.88,-.25,;7.37,-.65,;5.48,1.24,;6.39,2.48,;5.48,3.73,;4.02,3.25,;2.69,4.02,;1.35,3.25,;1.35,1.71,;2.69,.94,;2.69,-.6,;1.35,-1.37,;.02,-.6,;-1.32,-1.37,;-1.32,-2.91,;-2.65,-3.68,;.02,-3.68,;1.35,-2.91,;.02,-5.22,;-1.32,-5.99,;1.35,-5.99,;2.69,-5.22,;1.92,-3.88,;3.46,-3.88,;4.02,-5.99,;4.02,-7.53,;5.35,-5.22,;4.02,1.71,;.02,4.02,;.02,5.56,;-1.32,6.33,;-2.65,5.56,;-2.65,4.02,;-1.32,3.25,;-4.11,3.55,;-4.51,2.06,;-3.74,.73,;-5.08,-.04,;-5.85,1.29,;-5.48,-1.53,;-6.96,-1.93,;-7.37,-3.43,;-6.27,-4.54,;-4.77,-4.14,;-4.36,-2.63,;-5.02,4.79,;-6.56,4.79,;-4.11,6.04,;-3.72,7.53,;-5.45,6.81,)|
CC(C)n1cnc2cc(nc(Nc3ccc(C)c(c3)C(=O)NCC(C)(F)F)c12)-c1ccc2c(c1)N([C@H]1C[C@H](C1)N1CCCCC1)C(=O)C2(C)C |r,wU:35.38,37.43,(4.79,-1.44,;5.88,-.35,;7.37,-.75,;5.48,1.13,;6.39,2.38,;5.48,3.63,;4.02,3.15,;2.69,3.92,;1.35,3.15,;1.35,1.61,;2.69,.84,;2.69,-.7,;1.35,-1.47,;.02,-.7,;-1.32,-1.47,;-1.32,-3.01,;-2.65,-3.78,;.02,-3.78,;1.35,-3.01,;.02,-5.32,;-1.32,-6.09,;1.35,-6.09,;2.69,-5.32,;4.02,-6.09,;5.35,-5.32,;3.25,-7.42,;4.79,-7.42,;4.02,1.61,;.02,3.92,;.02,5.46,;-1.32,6.23,;-2.65,5.46,;-2.65,3.92,;-1.32,3.15,;-4.11,3.44,;-4.51,1.96,;-3.74,.62,;-5.08,-.15,;-5.85,1.19,;-5.48,-1.63,;-6.96,-2.03,;-7.37,-3.54,;-6.27,-4.64,;-4.77,-4.24,;-4.36,-2.74,;-5.02,4.69,;-6.56,4.69,;-4.11,5.94,;-3.72,7.42,;-5.45,6.71,)|
C[C@@H](CF)NC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C3(C)C)ccc1C |r,wU:30.32,32.37,1.0,(2.69,-4.45,;2.69,-5.99,;4.02,-6.76,;5.35,-5.99,;1.35,-6.76,;.02,-5.99,;-1.32,-6.76,;.02,-4.45,;1.35,-3.68,;1.35,-2.14,;2.69,-1.37,;2.69,.17,;1.35,.94,;1.35,2.48,;2.69,3.25,;4.02,2.48,;5.48,2.96,;6.39,1.71,;5.48,.47,;5.88,-1.02,;4.79,-2.11,;7.37,-1.42,;4.02,.94,;.02,3.25,;.02,4.79,;-1.32,5.56,;-2.65,4.79,;-2.65,3.25,;-1.32,2.48,;-4.11,2.78,;-4.51,1.29,;-3.74,-.04,;-5.08,-.81,;-5.85,.52,;-5.48,-2.3,;-6.96,-2.7,;-7.37,-4.2,;-6.27,-5.31,;-4.77,-4.91,;-4.36,-3.4,;-5.02,4.02,;-6.56,4.02,;-4.11,5.27,;-3.72,6.76,;-5.45,6.04,;.02,-1.37,;-1.32,-2.14,;-1.32,-3.68,;-2.65,-4.45,)|
C[C@H](CF)NC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C3(C)C)ccc1C |r,wU:30.32,32.37,wD:1.0,(2.69,-4.45,;2.69,-5.99,;4.02,-6.76,;5.35,-5.99,;1.35,-6.76,;.02,-5.99,;-1.32,-6.76,;.02,-4.45,;1.35,-3.68,;1.35,-2.14,;2.69,-1.37,;2.69,.17,;1.35,.94,;1.35,2.48,;2.69,3.25,;4.02,2.48,;5.48,2.96,;6.39,1.71,;5.48,.47,;5.88,-1.02,;4.79,-2.11,;7.37,-1.42,;4.02,.94,;.02,3.25,;.02,4.79,;-1.32,5.56,;-2.65,4.79,;-2.65,3.25,;-1.32,2.48,;-4.11,2.78,;-4.51,1.29,;-3.74,-.04,;-5.08,-.81,;-5.85,.52,;-5.48,-2.3,;-6.96,-2.7,;-7.37,-4.2,;-6.27,-5.31,;-4.77,-4.91,;-4.36,-3.4,;-5.02,4.02,;-6.56,4.02,;-4.11,5.27,;-3.72,6.76,;-5.45,6.04,;.02,-1.37,;-1.32,-2.14,;-1.32,-3.68,;-2.65,-4.45,)|
CC(C)n1cnc2cc(nc(Nc3ccc(C)c(c3)C(=O)NC(CF)CF)c12)-c1ccc2c(c1)N([C@H]1C[C@H](C1)N1CCCCC1)C(=O)C2(C)C |r,wU:35.38,37.43,(4.79,-2.11,;5.88,-1.02,;7.37,-1.42,;5.48,.47,;6.39,1.71,;5.48,2.96,;4.02,2.48,;2.69,3.25,;1.35,2.48,;1.35,.94,;2.69,.17,;2.69,-1.37,;1.35,-2.14,;.02,-1.37,;-1.32,-2.14,;-1.32,-3.68,;-2.65,-4.45,;.02,-4.45,;1.35,-3.68,;.02,-5.99,;-1.32,-6.76,;1.35,-6.76,;2.69,-5.99,;4.02,-6.76,;5.35,-5.99,;2.69,-4.45,;4.02,-3.68,;4.02,.94,;.02,3.25,;.02,4.79,;-1.32,5.56,;-2.65,4.79,;-2.65,3.25,;-1.32,2.48,;-4.11,2.78,;-4.51,1.29,;-3.74,-.04,;-5.08,-.81,;-5.85,.52,;-5.48,-2.3,;-6.96,-2.7,;-7.37,-4.2,;-6.27,-5.31,;-4.77,-4.91,;-4.36,-3.4,;-5.02,4.02,;-6.56,4.02,;-4.11,5.27,;-3.72,6.76,;-5.45,6.04,)|
CC(C)n1cnc2cc(nc(Nc3ccc(C)c(c3)C(=O)NC3(CC3)C(F)F)c12)-c1ccc2c(c1)N([C@H]1C[C@H](C1)N1CCCCC1)C(=O)C21CCOCC1 |r,wU:36.40,38.45,(4.79,-2.08,;5.88,-.99,;7.37,-1.39,;5.48,.49,;6.39,1.74,;5.48,2.99,;4.02,2.51,;2.69,3.28,;1.35,2.51,;1.35,.97,;2.69,.2,;2.69,-1.34,;1.35,-2.11,;.02,-1.34,;-1.32,-2.11,;-1.32,-3.65,;-2.65,-4.42,;.02,-4.42,;1.35,-3.65,;.02,-5.96,;-1.32,-6.73,;1.35,-6.73,;2.69,-5.96,;1.92,-4.63,;3.46,-4.63,;4.02,-6.73,;5.35,-5.96,;4.02,-8.27,;4.02,.97,;.02,3.28,;.02,4.82,;-1.32,5.59,;-2.65,4.82,;-2.65,3.28,;-1.32,2.51,;-4.11,2.8,;-4.51,1.32,;-3.74,-.02,;-5.08,-.79,;-5.85,.55,;-5.48,-2.28,;-6.96,-2.67,;-7.37,-4.18,;-6.27,-5.28,;-4.77,-4.88,;-4.36,-3.38,;-5.02,4.05,;-6.56,4.05,;-4.11,5.3,;-3.03,6.38,;-3.42,7.87,;-4.91,8.27,;-6,7.18,;-5.6,5.69,)|
Cc1ccc(Nc2nc(cc3ncn(C4CC4)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C3(C)C)cc1C(N)=O |r,wU:25.28,27.33,(-2.45,-4.45,;-1.12,-3.68,;-1.12,-2.14,;.22,-1.37,;1.55,-2.14,;2.88,-1.37,;2.88,.17,;1.55,.94,;1.55,2.48,;2.88,3.25,;4.22,2.48,;5.68,2.96,;6.59,1.71,;5.68,.47,;6.08,-1.02,;5.68,-2.51,;7.17,-2.11,;4.22,.94,;.22,3.25,;.22,4.79,;-1.12,5.56,;-2.45,4.79,;-2.45,3.25,;-1.12,2.48,;-3.91,2.78,;-4.31,1.29,;-3.54,-.04,;-4.88,-.81,;-5.65,.52,;-5.28,-2.3,;-6.76,-2.7,;-7.17,-4.2,;-6.07,-5.31,;-4.57,-4.91,;-4.16,-3.4,;-4.82,4.02,;-6.36,4.02,;-3.91,5.27,;-3.52,6.76,;-5.25,6.04,;1.55,-3.68,;.22,-4.45,;.22,-5.99,;-1.12,-6.76,;1.55,-6.76,)|
CNC(=O)c1cc(Oc2nc(cc3ncn(C4CC4)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C3(C)C)ccc1C |r,wU:27.30,29.35,(-1.12,-7.53,;-1.12,-5.99,;.22,-5.22,;1.55,-5.99,;.22,-3.68,;1.55,-2.91,;1.55,-1.37,;2.88,-.6,;2.88,.94,;1.55,1.71,;1.55,3.25,;2.88,4.02,;4.22,3.25,;5.68,3.73,;6.59,2.48,;5.68,1.24,;6.08,-.25,;5.68,-1.74,;7.17,-1.34,;4.22,1.71,;.22,4.02,;.22,5.56,;-1.12,6.33,;-2.45,5.56,;-2.45,4.02,;-1.12,3.25,;-3.91,3.55,;-4.31,2.06,;-3.54,.73,;-4.88,-.04,;-5.65,1.29,;-5.28,-1.53,;-6.76,-1.93,;-7.17,-3.43,;-6.07,-4.54,;-4.57,-4.14,;-4.16,-2.63,;-4.82,4.79,;-6.36,4.79,;-3.91,6.04,;-3.52,7.53,;-5.25,6.81,;.22,-.6,;-1.12,-1.37,;-1.12,-2.91,;-2.45,-3.68,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C32CCOCC2)c(F)cc1C |r,wU:27.29,29.34,(2.69,-6.73,;1.35,-7.5,;.02,-6.73,;-1.32,-7.5,;.02,-5.19,;1.35,-4.42,;1.35,-2.88,;2.69,-2.11,;2.69,-.57,;1.35,.2,;1.35,1.74,;2.69,2.51,;4.02,1.74,;5.48,2.22,;6.39,.97,;5.48,-.28,;5.88,-1.76,;7.37,-2.16,;4.79,-2.85,;4.02,.2,;.02,2.51,;.02,4.05,;-1.32,4.82,;-2.65,4.05,;-2.65,2.51,;-1.32,1.74,;-4.11,2.03,;-4.51,.55,;-3.74,-.79,;-5.08,-1.56,;-5.85,-.22,;-5.48,-3.05,;-6.96,-3.44,;-7.37,-4.95,;-6.27,-6.05,;-4.77,-5.65,;-4.36,-4.15,;-5.02,3.28,;-6.56,3.28,;-4.11,4.53,;-3.03,5.61,;-3.42,7.1,;-4.91,7.5,;-6,6.41,;-5.6,4.92,;.02,-2.11,;.02,-.57,;-1.32,-2.88,;-1.32,-4.42,;-2.65,-5.19,)|
Cc1ccc(Nc2nc(cc3ncn(C4CC4)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCC[C@H](O)C2)C(=O)C3(C)C)cc1C(N)=O |r,wU:25.28,27.33,wD:33.38,(-1.71,-4.45,;-.37,-3.68,;-.37,-2.14,;.96,-1.37,;2.3,-2.14,;3.63,-1.37,;3.63,.17,;2.3,.94,;2.3,2.48,;3.63,3.25,;4.96,2.48,;6.43,2.96,;7.33,1.71,;6.43,.47,;6.83,-1.02,;6.43,-2.51,;7.91,-2.11,;4.96,.94,;.96,3.25,;.96,4.79,;-.37,5.56,;-1.71,4.79,;-1.71,3.25,;-.37,2.48,;-3.17,2.78,;-3.57,1.29,;-2.8,-.04,;-4.13,-.81,;-4.9,.52,;-4.53,-2.3,;-3.42,-3.4,;-3.82,-4.91,;-5.33,-5.31,;-6.43,-4.2,;-7.91,-4.6,;-6.02,-2.7,;-4.08,4.02,;-5.62,4.02,;-3.17,5.27,;-2.77,6.76,;-4.26,6.36,;2.3,-3.68,;.96,-4.45,;.96,-5.99,;2.3,-6.76,;-.37,-6.76,)|
Cc1ccc(Nc2nc(cc3ncn(C4CC4)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCC[C@@H](O)C2)C(=O)C3(C)C)cc1C(N)=O |r,wU:25.28,27.33,33.38,(-1.71,-4.45,;-.37,-3.68,;-.37,-2.14,;.96,-1.37,;2.3,-2.14,;3.63,-1.37,;3.63,.17,;2.3,.94,;2.3,2.48,;3.63,3.25,;4.96,2.48,;6.43,2.96,;7.33,1.71,;6.43,.47,;6.83,-1.02,;6.43,-2.51,;7.91,-2.11,;4.96,.94,;.96,3.25,;.96,4.79,;-.37,5.56,;-1.71,4.79,;-1.71,3.25,;-.37,2.48,;-3.17,2.78,;-3.57,1.29,;-2.8,-.04,;-4.13,-.81,;-4.9,.52,;-4.53,-2.3,;-3.42,-3.4,;-3.82,-4.91,;-5.33,-5.31,;-6.43,-4.2,;-7.91,-4.6,;-6.02,-2.7,;-4.08,4.02,;-5.62,4.02,;-3.17,5.27,;-2.77,6.76,;-4.26,6.36,;2.3,-3.68,;.96,-4.45,;.96,-5.99,;2.3,-6.76,;-.37,-6.76,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C4CC4)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCC(C)(C)C2)C(=O)C3(C)C)ccc1C |r,wU:27.30,29.35,(3.63,-5.99,;2.29,-6.76,;.96,-5.99,;-.37,-6.76,;.96,-4.45,;2.29,-3.68,;2.29,-2.14,;3.63,-1.37,;3.63,.17,;2.29,.94,;2.29,2.48,;3.63,3.25,;4.96,2.48,;6.43,2.96,;7.33,1.71,;6.43,.47,;6.83,-1.02,;6.43,-2.51,;7.91,-2.11,;4.96,.94,;.96,3.25,;.96,4.79,;-.37,5.56,;-1.71,4.79,;-1.71,3.25,;-.37,2.48,;-3.17,2.78,;-3.57,1.29,;-2.8,-.04,;-4.13,-.81,;-4.9,.52,;-4.53,-2.3,;-3.42,-3.4,;-3.82,-4.91,;-5.33,-5.31,;-6.43,-4.2,;-7.91,-3.8,;-7.2,-5.54,;-6.02,-2.7,;-4.08,4.02,;-5.62,4.02,;-3.17,5.27,;-2.77,6.76,;-4.5,6.04,;.96,-1.37,;-.37,-2.14,;-.37,-3.68,;-1.71,-4.45,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCOCC2)C(=O)C3(C)C)ccc1C |r,wU:27.29,29.34,(1.35,-7.53,;1.35,-5.99,;.02,-5.22,;-1.32,-5.99,;.02,-3.68,;1.35,-2.91,;1.35,-1.37,;2.69,-.6,;2.69,.94,;1.35,1.71,;1.35,3.25,;2.69,4.02,;4.02,3.25,;5.48,3.73,;6.39,2.48,;5.48,1.24,;5.88,-.25,;7.37,-.65,;4.79,-1.34,;4.02,1.71,;.02,4.02,;.02,5.56,;-1.32,6.33,;-2.65,5.56,;-2.65,4.02,;-1.32,3.25,;-4.11,3.55,;-4.51,2.06,;-3.74,.73,;-5.08,-.04,;-5.85,1.29,;-5.48,-1.53,;-6.96,-1.93,;-7.37,-3.43,;-6.27,-4.54,;-4.77,-4.14,;-4.36,-2.63,;-5.02,4.79,;-6.56,4.79,;-4.11,6.04,;-3.72,7.53,;-5.2,7.13,;.02,-.6,;-1.32,-1.37,;-1.32,-2.91,;-2.65,-3.68,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C4CC4)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C3(C)C)ccc1Cl |r,wU:27.30,29.35,(1.55,-7.53,;1.55,-5.99,;.22,-5.22,;-1.12,-5.99,;.22,-3.68,;1.55,-2.91,;1.55,-1.37,;2.88,-.6,;2.88,.94,;1.55,1.71,;1.55,3.25,;2.88,4.02,;4.22,3.25,;5.68,3.73,;6.59,2.48,;5.68,1.24,;6.08,-.25,;5.68,-1.74,;7.17,-1.34,;4.22,1.71,;.22,4.02,;.22,5.56,;-1.12,6.33,;-2.45,5.56,;-2.45,4.02,;-1.12,3.25,;-3.91,3.55,;-4.31,2.06,;-3.54,.73,;-4.88,-.04,;-5.65,1.29,;-5.28,-1.53,;-6.76,-1.93,;-7.17,-3.43,;-6.07,-4.54,;-4.57,-4.14,;-4.16,-2.63,;-4.82,4.79,;-6.36,4.79,;-3.91,6.04,;-3.52,7.53,;-5,7.13,;.22,-.6,;-1.12,-1.37,;-1.12,-2.91,;-2.45,-3.68,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C4CC4)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C32CCN(CC2)C(=O)C23CC(C2)C3)ccc1Cl |r,wU:27.30,29.35,(2.88,-8.79,;1.55,-9.56,;.22,-8.79,;-1.12,-9.56,;.22,-7.25,;1.55,-6.48,;1.55,-4.94,;2.88,-4.17,;2.88,-2.63,;1.55,-1.86,;1.55,-.32,;2.88,.45,;4.22,-.32,;5.68,.16,;6.59,-1.09,;5.68,-2.33,;6.08,-3.82,;5.68,-5.31,;7.17,-4.91,;4.22,-1.86,;.22,.45,;.22,1.99,;-1.12,2.76,;-2.45,1.99,;-2.45,.45,;-1.12,-.32,;-3.91,-.02,;-4.31,-1.51,;-3.54,-2.85,;-4.88,-3.62,;-5.65,-2.28,;-5.28,-5.1,;-6.76,-5.5,;-7.17,-7,;-6.07,-8.11,;-4.57,-7.71,;-4.16,-6.21,;-4.82,1.22,;-6.36,1.22,;-3.91,2.47,;-2.83,3.56,;-3.22,5.04,;-4.71,5.44,;-5.8,4.35,;-5.4,2.87,;-5.11,6.93,;-6.6,7.33,;-4.02,8.02,;-2.48,8.02,;-2.48,9.56,;-4.02,9.56,;-3.47,8.97,;.22,-4.17,;-1.12,-4.94,;-1.12,-6.48,;-2.45,-7.25,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C4CC4)c23)-c2ccc3c(c2)N([C@@H]2C[C@@H](C2)N2C[C@H]4CC[C@@H]2C4)C(=O)C32CCN(CC2)C(=O)C2COC2)ccc1C |r,wU:27.30,29.35,wD:36.42,33.43,(2.88,-8.79,;1.55,-9.56,;.22,-8.79,;-1.12,-9.56,;.22,-7.25,;1.55,-6.48,;1.55,-4.94,;2.88,-4.17,;2.88,-2.63,;1.55,-1.86,;1.55,-.32,;2.88,.45,;4.22,-.32,;5.68,.16,;6.59,-1.09,;5.68,-2.33,;6.08,-3.82,;5.68,-5.31,;7.17,-4.91,;4.22,-1.86,;.22,.45,;.22,1.99,;-1.12,2.76,;-2.45,1.99,;-2.45,.45,;-1.12,-.32,;-3.91,-.02,;-4.31,-1.51,;-5.65,-2.28,;-4.88,-3.62,;-3.54,-2.85,;-5.28,-5.1,;-4.16,-6.21,;-4.57,-7.71,;-6.07,-8.11,;-7.17,-7,;-6.76,-5.5,;-5.99,-6.84,;-4.82,1.22,;-6.36,1.22,;-3.91,2.47,;-2.83,3.56,;-3.22,5.04,;-4.71,5.44,;-5.8,4.35,;-5.4,2.87,;-5.11,6.93,;-6.6,7.33,;-4.02,8.02,;-2.48,8.02,;-2.48,9.56,;-4.02,9.56,;.22,-4.17,;-1.12,-4.94,;-1.12,-6.48,;-2.45,-7.25,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C4CC4)c23)-c2ccc3c(c2)N([C@@H]2C[C@@H](C2)N2C[C@H]4CC[C@@H]2C4)C(=O)C32CCN(CC2)C(=O)C23CC(C2)C3)ccc1C |r,wU:27.30,29.35,wD:36.42,33.43,(2.88,-8.79,;1.55,-9.56,;.22,-8.79,;-1.12,-9.56,;.22,-7.25,;1.55,-6.48,;1.55,-4.94,;2.88,-4.17,;2.88,-2.63,;1.55,-1.86,;1.55,-.32,;2.88,.45,;4.22,-.32,;5.68,.16,;6.59,-1.09,;5.68,-2.33,;6.08,-3.82,;5.68,-5.31,;7.17,-4.91,;4.22,-1.86,;.22,.45,;.22,1.99,;-1.12,2.76,;-2.45,1.99,;-2.45,.45,;-1.12,-.32,;-3.91,-.02,;-4.31,-1.51,;-5.65,-2.28,;-4.88,-3.62,;-3.54,-2.85,;-5.28,-5.1,;-4.16,-6.21,;-4.57,-7.71,;-6.07,-8.11,;-7.17,-7,;-6.76,-5.5,;-5.99,-6.84,;-4.82,1.22,;-6.36,1.22,;-3.91,2.47,;-2.83,3.56,;-3.22,5.04,;-4.71,5.44,;-5.8,4.35,;-5.4,2.87,;-5.11,6.93,;-6.6,7.33,;-4.02,8.02,;-2.48,8.02,;-2.48,9.56,;-4.02,9.56,;-3.47,8.97,;.22,-4.17,;-1.12,-4.94,;-1.12,-6.48,;-2.45,-7.25,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C4CC4)c23)-c2ccc3c(c2)N([C@@H]2C[C@@H](C2)N2C[C@H]4CC[C@@H]2C4)C(=O)C32CCN(CC2)C(C)=O)ccc1C |r,wU:27.30,29.35,wD:36.42,33.43,(2.88,-8.02,;1.55,-8.79,;.22,-8.02,;-1.12,-8.79,;.22,-6.48,;1.55,-5.71,;1.55,-4.17,;2.88,-3.4,;2.88,-1.86,;1.55,-1.09,;1.55,.45,;2.88,1.22,;4.22,.45,;5.68,.93,;6.59,-.32,;5.68,-1.56,;6.08,-3.05,;5.68,-4.54,;7.17,-4.14,;4.22,-1.09,;.22,1.22,;.22,2.76,;-1.12,3.53,;-2.45,2.76,;-2.45,1.22,;-1.12,.45,;-3.91,.75,;-4.31,-.74,;-5.65,-1.51,;-4.88,-2.85,;-3.54,-2.08,;-5.28,-4.33,;-4.16,-5.44,;-4.57,-6.94,;-6.07,-7.34,;-7.17,-6.23,;-6.76,-4.73,;-5.99,-6.07,;-4.82,1.99,;-6.36,1.99,;-3.91,3.24,;-2.83,4.33,;-3.22,5.81,;-4.71,6.21,;-5.8,5.12,;-5.4,3.64,;-5.11,7.7,;-4.02,8.79,;-6.6,8.1,;.22,-3.4,;-1.12,-4.17,;-1.12,-5.71,;-2.45,-6.48,)|
CCC1(CC)C(=O)N([C@H]2C[C@H](C2)N2CCCCC2)c2cc(ccc12)-c1cc2ncn(C(C)C)c2c(Nc2ccc(C)c(c2)C(=O)NC)n1 |r,wU:8.7,10.12,(-6.69,6.53,;-5.2,6.93,;-4.11,5.84,;-3.72,7.33,;-2.23,7.73,;-5.02,4.59,;-6.56,4.59,;-4.11,3.35,;-4.51,1.86,;-3.74,.53,;-5.08,-.24,;-5.85,1.09,;-5.48,-1.73,;-6.96,-2.13,;-7.37,-3.63,;-6.27,-4.73,;-4.77,-4.34,;-4.36,-2.83,;-2.65,3.82,;-1.32,3.05,;.02,3.82,;.02,5.36,;-1.32,6.13,;-2.65,5.36,;1.35,3.05,;2.69,3.82,;4.02,3.05,;5.48,3.53,;6.39,2.28,;5.48,1.04,;5.88,-.45,;7.37,-.85,;4.79,-1.54,;4.02,1.51,;2.69,.74,;2.69,-.8,;1.35,-1.57,;.02,-.8,;-1.32,-1.57,;-1.32,-3.11,;-2.65,-3.88,;.02,-3.88,;1.35,-3.11,;.02,-5.42,;-1.32,-6.19,;1.35,-6.19,;1.35,-7.73,;1.35,1.51,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C32CCN(CC2)C(C)=O)ccc1C |r,wU:27.29,29.34,(2.69,-8.02,;1.35,-8.79,;.02,-8.02,;-1.32,-8.79,;.02,-6.48,;1.35,-5.71,;1.35,-4.17,;2.69,-3.4,;2.69,-1.86,;1.35,-1.09,;1.35,.45,;2.69,1.22,;4.02,.45,;5.48,.93,;6.39,-.32,;5.48,-1.56,;5.88,-3.05,;7.37,-3.45,;4.79,-4.14,;4.02,-1.09,;.02,1.22,;.02,2.76,;-1.32,3.53,;-2.65,2.76,;-2.65,1.22,;-1.32,.45,;-4.11,.75,;-4.51,-.74,;-3.74,-2.08,;-5.08,-2.85,;-5.85,-1.51,;-5.48,-4.33,;-6.96,-4.73,;-7.37,-6.23,;-6.27,-7.34,;-4.77,-6.94,;-4.36,-5.44,;-5.02,1.99,;-6.56,1.99,;-4.11,3.24,;-3.03,4.33,;-3.42,5.81,;-4.91,6.21,;-6,5.12,;-5.6,3.64,;-5.31,7.7,;-4.22,8.79,;-6.8,8.1,;.02,-3.4,;-1.32,-4.17,;-1.32,-5.71,;-2.65,-6.48,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C4CC4)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C32CCN(CC2)C(C)=O)ccc1Cl |r,wU:27.30,29.35,(2.88,-8.02,;1.55,-8.79,;.22,-8.02,;-1.12,-8.79,;.22,-6.48,;1.55,-5.71,;1.55,-4.17,;2.88,-3.4,;2.88,-1.86,;1.55,-1.09,;1.55,.45,;2.88,1.22,;4.22,.45,;5.68,.93,;6.59,-.32,;5.68,-1.56,;6.08,-3.05,;5.68,-4.54,;7.17,-4.14,;4.22,-1.09,;.22,1.22,;.22,2.76,;-1.12,3.53,;-2.45,2.76,;-2.45,1.22,;-1.12,.45,;-3.91,.75,;-4.31,-.74,;-3.54,-2.08,;-4.88,-2.85,;-5.65,-1.51,;-5.28,-4.33,;-6.76,-4.73,;-7.17,-6.23,;-6.07,-7.34,;-4.57,-6.94,;-4.16,-5.44,;-4.82,1.99,;-6.36,1.99,;-3.91,3.24,;-2.83,4.33,;-3.22,5.81,;-4.71,6.21,;-5.8,5.12,;-5.4,3.64,;-5.11,7.7,;-4.02,8.79,;-6.6,8.1,;.22,-3.4,;-1.12,-4.17,;-1.12,-5.71,;-2.45,-6.48,)|
CC[C@H](C)n1cnc2cc(nc(Nc3ccc(C)c(c3)C(=O)NC)c12)-c1ccc2c(c1)N([C@H]1C[C@H](C1)N1CCCCC1)C(=O)C21CCN(CC1)C(C)=O |r,wU:32.35,34.40,wD:2.2,(7.91,-2.36,;6.83,-3.45,;5.34,-3.05,;4.25,-4.14,;4.94,-1.56,;5.84,-.32,;4.94,.93,;3.47,.45,;2.14,1.22,;.81,.45,;.81,-1.09,;2.14,-1.86,;2.14,-3.4,;.81,-4.17,;-.53,-3.4,;-1.86,-4.17,;-1.86,-5.71,;-3.19,-6.48,;-.53,-6.48,;.81,-5.71,;-.53,-8.02,;-1.86,-8.79,;.81,-8.79,;2.14,-8.02,;3.47,-1.09,;-.53,1.22,;-.53,2.76,;-1.86,3.53,;-3.19,2.76,;-3.19,1.22,;-1.86,.45,;-4.66,.75,;-5.06,-.74,;-4.29,-2.08,;-5.62,-2.85,;-6.39,-1.51,;-6.02,-4.33,;-7.51,-4.73,;-7.91,-6.23,;-6.82,-7.34,;-5.31,-6.94,;-4.91,-5.44,;-5.56,1.99,;-7.1,1.99,;-4.66,3.24,;-3.57,4.33,;-3.97,5.81,;-5.46,6.21,;-6.54,5.12,;-6.15,3.64,;-5.85,7.7,;-4.77,8.79,;-7.34,8.1,)|
CCn1cnc2cc(nc(Nc3ccc(C)c(c3)C(=O)NC)c12)-c1ccc2c(c1)N([C@H]1C[C@H](C1)N1CCCCC1)C(=O)C21CCN(CC1)C(C)=O |r,wU:30.33,32.38,(7.37,-3.45,;5.88,-3.05,;5.48,-1.56,;6.39,-.32,;5.48,.93,;4.02,.45,;2.69,1.22,;1.35,.45,;1.35,-1.09,;2.69,-1.86,;2.69,-3.4,;1.35,-4.17,;.02,-3.4,;-1.32,-4.17,;-1.32,-5.71,;-2.65,-6.48,;.02,-6.48,;1.35,-5.71,;.02,-8.02,;-1.32,-8.79,;1.35,-8.79,;2.69,-8.02,;4.02,-1.09,;.02,1.22,;.02,2.76,;-1.32,3.53,;-2.65,2.76,;-2.65,1.22,;-1.32,.45,;-4.11,.75,;-4.51,-.74,;-3.74,-2.08,;-5.08,-2.85,;-5.85,-1.51,;-5.48,-4.33,;-6.96,-4.73,;-7.37,-6.23,;-6.27,-7.34,;-4.77,-6.94,;-4.36,-5.44,;-5.02,1.99,;-6.56,1.99,;-4.11,3.24,;-3.03,4.33,;-3.42,5.81,;-4.91,6.21,;-6,5.12,;-5.6,3.64,;-5.31,7.7,;-4.22,8.79,;-6.8,8.1,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C4CC4)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C32CCN(CC2)C(=O)OC)ccc1C |r,wU:27.30,29.35,(2.88,-8.02,;1.55,-8.79,;.22,-8.02,;-1.12,-8.79,;.22,-6.48,;1.55,-5.71,;1.55,-4.17,;2.88,-3.4,;2.88,-1.86,;1.55,-1.09,;1.55,.45,;2.88,1.22,;4.22,.45,;5.68,.93,;6.59,-.32,;5.68,-1.56,;6.08,-3.05,;5.68,-4.54,;7.17,-4.14,;4.22,-1.09,;.22,1.22,;.22,2.76,;-1.12,3.53,;-2.45,2.76,;-2.45,1.22,;-1.12,.45,;-3.91,.75,;-4.31,-.74,;-3.54,-2.08,;-4.88,-2.85,;-5.65,-1.51,;-5.28,-4.33,;-6.76,-4.73,;-7.17,-6.23,;-6.07,-7.34,;-4.57,-6.94,;-4.16,-5.44,;-4.82,1.99,;-6.36,1.99,;-3.91,3.24,;-2.83,4.33,;-3.22,5.81,;-4.71,6.21,;-5.8,5.12,;-5.4,3.64,;-5.11,7.7,;-6.6,8.1,;-4.02,8.79,;-2.53,8.39,;.22,-3.4,;-1.12,-4.17,;-1.12,-5.71,;-2.45,-6.48,)|
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CCn1cnc2cc(nc(Nc3cc(C(=O)NC(C)C)c(C)cc3F)c12)-c1ccc2c(c1)N([C@H]1C[C@H](C1)N1CCCCC1)C(=O)C21CCN(CC1)C(C)=O |r,wU:33.36,35.41,(7.37,-3.45,;5.88,-3.05,;5.48,-1.56,;6.39,-.32,;5.48,.93,;4.02,.45,;2.69,1.22,;1.35,.45,;1.35,-1.09,;2.69,-1.86,;2.69,-3.4,;1.35,-4.17,;1.35,-5.71,;.02,-6.48,;.02,-8.02,;-1.32,-8.79,;1.35,-8.79,;2.69,-8.02,;4.02,-8.79,;2.69,-6.48,;-1.32,-5.71,;-2.65,-6.48,;-1.32,-4.17,;.02,-3.4,;.02,-1.86,;4.02,-1.09,;.02,1.22,;.02,2.76,;-1.32,3.53,;-2.65,2.76,;-2.65,1.22,;-1.32,.45,;-4.11,.75,;-4.51,-.74,;-3.74,-2.08,;-5.08,-2.85,;-5.85,-1.51,;-5.48,-4.33,;-6.96,-4.73,;-7.37,-6.23,;-6.27,-7.34,;-4.77,-6.94,;-4.36,-5.44,;-5.02,1.99,;-6.56,1.99,;-4.11,3.24,;-3.03,4.33,;-3.42,5.81,;-4.91,6.21,;-6,5.12,;-5.6,3.64,;-5.31,7.7,;-4.22,8.79,;-6.8,8.1,)|
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CCNC(=O)c1cc(Nc2nc(cc3ncn(CC)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C32CCN(CC2)C(=O)CC)c(F)cc1C |r,wU:27.29,29.34,(2.69,-6.48,;2.69,-8.02,;1.35,-8.79,;.02,-8.02,;-1.32,-8.79,;.02,-6.48,;1.35,-5.71,;1.35,-4.17,;2.69,-3.4,;2.69,-1.86,;1.35,-1.09,;1.35,.45,;2.69,1.22,;4.02,.45,;5.48,.93,;6.39,-.32,;5.48,-1.56,;5.88,-3.05,;7.37,-3.45,;4.02,-1.09,;.02,1.22,;.02,2.76,;-1.32,3.53,;-2.65,2.76,;-2.65,1.22,;-1.32,.45,;-4.11,.75,;-4.51,-.74,;-3.74,-2.08,;-5.08,-2.85,;-5.85,-1.51,;-5.48,-4.33,;-6.96,-4.73,;-7.37,-6.23,;-6.27,-7.34,;-4.77,-6.94,;-4.36,-5.44,;-5.02,1.99,;-6.56,1.99,;-4.11,3.24,;-3.03,4.33,;-3.42,5.81,;-4.91,6.21,;-6,5.12,;-5.6,3.64,;-5.31,7.7,;-6.8,8.1,;-4.22,8.79,;-2.73,8.39,;.02,-3.4,;.02,-1.86,;-1.32,-4.17,;-1.32,-5.71,;-2.65,-6.48,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N(CC3(C)C)[C@H]2C[C@H](C2)N2CCCCC2)ccc1C |r,wU:31.34,33.39,(1.35,-7.53,;1.35,-5.99,;.02,-5.22,;-1.32,-5.99,;.02,-3.68,;1.35,-2.91,;1.35,-1.37,;2.69,-.6,;2.69,.94,;1.35,1.71,;1.35,3.25,;2.69,4.02,;4.02,3.25,;5.48,3.73,;6.39,2.48,;5.48,1.24,;5.88,-.25,;7.37,-.65,;4.79,-1.34,;4.02,1.71,;.02,4.02,;.02,5.56,;-1.32,6.33,;-2.65,5.56,;-2.65,4.02,;-1.32,3.25,;-4.11,3.55,;-5.02,4.79,;-4.11,6.04,;-3.72,7.53,;-5.2,7.13,;-4.51,2.06,;-3.74,.73,;-5.08,-.04,;-5.85,1.29,;-5.48,-1.53,;-6.96,-1.93,;-7.37,-3.43,;-6.27,-4.54,;-4.77,-4.14,;-4.36,-2.63,;.02,-.6,;-1.32,-1.37,;-1.32,-2.91,;-2.65,-3.68,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C4CC4)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C32CCN(CC2)C(C)=O)ccc1C |r,wU:27.30,29.35,(2.88,-8.02,;1.55,-8.79,;.22,-8.02,;-1.12,-8.79,;.22,-6.48,;1.55,-5.71,;1.55,-4.17,;2.88,-3.4,;2.88,-1.86,;1.55,-1.09,;1.55,.45,;2.88,1.22,;4.22,.45,;5.68,.93,;6.59,-.32,;5.68,-1.56,;6.08,-3.05,;5.68,-4.54,;7.17,-4.14,;4.22,-1.09,;.22,1.22,;.22,2.76,;-1.12,3.53,;-2.45,2.76,;-2.45,1.22,;-1.12,.45,;-3.91,.75,;-4.31,-.74,;-3.54,-2.08,;-4.88,-2.85,;-5.65,-1.51,;-5.28,-4.33,;-6.76,-4.73,;-7.17,-6.23,;-6.07,-7.34,;-4.57,-6.94,;-4.16,-5.44,;-4.82,1.99,;-6.36,1.99,;-3.91,3.24,;-2.83,4.33,;-3.22,5.81,;-4.71,6.21,;-5.8,5.12,;-5.4,3.64,;-5.11,7.7,;-6.6,8.1,;-4.02,8.79,;.22,-3.4,;-1.12,-4.17,;-1.12,-5.71,;-2.45,-6.48,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C4CC4)c23)-c2ccc3c(c2)N(CC3(C)C)[C@H]2C[C@H](C2)N2CCCCC2)ccc1C |r,wU:31.35,33.40,(1.55,-7.53,;1.55,-5.99,;.22,-5.22,;-1.12,-5.99,;.22,-3.68,;1.55,-2.91,;1.55,-1.37,;2.88,-.6,;2.88,.94,;1.55,1.71,;1.55,3.25,;2.88,4.02,;4.22,3.25,;5.68,3.73,;6.59,2.48,;5.68,1.24,;6.08,-.25,;5.68,-1.74,;7.17,-1.34,;4.22,1.71,;.22,4.02,;.22,5.56,;-1.12,6.33,;-2.45,5.56,;-2.45,4.02,;-1.12,3.25,;-3.91,3.55,;-4.82,4.79,;-3.91,6.04,;-3.52,7.53,;-5,7.13,;-4.31,2.06,;-3.54,.73,;-4.88,-.04,;-5.65,1.29,;-5.28,-1.53,;-6.76,-1.93,;-7.17,-3.43,;-6.07,-4.54,;-4.57,-4.14,;-4.16,-2.63,;.22,-.6,;-1.12,-1.37,;-1.12,-2.91,;-2.45,-3.68,)|
CC(C)n1cnc2cc(nc(Nc3cc(C(=O)NC(C)(C)C)c(C)cc3F)c12)-c1ccc2c(c1)N([C@H]1C[C@H](C1)N1CCCCC1)C(=O)C21CCN(CC1)C(C)=O |r,wU:35.38,37.43,(4.79,-4.14,;5.88,-3.05,;7.37,-3.45,;5.48,-1.56,;6.39,-.32,;5.48,.93,;4.02,.45,;2.69,1.22,;1.35,.45,;1.35,-1.09,;2.69,-1.86,;2.69,-3.4,;1.35,-4.17,;1.35,-5.71,;.02,-6.48,;.02,-8.02,;-1.32,-8.79,;1.35,-8.79,;2.69,-8.02,;1.92,-6.69,;4.02,-8.79,;3.46,-6.69,;-1.32,-5.71,;-2.65,-6.48,;-1.32,-4.17,;.02,-3.4,;.02,-1.86,;4.02,-1.09,;.02,1.22,;.02,2.76,;-1.32,3.53,;-2.65,2.76,;-2.65,1.22,;-1.32,.45,;-4.11,.75,;-4.51,-.74,;-3.74,-2.08,;-5.08,-2.85,;-5.85,-1.51,;-5.48,-4.33,;-6.96,-4.73,;-7.37,-6.23,;-6.27,-7.34,;-4.77,-6.94,;-4.36,-5.44,;-5.02,1.99,;-6.56,1.99,;-4.11,3.24,;-3.03,4.33,;-3.42,5.81,;-4.91,6.21,;-6,5.12,;-5.6,3.64,;-5.31,7.7,;-6.8,8.1,;-4.22,8.79,)|
CCNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C32CCN(CC2)C(=O)CC)c(F)cc1C |r,wU:28.30,30.35,(4.28,-8.79,;2.94,-8.02,;1.61,-8.79,;.28,-8.02,;-1.06,-8.79,;.28,-6.48,;1.61,-5.71,;1.61,-4.17,;2.94,-3.4,;2.94,-1.86,;1.61,-1.09,;1.61,.45,;2.94,1.22,;4.28,.45,;5.74,.93,;6.65,-.32,;5.74,-1.56,;6.14,-3.05,;5.05,-4.14,;7.63,-3.45,;4.28,-1.09,;.28,1.22,;.28,2.76,;-1.06,3.53,;-2.39,2.76,;-2.39,1.22,;-1.06,.45,;-3.86,.75,;-4.25,-.74,;-3.48,-2.08,;-4.82,-2.85,;-5.59,-1.51,;-5.22,-4.33,;-6.7,-4.73,;-7.11,-6.23,;-6.01,-7.34,;-4.51,-6.94,;-4.1,-5.44,;-4.76,1.99,;-6.3,1.99,;-3.86,3.24,;-2.77,4.33,;-3.17,5.81,;-4.65,6.21,;-5.74,5.12,;-5.34,3.64,;-5.05,7.7,;-3.96,8.79,;-6.54,8.1,;-7.63,7.01,;.28,-3.4,;.28,-1.86,;-1.06,-4.17,;-1.06,-5.71,;-2.39,-6.48,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C32CCN(CC(F)F)CC2)c(F)cc1C |r,wU:27.29,29.34,(2.94,-8.42,;1.61,-9.19,;.28,-8.42,;-1.06,-9.19,;.28,-6.88,;1.61,-6.11,;1.61,-4.57,;2.94,-3.8,;2.94,-2.26,;1.61,-1.49,;1.61,.05,;2.94,.82,;4.28,.05,;5.74,.53,;6.65,-.72,;5.74,-1.96,;6.14,-3.45,;5.05,-4.54,;7.63,-3.85,;4.28,-1.49,;.28,.82,;.28,2.36,;-1.06,3.13,;-2.39,2.36,;-2.39,.82,;-1.06,.05,;-3.86,.35,;-4.25,-1.14,;-3.48,-2.47,;-4.82,-3.24,;-5.59,-1.91,;-5.22,-4.73,;-6.7,-5.13,;-7.11,-6.63,;-6.01,-7.74,;-4.51,-7.34,;-4.1,-5.84,;-4.76,1.59,;-6.3,1.59,;-3.86,2.84,;-2.77,3.93,;-3.17,5.42,;-4.65,5.81,;-5.05,7.3,;-6.54,7.7,;-7.63,6.61,;-6.94,9.19,;-5.74,4.72,;-5.34,3.24,;.28,-3.8,;.28,-2.26,;-1.06,-4.57,;-1.06,-6.11,;-2.39,-6.88,)|
CC(C)NC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C32CCN(CC(F)F)CC2)ccc1C |r,wU:29.31,31.36,(4.02,-9.53,;2.69,-8.76,;2.69,-7.22,;1.35,-9.53,;.02,-8.76,;-1.32,-9.53,;.02,-7.22,;1.35,-6.45,;1.35,-4.91,;2.69,-4.14,;2.69,-2.6,;1.35,-1.83,;1.35,-.29,;2.69,.48,;4.02,-.29,;5.48,.18,;6.39,-1.06,;5.48,-2.31,;5.88,-3.8,;4.79,-4.88,;7.37,-4.19,;4.02,-1.83,;.02,.48,;.02,2.02,;-1.32,2.79,;-2.65,2.02,;-2.65,.48,;-1.32,-.29,;-4.11,0,;-4.51,-1.49,;-3.74,-2.82,;-5.08,-3.59,;-5.85,-2.26,;-5.48,-5.08,;-6.96,-5.48,;-7.37,-6.98,;-6.27,-8.08,;-4.77,-7.68,;-4.36,-6.18,;-5.02,1.25,;-6.56,1.25,;-4.11,2.49,;-3.03,3.58,;-3.42,5.07,;-4.91,5.47,;-5.31,6.96,;-4.22,8.04,;-2.73,7.65,;-4.62,9.53,;-6,4.38,;-5.6,2.89,;.02,-4.14,;-1.32,-4.91,;-1.32,-6.45,;-2.65,-7.22,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C3(C)O)ccc1Cl |r,wU:27.29,29.34,(2.69,-5.79,;1.35,-6.56,;.02,-5.79,;-1.32,-6.56,;.02,-4.25,;1.35,-3.48,;1.35,-1.94,;2.69,-1.17,;2.69,.37,;1.35,1.14,;1.35,2.68,;2.69,3.45,;4.02,2.68,;5.48,3.16,;6.39,1.91,;5.48,.67,;5.88,-.82,;4.79,-1.91,;7.37,-1.22,;4.02,1.14,;.02,3.45,;.02,4.99,;-1.32,5.76,;-2.65,4.99,;-2.65,3.45,;-1.32,2.68,;-4.11,2.98,;-4.51,1.49,;-3.74,.16,;-5.08,-.61,;-5.85,.72,;-5.48,-2.1,;-6.96,-2.5,;-7.37,-4,;-6.27,-5.11,;-4.77,-4.71,;-4.36,-3.21,;-5.02,4.22,;-6.56,4.22,;-4.11,5.47,;-3.03,6.56,;-5.6,5.87,;.02,-1.17,;-1.32,-1.94,;-1.32,-3.48,;-2.65,-4.25,)|
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CC(C)n1cnc2cc(nc(Nc3cc(C(=O)NC4(CC4)C(F)F)c(C)cc3F)c12)-c1ccc2c(c1)N([C@H]1C[C@H](C1)N1CCCCC1)C(=O)C2(C)C |r,wU:37.41,39.46,(4.79,-1.34,;5.88,-.25,;7.37,-.65,;5.48,1.24,;6.39,2.48,;5.48,3.73,;4.02,3.25,;2.69,4.02,;1.35,3.25,;1.35,1.71,;2.69,.94,;2.69,-.6,;1.35,-1.37,;1.35,-2.91,;.02,-3.68,;.02,-5.22,;-1.32,-5.99,;1.35,-5.99,;2.69,-5.22,;1.92,-3.88,;3.46,-3.88,;4.02,-5.99,;5.35,-5.22,;4.02,-7.53,;-1.32,-2.91,;-2.65,-3.68,;-1.32,-1.37,;.02,-.6,;.02,.94,;4.02,1.71,;.02,4.02,;.02,5.56,;-1.32,6.33,;-2.65,5.56,;-2.65,4.02,;-1.32,3.25,;-4.11,3.55,;-4.51,2.06,;-3.74,.73,;-5.08,-.04,;-5.85,1.29,;-5.48,-1.53,;-6.96,-1.93,;-7.37,-3.43,;-6.27,-4.54,;-4.77,-4.14,;-4.36,-2.63,;-5.02,4.79,;-6.56,4.79,;-4.11,6.04,;-3.72,7.53,;-5.2,7.13,)|
CC(C)n1cnc2cc(nc(Nc3cc(C(=O)NC4(CC4)C(F)F)c(C)cc3F)c12)-c1ccc2c(c1)N([C@@H]1C[C@@H](C1)N1C[C@H]3CC[C@@H]1C3)C(=O)C2(C)C |r,wU:37.41,39.46,wD:46.53,43.54,(4.79,-1.34,;5.88,-.25,;7.37,-.65,;5.48,1.24,;6.39,2.48,;5.48,3.73,;4.02,3.25,;2.69,4.02,;1.35,3.25,;1.35,1.71,;2.69,.94,;2.69,-.6,;1.35,-1.37,;1.35,-2.91,;.02,-3.68,;.02,-5.22,;-1.32,-5.99,;1.35,-5.99,;2.69,-5.22,;1.92,-3.88,;3.46,-3.88,;4.02,-5.99,;5.35,-5.22,;4.02,-7.53,;-1.32,-2.91,;-2.65,-3.68,;-1.32,-1.37,;.02,-.6,;.02,.94,;4.02,1.71,;.02,4.02,;.02,5.56,;-1.32,6.33,;-2.65,5.56,;-2.65,4.02,;-1.32,3.25,;-4.11,3.55,;-4.51,2.06,;-5.85,1.29,;-5.08,-.04,;-3.74,.73,;-5.48,-1.53,;-4.36,-2.63,;-4.77,-4.14,;-6.27,-4.54,;-7.37,-3.43,;-6.96,-1.93,;-6.19,-3.26,;-5.02,4.79,;-6.56,4.79,;-4.11,6.04,;-3.72,7.53,;-5.2,7.13,)|
CC(C)n1cnc2cc(nc(Nc3cc(C(=O)NC4(CC4)C(F)F)c(C)cc3F)c12)-c1cnc2c(c1)N([C@H]1C[C@H](C1)N1CCCCC1)C(=O)C2(C)C |r,wU:37.41,39.46,(4.79,-1.34,;5.88,-.25,;7.37,-.65,;5.48,1.24,;6.39,2.48,;5.48,3.73,;4.02,3.25,;2.69,4.02,;1.35,3.25,;1.35,1.71,;2.69,.94,;2.69,-.6,;1.35,-1.37,;1.35,-2.91,;.02,-3.68,;.02,-5.22,;-1.32,-5.99,;1.35,-5.99,;2.69,-5.22,;1.92,-3.88,;3.46,-3.88,;4.02,-5.99,;5.35,-5.22,;4.02,-7.53,;-1.32,-2.91,;-2.65,-3.68,;-1.32,-1.37,;.02,-.6,;.02,.94,;4.02,1.71,;.02,4.02,;.02,5.56,;-1.32,6.33,;-2.65,5.56,;-2.65,4.02,;-1.32,3.25,;-4.11,3.55,;-4.51,2.06,;-3.74,.73,;-5.08,-.04,;-5.85,1.29,;-5.48,-1.53,;-6.96,-1.93,;-7.37,-3.43,;-6.27,-4.54,;-4.77,-4.14,;-4.36,-2.63,;-5.02,4.79,;-6.56,4.79,;-4.11,6.04,;-3.72,7.53,;-5.2,7.13,)|
CCNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C32CCN(CC2)C2COC2)c(F)cc1C |r,wU:28.30,30.35,(4.01,-9.3,;2.68,-8.53,;1.35,-9.3,;.01,-8.53,;-1.32,-9.3,;.01,-6.99,;1.35,-6.22,;1.35,-4.68,;2.68,-3.91,;2.68,-2.37,;1.35,-1.6,;1.35,-.06,;2.68,.71,;4.01,-.06,;5.48,.42,;6.38,-.83,;5.48,-2.07,;5.88,-3.56,;4.79,-4.65,;7.37,-3.96,;4.01,-1.6,;.01,.71,;.01,2.25,;-1.32,3.02,;-2.65,2.25,;-2.65,.71,;-1.32,-.06,;-4.12,.24,;-4.52,-1.25,;-3.75,-2.58,;-5.08,-3.35,;-5.85,-2.02,;-5.48,-4.84,;-6.97,-5.24,;-7.37,-6.73,;-6.28,-7.82,;-4.79,-7.42,;-4.39,-5.93,;-5.02,1.48,;-6.56,1.48,;-4.12,2.73,;-3.03,3.82,;-3.43,5.31,;-4.92,5.7,;-6,4.62,;-5.61,3.13,;-5.31,7.19,;-4.54,8.53,;-5.88,9.3,;-6.65,7.96,;.01,-3.91,;.01,-2.37,;-1.32,-4.68,;-1.32,-6.22,;-2.65,-6.99,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@@H]2C[C@@H](C2)N2CC4C(C2)C4(F)F)C(=O)C32CCN(CC2)C2COC2)c(F)cc1C |r,wU:27.29,29.34,(2.98,-8.25,;1.64,-9.02,;.31,-8.25,;-1.02,-9.02,;.31,-6.71,;1.64,-5.94,;1.64,-4.4,;2.98,-3.63,;2.98,-2.09,;1.64,-1.32,;1.64,.22,;2.98,.99,;4.31,.22,;5.78,.7,;6.68,-.55,;5.78,-1.79,;6.17,-3.28,;5.08,-4.37,;7.66,-3.68,;4.31,-1.32,;.31,.99,;.31,2.53,;-1.02,3.3,;-2.36,2.53,;-2.36,.99,;-1.02,.22,;-3.82,.52,;-4.22,-.97,;-5.55,-1.74,;-4.78,-3.08,;-3.45,-2.31,;-5.18,-4.56,;-6.65,-5.04,;-6.65,-6.58,;-5.18,-7.06,;-4.28,-5.81,;-6.33,-8.09,;-7.66,-8.86,;-5.93,-9.57,;-4.73,1.76,;-6.27,1.76,;-3.82,3.01,;-2.73,4.1,;-3.13,5.58,;-4.62,5.98,;-5.71,4.89,;-5.31,3.41,;-5.02,7.47,;-4.25,8.8,;-5.58,9.57,;-6.35,8.24,;.31,-3.63,;.31,-2.09,;-1.02,-4.4,;-1.02,-5.94,;-2.36,-6.71,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@@H]2C[C@@H](C2)N2CC[C@@H](F)C2)C(=O)C32CCN(CC2)C2COC2)c(F)cc1C |r,wU:27.29,29.34,34.38,(3.14,-8.53,;1.8,-9.3,;.47,-8.53,;-.86,-9.3,;.47,-6.99,;1.8,-6.22,;1.8,-4.68,;3.14,-3.91,;3.14,-2.37,;1.8,-1.6,;1.8,-.06,;3.14,.71,;4.47,-.06,;5.94,.42,;6.84,-.83,;5.94,-2.07,;6.33,-3.56,;5.24,-4.65,;7.82,-3.96,;4.47,-1.6,;.47,.71,;.47,2.25,;-.86,3.02,;-2.2,2.25,;-2.2,.71,;-.86,-.06,;-3.66,.24,;-4.06,-1.25,;-5.39,-2.02,;-4.62,-3.35,;-3.29,-2.58,;-5.02,-4.84,;-4.12,-6.09,;-5.02,-7.33,;-6.49,-6.86,;-7.82,-7.63,;-6.49,-5.32,;-4.57,1.48,;-6.11,1.48,;-3.66,2.73,;-2.57,3.82,;-2.97,5.31,;-4.46,5.7,;-5.55,4.62,;-5.15,3.13,;-4.86,7.19,;-4.09,8.53,;-5.42,9.3,;-6.19,7.96,;.47,-3.91,;.47,-2.37,;-.86,-4.68,;-.86,-6.22,;-2.2,-6.99,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@@H]2C[C@@H](C2)N2CC[C@H](F)C2)C(=O)C32CCN(CC2)C2COC2)c(F)cc1C |r,wU:27.29,29.34,wD:34.38,(3.14,-8.53,;1.8,-9.3,;.47,-8.53,;-.86,-9.3,;.47,-6.99,;1.8,-6.22,;1.8,-4.68,;3.14,-3.91,;3.14,-2.37,;1.8,-1.6,;1.8,-.06,;3.14,.71,;4.47,-.06,;5.94,.42,;6.84,-.83,;5.94,-2.07,;6.33,-3.56,;5.24,-4.65,;7.82,-3.96,;4.47,-1.6,;.47,.71,;.47,2.25,;-.86,3.02,;-2.2,2.25,;-2.2,.71,;-.86,-.06,;-3.66,.24,;-4.06,-1.25,;-5.39,-2.02,;-4.62,-3.35,;-3.29,-2.58,;-5.02,-4.84,;-4.12,-6.09,;-5.02,-7.33,;-6.49,-6.86,;-7.82,-7.63,;-6.49,-5.32,;-4.57,1.48,;-6.11,1.48,;-3.66,2.73,;-2.57,3.82,;-2.97,5.31,;-4.46,5.7,;-5.55,4.62,;-5.15,3.13,;-4.86,7.19,;-4.09,8.53,;-5.42,9.3,;-6.19,7.96,;.47,-3.91,;.47,-2.37,;-.86,-4.68,;-.86,-6.22,;-2.2,-6.99,)|
CC(C)NC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C32CCN(CC2)C2COC2)ccc1C |r,wU:29.31,31.36,(4.01,-9.3,;2.68,-8.53,;2.68,-6.99,;1.35,-9.3,;.01,-8.53,;-1.32,-9.3,;.01,-6.99,;1.35,-6.22,;1.35,-4.68,;2.68,-3.91,;2.68,-2.37,;1.35,-1.6,;1.35,-.06,;2.68,.71,;4.01,-.06,;5.48,.42,;6.38,-.83,;5.48,-2.07,;5.88,-3.56,;4.79,-4.65,;7.37,-3.96,;4.01,-1.6,;.01,.71,;.01,2.25,;-1.32,3.02,;-2.65,2.25,;-2.65,.71,;-1.32,-.06,;-4.12,.24,;-4.52,-1.25,;-3.75,-2.58,;-5.08,-3.35,;-5.85,-2.02,;-5.48,-4.84,;-6.97,-5.24,;-7.37,-6.73,;-6.28,-7.82,;-4.79,-7.42,;-4.39,-5.93,;-5.02,1.48,;-6.56,1.48,;-4.12,2.73,;-3.03,3.82,;-3.43,5.31,;-4.92,5.7,;-6,4.62,;-5.61,3.13,;-5.31,7.19,;-4.54,8.53,;-5.88,9.3,;-6.65,7.96,;.01,-3.91,;-1.32,-4.68,;-1.32,-6.22,;-2.65,-6.99,)|
CCNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C32CCN(CC2)C(C)=O)c(F)cc1C |r,wU:28.30,30.35,(4.01,-8.79,;2.68,-8.02,;1.35,-8.79,;.01,-8.02,;-1.32,-8.79,;.01,-6.48,;1.35,-5.71,;1.35,-4.17,;2.68,-3.4,;2.68,-1.86,;1.35,-1.09,;1.35,.45,;2.68,1.22,;4.01,.45,;5.48,.93,;6.38,-.32,;5.48,-1.56,;5.88,-3.05,;4.79,-4.14,;7.37,-3.45,;4.01,-1.09,;.01,1.22,;.01,2.76,;-1.32,3.53,;-2.65,2.76,;-2.65,1.22,;-1.32,.45,;-4.12,.75,;-4.52,-.74,;-3.75,-2.08,;-5.08,-2.85,;-5.85,-1.51,;-5.48,-4.33,;-6.97,-4.73,;-7.37,-6.22,;-6.28,-7.31,;-4.79,-6.91,;-4.39,-5.42,;-5.02,1.99,;-6.56,1.99,;-4.12,3.24,;-3.03,4.33,;-3.43,5.81,;-4.92,6.21,;-6,5.12,;-5.61,3.64,;-5.31,7.7,;-6.8,8.1,;-4.23,8.79,;.01,-3.4,;.01,-1.86,;-1.32,-4.17,;-1.32,-5.71,;-2.65,-6.48,)|
CC(C)CNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C32CCN(CC2)C(C)=O)c(F)cc1C |r,wU:30.32,32.37,(4.01,-9.56,;4.01,-8.02,;5.35,-7.25,;2.68,-7.25,;1.35,-8.02,;.01,-7.25,;-1.32,-8.02,;.01,-5.71,;1.35,-4.94,;1.35,-3.4,;2.68,-2.63,;2.68,-1.09,;1.35,-.32,;1.35,1.22,;2.68,1.99,;4.01,1.22,;5.48,1.7,;6.38,.45,;5.48,-.79,;5.88,-2.28,;4.79,-3.37,;7.37,-2.68,;4.01,-.32,;.01,1.99,;.01,3.53,;-1.32,4.3,;-2.65,3.53,;-2.65,1.99,;-1.32,1.22,;-4.12,1.52,;-4.52,.03,;-3.75,-1.31,;-5.08,-2.08,;-5.85,-.74,;-5.48,-3.56,;-6.97,-3.96,;-7.37,-5.45,;-6.28,-6.54,;-4.79,-6.14,;-4.39,-4.65,;-5.02,2.76,;-6.56,2.76,;-4.12,4.01,;-3.03,5.1,;-3.43,6.58,;-4.92,6.98,;-6,5.89,;-5.61,4.41,;-5.31,8.47,;-6.8,8.87,;-4.23,9.56,;.01,-2.63,;.01,-1.09,;-1.32,-3.4,;-1.32,-4.94,;-2.65,-5.71,)|
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CC(C)NC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@@H]2C[C@@H](C2)N2C4CCC2COC4)C(=O)C32CCN(CC2)C(C)=O)c(F)cc1C |r,wU:29.31,31.36,(4.01,-8.79,;2.68,-8.02,;2.68,-6.48,;1.35,-8.79,;.01,-8.02,;-1.32,-8.79,;.01,-6.48,;1.35,-5.71,;1.35,-4.17,;2.68,-3.4,;2.68,-1.86,;1.35,-1.09,;1.35,.45,;2.68,1.22,;4.01,.45,;5.48,.93,;6.38,-.32,;5.48,-1.56,;5.88,-3.05,;4.79,-4.14,;7.37,-3.45,;4.01,-1.09,;.01,1.22,;.01,2.76,;-1.32,3.53,;-2.65,2.76,;-2.65,1.22,;-1.32,.45,;-4.12,.75,;-4.52,-.74,;-5.85,-1.51,;-5.08,-2.85,;-3.75,-2.08,;-5.48,-4.33,;-6.97,-4.73,;-6.57,-6.22,;-5.48,-6.51,;-4.39,-5.42,;-4.79,-6.91,;-6.28,-7.31,;-7.37,-6.22,;-5.02,1.99,;-6.56,1.99,;-4.12,3.24,;-3.03,4.33,;-3.43,5.81,;-4.92,6.21,;-6,5.12,;-5.61,3.64,;-5.31,7.7,;-4.23,8.79,;-6.8,8.1,;.01,-3.4,;.01,-1.86,;-1.32,-4.17,;-1.32,-5.71,;-2.65,-6.48,)|
CC(C)NC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CC4CCC(C2)O4)C(=O)C32CCN(CC2)C(C)=O)c(F)cc1C |r,wU:29.31,31.36,(4.01,-8.79,;2.68,-8.02,;2.68,-6.48,;1.35,-8.79,;.01,-8.02,;-1.32,-8.79,;.01,-6.48,;1.35,-5.71,;1.35,-4.17,;2.68,-3.4,;2.68,-1.86,;1.35,-1.09,;1.35,.45,;2.68,1.22,;4.01,.45,;5.48,.93,;6.38,-.32,;5.48,-1.56,;5.88,-3.05,;4.79,-4.14,;7.37,-3.45,;4.01,-1.09,;.01,1.22,;.01,2.76,;-1.32,3.53,;-2.65,2.76,;-2.65,1.22,;-1.32,.45,;-4.12,.75,;-4.52,-.74,;-3.75,-2.08,;-5.08,-2.85,;-5.85,-1.51,;-5.48,-4.33,;-4.39,-5.42,;-4.79,-6.91,;-5.19,-5.42,;-6.28,-5.13,;-7.37,-6.22,;-6.97,-4.73,;-6.28,-7.31,;-5.02,1.99,;-6.56,1.99,;-4.12,3.24,;-3.03,4.33,;-3.43,5.81,;-4.92,6.21,;-6,5.12,;-5.61,3.64,;-5.31,7.7,;-4.23,8.79,;-6.8,8.1,;.01,-3.4,;.01,-1.86,;-1.32,-4.17,;-1.32,-5.71,;-2.65,-6.48,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C4CC4)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C3(C)C)ccc1C |r,wU:27.30,29.35,(2.88,-5.99,;1.55,-6.76,;.21,-5.99,;-1.12,-6.76,;.21,-4.45,;1.55,-3.68,;1.55,-2.14,;2.88,-1.37,;2.88,.17,;1.55,.94,;1.55,2.48,;2.88,3.25,;4.21,2.48,;5.68,2.96,;6.58,1.71,;5.68,.47,;6.08,-1.02,;5.68,-2.51,;7.17,-2.11,;4.21,.94,;.21,3.25,;.21,4.79,;-1.12,5.56,;-2.45,4.79,;-2.45,3.25,;-1.12,2.48,;-3.92,2.78,;-4.32,1.29,;-3.55,-.04,;-4.88,-.81,;-5.65,.52,;-5.28,-2.3,;-4.19,-3.39,;-4.59,-4.88,;-6.08,-5.28,;-7.17,-4.19,;-6.77,-2.7,;-4.82,4.02,;-6.36,4.02,;-3.92,5.27,;-2.83,6.36,;-4.32,6.76,;.21,-1.37,;-1.12,-2.14,;-1.12,-3.68,;-2.45,-4.45,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@@H]2C[C@@H](C2)NC2CCC(F)(F)CC2)C(=O)C3(C)C)ccc1C |r,wU:27.29,29.34,(4.71,-5.91,;3.38,-6.68,;2.05,-5.91,;.71,-6.68,;2.05,-4.37,;3.38,-3.6,;3.38,-2.06,;4.71,-1.29,;4.71,.25,;3.38,1.02,;3.38,2.56,;4.71,3.33,;6.05,2.56,;7.51,3.04,;8.42,1.79,;7.51,.54,;7.91,-.94,;9.4,-1.34,;6.82,-2.03,;6.05,1.02,;2.05,3.33,;2.05,4.87,;.71,5.64,;-.62,4.87,;-.62,3.33,;.71,2.56,;-2.09,2.85,;-2.48,1.37,;-3.82,.6,;-3.05,-.74,;-1.71,.03,;-3.45,-2.22,;-4.93,-2.62,;-6.02,-1.53,;-7.51,-1.93,;-7.91,-3.42,;-9.4,-3.02,;-9,-4.51,;-6.82,-4.51,;-5.33,-4.11,;-2.99,4.1,;-4.53,4.1,;-2.09,5.35,;-1.32,6.68,;-3.18,6.43,;2.05,-1.29,;.71,-2.06,;.71,-3.6,;-.62,-4.37,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@@H]2C[C@@H](C2)NC2CC(F)(F)C2)C(=O)C3(C)C)ccc1C |r,wU:27.29,29.34,(4.28,-5.91,;2.94,-6.68,;1.61,-5.91,;.28,-6.68,;1.61,-4.37,;2.94,-3.6,;2.94,-2.06,;4.28,-1.29,;4.28,.25,;2.94,1.02,;2.94,2.56,;4.28,3.33,;5.61,2.56,;7.08,3.04,;7.98,1.79,;7.08,.54,;7.47,-.94,;8.96,-1.34,;6.39,-2.03,;5.61,1.02,;1.61,3.33,;1.61,4.87,;.28,5.64,;-1.06,4.87,;-1.06,3.33,;.28,2.56,;-2.52,2.85,;-2.92,1.37,;-4.25,.6,;-3.48,-.74,;-2.15,.03,;-3.88,-2.22,;-5.37,-2.62,;-6.7,-1.85,;-7.47,-3.19,;-8.96,-2.79,;-8.56,-4.28,;-6.14,-3.96,;-3.43,4.1,;-4.97,4.1,;-2.52,5.35,;-1.75,6.68,;-3.61,6.43,;1.61,-1.29,;.28,-2.06,;.28,-3.6,;-1.06,-4.37,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@@H]2C[C@@H](C2)NCC(C)(C)F)C(=O)C3(C)C)ccc1C |r,wU:27.29,29.34,(3.42,-5.91,;2.09,-6.68,;.76,-5.91,;-.58,-6.68,;.76,-4.37,;2.09,-3.6,;2.09,-2.06,;3.42,-1.29,;3.42,.25,;2.09,1.02,;2.09,2.56,;3.42,3.33,;4.76,2.56,;6.22,3.04,;7.13,1.79,;6.22,.54,;6.62,-.94,;8.11,-1.34,;5.53,-2.03,;4.76,1.02,;.76,3.33,;.76,4.87,;-.58,5.64,;-1.91,4.87,;-1.91,3.33,;-.58,2.56,;-3.37,2.85,;-3.77,1.37,;-5.11,.6,;-4.34,-.74,;-3,.03,;-4.74,-2.22,;-6.22,-2.62,;-6.62,-4.11,;-8.11,-3.71,;-7.71,-5.2,;-5.53,-5.2,;-4.28,4.1,;-5.82,4.1,;-3.37,5.35,;-2.6,6.68,;-4.46,6.43,;.76,-1.29,;-.58,-2.06,;-.58,-3.6,;-1.91,-4.37,)|
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CNC(=O)c1cc(Nc2nc(cc3ncn(C4CC4)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C32CCN(CC2)C(=O)C2(C)COC2)ccc1C |r,wU:27.30,29.35,(3.65,-8.34,;2.32,-9.11,;.98,-8.34,;-.35,-9.11,;.98,-6.8,;2.32,-6.03,;2.32,-4.49,;3.65,-3.72,;3.65,-2.18,;2.32,-1.41,;2.32,.13,;3.65,.9,;4.98,.13,;6.45,.61,;7.35,-.64,;6.45,-1.89,;6.85,-3.37,;6.45,-4.86,;7.94,-4.46,;4.98,-1.41,;.98,.9,;.98,2.44,;-.35,3.21,;-1.68,2.44,;-1.68,.9,;-.35,.13,;-3.15,.42,;-3.55,-1.06,;-2.78,-2.4,;-4.11,-3.17,;-4.88,-1.83,;-4.51,-4.65,;-6,-5.05,;-6.4,-6.54,;-5.31,-7.63,;-3.82,-7.23,;-3.42,-5.74,;-4.05,1.67,;-5.59,1.67,;-3.15,2.92,;-2.06,4,;-2.46,5.49,;-3.95,5.89,;-5.04,4.8,;-4.64,3.31,;-4.34,7.38,;-3.26,8.47,;-5.83,7.78,;-5.06,9.11,;-6.6,9.11,;-7.94,8.34,;-7.17,7.01,;.98,-3.72,;-.35,-4.49,;-.35,-6.03,;-1.68,-6.8,)|
COCCNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C32CCN(CC2)C(C)=O)c(F)cc1C |r,wU:30.32,32.37,(6.68,-8.79,;5.35,-8.02,;4.01,-8.79,;2.68,-8.02,;1.35,-8.79,;.01,-8.02,;-1.32,-8.79,;.01,-6.48,;1.35,-5.71,;1.35,-4.17,;2.68,-3.4,;2.68,-1.86,;1.35,-1.09,;1.35,.45,;2.68,1.22,;4.01,.45,;5.48,.93,;6.38,-.32,;5.48,-1.56,;5.88,-3.05,;4.79,-4.14,;7.37,-3.45,;4.01,-1.09,;.01,1.22,;.01,2.76,;-1.32,3.53,;-2.65,2.76,;-2.65,1.22,;-1.32,.45,;-4.12,.75,;-4.52,-.74,;-3.75,-2.08,;-5.08,-2.85,;-5.85,-1.51,;-5.48,-4.33,;-6.97,-4.73,;-7.37,-6.22,;-6.28,-7.31,;-4.79,-6.91,;-4.39,-5.42,;-5.02,1.99,;-6.56,1.99,;-4.12,3.24,;-3.03,4.33,;-3.43,5.81,;-4.92,6.21,;-6,5.12,;-5.61,3.64,;-5.31,7.7,;-6.8,8.1,;-4.23,8.79,;.01,-3.4,;.01,-1.86,;-1.32,-4.17,;-1.32,-5.71,;-2.65,-6.48,)|
CC[C@@H](C)NC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C32CCN(CC2)C(C)=O)c(F)cc1C |r,wU:30.32,32.37,wD:2.2,(5.35,-8.02,;4.01,-8.79,;2.68,-8.02,;2.68,-6.48,;1.35,-8.79,;.01,-8.02,;-1.32,-8.79,;.01,-6.48,;1.35,-5.71,;1.35,-4.17,;2.68,-3.4,;2.68,-1.86,;1.35,-1.09,;1.35,.45,;2.68,1.22,;4.01,.45,;5.48,.93,;6.38,-.32,;5.48,-1.56,;5.88,-3.05,;4.79,-4.14,;7.37,-3.45,;4.01,-1.09,;.01,1.22,;.01,2.76,;-1.32,3.53,;-2.65,2.76,;-2.65,1.22,;-1.32,.45,;-4.12,.75,;-4.52,-.74,;-3.75,-2.08,;-5.08,-2.85,;-5.85,-1.51,;-5.48,-4.33,;-6.97,-4.73,;-7.37,-6.22,;-6.28,-7.31,;-4.79,-6.91,;-4.39,-5.42,;-5.02,1.99,;-6.56,1.99,;-4.12,3.24,;-3.03,4.33,;-3.43,5.81,;-4.92,6.21,;-6,5.12,;-5.61,3.64,;-5.31,7.7,;-6.8,8.1,;-4.23,8.79,;.01,-3.4,;.01,-1.86,;-1.32,-4.17,;-1.32,-5.71,;-2.65,-6.48,)|
CC[C@H](C)NC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C32CCN(CC2)C(C)=O)c(F)cc1C |r,wU:30.32,32.37,2.2,(5.35,-8.02,;4.01,-8.79,;2.68,-8.02,;2.68,-6.48,;1.35,-8.79,;.01,-8.02,;-1.32,-8.79,;.01,-6.48,;1.35,-5.71,;1.35,-4.17,;2.68,-3.4,;2.68,-1.86,;1.35,-1.09,;1.35,.45,;2.68,1.22,;4.01,.45,;5.48,.93,;6.38,-.32,;5.48,-1.56,;5.88,-3.05,;4.79,-4.14,;7.37,-3.45,;4.01,-1.09,;.01,1.22,;.01,2.76,;-1.32,3.53,;-2.65,2.76,;-2.65,1.22,;-1.32,.45,;-4.12,.75,;-4.52,-.74,;-3.75,-2.08,;-5.08,-2.85,;-5.85,-1.51,;-5.48,-4.33,;-6.97,-4.73,;-7.37,-6.22,;-6.28,-7.31,;-4.79,-6.91,;-4.39,-5.42,;-5.02,1.99,;-6.56,1.99,;-4.12,3.24,;-3.03,4.33,;-3.43,5.81,;-4.92,6.21,;-6,5.12,;-5.61,3.64,;-5.31,7.7,;-6.8,8.1,;-4.23,8.79,;.01,-3.4,;.01,-1.86,;-1.32,-4.17,;-1.32,-5.71,;-2.65,-6.48,)|
CC(C)NC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C32CCN(CC2)C(C)=O)c(F)cc1Cl |r,wU:29.31,31.36,(4.01,-8.79,;2.68,-8.02,;2.68,-6.48,;1.35,-8.79,;.01,-8.02,;-1.32,-8.79,;.01,-6.48,;1.35,-5.71,;1.35,-4.17,;2.68,-3.4,;2.68,-1.86,;1.35,-1.09,;1.35,.45,;2.68,1.22,;4.01,.45,;5.48,.93,;6.38,-.32,;5.48,-1.56,;5.88,-3.05,;4.79,-4.14,;7.37,-3.45,;4.01,-1.09,;.01,1.22,;.01,2.76,;-1.32,3.53,;-2.65,2.76,;-2.65,1.22,;-1.32,.45,;-4.12,.75,;-4.52,-.74,;-3.75,-2.08,;-5.08,-2.85,;-5.85,-1.51,;-5.48,-4.33,;-6.97,-4.73,;-7.37,-6.22,;-6.28,-7.31,;-4.79,-6.91,;-4.39,-5.42,;-5.02,1.99,;-6.56,1.99,;-4.12,3.24,;-3.03,4.33,;-3.43,5.81,;-4.92,6.21,;-6,5.12,;-5.61,3.64,;-5.31,7.7,;-6.8,8.1,;-4.23,8.79,;.01,-3.4,;.01,-1.86,;-1.32,-4.17,;-1.32,-5.71,;-2.65,-6.48,)|
COCC1(CC1)NC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C32CCN(CC2)C(C)=O)c(F)cc1C |r,wU:32.35,34.40,(-2.72,-9.18,;-1.23,-9.58,;-.14,-8.49,;1.35,-8.89,;.58,-10.23,;2.12,-10.23,;1.35,-7.35,;.01,-6.58,;-1.32,-7.35,;.01,-5.04,;1.35,-4.27,;1.35,-2.73,;2.68,-1.96,;2.68,-.42,;1.35,.35,;1.35,1.89,;2.68,2.66,;4.01,1.89,;5.48,2.36,;6.38,1.12,;5.48,-.13,;5.88,-1.62,;4.79,-2.7,;7.37,-2.01,;4.01,.35,;.01,2.66,;.01,4.2,;-1.32,4.97,;-2.65,4.2,;-2.65,2.66,;-1.32,1.89,;-4.12,2.18,;-4.52,.69,;-3.75,-.64,;-5.08,-1.41,;-5.85,-.08,;-5.48,-2.9,;-6.97,-3.3,;-7.37,-4.78,;-6.28,-5.87,;-4.79,-5.47,;-4.39,-3.99,;-5.02,3.43,;-6.56,3.43,;-4.12,4.67,;-3.03,5.76,;-3.43,7.25,;-4.92,7.65,;-6,6.56,;-5.61,5.07,;-5.31,9.14,;-6.8,9.54,;-4.23,10.23,;.01,-1.96,;.01,-.42,;-1.32,-2.73,;-1.32,-4.27,;-2.65,-5.04,)|
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CNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C32CCN(CC2)C(C)=O)c(F)cc1C |r,wU:27.29,29.34,(1.35,-9.56,;1.35,-8.02,;.01,-7.25,;-1.32,-8.02,;.01,-5.71,;1.35,-4.94,;1.35,-3.4,;2.68,-2.63,;2.68,-1.09,;1.35,-.32,;1.35,1.22,;2.68,1.99,;4.01,1.22,;5.48,1.7,;6.38,.45,;5.48,-.79,;5.88,-2.28,;4.79,-3.37,;7.37,-2.68,;4.01,-.32,;.01,1.99,;.01,3.53,;-1.32,4.3,;-2.65,3.53,;-2.65,1.99,;-1.32,1.22,;-4.12,1.52,;-4.52,.03,;-3.75,-1.31,;-5.08,-2.08,;-5.85,-.74,;-5.48,-3.56,;-6.97,-3.96,;-7.37,-5.45,;-6.28,-6.54,;-4.79,-6.14,;-4.39,-4.65,;-5.02,2.76,;-6.56,2.76,;-4.12,4.01,;-3.03,5.1,;-3.43,6.58,;-4.92,6.98,;-6,5.89,;-5.61,4.41,;-5.31,8.47,;-6.8,8.87,;-4.23,9.56,;.01,-2.63,;.01,-1.09,;-1.32,-3.4,;-1.32,-4.94,;-2.65,-5.71,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C4CC4)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C32CCN(CC2)C(C)=O)c(F)cc1Cl |r,wU:27.30,29.35,(2.88,-8.02,;1.55,-8.79,;.21,-8.02,;-1.12,-8.79,;.21,-6.48,;1.55,-5.71,;1.55,-4.17,;2.88,-3.4,;2.88,-1.86,;1.55,-1.09,;1.55,.45,;2.88,1.22,;4.21,.45,;5.68,.93,;6.58,-.32,;5.68,-1.56,;6.08,-3.05,;5.68,-4.54,;7.17,-4.14,;4.21,-1.09,;.21,1.22,;.21,2.76,;-1.12,3.53,;-2.45,2.76,;-2.45,1.22,;-1.12,.45,;-3.92,.75,;-4.32,-.74,;-3.55,-2.08,;-4.88,-2.85,;-5.65,-1.51,;-5.28,-4.33,;-6.77,-4.73,;-7.17,-6.22,;-6.08,-7.31,;-4.59,-6.91,;-4.19,-5.42,;-4.82,1.99,;-6.36,1.99,;-3.92,3.24,;-2.83,4.33,;-3.23,5.81,;-4.72,6.21,;-5.81,5.12,;-5.41,3.64,;-5.11,7.7,;-6.6,8.1,;-4.03,8.79,;.21,-3.4,;.21,-1.86,;-1.12,-4.17,;-1.12,-5.71,;-2.45,-6.48,)|
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CNC(=O)c1ccc(F)c(Nc2nc(cc3ncn(C4CC4)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C32CCN(CC2)C(C)=O)c1 |r,wU:30.33,32.38,(2.88,-8.02,;1.55,-8.79,;.21,-8.02,;-1.12,-8.79,;.21,-6.48,;-1.12,-5.71,;-1.12,-4.17,;.21,-3.4,;.21,-1.86,;1.55,-4.17,;2.88,-3.4,;2.88,-1.86,;1.55,-1.09,;1.55,.45,;2.88,1.22,;4.21,.45,;5.68,.93,;6.58,-.32,;5.68,-1.56,;6.08,-3.05,;5.68,-4.54,;7.17,-4.14,;4.21,-1.09,;.21,1.22,;.21,2.76,;-1.12,3.53,;-2.45,2.76,;-2.45,1.22,;-1.12,.45,;-3.92,.75,;-4.32,-.74,;-3.55,-2.08,;-4.88,-2.85,;-5.65,-1.51,;-5.28,-4.33,;-6.77,-4.73,;-7.17,-6.22,;-6.08,-7.31,;-4.59,-6.91,;-4.19,-5.42,;-4.82,1.99,;-6.36,1.99,;-3.92,3.24,;-2.83,4.33,;-3.23,5.81,;-4.72,6.21,;-5.81,5.12,;-5.41,3.64,;-5.11,7.7,;-6.6,8.1,;-4.03,8.79,;1.55,-5.71,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C4CC4)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C32CCN(CC2)C(=O)C(C)(C)C)ccc1C |r,wU:27.30,29.35,(1.81,-9.96,;1.81,-8.42,;.48,-7.65,;-.86,-8.42,;.48,-6.11,;1.81,-5.34,;1.81,-3.8,;3.14,-3.03,;3.14,-1.49,;1.81,-.72,;1.81,.82,;3.14,1.59,;4.48,.82,;5.94,1.3,;6.85,.05,;5.94,-1.19,;6.34,-2.68,;5.94,-4.17,;7.43,-3.77,;4.48,-.72,;.48,1.59,;.48,3.13,;-.86,3.9,;-2.19,3.13,;-2.19,1.59,;-.86,.82,;-3.66,1.12,;-4.06,-.37,;-3.29,-1.7,;-4.62,-2.47,;-5.39,-1.14,;-5.02,-3.96,;-6.5,-4.36,;-6.9,-5.85,;-5.81,-6.94,;-4.33,-6.54,;-3.93,-5.05,;-4.56,2.36,;-6.1,2.36,;-3.66,3.61,;-2.57,4.7,;-2.97,6.19,;-4.45,6.58,;-5.54,5.49,;-5.14,4.01,;-4.85,8.07,;-3.76,9.16,;-6.34,8.47,;-7.43,7.38,;-6.74,9.96,;-5.25,9.56,;.48,-3.03,;-.86,-3.8,;-.86,-5.34,;-2.19,-6.11,)|
CC(C)NC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C32CCN(CC2)C2COC2)c(F)cc1C |r,wU:29.31,31.36,(-2.65,-10.45,;-1.32,-9.68,;.01,-10.45,;-1.32,-8.14,;.01,-7.37,;1.35,-8.14,;.01,-5.83,;1.35,-5.06,;1.35,-3.52,;2.68,-2.75,;2.68,-1.21,;1.35,-.44,;1.35,1.1,;2.68,1.87,;4.01,1.1,;5.48,1.57,;6.38,.33,;5.48,-.92,;5.88,-2.4,;4.79,-3.49,;7.37,-2.8,;4.01,-.44,;.01,1.87,;.01,3.41,;-1.32,4.18,;-2.65,3.41,;-2.65,1.87,;-1.32,1.1,;-4.12,1.39,;-4.52,-.09,;-3.75,-1.43,;-5.08,-2.2,;-5.85,-.86,;-5.48,-3.69,;-6.97,-4.08,;-7.37,-5.57,;-6.28,-6.66,;-4.79,-6.26,;-4.39,-4.77,;-5.02,2.64,;-6.56,2.64,;-4.12,3.88,;-3.03,4.97,;-3.43,6.46,;-4.92,6.86,;-6,5.77,;-5.61,4.28,;-5.31,8.35,;-4.54,9.68,;-5.88,10.45,;-6.65,9.12,;.01,-2.75,;.01,-1.21,;-1.32,-3.52,;-1.32,-5.06,;-2.65,-5.83,)|
CC(C)NC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@@H]2C[C@@H](C2)N2CCC(C)(C)C2)C(=O)C32CCN(CC2)C2COC2)c(F)cc1C |r,wU:29.31,31.36,(-2.09,-10.45,;-.76,-9.68,;.57,-10.45,;-.76,-8.14,;.57,-7.37,;1.91,-8.14,;.57,-5.83,;1.91,-5.06,;1.91,-3.52,;3.24,-2.75,;3.24,-1.21,;1.91,-.44,;1.91,1.1,;3.24,1.87,;4.57,1.1,;6.04,1.57,;6.94,.33,;6.04,-.92,;6.44,-2.4,;5.35,-3.49,;7.92,-2.8,;4.57,-.44,;.57,1.87,;.57,3.41,;-.76,4.18,;-2.09,3.41,;-2.09,1.87,;-.76,1.1,;-3.56,1.39,;-3.96,-.09,;-5.29,-.86,;-4.52,-2.2,;-3.19,-1.43,;-4.92,-3.69,;-4.01,-4.93,;-4.92,-6.18,;-6.38,-5.7,;-7.92,-5.7,;-6.78,-7.19,;-6.38,-4.16,;-4.46,2.64,;-6,2.64,;-3.56,3.88,;-2.47,4.97,;-2.87,6.46,;-4.36,6.86,;-5.45,5.77,;-5.05,4.28,;-4.75,8.35,;-3.98,9.68,;-5.32,10.45,;-6.09,9.12,;.57,-2.75,;.57,-1.21,;-.76,-3.52,;-.76,-5.06,;-2.09,-5.83,)|
CCn1cnc2cc(nc(Nc3cc(C(=O)NC)c(C)cc3F)c12)-c1ccc2c(c1)N([C@H]1C[C@H](C1)N1CCCCC1)C(=O)C2(C)C |r,wU:31.34,33.39,(7.37,-1.42,;5.88,-1.02,;5.48,.47,;6.38,1.71,;5.48,2.96,;4.01,2.48,;2.68,3.25,;1.35,2.48,;1.35,.94,;2.68,.17,;2.68,-1.37,;1.35,-2.14,;1.35,-3.68,;.01,-4.45,;.01,-5.99,;-1.32,-6.76,;1.35,-6.76,;2.68,-5.99,;-1.32,-3.68,;-2.65,-4.45,;-1.32,-2.14,;.01,-1.37,;.01,.17,;4.01,.94,;.01,3.25,;.01,4.79,;-1.32,5.56,;-2.65,4.79,;-2.65,3.25,;-1.32,2.48,;-4.12,2.78,;-4.52,1.29,;-3.75,-.04,;-5.08,-.81,;-5.85,.52,;-5.48,-2.3,;-6.97,-2.7,;-7.37,-4.19,;-6.28,-5.28,;-4.79,-4.88,;-4.39,-3.39,;-5.02,4.02,;-6.56,4.02,;-4.12,5.27,;-3.03,6.36,;-4.52,6.76,)|
CCn1cnc2cc(nc(Nc3ccc(C)c(c3)C(=O)NC)c12)-c1ccc2c(c1)N([C@H]1C[C@H](C1)N1CCCCC1)C(=O)C2(C)C |r,wU:30.33,32.38,(7.37,-1.42,;5.88,-1.02,;5.48,.47,;6.38,1.71,;5.48,2.96,;4.01,2.48,;2.68,3.25,;1.35,2.48,;1.35,.94,;2.68,.17,;2.68,-1.37,;1.35,-2.14,;.01,-1.37,;-1.32,-2.14,;-1.32,-3.68,;-2.65,-4.45,;.01,-4.45,;1.35,-3.68,;.01,-5.99,;-1.32,-6.76,;1.35,-6.76,;2.68,-5.99,;4.01,.94,;.01,3.25,;.01,4.79,;-1.32,5.56,;-2.65,4.79,;-2.65,3.25,;-1.32,2.48,;-4.12,2.78,;-4.52,1.29,;-3.75,-.04,;-5.08,-.81,;-5.85,.52,;-5.48,-2.3,;-6.97,-2.7,;-7.37,-4.19,;-6.28,-5.28,;-4.79,-4.88,;-4.39,-3.39,;-5.02,4.02,;-6.56,4.02,;-4.12,5.27,;-3.03,6.36,;-4.52,6.76,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@@H]2C[C@@H](C2)N2CCCC2)C(=O)C3(C)C)ccc1C |r,wU:27.29,29.34,(2.47,-5.99,;1.14,-6.76,;-.2,-5.99,;-1.53,-6.76,;-.2,-4.45,;1.14,-3.68,;1.14,-2.14,;2.47,-1.37,;2.47,.17,;1.14,.94,;1.14,2.48,;2.47,3.25,;3.8,2.48,;5.27,2.96,;6.17,1.71,;5.27,.47,;5.67,-1.02,;7.15,-1.42,;4.58,-2.11,;3.8,.94,;-.2,3.25,;-.2,4.79,;-1.53,5.56,;-2.86,4.79,;-2.86,3.25,;-1.53,2.48,;-4.33,2.78,;-4.73,1.29,;-6.06,.52,;-5.29,-.81,;-3.96,-.04,;-5.69,-2.3,;-7.15,-2.78,;-7.15,-4.32,;-5.69,-4.79,;-4.78,-3.55,;-5.23,4.02,;-6.77,4.02,;-4.33,5.27,;-3.93,6.76,;-5.42,6.36,;-.2,-1.37,;-1.53,-2.14,;-1.53,-3.68,;-2.86,-4.45,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@@H]2C[C@@H](C2)N2CCC(C2)C(F)F)C(=O)C3(C)C)ccc1C |r,wU:27.29,29.34,(3.8,-5.99,;2.47,-6.76,;1.14,-5.99,;-.2,-6.76,;1.14,-4.45,;2.47,-3.68,;2.47,-2.14,;3.8,-1.37,;3.8,.17,;2.47,.94,;2.47,2.48,;3.8,3.25,;5.14,2.48,;6.6,2.96,;7.51,1.71,;6.6,.47,;7,-1.02,;8.49,-1.42,;5.91,-2.11,;5.14,.94,;1.14,3.25,;1.14,4.79,;-.2,5.56,;-1.53,4.79,;-1.53,3.25,;-.2,2.48,;-3,2.78,;-3.39,1.29,;-4.73,.52,;-3.96,-.81,;-2.62,-.04,;-4.36,-2.3,;-3.45,-3.55,;-4.36,-4.79,;-5.82,-4.32,;-5.82,-2.78,;-7.15,-5.09,;-8.49,-4.32,;-7.15,-6.63,;-3.9,4.02,;-5.44,4.02,;-3,5.27,;-2.6,6.76,;-4.08,6.36,;1.14,-1.37,;-.2,-2.14,;-.2,-3.68,;-1.53,-4.45,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@@H]2C[C@@H](C2)N2CC[C@H](C2)C(F)F)C(=O)C3(C)C)ccc1C |r,wU:27.29,29.34,34.40,(3.8,-5.99,;2.47,-6.76,;1.14,-5.99,;-.2,-6.76,;1.14,-4.45,;2.47,-3.68,;2.47,-2.14,;3.8,-1.37,;3.8,.17,;2.47,.94,;2.47,2.48,;3.8,3.25,;5.14,2.48,;6.6,2.96,;7.51,1.71,;6.6,.47,;7,-1.02,;8.49,-1.42,;5.91,-2.11,;5.14,.94,;1.14,3.25,;1.14,4.79,;-.2,5.56,;-1.53,4.79,;-1.53,3.25,;-.2,2.48,;-3,2.78,;-3.39,1.29,;-4.73,.52,;-3.96,-.81,;-2.62,-.04,;-4.36,-2.3,;-3.45,-3.55,;-4.36,-4.79,;-5.82,-4.32,;-5.82,-2.78,;-7.15,-5.09,;-8.49,-4.32,;-7.15,-6.63,;-3.9,4.02,;-5.44,4.02,;-3,5.27,;-2.6,6.76,;-4.08,6.36,;1.14,-1.37,;-.2,-2.14,;-.2,-3.68,;-1.53,-4.45,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@@H]2C[C@@H](C2)N2CC[C@@H](C2)C(F)F)C(=O)C3(C)C)ccc1C |r,wU:27.29,29.34,wD:34.40,(3.8,-5.99,;2.47,-6.76,;1.14,-5.99,;-.2,-6.76,;1.14,-4.45,;2.47,-3.68,;2.47,-2.14,;3.8,-1.37,;3.8,.17,;2.47,.94,;2.47,2.48,;3.8,3.25,;5.14,2.48,;6.6,2.96,;7.51,1.71,;6.6,.47,;7,-1.02,;8.49,-1.42,;5.91,-2.11,;5.14,.94,;1.14,3.25,;1.14,4.79,;-.2,5.56,;-1.53,4.79,;-1.53,3.25,;-.2,2.48,;-3,2.78,;-3.39,1.29,;-4.73,.52,;-3.96,-.81,;-2.62,-.04,;-4.36,-2.3,;-3.45,-3.55,;-4.36,-4.79,;-5.82,-4.32,;-5.82,-2.78,;-7.15,-5.09,;-8.49,-4.32,;-7.15,-6.63,;-3.9,4.02,;-5.44,4.02,;-3,5.27,;-2.6,6.76,;-4.08,6.36,;1.14,-1.37,;-.2,-2.14,;-.2,-3.68,;-1.53,-4.45,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCC(C2)C(F)F)C(=O)C3(C)C)ccc1C |r,wU:27.29,29.34,(3.97,-5.99,;2.64,-6.76,;1.3,-5.99,;-.03,-6.76,;1.3,-4.45,;2.64,-3.68,;2.64,-2.14,;3.97,-1.37,;3.97,.17,;2.64,.94,;2.64,2.48,;3.97,3.25,;5.3,2.48,;6.77,2.96,;7.67,1.71,;6.77,.47,;7.17,-1.02,;8.65,-1.42,;6.08,-2.11,;5.3,.94,;1.3,3.25,;1.3,4.79,;-.03,5.56,;-1.37,4.79,;-1.37,3.25,;-.03,2.48,;-2.83,2.78,;-3.23,1.29,;-2.46,-.04,;-3.79,-.81,;-4.56,.52,;-4.19,-2.3,;-3.1,-3.39,;-3.5,-4.88,;-4.99,-5.28,;-6.08,-4.19,;-5.68,-2.7,;-7.56,-4.59,;-8.65,-3.5,;-7.96,-6.07,;-3.74,4.02,;-5.28,4.02,;-2.83,5.27,;-2.43,6.76,;-3.92,6.36,;1.3,-1.37,;-.03,-2.14,;-.03,-3.68,;-1.37,-4.45,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCC[C@H](C2)C(F)F)C(=O)C3(C)C)ccc1C |r,wU:27.29,29.34,35.41,(3.97,-5.99,;2.64,-6.76,;1.3,-5.99,;-.03,-6.76,;1.3,-4.45,;2.64,-3.68,;2.64,-2.14,;3.97,-1.37,;3.97,.17,;2.64,.94,;2.64,2.48,;3.97,3.25,;5.3,2.48,;6.77,2.96,;7.67,1.71,;6.77,.47,;7.17,-1.02,;8.65,-1.42,;6.08,-2.11,;5.3,.94,;1.3,3.25,;1.3,4.79,;-.03,5.56,;-1.37,4.79,;-1.37,3.25,;-.03,2.48,;-2.83,2.78,;-3.23,1.29,;-2.46,-.04,;-3.79,-.81,;-4.56,.52,;-4.19,-2.3,;-3.1,-3.39,;-3.5,-4.88,;-4.99,-5.28,;-6.08,-4.19,;-5.68,-2.7,;-7.56,-4.59,;-8.65,-3.5,;-7.96,-6.07,;-3.74,4.02,;-5.28,4.02,;-2.83,5.27,;-2.43,6.76,;-3.92,6.36,;1.3,-1.37,;-.03,-2.14,;-.03,-3.68,;-1.37,-4.45,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCC[C@@H](C2)C(F)F)C(=O)C3(C)C)ccc1C |r,wU:27.29,29.34,wD:35.41,(3.97,-5.99,;2.64,-6.76,;1.3,-5.99,;-.03,-6.76,;1.3,-4.45,;2.64,-3.68,;2.64,-2.14,;3.97,-1.37,;3.97,.17,;2.64,.94,;2.64,2.48,;3.97,3.25,;5.3,2.48,;6.77,2.96,;7.67,1.71,;6.77,.47,;7.17,-1.02,;8.65,-1.42,;6.08,-2.11,;5.3,.94,;1.3,3.25,;1.3,4.79,;-.03,5.56,;-1.37,4.79,;-1.37,3.25,;-.03,2.48,;-2.83,2.78,;-3.23,1.29,;-2.46,-.04,;-3.79,-.81,;-4.56,.52,;-4.19,-2.3,;-3.1,-3.39,;-3.5,-4.88,;-4.99,-5.28,;-6.08,-4.19,;-5.68,-2.7,;-7.56,-4.59,;-8.65,-3.5,;-7.96,-6.07,;-3.74,4.02,;-5.28,4.02,;-2.83,5.27,;-2.43,6.76,;-3.92,6.36,;1.3,-1.37,;-.03,-2.14,;-.03,-3.68,;-1.37,-4.45,)|
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CNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCC[C@@H](F)C2)C(=O)C3(C)C)c(F)cc1C |r,wU:27.29,29.34,35.39,(3.42,-5.99,;2.09,-6.76,;.76,-5.99,;-.58,-6.76,;.76,-4.45,;2.09,-3.68,;2.09,-2.14,;3.42,-1.37,;3.42,.17,;2.09,.94,;2.09,2.48,;3.42,3.25,;4.76,2.48,;6.22,2.96,;7.13,1.71,;6.22,.47,;6.62,-1.02,;8.11,-1.42,;5.53,-2.11,;4.76,.94,;.76,3.25,;.76,4.79,;-.58,5.56,;-1.91,4.79,;-1.91,3.25,;-.58,2.48,;-3.37,2.78,;-3.77,1.29,;-3,-.04,;-4.34,-.81,;-5.11,.52,;-4.74,-2.3,;-3.65,-3.39,;-4.05,-4.88,;-5.53,-5.28,;-6.62,-4.19,;-8.11,-4.59,;-6.22,-2.7,;-4.28,4.02,;-5.82,4.02,;-3.37,5.27,;-2.98,6.76,;-4.46,6.36,;.76,-1.37,;.76,.17,;-.58,-2.14,;-.58,-3.68,;-1.91,-4.45,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@@H]2C[C@@H](C2)N2CC[C@@H](F)C2)C(=O)C3(C)C)c(F)cc1C |r,wU:27.29,29.34,34.38,(3.14,-5.99,;1.8,-6.76,;.47,-5.99,;-.86,-6.76,;.47,-4.45,;1.8,-3.68,;1.8,-2.14,;3.14,-1.37,;3.14,.17,;1.8,.94,;1.8,2.48,;3.14,3.25,;4.47,2.48,;5.94,2.96,;6.84,1.71,;5.94,.47,;6.33,-1.02,;7.82,-1.42,;5.24,-2.11,;4.47,.94,;.47,3.25,;.47,4.79,;-.86,5.56,;-2.2,4.79,;-2.2,3.25,;-.86,2.48,;-3.66,2.78,;-4.06,1.29,;-5.39,.52,;-4.62,-.81,;-3.29,-.04,;-5.02,-2.3,;-4.12,-3.55,;-5.02,-4.79,;-6.49,-4.32,;-7.82,-5.09,;-6.49,-2.78,;-4.57,4.02,;-6.11,4.02,;-3.66,5.27,;-3.26,6.76,;-4.75,6.36,;.47,-1.37,;.47,.17,;-.86,-2.14,;-.86,-3.68,;-2.2,-4.45,)|
CC[C@H](C)n1cnc2cc(nc(Nc3cc(C(=O)NC)c(C)cc3F)c12)-c1ccc2c(c1)N([C@@H]1C[C@@H](C1)N1CC[C@@H](F)C1)C(=O)C2(C)C |r,wU:33.36,35.41,40.45,wD:2.2,(8.37,-.33,;7.28,-1.42,;5.79,-1.02,;4.7,-2.11,;5.39,.47,;6.3,1.71,;5.39,2.96,;3.93,2.48,;2.59,3.25,;1.26,2.48,;1.26,.94,;2.59,.17,;2.59,-1.37,;1.26,-2.14,;1.26,-3.68,;-.07,-4.45,;-.07,-5.99,;-1.41,-6.76,;1.26,-6.76,;2.59,-5.99,;-1.41,-3.68,;-2.74,-4.45,;-1.41,-2.14,;-.07,-1.37,;-.07,.17,;3.93,.94,;-.07,3.25,;-.07,4.79,;-1.41,5.56,;-2.74,4.79,;-2.74,3.25,;-1.41,2.48,;-4.21,2.78,;-4.61,1.29,;-5.94,.52,;-5.17,-.81,;-3.84,-.04,;-5.57,-2.3,;-4.66,-3.55,;-5.57,-4.79,;-7.03,-4.32,;-8.37,-5.09,;-7.03,-2.78,;-5.11,4.02,;-6.65,4.02,;-4.21,5.27,;-3.81,6.76,;-5.3,6.36,)|
CC(C)NC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCC[C@@H](F)C2)C(=O)C3(C)C)c(F)cc1C |r,wU:29.31,31.36,37.41,(4.76,-6.76,;3.42,-5.99,;3.42,-4.45,;2.09,-6.76,;.76,-5.99,;-.58,-6.76,;.76,-4.45,;2.09,-3.68,;2.09,-2.14,;3.42,-1.37,;3.42,.17,;2.09,.94,;2.09,2.48,;3.42,3.25,;4.76,2.48,;6.22,2.96,;7.13,1.71,;6.22,.47,;6.62,-1.02,;8.11,-1.42,;5.53,-2.11,;4.76,.94,;.76,3.25,;.76,4.79,;-.58,5.56,;-1.91,4.79,;-1.91,3.25,;-.58,2.48,;-3.37,2.78,;-3.77,1.29,;-3,-.04,;-4.34,-.81,;-5.11,.52,;-4.74,-2.3,;-3.65,-3.39,;-4.05,-4.88,;-5.53,-5.28,;-6.62,-4.19,;-8.11,-4.59,;-6.22,-2.7,;-4.28,4.02,;-5.82,4.02,;-3.37,5.27,;-2.98,6.76,;-4.46,6.36,;.76,-1.37,;.76,.17,;-.58,-2.14,;-.58,-3.68,;-1.91,-4.45,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2cnc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C3(C)C)c(F)cc1C |r,wU:27.29,29.34,(2.68,-5.99,;1.35,-6.76,;.01,-5.99,;-1.32,-6.76,;.01,-4.45,;1.35,-3.68,;1.35,-2.14,;2.68,-1.37,;2.68,.17,;1.35,.94,;1.35,2.48,;2.68,3.25,;4.01,2.48,;5.48,2.96,;6.38,1.71,;5.48,.47,;5.88,-1.02,;7.37,-1.42,;4.79,-2.11,;4.01,.94,;.01,3.25,;.01,4.79,;-1.32,5.56,;-2.65,4.79,;-2.65,3.25,;-1.32,2.48,;-4.12,2.78,;-4.52,1.29,;-3.75,-.04,;-5.08,-.81,;-5.85,.52,;-5.48,-2.3,;-6.97,-2.7,;-7.37,-4.19,;-6.28,-5.28,;-4.79,-4.88,;-4.39,-3.39,;-5.02,4.02,;-6.56,4.02,;-4.12,5.27,;-3.72,6.76,;-5.21,6.36,;.01,-1.37,;.01,.17,;-1.32,-2.14,;-1.32,-3.68,;-2.65,-4.45,)|
Cc1ccc(Nc2nc(cc3ncn(C4CC4)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C3(C)C)cc1C(N)=O |r,wU:25.28,27.33,(-2.45,-4.45,;-1.12,-3.68,;-1.12,-2.14,;.21,-1.37,;1.55,-2.14,;2.88,-1.37,;2.88,.17,;1.55,.94,;1.55,2.48,;2.88,3.25,;4.21,2.48,;5.68,2.96,;6.58,1.71,;5.68,.47,;6.08,-1.02,;5.68,-2.51,;7.17,-2.11,;4.21,.94,;.21,3.25,;.21,4.79,;-1.12,5.56,;-2.45,4.79,;-2.45,3.25,;-1.12,2.48,;-3.92,2.78,;-4.32,1.29,;-3.55,-.04,;-4.88,-.81,;-5.65,.52,;-5.28,-2.3,;-6.77,-2.7,;-7.17,-4.19,;-6.08,-5.28,;-4.59,-4.88,;-4.19,-3.39,;-4.82,4.02,;-6.36,4.02,;-3.92,5.27,;-3.52,6.76,;-5.01,6.36,;1.55,-3.68,;.21,-4.45,;.21,-5.99,;-1.12,-6.76,;1.55,-6.76,)|
CC[C@H](C)n1cnc2cc(nc(Nc3cc(C(=O)NC)c(C)cc3F)c12)-c1ccc2c(c1)N([C@H]1C[C@H](C1)N1CCC[C@@H](F)C1)C(=O)C2(C)C |r,wU:33.36,35.41,41.46,wD:2.2,(8.65,.44,;7.56,-.65,;6.08,-.25,;4.99,-1.34,;5.68,1.24,;6.58,2.48,;5.68,3.73,;4.21,3.25,;2.88,4.02,;1.55,3.25,;1.55,1.71,;2.88,.94,;2.88,-.6,;1.55,-1.37,;1.55,-2.91,;.21,-3.68,;.21,-5.22,;-1.12,-5.99,;1.55,-5.99,;1.55,-7.53,;-1.12,-2.91,;-2.45,-3.68,;-1.12,-1.37,;.21,-.6,;.21,.94,;4.21,1.71,;.21,4.02,;.21,5.56,;-1.12,6.33,;-2.45,5.56,;-2.45,4.02,;-1.12,3.25,;-3.92,3.55,;-4.32,2.06,;-3.55,.73,;-4.88,-.04,;-5.65,1.29,;-5.28,-1.53,;-4.19,-2.62,;-4.59,-4.11,;-6.08,-4.51,;-7.17,-3.42,;-8.65,-3.82,;-6.77,-1.93,;-4.82,4.79,;-6.36,4.79,;-3.92,6.04,;-3.52,7.53,;-5.01,7.13,)|
CC[C@H](C)n1cnc2cc(nc(Nc3ccc(Cl)c(c3)C(=O)NC)c12)-c1ccc2c(c1)N([C@H]1C[C@H](C1)N1CCCCC1)C(=O)C2(C)C |r,wU:32.35,34.40,wD:2.2,(7.91,-.33,;6.82,-1.42,;5.33,-1.02,;4.24,-2.11,;4.93,.47,;5.84,1.71,;4.93,2.96,;3.47,2.48,;2.14,3.25,;.8,2.48,;.8,.94,;2.14,.17,;2.14,-1.37,;.8,-2.14,;-.53,-1.37,;-1.86,-2.14,;-1.86,-3.68,;-3.2,-4.45,;-.53,-4.45,;.8,-3.68,;-.53,-5.99,;-1.86,-6.76,;.8,-6.76,;2.14,-5.99,;3.47,.94,;-.53,3.25,;-.53,4.79,;-1.86,5.56,;-3.2,4.79,;-3.2,3.25,;-1.86,2.48,;-4.66,2.78,;-5.06,1.29,;-4.29,-.04,;-5.63,-.81,;-6.4,.52,;-6.02,-2.3,;-7.51,-2.7,;-7.91,-4.19,;-6.82,-5.28,;-5.33,-4.88,;-4.93,-3.39,;-5.57,4.02,;-7.11,4.02,;-4.66,5.27,;-4.26,6.76,;-5.75,6.36,)|
CC(C)NC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C3(C)C)ccc1Cl |r,wU:29.31,31.36,(4.01,-6.76,;2.68,-5.99,;2.68,-4.45,;1.35,-6.76,;.01,-5.99,;-1.32,-6.76,;.01,-4.45,;1.35,-3.68,;1.35,-2.14,;2.68,-1.37,;2.68,.17,;1.35,.94,;1.35,2.48,;2.68,3.25,;4.01,2.48,;5.48,2.96,;6.38,1.71,;5.48,.47,;5.88,-1.02,;4.79,-2.11,;7.37,-1.42,;4.01,.94,;.01,3.25,;.01,4.79,;-1.32,5.56,;-2.65,4.79,;-2.65,3.25,;-1.32,2.48,;-4.12,2.78,;-4.52,1.29,;-3.75,-.04,;-5.08,-.81,;-5.85,.52,;-5.48,-2.3,;-6.97,-2.7,;-7.37,-4.19,;-6.28,-5.28,;-4.79,-4.88,;-4.39,-3.39,;-5.02,4.02,;-6.56,4.02,;-4.12,5.27,;-3.72,6.76,;-5.21,6.36,;.01,-1.37,;-1.32,-2.14,;-1.32,-3.68,;-2.65,-4.45,)|
COCCNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C3(C)C)c(F)cc1C |r,wU:30.32,32.37,(6.68,-6.76,;5.35,-5.99,;4.01,-6.76,;2.68,-5.99,;1.35,-6.76,;.01,-5.99,;-1.32,-6.76,;.01,-4.45,;1.35,-3.68,;1.35,-2.14,;2.68,-1.37,;2.68,.17,;1.35,.94,;1.35,2.48,;2.68,3.25,;4.01,2.48,;5.48,2.96,;6.38,1.71,;5.48,.47,;5.88,-1.02,;4.79,-2.11,;7.37,-1.42,;4.01,.94,;.01,3.25,;.01,4.79,;-1.32,5.56,;-2.65,4.79,;-2.65,3.25,;-1.32,2.48,;-4.12,2.78,;-4.52,1.29,;-3.75,-.04,;-5.08,-.81,;-5.85,.52,;-5.48,-2.3,;-6.97,-2.7,;-7.37,-4.19,;-6.28,-5.28,;-4.79,-4.88,;-4.39,-3.39,;-5.02,4.02,;-6.56,4.02,;-4.12,5.27,;-3.72,6.76,;-5.21,6.36,;.01,-1.37,;.01,.17,;-1.32,-2.14,;-1.32,-3.68,;-2.65,-4.45,)|
CC(C)NC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C3(C)C)c(F)cc1Cl |r,wU:29.31,31.36,(4.01,-6.76,;2.68,-5.99,;2.68,-4.45,;1.35,-6.76,;.01,-5.99,;-1.32,-6.76,;.01,-4.45,;1.35,-3.68,;1.35,-2.14,;2.68,-1.37,;2.68,.17,;1.35,.94,;1.35,2.48,;2.68,3.25,;4.01,2.48,;5.48,2.96,;6.38,1.71,;5.48,.47,;5.88,-1.02,;4.79,-2.11,;7.37,-1.42,;4.01,.94,;.01,3.25,;.01,4.79,;-1.32,5.56,;-2.65,4.79,;-2.65,3.25,;-1.32,2.48,;-4.12,2.78,;-4.52,1.29,;-3.75,-.04,;-5.08,-.81,;-5.85,.52,;-5.48,-2.3,;-6.97,-2.7,;-7.37,-4.19,;-6.28,-5.28,;-4.79,-4.88,;-4.39,-3.39,;-5.02,4.02,;-6.56,4.02,;-4.12,5.27,;-3.72,6.76,;-5.21,6.36,;.01,-1.37,;.01,.17,;-1.32,-2.14,;-1.32,-3.68,;-2.65,-4.45,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C3(C)C)c(F)cc1Cl |r,wU:27.29,29.34,(2.68,-5.99,;1.35,-6.76,;.01,-5.99,;-1.32,-6.76,;.01,-4.45,;1.35,-3.68,;1.35,-2.14,;2.68,-1.37,;2.68,.17,;1.35,.94,;1.35,2.48,;2.68,3.25,;4.01,2.48,;5.48,2.96,;6.38,1.71,;5.48,.47,;5.88,-1.02,;4.79,-2.11,;7.37,-1.42,;4.01,.94,;.01,3.25,;.01,4.79,;-1.32,5.56,;-2.65,4.79,;-2.65,3.25,;-1.32,2.48,;-4.12,2.78,;-4.52,1.29,;-3.75,-.04,;-5.08,-.81,;-5.85,.52,;-5.48,-2.3,;-6.97,-2.7,;-7.37,-4.19,;-6.28,-5.28,;-4.79,-4.88,;-4.39,-3.39,;-5.02,4.02,;-6.56,4.02,;-4.12,5.27,;-3.72,6.76,;-5.21,6.36,;.01,-1.37,;.01,.17,;-1.32,-2.14,;-1.32,-3.68,;-2.65,-4.45,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C3(C)C)ccc1Cl |r,wU:27.29,29.34,(2.68,-5.99,;1.35,-6.76,;.01,-5.99,;-1.32,-6.76,;.01,-4.45,;1.35,-3.68,;1.35,-2.14,;2.68,-1.37,;2.68,.17,;1.35,.94,;1.35,2.48,;2.68,3.25,;4.01,2.48,;5.48,2.96,;6.38,1.71,;5.48,.47,;5.88,-1.02,;4.79,-2.11,;7.37,-1.42,;4.01,.94,;.01,3.25,;.01,4.79,;-1.32,5.56,;-2.65,4.79,;-2.65,3.25,;-1.32,2.48,;-4.12,2.78,;-4.52,1.29,;-3.75,-.04,;-5.08,-.81,;-5.85,.52,;-5.48,-2.3,;-6.97,-2.7,;-7.37,-4.19,;-6.28,-5.28,;-4.79,-4.88,;-4.39,-3.39,;-5.02,4.02,;-6.56,4.02,;-4.12,5.27,;-3.72,6.76,;-5.21,6.36,;.01,-1.37,;-1.32,-2.14,;-1.32,-3.68,;-2.65,-4.45,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@@H]2C[C@@H](C2)N2CC(C)(C)C2)C(=O)C3(C)C)c(F)cc1C |r,wU:27.29,29.34,(2.56,-5.99,;1.23,-6.76,;-.1,-5.99,;-1.44,-6.76,;-.1,-4.45,;1.23,-3.68,;1.23,-2.14,;2.56,-1.37,;2.56,.17,;1.23,.94,;1.23,2.48,;2.56,3.25,;3.9,2.48,;5.36,2.96,;6.27,1.71,;5.36,.47,;5.76,-1.02,;4.67,-2.11,;7.25,-1.42,;3.9,.94,;-.1,3.25,;-.1,4.79,;-1.44,5.56,;-2.77,4.79,;-2.77,3.25,;-1.44,2.48,;-4.24,2.78,;-4.63,1.29,;-5.97,.52,;-5.2,-.81,;-3.86,-.04,;-5.6,-2.3,;-6.93,-3.07,;-6.16,-4.4,;-5.76,-5.89,;-7.25,-5.49,;-4.83,-3.63,;-5.14,4.02,;-6.68,4.02,;-4.24,5.27,;-3.84,6.76,;-5.32,6.36,;-.1,-1.37,;-.1,.17,;-1.44,-2.14,;-1.44,-3.68,;-2.77,-4.45,)|
CC(C)n1cnc2cc(nc(Nc3ccc(C)c(c3)C(=O)NC3CC3)c12)-c1ccc2c(c1)N([C@@H]1C[C@@H](C1)N1CC(C)(C)C1)C(=O)C2(C)C |r,wU:33.37,35.42,(4.67,-2.11,;5.76,-1.02,;7.25,-1.42,;5.36,.47,;6.27,1.71,;5.36,2.96,;3.9,2.48,;2.56,3.25,;1.23,2.48,;1.23,.94,;2.56,.17,;2.56,-1.37,;1.23,-2.14,;-.1,-1.37,;-1.44,-2.14,;-1.44,-3.68,;-2.77,-4.45,;-.1,-4.45,;1.23,-3.68,;-.1,-5.99,;-1.44,-6.76,;1.23,-6.76,;2.56,-5.99,;4.1,-5.99,;3.33,-4.65,;3.9,.94,;-.1,3.25,;-.1,4.79,;-1.44,5.56,;-2.77,4.79,;-2.77,3.25,;-1.44,2.48,;-4.24,2.78,;-4.63,1.29,;-5.97,.52,;-5.2,-.81,;-3.86,-.04,;-5.6,-2.3,;-6.93,-3.07,;-6.16,-4.4,;-5.76,-5.89,;-7.25,-5.49,;-4.83,-3.63,;-5.14,4.02,;-6.68,4.02,;-4.24,5.27,;-3.84,6.76,;-5.32,6.36,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@@H]2C[C@@H](C2)N2CC(C)(C)C2)C(=O)C3(C)C)ccc1C |r,wU:27.29,29.34,(2.56,-5.99,;1.23,-6.76,;-.1,-5.99,;-1.44,-6.76,;-.1,-4.45,;1.23,-3.68,;1.23,-2.14,;2.56,-1.37,;2.56,.17,;1.23,.94,;1.23,2.48,;2.56,3.25,;3.9,2.48,;5.36,2.96,;6.27,1.71,;5.36,.47,;5.76,-1.02,;4.67,-2.11,;7.25,-1.42,;3.9,.94,;-.1,3.25,;-.1,4.79,;-1.44,5.56,;-2.77,4.79,;-2.77,3.25,;-1.44,2.48,;-4.24,2.78,;-4.63,1.29,;-5.97,.52,;-5.2,-.81,;-3.86,-.04,;-5.6,-2.3,;-6.93,-3.07,;-6.16,-4.4,;-5.76,-5.89,;-7.25,-5.49,;-4.83,-3.63,;-5.14,4.02,;-6.68,4.02,;-4.24,5.27,;-3.84,6.76,;-5.32,6.36,;-.1,-1.37,;-1.44,-2.14,;-1.44,-3.68,;-2.77,-4.45,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C32CCOCC2)ccc1C |r,wU:27.29,29.34,(2.68,-6.73,;1.35,-7.5,;.01,-6.73,;-1.32,-7.5,;.01,-5.19,;1.35,-4.42,;1.35,-2.88,;2.68,-2.11,;2.68,-.57,;1.35,.2,;1.35,1.74,;2.68,2.51,;4.01,1.74,;5.48,2.22,;6.38,.97,;5.48,-.28,;5.88,-1.76,;4.79,-2.85,;7.37,-2.16,;4.01,.2,;.01,2.51,;.01,4.05,;-1.32,4.82,;-2.65,4.05,;-2.65,2.51,;-1.32,1.74,;-4.12,2.03,;-4.52,.55,;-3.75,-.79,;-5.08,-1.56,;-5.85,-.22,;-5.48,-3.05,;-6.97,-3.44,;-7.37,-4.93,;-6.28,-6.02,;-4.79,-5.62,;-4.39,-4.13,;-5.02,3.28,;-6.56,3.28,;-4.12,4.53,;-3.03,5.61,;-3.43,7.1,;-4.92,7.5,;-6,6.41,;-5.61,4.92,;.01,-2.11,;-1.32,-2.88,;-1.32,-4.42,;-2.65,-5.19,)|
CC(C)NC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C32CCOCC2)ccc1C |r,wU:29.31,31.36,(4.01,-7.5,;2.68,-6.73,;2.68,-5.19,;1.35,-7.5,;.01,-6.73,;-1.32,-7.5,;.01,-5.19,;1.35,-4.42,;1.35,-2.88,;2.68,-2.11,;2.68,-.57,;1.35,.2,;1.35,1.74,;2.68,2.51,;4.01,1.74,;5.48,2.22,;6.38,.97,;5.48,-.28,;5.88,-1.76,;4.79,-2.85,;7.37,-2.16,;4.01,.2,;.01,2.51,;.01,4.05,;-1.32,4.82,;-2.65,4.05,;-2.65,2.51,;-1.32,1.74,;-4.12,2.03,;-4.52,.55,;-3.75,-.79,;-5.08,-1.56,;-5.85,-.22,;-5.48,-3.05,;-6.97,-3.44,;-7.37,-4.93,;-6.28,-6.02,;-4.79,-5.62,;-4.39,-4.13,;-5.02,3.28,;-6.56,3.28,;-4.12,4.53,;-3.03,5.61,;-3.43,7.1,;-4.92,7.5,;-6,6.41,;-5.61,4.92,;.01,-2.11,;-1.32,-2.88,;-1.32,-4.42,;-2.65,-5.19,)|
CC(C)NC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C32CCOCC2)c(F)cc1C |r,wU:29.31,31.36,(4.01,-7.5,;2.68,-6.73,;2.68,-5.19,;1.35,-7.5,;.01,-6.73,;-1.32,-7.5,;.01,-5.19,;1.35,-4.42,;1.35,-2.88,;2.68,-2.11,;2.68,-.57,;1.35,.2,;1.35,1.74,;2.68,2.51,;4.01,1.74,;5.48,2.22,;6.38,.97,;5.48,-.28,;5.88,-1.76,;4.79,-2.85,;7.37,-2.16,;4.01,.2,;.01,2.51,;.01,4.05,;-1.32,4.82,;-2.65,4.05,;-2.65,2.51,;-1.32,1.74,;-4.12,2.03,;-4.52,.55,;-3.75,-.79,;-5.08,-1.56,;-5.85,-.22,;-5.48,-3.05,;-6.97,-3.44,;-7.37,-4.93,;-6.28,-6.02,;-4.79,-5.62,;-4.39,-4.13,;-5.02,3.28,;-6.56,3.28,;-4.12,4.53,;-3.03,5.61,;-3.43,7.1,;-4.92,7.5,;-6,6.41,;-5.61,4.92,;.01,-2.11,;.01,-.57,;-1.32,-2.88,;-1.32,-4.42,;-2.65,-5.19,)|
Cc1ccc(Nc2nc(cc3ncn(C4CC4)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C32CCOCC2)cc1C(N)=O |r,wU:25.28,27.33,(-2.45,-5.19,;-1.12,-4.42,;-1.12,-2.88,;.21,-2.11,;1.55,-2.88,;2.88,-2.11,;2.88,-.57,;1.55,.2,;1.55,1.74,;2.88,2.51,;4.21,1.74,;5.68,2.22,;6.58,.97,;5.68,-.28,;6.08,-1.76,;5.68,-3.25,;7.17,-2.85,;4.21,.2,;.21,2.51,;.21,4.05,;-1.12,4.82,;-2.45,4.05,;-2.45,2.51,;-1.12,1.74,;-3.92,2.03,;-4.32,.55,;-3.55,-.79,;-4.88,-1.56,;-5.65,-.22,;-5.28,-3.05,;-6.77,-3.44,;-7.17,-4.93,;-6.08,-6.02,;-4.59,-5.62,;-4.19,-4.13,;-4.82,3.28,;-6.36,3.28,;-3.92,4.53,;-2.83,5.61,;-3.23,7.1,;-4.72,7.5,;-5.81,6.41,;-5.41,4.92,;1.55,-4.42,;.21,-5.19,;.21,-6.73,;1.55,-7.5,;-1.12,-7.5,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C4CC4)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C32CCOCC2)ccc1C |r,wU:27.30,29.35,(2.88,-6.73,;1.55,-7.5,;.21,-6.73,;-1.12,-7.5,;.21,-5.19,;1.55,-4.42,;1.55,-2.88,;2.88,-2.11,;2.88,-.57,;1.55,.2,;1.55,1.74,;2.88,2.51,;4.21,1.74,;5.68,2.22,;6.58,.97,;5.68,-.28,;6.08,-1.76,;5.68,-3.25,;7.17,-2.85,;4.21,.2,;.21,2.51,;.21,4.05,;-1.12,4.82,;-2.45,4.05,;-2.45,2.51,;-1.12,1.74,;-3.92,2.03,;-4.32,.55,;-3.55,-.79,;-4.88,-1.56,;-5.65,-.22,;-5.28,-3.05,;-6.77,-3.44,;-7.17,-4.93,;-6.08,-6.02,;-4.59,-5.62,;-4.19,-4.13,;-4.82,3.28,;-6.36,3.28,;-3.92,4.53,;-2.83,5.61,;-3.23,7.1,;-4.72,7.5,;-5.81,6.41,;-5.41,4.92,;.21,-2.11,;-1.12,-2.88,;-1.12,-4.42,;-2.45,-5.19,)|
CC[C@H](C)n1cnc2cc(nc(Nc3ccc(C)c(c3)C(=O)NC)c12)-c1ccc2c(c1)N([C@H]1C[C@H](C1)N1CCCCC1)C(=O)C2(C)C |r,wU:32.35,34.40,wD:2.2,(7.91,.44,;6.82,-.65,;5.33,-.25,;4.24,-1.34,;4.93,1.24,;5.84,2.48,;4.93,3.73,;3.47,3.25,;2.14,4.02,;.8,3.25,;.8,1.71,;2.14,.94,;2.14,-.6,;.8,-1.37,;-.53,-.6,;-1.86,-1.37,;-1.86,-2.91,;-3.2,-3.68,;-.53,-3.68,;.8,-2.91,;-.53,-5.22,;-1.86,-5.99,;.8,-5.99,;.8,-7.53,;3.47,1.71,;-.53,4.02,;-.53,5.56,;-1.86,6.33,;-3.2,5.56,;-3.2,4.02,;-1.86,3.25,;-4.66,3.55,;-5.06,2.06,;-4.29,.73,;-5.63,-.04,;-6.4,1.29,;-6.02,-1.53,;-7.51,-1.93,;-7.91,-3.42,;-6.82,-4.51,;-5.33,-4.11,;-4.93,-2.62,;-5.57,4.79,;-7.11,4.79,;-4.66,6.04,;-4.26,7.53,;-5.75,7.13,)|
CC(C)NC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C32CCN(CC2)C(C)=O)c(F)cc1C |r,wU:29.31,31.36,(-3.63,-6.79,;-2.86,-8.12,;-3.63,-9.46,;-1.32,-8.12,;.01,-7.35,;1.35,-8.12,;.01,-5.81,;1.35,-5.04,;1.35,-3.5,;2.68,-2.73,;2.68,-1.19,;1.35,-.42,;1.35,1.12,;2.68,1.89,;4.01,1.12,;5.48,1.59,;6.38,.35,;5.48,-.9,;5.88,-2.39,;7.37,-2.78,;4.79,-3.47,;4.01,-.42,;.01,1.89,;.01,3.43,;-1.32,4.2,;-2.65,3.43,;-2.65,1.89,;-1.32,1.12,;-4.12,1.41,;-4.52,-.08,;-3.75,-1.41,;-5.08,-2.18,;-5.85,-.85,;-5.48,-3.67,;-6.97,-4.07,;-7.37,-5.55,;-6.28,-6.64,;-4.79,-6.24,;-4.39,-4.76,;-5.02,2.66,;-6.56,2.66,;-4.12,3.9,;-3.03,4.99,;-3.43,6.48,;-4.92,6.88,;-6,5.79,;-5.61,4.3,;-5.31,8.37,;-6.8,8.77,;-4.23,9.46,;.01,-2.73,;.01,-1.19,;-1.32,-3.5,;-1.32,-5.04,;-2.65,-5.81,)|
CCNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C32CCN(CC2)C(C)=O)ccc1C |r,wU:28.30,30.35,(4.01,-8.79,;2.68,-8.02,;1.35,-8.79,;.01,-8.02,;-1.32,-8.79,;.01,-6.48,;1.35,-5.71,;1.35,-4.17,;2.68,-3.4,;2.68,-1.86,;1.35,-1.09,;1.35,.45,;2.68,1.22,;4.01,.45,;5.48,.93,;6.38,-.32,;5.48,-1.56,;5.88,-3.05,;7.37,-3.45,;4.79,-4.14,;4.01,-1.09,;.01,1.22,;.01,2.76,;-1.32,3.53,;-2.65,2.76,;-2.65,1.22,;-1.32,.45,;-4.12,.75,;-4.52,-.74,;-3.75,-2.08,;-5.08,-2.85,;-5.85,-1.51,;-5.48,-4.33,;-6.97,-4.73,;-7.37,-6.22,;-6.28,-7.31,;-4.79,-6.91,;-4.39,-5.42,;-5.02,1.99,;-6.56,1.99,;-4.12,3.24,;-3.03,4.33,;-3.43,5.81,;-4.92,6.21,;-6,5.12,;-5.61,3.64,;-5.31,7.7,;-6.8,8.1,;-4.23,8.79,;.01,-3.4,;-1.32,-4.17,;-1.32,-5.71,;-2.65,-6.48,)|
COCCNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C32CCN(CC2)C(C)=O)ccc1C |r,wU:30.32,32.37,(6.68,-8.79,;5.35,-8.02,;4.01,-8.79,;2.68,-8.02,;1.35,-8.79,;.01,-8.02,;-1.32,-8.79,;.01,-6.48,;1.35,-5.71,;1.35,-4.17,;2.68,-3.4,;2.68,-1.86,;1.35,-1.09,;1.35,.45,;2.68,1.22,;4.01,.45,;5.48,.93,;6.38,-.32,;5.48,-1.56,;5.88,-3.05,;7.37,-3.45,;4.79,-4.14,;4.01,-1.09,;.01,1.22,;.01,2.76,;-1.32,3.53,;-2.65,2.76,;-2.65,1.22,;-1.32,.45,;-4.12,.75,;-4.52,-.74,;-3.75,-2.08,;-5.08,-2.85,;-5.85,-1.51,;-5.48,-4.33,;-6.97,-4.73,;-7.37,-6.22,;-6.28,-7.31,;-4.79,-6.91,;-4.39,-5.42,;-5.02,1.99,;-6.56,1.99,;-4.12,3.24,;-3.03,4.33,;-3.43,5.81,;-4.92,6.21,;-6,5.12,;-5.61,3.64,;-5.31,7.7,;-6.8,8.1,;-4.23,8.79,;.01,-3.4,;-1.32,-4.17,;-1.32,-5.71,;-2.65,-6.48,)|
CC(C)n1cnc2cc(nc(Nc3ccc(C)c(c3)C(=O)NCCO)c12)-c1ccc2c(c1)N([C@H]1C[C@H](C1)N1CCCCC1)C(=O)C21CCN(CC1)C(C)=O |r,wU:33.36,35.41,(7.37,-3.45,;5.88,-3.05,;4.79,-4.14,;5.48,-1.56,;6.38,-.32,;5.48,.93,;4.01,.45,;2.68,1.22,;1.35,.45,;1.35,-1.09,;2.68,-1.86,;2.68,-3.4,;1.35,-4.17,;.01,-3.4,;-1.32,-4.17,;-1.32,-5.71,;-2.65,-6.48,;.01,-6.48,;1.35,-5.71,;.01,-8.02,;-1.32,-8.79,;1.35,-8.79,;2.68,-8.02,;4.01,-8.79,;5.35,-8.02,;4.01,-1.09,;.01,1.22,;.01,2.76,;-1.32,3.53,;-2.65,2.76,;-2.65,1.22,;-1.32,.45,;-4.12,.75,;-4.52,-.74,;-3.75,-2.08,;-5.08,-2.85,;-5.85,-1.51,;-5.48,-4.33,;-6.97,-4.73,;-7.37,-6.22,;-6.28,-7.31,;-4.79,-6.91,;-4.39,-5.42,;-5.02,1.99,;-6.56,1.99,;-4.12,3.24,;-3.03,4.33,;-3.43,5.81,;-4.92,6.21,;-6,5.12,;-5.61,3.64,;-5.31,7.7,;-6.8,8.1,;-4.23,8.79,)|
CCn1cnc2cc(nc(Nc3ccc(C)c(c3)C(N)=O)c12)-c1ccc2c(c1)N([C@@H]1C[C@@H](C1)NC(=O)C(C)(C)C)C(=O)C2(C)C |r,wU:29.32,31.37,(6.99,-1.02,;5.45,-1.02,;5.05,.47,;5.96,1.71,;5.05,2.96,;3.59,2.48,;2.25,3.25,;.92,2.48,;.92,.94,;2.25,.17,;2.25,-1.37,;.92,-2.14,;-.41,-1.37,;-1.75,-2.14,;-1.75,-3.68,;-3.08,-4.45,;-.41,-4.45,;.92,-3.68,;-.41,-5.99,;.92,-6.76,;-1.75,-6.76,;3.59,.94,;-.41,3.25,;-.41,4.79,;-1.75,5.56,;-3.08,4.79,;-3.08,3.25,;-1.75,2.48,;-4.55,2.78,;-4.94,1.29,;-6.28,.52,;-5.51,-.81,;-4.17,-.04,;-5.91,-2.3,;-4.82,-3.39,;-3.33,-2.99,;-5.22,-4.88,;-6.7,-5.28,;-4.82,-6.37,;-3.68,-4.88,;-5.45,4.02,;-6.99,4.02,;-4.55,5.27,;-4.15,6.76,;-5.63,6.36,)|
CC(C)n1cnc2cc(nc(Nc3cc(C(=O)NC4(CF)CC4)c(C)cc3F)c12)-c1cnc2c(c1)N([C@H]1C[C@H](C1)N1CCCCC1)C(=O)C2(C)C |r,wU:36.40,38.45,(7.37,-1.42,;5.88,-1.02,;4.79,-2.11,;5.48,.47,;6.38,1.71,;5.48,2.96,;4.01,2.48,;2.68,3.25,;1.35,2.48,;1.35,.94,;2.68,.17,;2.68,-1.37,;1.35,-2.14,;1.35,-3.68,;.01,-4.45,;.01,-5.99,;-1.32,-6.76,;1.35,-6.76,;2.68,-5.99,;4.01,-6.76,;5.35,-5.99,;1.91,-4.65,;3.45,-4.65,;-1.32,-3.68,;-2.65,-4.45,;-1.32,-2.14,;.01,-1.37,;.01,.17,;4.01,.94,;.01,3.25,;.01,4.79,;-1.32,5.56,;-2.65,4.79,;-2.65,3.25,;-1.32,2.48,;-4.12,2.78,;-4.52,1.29,;-3.75,-.04,;-5.08,-.81,;-5.85,.52,;-5.48,-2.3,;-6.97,-2.7,;-7.37,-4.19,;-6.28,-5.28,;-4.79,-4.88,;-4.39,-3.39,;-5.02,4.02,;-6.56,4.02,;-4.12,5.27,;-3.72,6.76,;-5.21,6.36,)|
CC(C)n1cnc2cc(nc(Nc3ccc(C)c(c3)C(N)=O)c12)-c1ccc2c(c1)N(C1CC(C1)NC(=O)C(C)(C)C)C(=O)C2(C)C |(-2.25,5.87,;-.74,5.55,;.29,6.7,;-.27,4.09,;-1.17,2.84,;-.27,1.6,;1.2,2.07,;2.53,1.3,;3.86,2.07,;3.86,3.61,;2.53,4.38,;2.53,5.92,;3.86,6.69,;3.86,8.23,;5.2,9,;6.53,8.23,;7.87,9,;6.53,6.69,;5.2,5.92,;7.87,5.92,;7.87,4.38,;9.2,6.69,;1.2,3.61,;5.2,1.3,;5.2,-.24,;6.53,-1.01,;7.87,-.24,;7.87,1.3,;6.53,2.07,;9.33,1.78,;9.81,3.24,;9.11,4.62,;10.48,5.31,;11.18,3.94,;10.95,6.78,;12.46,7.1,;13.49,5.96,;12.94,8.56,;13.41,10.03,;14.4,8.09,;11.47,9.04,;10.23,.53,;11.77,.53,;9.33,-.71,;8.7,-2.12,;10.66,-1.48,)|
CC(C)NC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N(C2CC(C2)N2CCCCC2)C(=O)C3(C)C)ccc1C |(2.53,13.62,;3.86,12.85,;5.2,13.62,;3.86,11.31,;5.2,10.54,;6.53,11.31,;5.2,9,;3.86,8.23,;3.86,6.69,;2.53,5.92,;2.53,4.38,;3.86,3.61,;3.86,2.07,;2.53,1.3,;1.2,2.07,;-.27,1.6,;-1.17,2.84,;-.27,4.09,;-.74,5.55,;-2.25,5.87,;.29,6.7,;1.2,3.61,;5.2,1.3,;5.2,-.24,;6.53,-1.01,;7.87,-.24,;7.87,1.3,;6.53,2.07,;9.33,1.78,;9.81,3.24,;9.11,4.62,;10.48,5.31,;11.18,3.94,;10.95,6.78,;9.92,7.92,;10.4,9.39,;11.91,9.71,;12.94,8.56,;12.46,7.1,;10.23,.53,;11.77,.53,;9.33,-.71,;10.66,-1.48,;8.7,-2.12,;5.2,5.92,;6.53,6.69,;6.53,8.23,;7.87,9,)|
COCCNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C3(C)C)ccc1C |r,wU:30.32,32.37,(6.68,-6.76,;5.35,-5.99,;4.01,-6.76,;2.68,-5.99,;1.35,-6.76,;.01,-5.99,;-1.32,-6.76,;.01,-4.45,;1.35,-3.68,;1.35,-2.14,;2.68,-1.37,;2.68,.17,;1.35,.94,;1.35,2.48,;2.68,3.25,;4.01,2.48,;5.48,2.96,;6.38,1.71,;5.48,.47,;5.88,-1.02,;7.37,-1.42,;4.79,-2.11,;4.01,.94,;.01,3.25,;.01,4.79,;-1.32,5.56,;-2.65,4.79,;-2.65,3.25,;-1.32,2.48,;-4.12,2.78,;-4.52,1.29,;-3.75,-.04,;-5.08,-.81,;-5.85,.52,;-5.48,-2.3,;-6.97,-2.7,;-7.37,-4.19,;-6.28,-5.28,;-4.79,-4.88,;-4.39,-3.39,;-5.02,4.02,;-6.56,4.02,;-4.12,5.27,;-5.21,6.36,;-3.72,6.76,;.01,-1.37,;-1.32,-2.14,;-1.32,-3.68,;-2.65,-4.45,)|
CCNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C3(C)C)ccc1C |r,wU:28.30,30.35,(4.01,-6.76,;2.68,-5.99,;1.35,-6.76,;.01,-5.99,;-1.32,-6.76,;.01,-4.45,;1.35,-3.68,;1.35,-2.14,;2.68,-1.37,;2.68,.17,;1.35,.94,;1.35,2.48,;2.68,3.25,;4.01,2.48,;5.48,2.96,;6.38,1.71,;5.48,.47,;5.88,-1.02,;7.37,-1.42,;4.79,-2.11,;4.01,.94,;.01,3.25,;.01,4.79,;-1.32,5.56,;-2.65,4.79,;-2.65,3.25,;-1.32,2.48,;-4.12,2.78,;-4.52,1.29,;-3.75,-.04,;-5.08,-.81,;-5.85,.52,;-5.48,-2.3,;-6.97,-2.7,;-7.37,-4.19,;-6.28,-5.28,;-4.79,-4.88,;-4.39,-3.39,;-5.02,4.02,;-6.56,4.02,;-4.12,5.27,;-5.21,6.36,;-3.72,6.76,;.01,-1.37,;-1.32,-2.14,;-1.32,-3.68,;-2.65,-4.45,)|
CC(C)CNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C3(C)C)ccc1C |r,wU:30.32,32.37,(4.01,-7.53,;4.01,-5.99,;5.35,-5.22,;2.68,-5.22,;1.35,-5.99,;.01,-5.22,;-1.32,-5.99,;.01,-3.68,;1.35,-2.91,;1.35,-1.37,;2.68,-.6,;2.68,.94,;1.35,1.71,;1.35,3.25,;2.68,4.02,;4.01,3.25,;5.48,3.73,;6.38,2.48,;5.48,1.24,;5.88,-.25,;7.37,-.65,;4.79,-1.34,;4.01,1.71,;.01,4.02,;.01,5.56,;-1.32,6.33,;-2.65,5.56,;-2.65,4.02,;-1.32,3.25,;-4.12,3.55,;-4.52,2.06,;-3.75,.73,;-5.08,-.04,;-5.85,1.29,;-5.48,-1.53,;-6.97,-1.93,;-7.37,-3.42,;-6.28,-4.51,;-4.79,-4.11,;-4.39,-2.62,;-5.02,4.79,;-6.56,4.79,;-4.12,6.04,;-5.21,7.13,;-3.72,7.53,;.01,-.6,;-1.32,-1.37,;-1.32,-2.91,;-2.65,-3.68,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C3(C)C)ccc1OC(F)(F)F |r,wU:27.29,29.34,(2.68,-5.39,;1.35,-6.16,;.01,-5.39,;-1.32,-6.16,;.01,-3.85,;1.35,-3.08,;1.35,-1.54,;2.68,-.77,;2.68,.77,;1.35,1.54,;1.35,3.08,;2.68,3.85,;4.01,3.08,;5.48,3.56,;6.38,2.31,;5.48,1.07,;5.88,-.42,;7.37,-.82,;4.79,-1.51,;4.01,1.54,;.01,3.85,;.01,5.39,;-1.32,6.16,;-2.65,5.39,;-2.65,3.85,;-1.32,3.08,;-4.12,3.38,;-4.52,1.89,;-3.75,.56,;-5.08,-.21,;-5.85,1.12,;-5.48,-1.7,;-6.97,-2.1,;-7.37,-3.59,;-6.28,-4.67,;-4.79,-4.28,;-4.39,-2.79,;-5.02,4.62,;-6.56,4.62,;-4.12,5.87,;-5.21,6.96,;-3.72,7.36,;.01,-.77,;-1.32,-1.54,;-1.32,-3.08,;-3.4,-4.28,;-3.4,-5.82,;-2.07,-6.59,;-4.74,-6.59,;-3.4,-7.36,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C3(C)C)ccc1C(F)(F)F |r,wU:27.29,29.34,(2.68,-5.99,;1.35,-6.76,;.01,-5.99,;-1.32,-6.76,;.01,-4.45,;1.35,-3.68,;1.35,-2.14,;2.68,-1.37,;2.68,.17,;1.35,.94,;1.35,2.48,;2.68,3.25,;4.01,2.48,;5.48,2.96,;6.38,1.71,;5.48,.47,;5.88,-1.02,;7.37,-1.42,;4.79,-2.11,;4.01,.94,;.01,3.25,;.01,4.79,;-1.32,5.56,;-2.65,4.79,;-2.65,3.25,;-1.32,2.48,;-4.12,2.78,;-4.52,1.29,;-3.75,-.04,;-5.08,-.81,;-5.85,.52,;-5.48,-2.3,;-6.97,-2.7,;-7.37,-4.19,;-6.28,-5.28,;-4.79,-4.88,;-4.39,-3.39,;-5.02,4.02,;-6.56,4.02,;-4.12,5.27,;-5.21,6.36,;-3.72,6.76,;.01,-1.37,;-1.32,-2.14,;-1.32,-3.68,;-2.65,-4.45,;-2.65,-5.99,;-3.99,-3.68,;-3.99,-5.22,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C3(C)C)ccc1C1CC1 |r,wU:27.29,29.34,(2.68,-5.99,;1.35,-6.76,;.01,-5.99,;-1.32,-6.76,;.01,-4.45,;1.35,-3.68,;1.35,-2.14,;2.68,-1.37,;2.68,.17,;1.35,.94,;1.35,2.48,;2.68,3.25,;4.01,2.48,;5.48,2.96,;6.38,1.71,;5.48,.47,;5.88,-1.02,;7.37,-1.42,;4.79,-2.11,;4.01,.94,;.01,3.25,;.01,4.79,;-1.32,5.56,;-2.65,4.79,;-2.65,3.25,;-1.32,2.48,;-4.12,2.78,;-4.52,1.29,;-3.75,-.04,;-5.08,-.81,;-5.85,.52,;-5.48,-2.3,;-6.97,-2.7,;-7.37,-4.19,;-6.28,-5.28,;-4.79,-4.88,;-4.39,-3.39,;-5.02,4.02,;-6.56,4.02,;-4.12,5.27,;-5.21,6.36,;-3.72,6.76,;.01,-1.37,;-1.32,-2.14,;-1.32,-3.68,;-2.65,-4.45,;-4.19,-4.45,;-3.42,-5.78,)|
CCc1ccc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C3(C)C)cc1C(=O)NC |r,wU:26.28,28.33,(-3.99,-3.68,;-2.65,-4.45,;-1.32,-3.68,;-1.32,-2.14,;.01,-1.37,;1.35,-2.14,;2.68,-1.37,;2.68,.17,;1.35,.94,;1.35,2.48,;2.68,3.25,;4.01,2.48,;5.48,2.96,;6.38,1.71,;5.48,.47,;5.88,-1.02,;7.37,-1.42,;4.79,-2.11,;4.01,.94,;.01,3.25,;.01,4.79,;-1.32,5.56,;-2.65,4.79,;-2.65,3.25,;-1.32,2.48,;-4.12,2.78,;-4.52,1.29,;-3.75,-.04,;-5.08,-.81,;-5.85,.52,;-5.48,-2.3,;-6.97,-2.7,;-7.37,-4.19,;-6.28,-5.28,;-4.79,-4.88,;-4.39,-3.39,;-5.02,4.02,;-6.56,4.02,;-4.12,5.27,;-5.21,6.36,;-3.72,6.76,;1.35,-3.68,;.01,-4.45,;.01,-5.99,;-1.32,-6.76,;1.35,-6.76,;2.68,-5.99,)|
CC(C)n1cnc2cc(nc(Nc3cc(C(=O)NC4(CC4)C(F)F)c(C)c(F)c3F)c12)-c1ccc2c(c1)N([C@H]1C[C@H](C1)N1CCCCC1)C(=O)C2(C)C |r,wU:38.42,40.47,(7.37,-.65,;5.88,-.25,;4.79,-1.34,;5.48,1.24,;6.38,2.48,;5.48,3.73,;4.01,3.25,;2.68,4.02,;1.35,3.25,;1.35,1.71,;2.68,.94,;2.68,-.6,;1.35,-1.37,;1.35,-2.91,;.01,-3.68,;.01,-5.22,;-1.32,-5.99,;1.35,-5.99,;2.68,-5.22,;1.91,-3.88,;3.45,-3.88,;4.01,-5.99,;4.01,-7.53,;5.35,-5.22,;-1.32,-2.91,;-2.65,-3.68,;-1.32,-1.37,;-2.65,-.6,;.01,-.6,;.01,.94,;4.01,1.71,;.01,4.02,;.01,5.56,;-1.32,6.33,;-2.65,5.56,;-2.65,4.02,;-1.32,3.25,;-4.12,3.55,;-4.52,2.06,;-3.75,.73,;-5.08,-.04,;-5.85,1.29,;-5.48,-1.53,;-6.97,-1.93,;-7.37,-3.42,;-6.28,-4.51,;-4.79,-4.11,;-4.39,-2.62,;-5.02,4.79,;-6.56,4.79,;-4.12,6.04,;-5.21,7.13,;-3.72,7.53,)|
CC(C)n1cnc2cc(nc(Nc3cc(C(=O)NC4(CC4)C(F)F)c(C)c(F)c3F)c12)-c1ccc2c(c1)N(C1CC(C1)N1CC3CCC1C3)C(=O)C2(C)C |(-2.25,5.87,;-.74,5.55,;.29,6.7,;-.27,4.09,;-1.17,2.84,;-.27,1.6,;1.2,2.07,;2.53,1.3,;3.86,2.07,;3.86,3.61,;2.53,4.38,;2.53,5.92,;3.86,6.69,;5.2,5.92,;6.53,6.69,;7.87,5.92,;7.87,4.38,;9.2,6.69,;10.53,5.92,;11.52,4.74,;10.01,4.48,;11.52,7.1,;11,8.55,;13.04,6.84,;6.53,8.23,;7.87,9,;5.2,9,;5.2,10.54,;3.86,8.23,;2.53,9,;1.2,3.61,;5.2,1.3,;6.53,2.07,;7.87,1.3,;7.87,-.24,;6.53,-1.01,;5.2,-.24,;6.85,-2.51,;5.82,-3.66,;4.28,-3.74,;4.36,-5.28,;5.9,-5.2,;3.33,-6.42,;1.83,-6.1,;.8,-7.25,;1.27,-8.71,;2.78,-9.03,;3.81,-7.89,;2.22,-7.94,;8.38,-2.67,;9.15,-4.01,;9.01,-1.27,;10.48,-1.73,;10.16,-.25,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N(C2CC(C2)N2CCCCC2)C(=O)C32CCN(CC2)C(=O)C(C)(C)O)ccc1C |(1.33,13.09,;1.33,11.55,;,10.78,;-1.33,11.55,;,9.24,;-1.33,8.47,;-1.33,6.93,;-2.67,6.16,;-2.67,4.62,;-1.33,3.85,;-1.33,2.31,;-2.67,1.54,;-4,2.31,;-5.47,1.83,;-6.37,3.08,;-5.47,4.33,;-5.94,5.79,;-7.45,6.11,;-4.91,6.94,;-4,3.85,;,1.54,;1.33,2.31,;2.67,1.54,;2.67,,;1.33,-.77,;;1.65,-2.28,;.62,-3.42,;.7,-4.96,;-.83,-5.04,;-.91,-3.5,;-1.86,-6.18,;-1.39,-7.65,;-2.42,-8.79,;-3.93,-8.47,;-4.4,-7.01,;-3.37,-5.86,;3.19,-2.44,;3.96,-3.77,;3.81,-1.03,;4.84,-2.17,;6.35,-1.85,;6.82,-.39,;5.79,.75,;4.29,.43,;8.33,-.07,;9.36,-1.21,;8.81,1.39,;10.27,.92,;9.28,2.86,;7.34,1.87,;,6.16,;1.33,6.93,;1.33,8.47,;2.67,9.24,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C32CCN(CC2)C(=O)[C@@H](C)O)ccc1C |r,wU:27.29,29.34,47.55,(2.68,-8.76,;1.35,-9.53,;.01,-8.76,;-1.32,-9.53,;.01,-7.22,;1.35,-6.45,;1.35,-4.91,;2.68,-4.14,;2.68,-2.6,;1.35,-1.83,;1.35,-.29,;2.68,.48,;4.01,-.29,;5.48,.18,;6.38,-1.06,;5.48,-2.31,;5.88,-3.8,;7.37,-4.19,;4.79,-4.88,;4.01,-1.83,;.01,.48,;.01,2.02,;-1.32,2.79,;-2.65,2.02,;-2.65,.48,;-1.32,-.29,;-4.12,0,;-4.52,-1.49,;-3.75,-2.82,;-5.08,-3.59,;-5.85,-2.26,;-5.48,-5.08,;-6.97,-5.48,;-7.37,-6.96,;-6.28,-8.05,;-4.79,-7.65,;-4.39,-6.17,;-5.02,1.25,;-6.56,1.25,;-4.12,2.49,;-3.03,3.58,;-3.43,5.07,;-4.92,5.47,;-6,4.38,;-5.61,2.89,;-5.31,6.96,;-6.8,7.35,;-4.23,8.04,;-4.62,9.53,;-2.74,7.65,;.01,-4.14,;-1.32,-4.91,;-1.32,-6.45,;-2.65,-7.22,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C32CCN(CC2)C(=O)C23CC(O)(C2)C3)ccc1C |r,wU:27.29,29.34,(2.68,-9.33,;1.35,-10.1,;.01,-9.33,;-1.32,-10.1,;.01,-7.79,;1.35,-7.02,;1.35,-5.48,;2.68,-4.71,;2.68,-3.17,;1.35,-2.4,;1.35,-.86,;2.68,-.09,;4.01,-.86,;5.48,-.39,;6.38,-1.63,;5.48,-2.88,;5.88,-4.37,;7.37,-4.77,;4.79,-5.46,;4.01,-2.4,;.01,-.09,;.01,1.45,;-1.32,2.22,;-2.65,1.45,;-2.65,-.09,;-1.32,-.86,;-4.12,-.57,;-4.52,-2.06,;-3.75,-3.39,;-5.08,-4.16,;-5.85,-2.83,;-5.48,-5.65,;-6.97,-6.05,;-7.37,-7.53,;-6.28,-8.62,;-4.79,-8.22,;-4.39,-6.74,;-5.02,.68,;-6.56,.68,;-4.12,1.92,;-3.03,3.01,;-3.43,4.5,;-4.92,4.9,;-6,3.81,;-5.61,2.32,;-5.31,6.39,;-6.8,6.78,;-4.23,7.47,;-2.69,7.47,;-2.69,9.01,;-1.6,10.1,;-4.23,9.01,;-3.68,8.42,;.01,-4.71,;-1.32,-5.48,;-1.32,-7.02,;-2.65,-7.79,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C4CC4)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C32CCN(CC2)C(=O)C2(C)CCC2)ccc1C |r,wU:27.30,29.35,(2.88,-8.69,;1.55,-9.46,;.21,-8.69,;-1.12,-9.46,;.21,-7.15,;1.55,-6.38,;1.55,-4.84,;2.88,-4.07,;2.88,-2.53,;1.55,-1.76,;1.55,-.22,;2.88,.55,;4.21,-.22,;5.68,.26,;6.58,-.99,;5.68,-2.23,;6.08,-3.72,;5.68,-5.21,;7.17,-4.81,;4.21,-1.76,;.21,.55,;.21,2.09,;-1.12,2.86,;-2.45,2.09,;-2.45,.55,;-1.12,-.22,;-3.92,.08,;-4.32,-1.41,;-3.55,-2.74,;-4.88,-3.51,;-5.65,-2.18,;-5.28,-5,;-6.77,-5.4,;-7.17,-6.89,;-6.08,-7.98,;-4.59,-7.58,;-4.19,-6.09,;-4.82,1.32,;-6.36,1.32,;-3.92,2.57,;-2.83,3.66,;-3.23,5.15,;-4.72,5.55,;-5.81,4.46,;-5.41,2.97,;-5.11,7.03,;-6.6,7.43,;-4.03,8.12,;-5.36,8.89,;-2.69,7.35,;-1.92,8.69,;-3.26,9.46,;.21,-4.07,;-1.12,-4.84,;-1.12,-6.38,;-2.45,-7.15,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C4CC4)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C32CCN(CC2)C(=O)C2(C)CC2)ccc1C |r,wU:27.30,29.35,(2.88,-8.76,;1.55,-9.53,;.21,-8.76,;-1.12,-9.53,;.21,-7.22,;1.55,-6.45,;1.55,-4.91,;2.88,-4.14,;2.88,-2.6,;1.55,-1.83,;1.55,-.29,;2.88,.48,;4.21,-.29,;5.68,.18,;6.58,-1.06,;5.68,-2.31,;6.08,-3.8,;5.68,-5.28,;7.17,-4.88,;4.21,-1.83,;.21,.48,;.21,2.02,;-1.12,2.79,;-2.45,2.02,;-2.45,.48,;-1.12,-.29,;-3.92,0,;-4.32,-1.49,;-3.55,-2.82,;-4.88,-3.59,;-5.65,-2.26,;-5.28,-5.08,;-6.77,-5.48,;-7.17,-6.96,;-6.08,-8.05,;-4.59,-7.65,;-4.19,-6.17,;-4.82,1.25,;-6.36,1.25,;-3.92,2.49,;-2.83,3.58,;-3.23,5.07,;-4.72,5.47,;-5.81,4.38,;-5.41,2.89,;-5.11,6.96,;-6.6,7.35,;-4.03,8.04,;-5.36,8.81,;-2.54,8.44,;-3.63,9.53,;.21,-4.14,;-1.12,-4.91,;-1.12,-6.45,;-2.45,-7.22,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C4CC4)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C32CCN(CC2)C(=O)[C@@H](C)O)ccc1C |r,wU:27.30,29.35,47.56,(1.81,-9.96,;1.81,-8.42,;.48,-7.65,;-.86,-8.42,;.48,-6.11,;1.81,-5.34,;1.81,-3.8,;3.14,-3.03,;3.14,-1.49,;1.81,-.72,;1.81,.82,;3.14,1.59,;4.48,.82,;5.94,1.3,;6.85,.05,;5.94,-1.19,;6.34,-2.68,;5.94,-4.17,;7.43,-3.77,;4.48,-.72,;.48,1.59,;.48,3.13,;-.86,3.9,;-2.19,3.13,;-2.19,1.59,;-.86,.82,;-3.66,1.12,;-4.06,-.37,;-3.29,-1.7,;-4.62,-2.47,;-5.39,-1.14,;-5.02,-3.96,;-6.5,-4.36,;-6.9,-5.85,;-5.81,-6.94,;-4.33,-6.54,;-3.93,-5.05,;-4.56,2.36,;-6.1,2.36,;-3.66,3.61,;-2.57,4.7,;-2.97,6.19,;-4.45,6.58,;-5.54,5.49,;-5.14,4.01,;-4.85,8.07,;-3.76,9.16,;-6.34,8.47,;-7.43,7.38,;-6.74,9.96,;.48,-3.03,;-.86,-3.8,;-.86,-5.34,;-2.19,-6.11,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N(C2CC(C2)N2CCCCC2)C(=O)C32CCN(CC2)C(=O)C2(C)CC2)ccc1C |(9.16,-6.59,;8.63,-5.14,;9.61,-3.96,;11.13,-4.22,;9.07,-2.51,;10.06,-1.33,;9.52,.12,;10.5,1.3,;9.97,2.75,;8.45,3,;7.91,4.45,;8.89,5.63,;10.41,5.38,;11.62,6.33,;12.9,5.48,;12.49,4,;13.44,2.79,;12.87,1.36,;14.97,3.01,;10.95,3.93,;6.39,4.7,;5.41,3.52,;3.89,3.77,;3.36,5.22,;4.34,6.4,;5.86,6.15,;3.51,7.7,;4.08,9.14,;3.47,10.55,;4.88,11.16,;5.49,9.75,;5.45,12.59,;4.49,13.8,;5.06,15.23,;6.58,15.46,;7.54,14.25,;6.97,12.82,;2.02,7.32,;.83,8.3,;1.92,5.79,;1.99,4.25,;.69,3.42,;-.68,4.14,;-.74,5.67,;.56,6.5,;-1.98,3.31,;-1.91,1.77,;-3.34,4.03,;-4.28,2.81,;-4.38,5.16,;-2.88,5.49,;8,.37,;7.02,-.81,;7.56,-2.26,;6.57,-3.44,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C4CC4)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C32CCN(CC2)C(=O)C2COC2)ccc1C |r,wU:27.30,29.35,(1.55,-10.33,;1.55,-8.79,;.21,-8.02,;-1.12,-8.79,;.21,-6.48,;1.55,-5.71,;1.55,-4.17,;2.88,-3.4,;2.88,-1.86,;1.55,-1.09,;1.55,.45,;2.88,1.22,;4.21,.45,;5.68,.93,;6.58,-.32,;5.68,-1.56,;6.08,-3.05,;5.68,-4.54,;7.17,-4.14,;4.21,-1.09,;.21,1.22,;.21,2.76,;-1.12,3.53,;-2.45,2.76,;-2.45,1.22,;-1.12,.45,;-3.92,.75,;-4.32,-.74,;-3.55,-2.08,;-4.88,-2.85,;-5.65,-1.51,;-5.28,-4.33,;-6.77,-4.73,;-7.17,-6.22,;-6.08,-7.31,;-4.59,-6.91,;-4.19,-5.42,;-4.82,1.99,;-6.36,1.99,;-3.92,3.24,;-2.83,4.33,;-3.23,5.81,;-4.72,6.21,;-5.81,5.12,;-5.41,3.64,;-5.11,7.7,;-6.6,8.1,;-4.03,8.79,;-2.49,8.79,;-2.49,10.33,;-4.03,10.33,;.21,-3.4,;-1.12,-4.17,;-1.12,-5.71,;-2.45,-6.48,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C4CC4)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C32CCN(CC2)C(=O)C23CC(F)(C2)C3)ccc1C |r,wU:27.30,29.35,(1.55,-10.87,;1.55,-9.33,;.21,-8.56,;-1.12,-9.33,;.21,-7.02,;1.55,-6.25,;1.55,-4.71,;2.88,-3.94,;2.88,-2.4,;1.55,-1.63,;1.55,-.09,;2.88,.68,;4.21,-.09,;5.68,.38,;6.58,-.86,;5.68,-2.11,;6.08,-3.6,;5.68,-5.08,;7.17,-4.69,;4.21,-1.63,;.21,.68,;.21,2.22,;-1.12,2.99,;-2.45,2.22,;-2.45,.68,;-1.12,-.09,;-3.92,.2,;-4.32,-1.29,;-3.55,-2.62,;-4.88,-3.39,;-5.65,-2.06,;-5.28,-4.88,;-6.77,-5.28,;-7.17,-6.76,;-6.08,-7.85,;-4.59,-7.45,;-4.19,-5.97,;-4.82,1.45,;-6.36,1.45,;-3.92,2.69,;-2.83,3.78,;-3.23,5.27,;-4.72,5.67,;-5.81,4.58,;-5.41,3.09,;-5.11,7.16,;-6.6,7.55,;-4.03,8.24,;-2.49,8.24,;-2.49,9.78,;-1.4,10.87,;-4.03,9.78,;-3.48,9.19,;.21,-3.94,;-1.12,-4.71,;-1.12,-6.25,;-2.45,-7.02,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C4CC4)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C32CCN(CC2)C(=O)C2CCC2)ccc1C |r,wU:27.30,29.35,(2.88,-8.79,;1.55,-9.56,;.21,-8.79,;-1.12,-9.56,;.21,-7.25,;1.55,-6.48,;1.55,-4.94,;2.88,-4.17,;2.88,-2.63,;1.55,-1.86,;1.55,-.32,;2.88,.45,;4.21,-.32,;5.68,.16,;6.58,-1.09,;5.68,-2.33,;6.08,-3.82,;5.68,-5.31,;7.17,-4.91,;4.21,-1.86,;.21,.45,;.21,1.99,;-1.12,2.76,;-2.45,1.99,;-2.45,.45,;-1.12,-.32,;-3.92,-.02,;-4.32,-1.51,;-3.55,-2.85,;-4.88,-3.62,;-5.65,-2.28,;-5.28,-5.1,;-6.77,-5.5,;-7.17,-6.99,;-6.08,-8.08,;-4.59,-7.68,;-4.19,-6.19,;-4.82,1.22,;-6.36,1.22,;-3.92,2.47,;-2.83,3.56,;-3.23,5.04,;-4.72,5.44,;-5.81,4.35,;-5.41,2.87,;-5.11,6.93,;-6.6,7.33,;-4.03,8.02,;-2.49,8.02,;-2.49,9.56,;-4.03,9.56,;.21,-4.17,;-1.12,-4.94,;-1.12,-6.48,;-2.45,-7.25,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C4CC4)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C32CCN(CC2)C(=O)C23CC(C2)C3)ccc1C |r,wU:27.30,29.35,(2.88,-8.79,;1.55,-9.56,;.21,-8.79,;-1.12,-9.56,;.21,-7.25,;1.55,-6.48,;1.55,-4.94,;2.88,-4.17,;2.88,-2.63,;1.55,-1.86,;1.55,-.32,;2.88,.45,;4.21,-.32,;5.68,.16,;6.58,-1.09,;5.68,-2.33,;6.08,-3.82,;5.68,-5.31,;7.17,-4.91,;4.21,-1.86,;.21,.45,;.21,1.99,;-1.12,2.76,;-2.45,1.99,;-2.45,.45,;-1.12,-.32,;-3.92,-.02,;-4.32,-1.51,;-3.55,-2.85,;-4.88,-3.62,;-5.65,-2.28,;-5.28,-5.1,;-6.77,-5.5,;-7.17,-6.99,;-6.08,-8.08,;-4.59,-7.68,;-4.19,-6.19,;-4.82,1.22,;-6.36,1.22,;-3.92,2.47,;-2.83,3.56,;-3.23,5.04,;-4.72,5.44,;-5.81,4.35,;-5.41,2.87,;-5.11,6.93,;-6.6,7.33,;-4.03,8.02,;-2.49,8.02,;-2.49,9.56,;-4.03,9.56,;-3.48,8.96,;.21,-4.17,;-1.12,-4.94,;-1.12,-6.48,;-2.45,-7.25,)|
CC[C@H](C)n1cnc2cc(nc(Nc3ccc(C)c(c3)C(=O)NC)c12)-c1ccc2c(c1)N(C1CC(C1)N1CCC[C@@H](F)C1)C(=O)C21CCN(CC1)C(C)=O |wD:2.2,40.45,(-8.48,4.97,;-7.45,6.11,;-5.94,5.79,;-4.91,6.94,;-5.47,4.33,;-6.37,3.08,;-5.47,1.83,;-4,2.31,;-2.67,1.54,;-1.33,2.31,;-1.33,3.85,;-2.67,4.62,;-2.67,6.16,;-1.33,6.93,;-1.33,8.47,;,9.24,;1.33,8.47,;2.67,9.24,;1.33,6.93,;,6.16,;2.67,6.16,;2.67,4.62,;4,6.93,;5.33,6.16,;-4,3.85,;,1.54,;1.33,2.31,;2.67,1.54,;2.67,,;1.33,-.77,;;1.65,-2.28,;.62,-3.42,;.7,-4.96,;-.83,-5.04,;-.91,-3.5,;-1.86,-6.18,;-3.37,-5.86,;-4.4,-7.01,;-3.93,-8.47,;-2.42,-8.79,;-1.94,-10.26,;-1.39,-7.65,;3.19,-2.44,;3.96,-3.77,;3.81,-1.03,;4.84,-2.17,;6.35,-1.85,;6.82,-.39,;5.79,.75,;4.29,.43,;8.33,-.07,;8.81,1.39,;9.36,-1.21,)|
CC[C@H](C)n1cnc2cc(nc(Nc3ccc(C)c(c3)C(=O)NC)c12)-c1ccc2c(c1)N([C@@H]1C[C@@H](C1)N1CCC3(CC3(F)F)C1)C(=O)C21CCN(CC1)C(C)=O |r,wU:32.35,34.40,wD:2.2,(8.47,-1.59,;7.38,-2.68,;5.89,-2.28,;4.8,-3.37,;5.49,-.79,;6.4,.45,;5.49,1.7,;4.03,1.22,;2.7,1.99,;1.36,1.22,;1.36,-.32,;2.7,-1.09,;2.7,-2.63,;1.36,-3.4,;.03,-2.63,;-1.31,-3.4,;-1.31,-4.94,;-2.64,-5.71,;.03,-5.71,;1.36,-4.94,;.03,-7.25,;-1.31,-8.02,;1.36,-8.02,;1.36,-9.56,;4.03,-.32,;.03,1.99,;.03,3.53,;-1.31,4.3,;-2.64,3.53,;-2.64,1.99,;-1.31,1.22,;-4.1,1.52,;-4.5,.03,;-5.84,-.74,;-5.07,-2.08,;-3.73,-1.31,;-5.46,-3.56,;-4.56,-4.81,;-5.46,-6.06,;-6.93,-5.58,;-8.47,-5.58,;-7.7,-6.91,;-8.47,-8.25,;-6.93,-8.25,;-6.93,-4.04,;-5.01,2.76,;-6.55,2.76,;-4.1,4.01,;-3.01,5.1,;-3.41,6.58,;-4.9,6.98,;-5.99,5.89,;-5.59,4.41,;-5.3,8.47,;-6.79,8.87,;-4.21,9.56,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C4CC4)c23)-c2ccc3c(c2)N([C@@H]2C[C@@H](C2)N2CCC(C)(C)C2)C(=O)C32CCN(CC2)C(C)=O)ccc1C |r,wU:27.30,29.35,(3.34,-8.02,;2,-8.79,;.67,-8.02,;-.66,-8.79,;.67,-6.48,;2,-5.71,;2,-4.17,;3.34,-3.4,;3.34,-1.86,;2,-1.09,;2,.45,;3.34,1.22,;4.67,.45,;6.13,.93,;7.04,-.32,;6.13,-1.56,;6.53,-3.05,;6.13,-4.54,;7.62,-4.14,;4.67,-1.09,;.67,1.22,;.67,2.76,;-.66,3.53,;-2,2.76,;-2,1.22,;-.66,.45,;-3.46,.75,;-3.86,-.74,;-5.2,-1.51,;-4.43,-2.85,;-3.09,-2.08,;-4.82,-4.33,;-3.92,-5.58,;-4.82,-6.83,;-6.29,-6.35,;-7.62,-7.12,;-7.62,-5.58,;-6.29,-4.81,;-4.37,1.99,;-5.91,1.99,;-3.46,3.24,;-2.37,4.33,;-2.77,5.81,;-4.26,6.21,;-5.35,5.12,;-4.95,3.64,;-4.66,7.7,;-3.57,8.79,;-6.15,8.1,;.67,-3.4,;-.66,-4.17,;-.66,-5.71,;-2,-6.48,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C4CC4)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CC(C)(C)CC(C)(C)C2)C(=O)C32CCN(CC2)C(C)=O)ccc1C |r,wU:27.30,29.35,(3.62,-8.02,;2.29,-8.79,;.96,-8.02,;-.38,-8.79,;.96,-6.48,;2.29,-5.71,;2.29,-4.17,;3.62,-3.4,;3.62,-1.86,;2.29,-1.09,;2.29,.45,;3.62,1.22,;4.96,.45,;6.42,.93,;7.33,-.32,;6.42,-1.56,;6.82,-3.05,;6.42,-4.54,;7.91,-4.14,;4.96,-1.09,;.96,1.22,;.96,2.76,;-.38,3.53,;-1.71,2.76,;-1.71,1.22,;-.38,.45,;-3.18,.75,;-3.57,-.74,;-2.8,-2.08,;-4.14,-2.85,;-4.91,-1.51,;-4.54,-4.33,;-3.45,-5.42,;-3.85,-6.91,;-3.85,-8.45,;-2.36,-7.31,;-5.33,-7.31,;-6.42,-6.22,;-7.91,-5.82,;-7.19,-7.55,;-6.02,-4.73,;-4.08,1.99,;-5.62,1.99,;-3.18,3.24,;-2.09,4.33,;-2.48,5.81,;-3.97,6.21,;-5.06,5.12,;-4.66,3.64,;-4.37,7.7,;-5.86,8.1,;-3.28,8.79,;.96,-3.4,;-.38,-4.17,;-.38,-5.71,;-1.71,-6.48,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C4CC4)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCC(C)(C)C2)C(=O)C32CCN(CC2)C(C)=O)ccc1C |r,wU:27.30,29.35,(3.62,-8.02,;2.29,-8.79,;.96,-8.02,;-.38,-8.79,;.96,-6.48,;2.29,-5.71,;2.29,-4.17,;3.62,-3.4,;3.62,-1.86,;2.29,-1.09,;2.29,.45,;3.62,1.22,;4.96,.45,;6.42,.93,;7.33,-.32,;6.42,-1.56,;6.82,-3.05,;6.42,-4.54,;7.91,-4.14,;4.96,-1.09,;.96,1.22,;.96,2.76,;-.38,3.53,;-1.71,2.76,;-1.71,1.22,;-.38,.45,;-3.18,.75,;-3.57,-.74,;-2.8,-2.08,;-4.14,-2.85,;-4.91,-1.51,;-4.54,-4.33,;-3.45,-5.42,;-3.85,-6.91,;-5.33,-7.31,;-6.42,-6.22,;-7.91,-5.82,;-7.19,-7.55,;-6.02,-4.73,;-4.08,1.99,;-5.62,1.99,;-3.18,3.24,;-2.09,4.33,;-2.48,5.81,;-3.97,6.21,;-5.06,5.12,;-4.66,3.64,;-4.37,7.7,;-5.86,8.1,;-3.28,8.79,;.96,-3.4,;-.38,-4.17,;-.38,-5.71,;-1.71,-6.48,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCC[C@@H](F)C2)C(=O)C32CCN(CC2)C(C)=O)ccc1C |r,wU:27.29,29.34,35.39,(3.42,-8.02,;2.09,-8.79,;.76,-8.02,;-.58,-8.79,;.76,-6.48,;2.09,-5.71,;2.09,-4.17,;3.42,-3.4,;3.42,-1.86,;2.09,-1.09,;2.09,.45,;3.42,1.22,;4.76,.45,;6.22,.93,;7.13,-.32,;6.22,-1.56,;6.62,-3.05,;5.53,-4.14,;8.11,-3.45,;4.76,-1.09,;.76,1.22,;.76,2.76,;-.58,3.53,;-1.91,2.76,;-1.91,1.22,;-.58,.45,;-3.37,.75,;-3.77,-.74,;-3,-2.08,;-4.34,-2.85,;-5.11,-1.51,;-4.74,-4.33,;-3.65,-5.42,;-4.05,-6.91,;-5.53,-7.31,;-6.62,-6.22,;-8.11,-6.62,;-6.22,-4.73,;-4.28,1.99,;-5.82,1.99,;-3.37,3.24,;-2.29,4.33,;-2.68,5.81,;-4.17,6.21,;-5.26,5.12,;-4.86,3.64,;-4.57,7.7,;-6.06,8.1,;-3.48,8.79,;.76,-3.4,;-.58,-4.17,;-.58,-5.71,;-1.91,-6.48,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C4CC4)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCC4(CC4(F)F)C2)C(=O)C32CCN(CC2)C(C)=O)ccc1C |r,wU:27.30,29.35,(2.76,-9.56,;2.76,-8.02,;1.42,-7.25,;.09,-8.02,;1.42,-5.71,;2.76,-4.94,;2.76,-3.4,;4.09,-2.63,;4.09,-1.09,;2.76,-.32,;2.76,1.22,;4.09,1.99,;5.43,1.22,;6.89,1.7,;7.8,.45,;6.89,-.79,;7.29,-2.28,;6.89,-3.77,;8.38,-3.37,;5.43,-.32,;1.42,1.99,;1.42,3.53,;.09,4.3,;-1.24,3.53,;-1.24,1.99,;.09,1.22,;-2.71,1.52,;-3.11,.03,;-2.34,-1.31,;-3.67,-2.08,;-4.44,-.74,;-4.07,-3.56,;-2.98,-4.65,;-3.38,-6.14,;-4.87,-6.54,;-5.95,-5.45,;-7.44,-5.05,;-7.04,-6.54,;-8.38,-7.31,;-6.27,-7.87,;-5.56,-3.96,;-3.61,2.76,;-5.15,2.76,;-2.71,4.01,;-1.62,5.1,;-2.02,6.58,;-3.51,6.98,;-4.59,5.89,;-4.2,4.41,;-3.9,8.47,;-5.39,8.87,;-2.81,9.56,;1.42,-2.63,;.09,-3.4,;.09,-4.94,;-1.24,-5.71,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@@H]2C[C@@H](C2)N2CCC4(CC4(F)F)C2)C(=O)C32CCN(CC2)C(C)=O)ccc1C |r,wU:27.29,29.34,(1.91,-9.56,;1.91,-8.02,;.57,-7.25,;-.76,-8.02,;.57,-5.71,;1.91,-4.94,;1.91,-3.4,;3.24,-2.63,;3.24,-1.09,;1.91,-.32,;1.91,1.22,;3.24,1.99,;4.57,1.22,;6.04,1.7,;6.94,.45,;6.04,-.79,;6.44,-2.28,;5.35,-3.37,;7.92,-2.68,;4.57,-.32,;.57,1.99,;.57,3.53,;-.76,4.3,;-2.09,3.53,;-2.09,1.99,;-.76,1.22,;-3.56,1.52,;-3.96,.03,;-5.29,-.74,;-4.52,-2.08,;-3.19,-1.31,;-4.92,-3.56,;-4.01,-4.81,;-4.92,-6.06,;-6.38,-5.58,;-7.92,-5.58,;-7.15,-6.91,;-7.92,-8.25,;-6.38,-8.25,;-6.38,-4.04,;-4.46,2.76,;-6,2.76,;-3.56,4.01,;-2.47,5.1,;-2.87,6.58,;-4.36,6.98,;-5.45,5.89,;-5.05,4.41,;-4.75,8.47,;-6.24,8.87,;-3.67,9.56,;.57,-2.63,;-.76,-3.4,;-.76,-4.94,;-2.09,-5.71,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@@H]2C[C@@H](C2)N2CCC(C)(C)C2)C(=O)C32CCN(CC2)C(C)=O)ccc1C |r,wU:27.29,29.34,(3.21,-8.02,;1.88,-8.79,;.55,-8.02,;-.79,-8.79,;.55,-6.48,;1.88,-5.71,;1.88,-4.17,;3.21,-3.4,;3.21,-1.86,;1.88,-1.09,;1.88,.45,;3.21,1.22,;4.55,.45,;6.01,.93,;6.92,-.32,;6.01,-1.56,;6.41,-3.05,;5.32,-4.14,;7.9,-3.45,;4.55,-1.09,;.55,1.22,;.55,2.76,;-.79,3.53,;-2.12,2.76,;-2.12,1.22,;-.79,.45,;-3.59,.75,;-3.98,-.74,;-5.32,-1.51,;-4.55,-2.85,;-3.21,-2.08,;-4.95,-4.33,;-4.04,-5.58,;-4.95,-6.83,;-6.41,-6.35,;-7.9,-6.75,;-6.41,-7.89,;-6.41,-4.81,;-4.49,1.99,;-6.03,1.99,;-3.59,3.24,;-2.5,4.33,;-2.9,5.81,;-4.38,6.21,;-5.47,5.12,;-5.07,3.64,;-4.78,7.7,;-6.27,8.1,;-3.69,8.79,;.55,-3.4,;-.79,-4.17,;-.79,-5.71,;-2.12,-6.48,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C4CC4)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCC4(CC4)C2)C(=O)C32CCN(CC2)C(C)=O)ccc1C |r,wU:27.30,29.35,(2.29,-9.56,;2.29,-8.02,;.96,-7.25,;-.38,-8.02,;.96,-5.71,;2.29,-4.94,;2.29,-3.4,;3.62,-2.63,;3.62,-1.09,;2.29,-.32,;2.29,1.22,;3.62,1.99,;4.96,1.22,;6.42,1.7,;7.33,.45,;6.42,-.79,;6.82,-2.28,;6.42,-3.77,;7.91,-3.37,;4.96,-.32,;.96,1.99,;.96,3.53,;-.38,4.3,;-1.71,3.53,;-1.71,1.99,;-.38,1.22,;-3.18,1.52,;-3.57,.03,;-2.8,-1.31,;-4.14,-2.08,;-4.91,-.74,;-4.54,-3.56,;-3.45,-4.65,;-3.85,-6.14,;-5.33,-6.54,;-6.42,-5.45,;-7.91,-5.05,;-7.51,-6.54,;-6.02,-3.96,;-4.08,2.76,;-5.62,2.76,;-3.18,4.01,;-2.09,5.1,;-2.48,6.58,;-3.97,6.98,;-5.06,5.89,;-4.66,4.41,;-4.37,8.47,;-5.86,8.87,;-3.28,9.56,;.96,-2.63,;-.38,-3.4,;-.38,-4.94,;-1.71,-5.71,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C4CC4)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C32CCN(CC2)S(=O)(=O)C2CC2)ccc1C |r,wU:27.30,29.35,(2.01,-9.76,;2.01,-8.22,;.67,-7.45,;-.66,-8.22,;.67,-5.91,;2.01,-5.14,;2.01,-3.6,;3.34,-2.83,;3.34,-1.29,;2.01,-.52,;2.01,1.02,;3.34,1.79,;4.68,1.02,;6.14,1.5,;7.05,.25,;6.14,-.99,;6.54,-2.48,;6.14,-3.97,;7.63,-3.57,;4.68,-.52,;.67,1.79,;.67,3.33,;-.66,4.1,;-1.99,3.33,;-1.99,1.79,;-.66,1.02,;-3.46,1.32,;-3.86,-.17,;-3.09,-1.51,;-4.42,-2.28,;-5.19,-.94,;-4.82,-3.76,;-6.31,-4.16,;-6.7,-5.65,;-5.62,-6.74,;-4.13,-6.34,;-3.73,-4.85,;-4.36,2.56,;-5.9,2.56,;-3.46,3.81,;-2.37,4.9,;-2.77,6.38,;-4.25,6.78,;-5.34,5.69,;-4.94,4.21,;-4.65,8.27,;-5.05,9.76,;-3.17,8.67,;-6.14,7.87,;-7.63,8.27,;-7.23,6.78,;.67,-2.83,;-.66,-3.6,;-.66,-5.14,;-1.99,-5.91,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C4CC4)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C32CCN(CC2)S(C)(=O)=O)ccc1C |r,wU:27.30,29.35,(1.55,-9.76,;1.55,-8.22,;.21,-7.45,;-1.12,-8.22,;.21,-5.91,;1.55,-5.14,;1.55,-3.6,;2.88,-2.83,;2.88,-1.29,;1.55,-.52,;1.55,1.02,;2.88,1.79,;4.21,1.02,;5.68,1.5,;6.58,.25,;5.68,-.99,;6.08,-2.48,;5.68,-3.97,;7.17,-3.57,;4.21,-.52,;.21,1.79,;.21,3.33,;-1.12,4.1,;-2.45,3.33,;-2.45,1.79,;-1.12,1.02,;-3.92,1.32,;-4.32,-.17,;-3.55,-1.51,;-4.88,-2.28,;-5.65,-.94,;-5.28,-3.76,;-6.77,-4.16,;-7.17,-5.65,;-6.08,-6.74,;-4.59,-6.34,;-4.19,-4.85,;-4.82,2.56,;-6.36,2.56,;-3.92,3.81,;-2.83,4.9,;-3.23,6.38,;-4.72,6.78,;-5.81,5.69,;-5.41,4.21,;-5.11,8.27,;-6.6,7.87,;-5.51,9.76,;-3.63,8.67,;.21,-2.83,;-1.12,-3.6,;-1.12,-5.14,;-2.45,-5.91,)|
CC[C@H](C)n1cnc2cc(nc(Nc3ccc(C)c(c3)C(=O)NC)c12)-c1ccc2c(c1)N([C@H]1C[C@H](C1)N1CCCCC1)C(=O)C21CCN(CC1)C(=O)OC |r,wU:32.35,34.40,wD:2.2,(7.91,-1.99,;6.82,-3.08,;5.33,-2.68,;4.24,-3.77,;4.93,-1.19,;5.84,.05,;4.93,1.3,;3.47,.82,;2.14,1.59,;.8,.82,;.8,-.72,;2.14,-1.49,;2.14,-3.03,;.8,-3.8,;-.53,-3.03,;-1.86,-3.8,;-1.86,-5.34,;-3.2,-6.11,;-.53,-6.11,;.8,-5.34,;-.53,-7.65,;.8,-8.42,;-1.86,-8.42,;-1.86,-9.96,;3.47,-.72,;-.53,1.59,;-.53,3.13,;-1.86,3.9,;-3.2,3.13,;-3.2,1.59,;-1.86,.82,;-4.66,1.12,;-5.06,-.37,;-4.29,-1.7,;-5.63,-2.47,;-6.4,-1.14,;-6.02,-3.96,;-7.51,-4.36,;-7.91,-5.85,;-6.82,-6.94,;-5.33,-6.54,;-4.93,-5.05,;-5.57,2.36,;-7.11,2.36,;-4.66,3.61,;-3.57,4.7,;-3.97,6.19,;-5.46,6.58,;-6.55,5.49,;-6.15,4.01,;-5.86,8.07,;-4.77,9.16,;-7.35,8.47,;-7.74,9.96,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N(C2CC(C2)N2CCC[C@@H](F)C2)C(=O)C32CCN(CC2)C2COC2)c(F)cc1C |wD:35.39,(11.66,-5.66,;11.13,-4.22,;9.61,-3.96,;8.63,-5.14,;9.07,-2.51,;10.06,-1.33,;9.52,.12,;10.5,1.3,;9.97,2.75,;8.45,3,;7.91,4.45,;8.89,5.63,;10.41,5.38,;11.62,6.33,;12.9,5.48,;12.49,4,;13.44,2.79,;14.97,3.01,;12.87,1.36,;10.95,3.93,;6.39,4.7,;5.41,3.52,;3.89,3.77,;3.36,5.22,;4.34,6.4,;5.86,6.15,;3.51,7.7,;4.08,9.14,;3.47,10.55,;4.88,11.16,;5.49,9.75,;5.45,12.59,;6.97,12.82,;7.54,14.25,;6.58,15.46,;5.06,15.23,;4.11,16.44,;4.49,13.8,;2.02,7.32,;.83,8.3,;1.92,5.79,;1.99,4.25,;.69,3.42,;-.68,4.14,;-.74,5.67,;.56,6.5,;-1.98,3.31,;-2.31,1.81,;-3.82,2.14,;-3.48,3.65,;8,.37,;7.46,1.82,;7.02,-.81,;7.56,-2.26,;6.57,-3.44,)|
CCNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCC[C@@H](F)C2)C(=O)C32CCN(CC2)C2COC2)c(F)cc1C |r,wU:28.30,30.35,36.40,(3.42,-10.45,;2.09,-9.68,;2.09,-8.14,;.76,-7.37,;-.58,-8.14,;.76,-5.83,;2.09,-5.06,;2.09,-3.52,;3.42,-2.75,;3.42,-1.21,;2.09,-.44,;2.09,1.1,;3.42,1.87,;4.76,1.1,;6.22,1.57,;7.13,.33,;6.22,-.92,;6.62,-2.4,;5.53,-3.49,;8.11,-2.8,;4.76,-.44,;.76,1.87,;.76,3.41,;-.58,4.18,;-1.91,3.41,;-1.91,1.87,;-.58,1.1,;-3.37,1.39,;-3.77,-.09,;-3,-1.43,;-4.34,-2.2,;-5.11,-.86,;-4.74,-3.69,;-3.65,-4.77,;-4.05,-6.26,;-5.53,-6.66,;-6.62,-5.57,;-8.11,-5.97,;-6.22,-4.08,;-4.28,2.64,;-5.82,2.64,;-3.37,3.88,;-2.29,4.97,;-2.68,6.46,;-4.17,6.86,;-5.26,5.77,;-4.86,4.28,;-4.57,8.35,;-3.8,9.68,;-5.13,10.45,;-5.9,9.12,;.76,-2.75,;.76,-1.21,;-.58,-3.52,;-.58,-5.06,;-1.91,-5.83,)|
CC(C)NC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCC[C@@H](F)C2)C(=O)C32CCN(CC2)C2COC2)c(F)cc1C |r,wU:29.31,31.36,37.41,(3.42,-10.45,;2.09,-9.68,;.76,-10.45,;2.09,-8.14,;.76,-7.37,;-.58,-8.14,;.76,-5.83,;2.09,-5.06,;2.09,-3.52,;3.42,-2.75,;3.42,-1.21,;2.09,-.44,;2.09,1.1,;3.42,1.87,;4.76,1.1,;6.22,1.57,;7.13,.33,;6.22,-.92,;6.62,-2.4,;5.53,-3.49,;8.11,-2.8,;4.76,-.44,;.76,1.87,;.76,3.41,;-.58,4.18,;-1.91,3.41,;-1.91,1.87,;-.58,1.1,;-3.37,1.39,;-3.77,-.09,;-3,-1.43,;-4.34,-2.2,;-5.11,-.86,;-4.74,-3.69,;-3.65,-4.77,;-4.05,-6.26,;-5.53,-6.66,;-6.62,-5.57,;-8.11,-5.97,;-6.22,-4.08,;-4.28,2.64,;-5.82,2.64,;-3.37,3.88,;-2.29,4.97,;-2.68,6.46,;-4.17,6.86,;-5.26,5.77,;-4.86,4.28,;-4.57,8.35,;-3.8,9.68,;-5.13,10.45,;-5.9,9.12,;.76,-2.75,;.76,-1.21,;-.58,-3.52,;-.58,-5.06,;-1.91,-5.83,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C4CC4)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C32CCN(CC2)C2COC2)ccc1C |r,wU:27.30,29.35,(2.88,-8.53,;1.55,-9.3,;.21,-8.53,;-1.12,-9.3,;.21,-6.99,;1.55,-6.22,;1.55,-4.68,;2.88,-3.91,;2.88,-2.37,;1.55,-1.6,;1.55,-.06,;2.88,.71,;4.21,-.06,;5.68,.42,;6.58,-.83,;5.68,-2.07,;6.08,-3.56,;5.68,-5.05,;7.17,-4.65,;4.21,-1.6,;.21,.71,;.21,2.25,;-1.12,3.02,;-2.45,2.25,;-2.45,.71,;-1.12,-.06,;-3.92,.24,;-4.32,-1.25,;-3.55,-2.58,;-4.88,-3.35,;-5.65,-2.02,;-5.28,-4.84,;-6.77,-5.24,;-7.17,-6.73,;-6.08,-7.82,;-4.59,-7.42,;-4.19,-5.93,;-4.82,1.48,;-6.36,1.48,;-3.92,2.73,;-2.83,3.82,;-3.23,5.31,;-4.72,5.7,;-5.81,4.62,;-5.41,3.13,;-5.11,7.19,;-4.34,8.53,;-5.68,9.3,;-6.45,7.96,;.21,-3.91,;-1.12,-4.68,;-1.12,-6.22,;-2.45,-6.99,)|
CC(C)n1cnc2cc(nc(Nc3ccc(C)c(c3)C(=O)NC3(CF)CC3)c12)-c1ccc2c(c1)N(C1CC(C1)N1CCCCC1)C(=O)C2(C)C |(-2.25,5.87,;-.74,5.55,;.29,6.7,;-.27,4.09,;-1.17,2.84,;-.27,1.6,;1.2,2.07,;2.53,1.3,;3.86,2.07,;3.86,3.61,;2.53,4.38,;2.53,5.92,;3.86,6.69,;5.2,5.92,;6.53,6.69,;6.53,8.23,;7.87,9,;5.2,9,;3.86,8.23,;5.2,10.54,;6.53,11.31,;3.86,11.31,;3.86,12.85,;2.35,13.12,;1.36,11.94,;4.39,14.3,;5.38,13.12,;1.2,3.61,;5.2,1.3,;5.2,-.24,;6.53,-1.01,;7.87,-.24,;7.87,1.3,;6.53,2.07,;9.33,1.78,;9.81,3.24,;9.11,4.62,;10.48,5.31,;11.18,3.94,;10.95,6.78,;9.92,7.92,;10.4,9.39,;11.91,9.71,;12.94,8.56,;12.46,7.1,;10.23,.53,;11.77,.53,;9.33,-.71,;10.66,-1.48,;8.7,-2.12,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C3(C)C)c(F)cc1C |r,wU:27.29,29.34,(2.68,-5.99,;1.35,-6.76,;.01,-5.99,;-1.32,-6.76,;.01,-4.45,;1.35,-3.68,;1.35,-2.14,;2.68,-1.37,;2.68,.17,;1.35,.94,;1.35,2.48,;2.68,3.25,;4.01,2.48,;5.48,2.96,;6.38,1.71,;5.48,.47,;5.88,-1.02,;4.79,-2.11,;7.37,-1.42,;4.01,.94,;.01,3.25,;.01,4.79,;-1.32,5.56,;-2.65,4.79,;-2.65,3.25,;-1.32,2.48,;-4.12,2.78,;-4.52,1.29,;-3.75,-.04,;-5.08,-.81,;-5.85,.52,;-5.48,-2.3,;-6.97,-2.7,;-7.37,-4.19,;-6.28,-5.28,;-4.79,-4.88,;-4.39,-3.39,;-5.02,4.02,;-6.56,4.02,;-4.12,5.27,;-3.03,6.36,;-4.52,6.76,;.01,-1.37,;.01,.17,;-1.32,-2.14,;-1.32,-3.68,;-2.65,-4.45,)|
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CCNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N([C@H]2C[C@H](C2)N2CCCCC2)C(=O)C32CN(C2)C(C)=O)c(F)cc1C |r,wU:28.30,30.35,(4.01,-8.35,;2.68,-7.58,;1.35,-8.35,;.01,-7.58,;-1.32,-8.35,;.01,-6.04,;1.35,-5.27,;1.35,-3.73,;2.68,-2.96,;2.68,-1.42,;1.35,-.65,;1.35,.89,;2.68,1.66,;4.01,.89,;5.48,1.36,;6.38,.12,;5.48,-1.13,;5.88,-2.62,;4.79,-3.71,;7.37,-3.02,;4.01,-.65,;.01,1.66,;.01,3.2,;-1.32,3.97,;-2.65,3.2,;-2.65,1.66,;-1.32,.89,;-4.12,1.18,;-4.52,-.31,;-3.75,-1.64,;-5.08,-2.41,;-5.85,-1.08,;-5.48,-3.9,;-6.97,-4.3,;-7.37,-5.78,;-6.28,-6.87,;-4.79,-6.47,;-4.39,-4.99,;-5.02,2.43,;-6.56,2.43,;-4.12,3.67,;-3.35,5.01,;-4.68,5.78,;-5.45,4.44,;-5.08,7.26,;-3.99,8.35,;-6.57,7.66,;.01,-2.96,;.01,-1.42,;-1.32,-3.73,;-1.32,-5.27,;-2.65,-6.04,)|
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CC(C)n1cnc2cc(nc(Nc3cc(C(=O)NC4(CC4)C(F)F)c(C)c(F)c3F)c12)-c1cnc2c(c1)N([C@H]1C[C@](C)(C1)N1CC3CCC1CO3)C(=O)C2(C)C |r,wU:38.42,wD:40.45,(5.01,-1.32,;6.1,-.23,;7.58,-.63,;5.62,1.24,;6.53,2.48,;5.62,3.73,;4.16,3.25,;2.82,4.02,;1.49,3.25,;1.49,1.71,;2.82,.94,;2.82,-.6,;1.49,-1.37,;1.49,-2.91,;.15,-3.68,;.15,-5.22,;-1.18,-5.99,;1.49,-5.99,;2.82,-5.22,;3.59,-3.88,;2.05,-3.88,;4.16,-5.99,;5.49,-5.22,;4.16,-7.53,;-1.18,-2.91,;-2.51,-3.68,;-1.18,-1.37,;-2.51,-.6,;.15,-.6,;.15,.94,;4.16,1.71,;.15,4.02,;.15,5.56,;-1.18,6.33,;-2.51,5.56,;-2.51,4.02,;-1.18,3.25,;-3.98,3.55,;-4.45,2.08,;-3.75,.71,;-5.13,.01,;-4.04,-1.08,;-5.83,1.38,;-5.6,-1.45,;-4.57,-2.6,;-5.05,-4.06,;-5.34,-3,;-6.84,-2.8,;-7.11,-1.77,;-7.58,-3.24,;-6.55,-4.38,;-4.88,4.79,;-6.42,4.79,;-3.98,6.04,;-4.38,7.53,;-2.89,7.13,)|
CC(C)n1cnc2cc(nc(Nc3cc(C(=O)NC4(CC4)C(F)F)c(Cl)c(F)c3F)c12)-c1cnc2c(c1)N(C1CC(C)(C1)N1CCC3CC3C1)C(=O)C2(C)C |(-2.25,5.87,;-.74,5.55,;.29,6.7,;-.27,4.09,;-1.17,2.84,;-.27,1.6,;1.2,2.07,;2.53,1.3,;3.86,2.07,;3.86,3.61,;2.53,4.38,;2.53,5.92,;3.86,6.69,;5.2,5.92,;6.53,6.69,;7.87,5.92,;7.87,4.38,;9.2,6.69,;10.53,5.92,;11.52,4.74,;10.01,4.48,;11.52,7.1,;11,8.55,;13.04,6.84,;6.53,8.23,;7.87,9,;5.2,9,;5.2,10.54,;3.86,8.23,;2.53,9,;1.2,3.61,;5.2,1.3,;6.53,2.07,;7.87,1.3,;7.87,-.24,;6.53,-1.01,;5.2,-.24,;6.85,-2.51,;5.82,-3.66,;4.28,-3.74,;4.36,-5.28,;2.83,-5.36,;5.9,-5.2,;4.44,-6.81,;5.82,-7.51,;5.9,-9.05,;4.61,-9.89,;3.31,-10.73,;3.23,-9.19,;3.15,-7.65,;8.38,-2.67,;9.15,-4.01,;9.01,-1.27,;10.48,-1.73,;10.16,-.25,)|
CC(C)n1cnc2cc(nc(Nc3cc(C(=O)NC4(CC4)C(F)F)c(Cl)c(F)c3F)c12)-c1cnc2c(c1)N(C1CC(C)(C1)N1CCCCCC1)C(=O)C2(C)C |(-2.25,5.87,;-.74,5.55,;.29,6.7,;-.27,4.09,;-1.17,2.84,;-.27,1.6,;1.2,2.07,;2.53,1.3,;3.86,2.07,;3.86,3.61,;2.53,4.38,;2.53,5.92,;3.86,6.69,;5.2,5.92,;6.53,6.69,;7.87,5.92,;7.87,4.38,;9.2,6.69,;10.53,5.92,;11.52,4.74,;10.01,4.48,;11.52,7.1,;11,8.55,;13.04,6.84,;6.53,8.23,;7.87,9,;5.2,9,;5.2,10.54,;3.86,8.23,;2.53,9,;1.2,3.61,;5.2,1.3,;6.53,2.07,;7.87,1.3,;7.87,-.24,;6.53,-1.01,;5.2,-.24,;6.85,-2.51,;5.82,-3.66,;4.28,-3.74,;4.36,-5.28,;2.83,-5.36,;5.9,-5.2,;4.44,-6.81,;5.87,-7.41,;6.29,-8.89,;5.39,-10.14,;3.85,-10.22,;2.83,-9.07,;3.09,-7.55,;8.38,-2.67,;9.15,-4.01,;9.01,-1.27,;10.48,-1.73,;10.16,-.25,)|
CC(C)n1cnc2cc(nc(Nc3cc(C(=O)NC4(CF)CC4)c(Cl)c(F)c3F)c12)-c1cnc2c(c1)N(C1CC(C)(C1)N1CCC3CC3C1)C(=O)C2(C)C |(-2.25,5.87,;-.74,5.55,;.29,6.7,;-.27,4.09,;-1.17,2.84,;-.27,1.6,;1.2,2.07,;2.53,1.3,;3.86,2.07,;3.86,3.61,;2.53,4.38,;2.53,5.92,;3.86,6.69,;5.2,5.92,;6.53,6.69,;7.87,5.92,;7.87,4.38,;9.2,6.69,;10.53,5.92,;11.52,7.1,;11,8.55,;11.52,4.74,;10.01,4.48,;6.53,8.23,;7.87,9,;5.2,9,;5.2,10.54,;3.86,8.23,;2.53,9,;1.2,3.61,;5.2,1.3,;6.53,2.07,;7.87,1.3,;7.87,-.24,;6.53,-1.01,;5.2,-.24,;6.85,-2.51,;5.82,-3.66,;4.28,-3.74,;4.36,-5.28,;2.83,-5.36,;5.9,-5.2,;4.44,-6.81,;5.82,-7.51,;5.9,-9.05,;4.61,-9.89,;3.31,-10.73,;3.23,-9.19,;3.15,-7.65,;8.38,-2.67,;9.15,-4.01,;9.01,-1.27,;10.48,-1.73,;10.16,-.25,)|
CC(C)n1cnc2cc(nc(Nc3cc(C(=O)NC4(CC4)C(F)F)c(C)c(F)c3F)c12)-c1cnc2c(c1)N(C1CC(C)(C1)N1CC3CCC(C1)O3)C(=O)C2(C)C |(-2.25,5.87,;-.74,5.55,;.29,6.7,;-.27,4.09,;-1.17,2.84,;-.27,1.6,;1.2,2.07,;2.53,1.3,;3.86,2.07,;3.86,3.61,;2.53,4.38,;2.53,5.92,;3.86,6.69,;5.2,5.92,;6.53,6.69,;7.87,5.92,;7.87,4.38,;9.2,6.69,;10.53,5.92,;11.52,4.74,;10.01,4.48,;11.52,7.1,;11,8.55,;13.04,6.84,;6.53,8.23,;7.87,9,;5.2,9,;5.2,10.54,;3.86,8.23,;2.53,9,;1.2,3.61,;5.2,1.3,;6.53,2.07,;7.87,1.3,;7.87,-.24,;6.53,-1.01,;5.2,-.24,;6.85,-2.51,;5.82,-3.66,;4.28,-3.74,;4.36,-5.28,;2.83,-5.36,;5.9,-5.2,;4.44,-6.81,;3.09,-7.55,;2.83,-9.07,;3.85,-10.22,;5.39,-10.14,;6.29,-8.89,;5.87,-7.41,;4.54,-8.55,;8.38,-2.67,;9.15,-4.01,;9.01,-1.27,;10.48,-1.73,;10.16,-.25,)|
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CC(C)n1cnc2cc(nc(Nc3cc(C(=O)NC4(CC4)C(F)F)c(C)c(F)c3F)c12)-c1cnc2c(c1)N(C1CC(C)(C1)N1CC3CCC(C3)C1)C(=O)C2(C)C |(-2.25,5.87,;-.74,5.55,;.29,6.7,;-.27,4.09,;-1.17,2.84,;-.27,1.6,;1.2,2.07,;2.53,1.3,;3.86,2.07,;3.86,3.61,;2.53,4.38,;2.53,5.92,;3.86,6.69,;5.2,5.92,;6.53,6.69,;7.87,5.92,;7.87,4.38,;9.2,6.69,;10.53,5.92,;11.52,4.74,;10.01,4.48,;11.52,7.1,;11,8.55,;13.04,6.84,;6.53,8.23,;7.87,9,;5.2,9,;5.2,10.54,;3.86,8.23,;2.53,9,;1.2,3.61,;5.2,1.3,;6.53,2.07,;7.87,1.3,;7.87,-.24,;6.53,-1.01,;5.2,-.24,;6.85,-2.51,;5.82,-3.66,;4.28,-3.74,;4.36,-5.28,;2.83,-5.36,;5.9,-5.2,;4.44,-6.81,;3.09,-7.55,;2.83,-9.07,;3.85,-10.22,;5.39,-10.14,;6.29,-8.89,;4.54,-8.55,;5.87,-7.41,;8.38,-2.67,;9.15,-4.01,;9.01,-1.27,;10.48,-1.73,;10.16,-.25,)|
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CC(C)n1cnc2cc(nc(Nc3cc(C(=O)NC4(CC4)C(F)F)c(Cl)c(F)c3F)c12)-c1cnc2c(c1)N(C1CC(C)(C1)N1CC3CC3C1)C(=O)C2(C)C |(-2.25,5.87,;-.74,5.55,;.29,6.7,;-.27,4.09,;-1.17,2.84,;-.27,1.6,;1.2,2.07,;2.53,1.3,;3.86,2.07,;3.86,3.61,;2.53,4.38,;2.53,5.92,;3.86,6.69,;5.2,5.92,;6.53,6.69,;7.87,5.92,;7.87,4.38,;9.2,6.69,;10.53,5.92,;11.52,4.74,;10.01,4.48,;11.52,7.1,;11,8.55,;13.04,6.84,;6.53,8.23,;7.87,9,;5.2,9,;5.2,10.54,;3.86,8.23,;2.53,9,;1.2,3.61,;5.2,1.3,;6.53,2.07,;7.87,1.3,;7.87,-.24,;6.53,-1.01,;5.2,-.24,;6.85,-2.51,;5.82,-3.66,;4.28,-3.74,;4.36,-5.28,;2.83,-5.36,;5.9,-5.2,;4.44,-6.81,;3.25,-7.78,;3.8,-9.22,;4.64,-10.51,;5.34,-9.14,;5.74,-7.65,;8.38,-2.67,;9.15,-4.01,;9.01,-1.27,;10.48,-1.73,;10.16,-.25,)|
CC(C)n1cnc2cc(nc(Nc3cc(C(=O)NC4(CC4)C(F)F)c(C)cc3F)c12)-c1ccc2c(c1)N(C1CC(C)(C1)N1CCCCC1)C(=O)C2(C)C |(13.94,7.78,;12.91,6.63,;13.39,5.17,;11.4,6.95,;10.78,8.36,;9.25,8.2,;8.93,6.69,;7.59,5.92,;7.59,4.38,;8.93,3.61,;10.26,4.38,;11.59,3.61,;11.59,2.07,;10.26,1.3,;10.26,-.24,;8.93,-1.01,;7.59,-.24,;8.93,-2.55,;7.59,-3.32,;6.6,-2.14,;6.07,-3.58,;8.12,-4.76,;7.13,-5.94,;9.63,-5.03,;11.59,-1.01,;11.59,-2.55,;12.93,-.24,;12.93,1.3,;14.26,2.07,;10.26,5.92,;6.26,3.61,;6.26,2.07,;4.92,1.3,;3.59,2.07,;3.59,3.61,;4.92,4.38,;2.13,4.09,;1.65,5.55,;.28,6.25,;.98,7.62,;1.34,9.12,;2.35,6.93,;-.19,8.62,;-1.65,8.11,;-2.82,9.11,;-2.54,10.63,;-1.08,11.14,;.09,10.14,;1.22,2.84,;-.32,2.84,;2.13,1.6,;2.43,.09,;.99,.55,)|
CC(C)n1cnc2cc(nc(Nc3cc(C(=O)NC4(CC4)C(F)F)c(C)c(F)c3F)c12)-c1ccc2c(c1)N(C1CC(C)(C1)N1CCCCC1)C(=O)C2(C)C |(13.94,7.78,;12.91,6.63,;13.39,5.17,;11.4,6.95,;10.78,8.36,;9.25,8.2,;8.93,6.69,;7.59,5.92,;7.59,4.38,;8.93,3.61,;10.26,4.38,;11.59,3.61,;11.59,2.07,;10.26,1.3,;10.26,-.24,;8.93,-1.01,;7.59,-.24,;8.93,-2.55,;7.59,-3.32,;6.6,-2.14,;6.07,-3.58,;8.12,-4.76,;7.13,-5.94,;9.63,-5.03,;11.59,-1.01,;11.59,-2.55,;12.93,-.24,;14.26,-1.01,;12.93,1.3,;14.26,2.07,;10.26,5.92,;6.26,3.61,;6.26,2.07,;4.92,1.3,;3.59,2.07,;3.59,3.61,;4.92,4.38,;2.13,4.09,;1.65,5.55,;.28,6.25,;.98,7.62,;1.34,9.12,;2.35,6.93,;-.19,8.62,;-1.65,8.11,;-2.82,9.11,;-2.54,10.63,;-1.08,11.14,;.09,10.14,;1.22,2.84,;-.32,2.84,;2.13,1.6,;2.43,.09,;.99,.55,)|
CC(C)n1cnc2cc(nc(Nc3cc(C(=O)NC4(CC4)C(F)F)c(C)c(F)c3F)c12)-c1ccc2c(c1)N(CC2(C)C)C1CC(C)(C1)N1CCCCC1 |(13.94,7.78,;12.91,6.63,;13.39,5.17,;11.4,6.95,;10.78,8.36,;9.25,8.2,;8.93,6.69,;7.59,5.92,;7.59,4.38,;8.93,3.61,;10.26,4.38,;11.59,3.61,;11.59,2.07,;10.26,1.3,;10.26,-.24,;8.93,-1.01,;7.59,-.24,;8.93,-2.55,;7.59,-3.32,;6.6,-2.14,;6.07,-3.58,;8.12,-4.76,;7.13,-5.94,;9.63,-5.03,;11.59,-1.01,;11.59,-2.55,;12.93,-.24,;14.26,-1.01,;12.93,1.3,;14.26,2.07,;10.26,5.92,;6.26,3.61,;6.26,2.07,;4.92,1.3,;3.59,2.07,;3.59,3.61,;4.92,4.38,;2.13,4.09,;1.22,2.84,;2.13,1.6,;2.43,.09,;.99,.55,;1.65,5.55,;.28,6.25,;.98,7.62,;1.34,9.12,;2.35,6.93,;-.19,8.62,;-1.65,8.11,;-2.82,9.11,;-2.54,10.63,;-1.08,11.14,;.09,10.14,)|
CC(C)n1cnc2cc(nc(Nc3cc(ccc3F)C(=O)NC3(CC3)C(F)F)c12)-c1ccc2c(c1)N(C1CC(C)(C1)N1CCCCC1)C(=O)C2(C)C |(13.94,7.78,;12.91,6.63,;13.39,5.17,;11.4,6.95,;10.78,8.36,;9.25,8.2,;8.93,6.69,;7.59,5.92,;7.59,4.38,;8.93,3.61,;10.26,4.38,;11.59,3.61,;11.59,2.07,;12.93,1.3,;12.93,-.24,;11.59,-1.01,;10.26,-.24,;10.26,1.3,;8.93,2.07,;14.26,-1.01,;14.26,-2.55,;15.59,-.24,;16.93,-1.01,;16.4,-2.45,;17.92,-2.19,;17.92,.17,;17.39,1.62,;19.43,-.09,;10.26,5.92,;6.26,3.61,;6.26,2.07,;4.92,1.3,;3.59,2.07,;3.59,3.61,;4.92,4.38,;2.13,4.09,;1.65,5.55,;.28,6.25,;.98,7.62,;1.34,9.12,;2.35,6.93,;-.19,8.62,;-1.65,8.11,;-2.82,9.11,;-2.54,10.63,;-1.08,11.14,;.09,10.14,;1.22,2.84,;-.32,2.84,;2.13,1.6,;2.43,.09,;.99,.55,)|
CCNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N(C2CC(C)(C2)N2CCCCC2)C(=O)C3(C)C)c(F)c(F)c1C |(5.2,4.38,;6.53,3.61,;7.87,4.38,;7.87,5.92,;9.2,6.69,;6.53,6.69,;5.2,5.92,;3.86,6.69,;2.53,5.92,;2.53,4.38,;3.86,3.61,;3.86,2.07,;2.53,1.3,;1.2,2.07,;-.27,1.6,;-1.17,2.84,;-.27,4.09,;-.74,5.55,;-2.25,5.87,;.29,6.7,;1.2,3.61,;5.2,1.3,;5.2,-.24,;6.53,-1.01,;7.87,-.24,;7.87,1.3,;6.53,2.07,;9.33,1.78,;9.81,3.24,;9.11,4.62,;10.48,5.31,;10.12,6.81,;11.18,3.94,;11.65,6.31,;11.37,7.83,;12.54,8.83,;13.99,8.32,;14.27,6.8,;13.1,5.8,;10.23,.53,;11.77,.53,;9.33,-.71,;8.7,-2.12,;10.66,-1.48,;3.86,8.23,;2.53,9,;5.2,9,;5.2,10.54,;6.53,8.23,;7.87,9,)|
CCNC(=O)c1ccc(F)c(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N(C2CC(C)(C2)N2CCCCC2)C(=O)C3(C)C)c1 |(7.87,13.62,;6.53,12.85,;6.53,11.31,;5.2,10.54,;3.86,11.31,;5.2,9,;6.53,8.23,;6.53,6.69,;5.2,5.92,;5.2,4.38,;3.86,6.69,;2.53,5.92,;2.53,4.38,;3.86,3.61,;3.86,2.07,;2.53,1.3,;1.2,2.07,;-.27,1.6,;-1.17,2.84,;-.27,4.09,;-.74,5.55,;-2.25,5.87,;.29,6.7,;1.2,3.61,;5.2,1.3,;5.2,-.24,;6.53,-1.01,;7.87,-.24,;7.87,1.3,;6.53,2.07,;9.33,1.78,;9.81,3.24,;9.11,4.62,;10.48,5.31,;11.65,6.31,;11.18,3.94,;10.12,6.81,;8.64,7.25,;8.28,8.75,;9.4,9.81,;10.88,9.37,;11.24,7.87,;10.23,.53,;11.77,.53,;9.33,-.71,;8.7,-2.12,;10.66,-1.48,;3.86,8.23,)|
CC(C)n1cnc2cc(nc(Nc3cc(C(=O)NC4(CC4)C(F)F)c(Cl)c(F)c3F)c12)-c1ccc2c(c1)N(C1CC(C)(C1)N1CCCCC1)C(=O)C2(C)C |(13.94,7.78,;12.91,6.63,;13.39,5.17,;11.4,6.95,;10.78,8.36,;9.25,8.2,;8.93,6.69,;7.59,5.92,;7.59,4.38,;8.93,3.61,;10.26,4.38,;11.59,3.61,;11.59,2.07,;12.93,1.3,;12.93,-.24,;14.26,-1.01,;14.26,-2.55,;15.59,-.24,;16.93,-1.01,;17.92,-2.19,;16.4,-2.45,;17.92,.17,;17.39,1.62,;19.43,-.09,;11.59,-1.01,;11.59,-2.55,;10.26,-.24,;8.93,-1.01,;10.26,1.3,;8.93,2.07,;10.26,5.92,;6.26,3.61,;6.26,2.07,;4.92,1.3,;3.59,2.07,;3.59,3.61,;4.92,4.38,;2.13,4.09,;1.65,5.55,;.28,6.25,;.98,7.62,;1.34,9.12,;2.35,6.93,;-.19,8.62,;-1.65,8.11,;-2.82,9.11,;-2.54,10.63,;-1.08,11.14,;.09,10.14,;1.22,2.84,;-.32,2.84,;2.13,1.6,;2.43,.09,;.99,.55,)|
CC(C)n1cnc2cc(nc(Nc3cc(cc(F)c3F)C(=O)NC3(CC3)C(F)F)c12)-c1cnc2c(c1)N(C(=O)C2(C)C)C1(C)CC(C1)N1CCCCC1
CC(C)n1cnc2cc(nc(Nc3c(F)c(F)cc(C(N)=O)c3C3(CC3)C(F)F)c12)-c1ccc2c(c1)N(C1CC(C)(C1)N1CCCCC1)C(=O)C2(C)C |(13.94,7.78,;12.91,6.63,;13.39,5.17,;11.4,6.95,;10.78,8.36,;9.25,8.2,;8.93,6.69,;7.59,5.92,;7.59,4.38,;8.93,3.61,;10.26,4.38,;11.59,3.61,;11.59,2.07,;10.26,1.3,;8.93,2.07,;10.26,-.24,;8.93,-1.01,;11.59,-1.01,;12.93,-.24,;14.26,-1.01,;15.77,-.69,;14.26,-2.55,;12.93,1.3,;14.26,2.07,;13.73,3.52,;15.25,3.25,;15.25,.89,;14.72,-.55,;16.77,1.16,;10.26,5.92,;6.26,3.61,;6.26,2.07,;4.92,1.3,;3.59,2.07,;3.59,3.61,;4.92,4.38,;2.13,4.09,;1.65,5.55,;.28,6.25,;.98,7.62,;1.34,9.12,;2.35,6.93,;-.19,8.62,;-1.65,8.11,;-2.82,9.11,;-2.54,10.63,;-1.08,11.14,;.09,10.14,;1.22,2.84,;-.32,2.84,;2.13,1.6,;2.43,.09,;.99,.55,)|
CC(C)n1cnc2cc(nc(Nc3cc(C(=O)NC4(CC4)C(F)F)c(Cl)c(F)c3F)c12)-c1ccc2c(c1)N(C1CC(C1)N1CCCCC1)C(=O)C2(C)C |(13.94,7.78,;12.91,6.63,;13.39,5.17,;11.4,6.95,;10.78,8.36,;9.25,8.2,;8.93,6.69,;7.59,5.92,;7.59,4.38,;8.93,3.61,;10.26,4.38,;11.59,3.61,;11.59,2.07,;12.93,1.3,;12.93,-.24,;14.26,-1.01,;14.26,-2.55,;15.59,-.24,;16.93,-1.01,;17.92,-2.19,;16.4,-2.45,;17.92,.17,;17.39,1.62,;19.43,-.09,;11.59,-1.01,;11.59,-2.55,;10.26,-.24,;8.93,-1.01,;10.26,1.3,;8.93,2.07,;10.26,5.92,;6.26,3.61,;6.26,2.07,;4.92,1.3,;3.59,2.07,;3.59,3.61,;4.92,4.38,;2.13,4.09,;1.65,5.55,;.28,6.25,;.98,7.62,;2.35,6.93,;.5,9.09,;-1.01,9.41,;-1.48,10.87,;-.45,12.02,;1.06,11.7,;1.53,10.23,;1.22,2.84,;-.32,2.84,;2.13,1.6,;2.43,.09,;.99,.55,)|
CC(C)n1cnc2cc(nc(Nc3cc(C(=O)NC4(CC4)C(F)F)c(Cl)c(F)c3F)c12)-c1cnc2c(c1)N(C1CC(C1)N1CCCCC1)C(=O)C2(C)C |(11.31,-2.5,;9.81,-2.18,;8.78,-3.32,;9.33,-.71,;10.23,.53,;9.33,1.78,;7.87,1.3,;6.53,2.07,;5.2,1.3,;5.2,-.24,;6.53,-1.01,;6.53,-2.55,;5.2,-3.32,;5.2,-4.86,;3.86,-5.63,;3.86,-7.17,;2.53,-7.94,;5.2,-7.94,;5.2,-9.48,;4.67,-10.92,;3.68,-9.74,;6.71,-9.74,;7.7,-8.56,;7.24,-11.19,;2.53,-4.86,;1.2,-5.63,;2.53,-3.32,;1.2,-2.55,;3.86,-2.55,;3.86,-1.01,;7.87,-.24,;3.86,2.07,;3.86,3.61,;2.53,4.38,;1.2,3.61,;1.2,2.07,;2.53,1.3,;-.27,1.6,;-.74,.13,;-.04,-1.24,;-1.42,-1.94,;-2.12,-.57,;-1.89,-3.4,;-.86,-4.55,;-1.34,-6.01,;-2.84,-6.33,;-3.87,-5.19,;-3.4,-3.72,;-1.17,2.84,;-2.71,2.84,;-.27,4.09,;.04,5.6,;-1.4,5.13,)|
CC(C)n1cnc2cc(nc(Nc3cc(C(=O)NC4(CC4)C(F)F)c(C)c(F)c3F)c12)-c1cnc2c(c1)N(C1CC(C1)N1CCCCC1)C(=O)C2(C)C |(11.31,-2.5,;9.81,-2.18,;8.78,-3.32,;9.33,-.71,;10.23,.53,;9.33,1.78,;7.87,1.3,;6.53,2.07,;5.2,1.3,;5.2,-.24,;6.53,-1.01,;6.53,-2.55,;5.2,-3.32,;5.2,-4.86,;3.86,-5.63,;3.86,-7.17,;2.53,-7.94,;5.2,-7.94,;6.53,-7.17,;6,-5.72,;7.52,-5.99,;7.52,-8.35,;6.99,-9.79,;9.04,-8.08,;2.53,-4.86,;1.2,-5.63,;2.53,-3.32,;1.2,-2.55,;3.86,-2.55,;3.86,-1.01,;7.87,-.24,;3.86,2.07,;3.86,3.61,;2.53,4.38,;1.2,3.61,;1.2,2.07,;2.53,1.3,;-.27,1.6,;-.74,.13,;-.04,-1.24,;-1.42,-1.94,;-2.12,-.57,;-1.89,-3.4,;-.86,-4.55,;-1.34,-6.01,;-2.84,-6.33,;-3.87,-5.19,;-3.4,-3.72,;-1.17,2.84,;-2.71,2.84,;-.27,4.09,;.04,5.6,;-1.4,5.13,)|
CCNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2cnc3c(c2)N(C2CC(C)(C2)N2CCCCCC2)C(=O)C3(C)C)c(F)c(F)c1Cl |(11.87,6.69,;10.53,5.92,;9.2,6.69,;7.87,5.92,;7.87,4.38,;6.53,6.69,;5.2,5.92,;3.86,6.69,;2.53,5.92,;2.53,4.38,;3.86,3.61,;3.86,2.07,;2.53,1.3,;1.2,2.07,;-.27,1.6,;-1.17,2.84,;-.27,4.09,;-.74,5.55,;-2.25,5.87,;.29,6.7,;1.2,3.61,;5.2,1.3,;6.53,2.07,;7.87,1.3,;7.87,-.24,;6.53,-1.01,;5.2,-.24,;6.85,-2.51,;5.82,-3.66,;4.28,-3.74,;4.36,-5.28,;2.83,-5.36,;5.9,-5.2,;4.44,-6.81,;5.87,-7.41,;6.29,-8.89,;5.39,-10.14,;3.85,-10.22,;2.83,-9.07,;3.09,-7.55,;8.38,-2.67,;9.15,-4.01,;9.01,-1.27,;10.48,-1.73,;10.16,-.25,;3.86,8.23,;2.53,9,;5.2,9,;5.2,10.54,;6.53,8.23,;7.87,9,)|
CC(C)n1cnc2cc(nc(Nc3cc(C(=O)NCC(F)F)c(Cl)c(F)c3F)c12)-c1cnc2c(c1)N(C(=O)C2(C)C)C1(CC(C)C1)N1CCCCCC1 |(-2.25,5.87,;-.74,5.55,;.29,6.7,;-.27,4.09,;-1.17,2.84,;-.27,1.6,;1.2,2.07,;2.53,1.3,;3.86,2.07,;3.86,3.61,;2.53,4.38,;2.53,5.92,;3.86,6.69,;5.2,5.92,;6.53,6.69,;7.87,5.92,;7.87,4.38,;9.2,6.69,;9.2,8.23,;10.53,9,;10.53,10.54,;11.87,8.23,;6.53,8.23,;7.87,9,;5.2,9,;5.2,10.54,;3.86,8.23,;2.53,9,;1.2,3.61,;5.2,1.3,;6.53,2.07,;7.87,1.3,;7.87,-.24,;6.53,-1.01,;5.2,-.24,;6.85,-2.51,;8.38,-2.67,;9.15,-4.01,;9.01,-1.27,;10.48,-1.73,;10.16,-.25,;5.82,-3.66,;6.97,-4.69,;5.94,-5.83,;6.02,-7.37,;4.79,-4.8,;4.68,-2.63,;3.25,-3.21,;1.91,-2.46,;1.65,-.94,;2.68,.2,;4.22,.11,;5.11,-1.15,)|
CC(C)n1cnc2cc(nc(Nc3cc(C(=O)NC4(CF)CC4)c(Cl)c(F)c3F)c12)-c1cnc2c(c1)N(C1CC(C)(C1)N1CCCCCC1)C(=O)C2(C)C |(-2.25,5.87,;-.74,5.55,;.29,6.7,;-.27,4.09,;-1.17,2.84,;-.27,1.6,;1.2,2.07,;2.53,1.3,;3.86,2.07,;3.86,3.61,;2.53,4.38,;2.53,5.92,;3.86,6.69,;5.2,5.92,;6.53,6.69,;7.87,5.92,;7.87,4.38,;9.2,6.69,;10.53,5.92,;11.52,7.1,;11,8.55,;11.52,4.74,;10.01,4.48,;6.53,8.23,;7.87,9,;5.2,9,;5.2,10.54,;3.86,8.23,;2.53,9,;1.2,3.61,;5.2,1.3,;6.53,2.07,;7.87,1.3,;7.87,-.24,;6.53,-1.01,;5.2,-.24,;6.85,-2.51,;5.82,-3.66,;4.28,-3.74,;4.36,-5.28,;2.83,-5.36,;5.9,-5.2,;4.44,-6.81,;5.87,-7.41,;6.29,-8.89,;5.39,-10.14,;3.85,-10.22,;2.83,-9.07,;3.09,-7.55,;8.38,-2.67,;9.15,-4.01,;9.01,-1.27,;10.48,-1.73,;10.16,-.25,)|
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CC(C)n1cnc2cc(nc(Nc3cc(C(=O)NCC(F)F)c(Cl)c(F)c3F)c12)-c1cnc2c(c1)N(C1CC(C)(C1)N1CCC3CC3C1)C(=O)C2(C)C |(-2.25,5.87,;-.74,5.55,;.29,6.7,;-.27,4.09,;-1.17,2.84,;-.27,1.6,;1.2,2.07,;2.53,1.3,;3.86,2.07,;3.86,3.61,;2.53,4.38,;2.53,5.92,;3.86,6.69,;5.2,5.92,;6.53,6.69,;7.87,5.92,;7.87,4.38,;9.2,6.69,;9.2,8.23,;10.53,9,;10.53,10.54,;11.87,8.23,;6.53,8.23,;7.87,9,;5.2,9,;5.2,10.54,;3.86,8.23,;2.53,9,;1.2,3.61,;5.2,1.3,;6.53,2.07,;7.87,1.3,;7.87,-.24,;6.53,-1.01,;5.2,-.24,;6.85,-2.51,;5.82,-3.66,;4.28,-3.74,;4.36,-5.28,;4.44,-6.81,;5.9,-5.2,;2.83,-5.36,;2.13,-6.73,;.59,-6.81,;-.25,-5.52,;-1.09,-4.23,;.45,-4.15,;1.99,-4.07,;8.38,-2.67,;9.15,-4.01,;9.01,-1.27,;10.48,-1.73,;10.16,-.25,)|
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CC(C)n1cnc2cc(nc(Nc3cc(C(=O)NCC(F)F)c(F)c(F)c3F)c12)-c1cnc2c(c1)N(C1CC(C)(C1)N1CCCCC1)C(=O)C2(C)C |(11.31,-2.5,;9.81,-2.18,;8.78,-3.32,;9.33,-.71,;10.23,.53,;9.33,1.78,;7.87,1.3,;6.53,2.07,;5.2,1.3,;5.2,-.24,;6.53,-1.01,;6.53,-2.55,;5.2,-3.32,;5.2,-4.86,;3.86,-5.63,;3.86,-7.17,;5.2,-7.94,;2.53,-7.94,;2.53,-9.48,;1.2,-10.25,;1.2,-11.79,;-.14,-9.48,;2.53,-4.86,;1.2,-5.63,;2.53,-3.32,;1.2,-2.55,;3.86,-2.55,;3.86,-1.01,;7.87,-.24,;3.86,2.07,;3.86,3.61,;2.53,4.38,;1.2,3.61,;1.2,2.07,;2.53,1.3,;-.27,1.6,;-.74,.13,;-.04,-1.24,;-1.42,-1.94,;-1.06,-3.44,;-2.12,-.57,;-2.59,-2.94,;-2.31,-4.45,;-3.48,-5.45,;-4.93,-4.94,;-5.21,-3.43,;-4.04,-2.43,;-1.17,2.84,;-2.71,2.84,;-.27,4.09,;.04,5.6,;-1.4,5.13,)|
CC(C)n1cnc2cc(nc(Nc3cc(C(=O)NCC(F)F)c(Cl)c(F)c3F)c12)-c1ccc2c(c1)N(C(=O)C21CC1)C1(C)CC(C1)N1CCCCC1 |(-8.9,1.76,;-7.4,2.13,;-6.97,3.61,;-6.34,1.02,;-6.61,-.5,;-5.25,-1.23,;-4.14,-.16,;-2.6,-.28,;-1.74,1,;-2.41,2.38,;-3.94,2.5,;-4.61,3.89,;-3.75,5.16,;-4.42,6.55,;-3.55,7.82,;-4.22,9.21,;-3.35,10.48,;-5.75,9.32,;-6.42,10.71,;-7.96,10.82,;-8.63,12.21,;-8.83,9.55,;-2.01,7.7,;-1.15,8.98,;-1.34,6.32,;.19,6.2,;-2.21,5.04,;-1.54,3.66,;-4.81,1.23,;-.2,.88,;.66,2.16,;2.2,2.04,;2.87,.66,;2,-.62,;.47,-.5,;2.95,-1.83,;4.4,-1.31,;5.67,-2.18,;4.35,.23,;4.93,1.65,;5.87,.43,;2.52,-3.31,;3.99,-3.74,;2.08,-4.79,;.61,-4.36,;1.04,-2.88,;-.74,-5.1,;-.78,-6.64,;-2.13,-7.38,;-3.44,-6.58,;-3.41,-5.04,;-2.06,-4.3,)|
CCNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N(C2CC(C)(C2)N2CCCCC2)C(=O)C3(C)C)c(F)cc1C |(5.2,4.38,;6.53,3.61,;7.87,4.38,;7.87,5.92,;9.2,6.69,;6.53,6.69,;5.2,5.92,;3.86,6.69,;2.53,5.92,;2.53,4.38,;3.86,3.61,;3.86,2.07,;2.53,1.3,;1.2,2.07,;-.27,1.6,;-1.17,2.84,;-.27,4.09,;-.74,5.55,;-2.25,5.87,;.29,6.7,;1.2,3.61,;5.2,1.3,;5.2,-.24,;6.53,-1.01,;7.87,-.24,;7.87,1.3,;6.53,2.07,;9.33,1.78,;9.81,3.24,;9.11,4.62,;10.48,5.31,;10.12,6.81,;11.18,3.94,;11.65,6.31,;11.37,7.83,;12.54,8.83,;13.99,8.32,;14.27,6.8,;13.1,5.8,;10.23,.53,;11.77,.53,;9.33,-.71,;8.7,-2.12,;10.66,-1.48,;3.86,8.23,;2.53,9,;5.2,9,;6.53,8.23,;7.87,9,)|
CC(C)n1cnc2cc(nc(Nc3cc(C(=O)NCC(F)F)c(C)c(F)c3F)c12)-c1cc2N(C3CC(C)(C3)N3CCCC4(CC4)C3)C(=O)C(C)(C)c2nc1F
CCNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2cnc3c(c2)N(C2CC(C)(C2)N2CCCCC2)C(=O)C3(C)C)c(F)c(F)c1F |(11.87,6.69,;10.53,5.92,;9.2,6.69,;7.87,5.92,;7.87,4.38,;6.53,6.69,;5.2,5.92,;3.86,6.69,;2.53,5.92,;2.53,4.38,;3.86,3.61,;3.86,2.07,;2.53,1.3,;1.2,2.07,;-.27,1.6,;-1.17,2.84,;-.27,4.09,;-.74,5.55,;-2.25,5.87,;.29,6.7,;1.2,3.61,;5.2,1.3,;6.53,2.07,;7.87,1.3,;7.87,-.24,;6.53,-1.01,;5.2,-.24,;6.85,-2.51,;5.82,-3.66,;5.9,-5.2,;4.36,-5.28,;2.89,-5.71,;4.28,-3.74,;4.08,-6.79,;5.25,-7.79,;4.97,-9.3,;3.52,-9.82,;2.35,-8.82,;2.63,-7.3,;8.38,-2.67,;9.15,-4.01,;9.01,-1.27,;9.91,-.02,;10.34,-2.04,;3.86,8.23,;2.53,9,;5.2,9,;5.2,10.54,;6.53,8.23,;7.87,9,)|
CCNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2cc3N(C4CC(C)(C4)N4CCCC5(CC5)C4)C(=O)C(C)(C)c3nc2F)c(F)c(F)c1C
CC(C)n1cnc2cc(nc(Nc3cc(C(=O)NC4(CC4)C(F)F)c(F)c(F)c3F)c12)-c1cnc2c(c1)N(C1CC(C)(C1)N1CCCCC1)C(=O)C2(C)C |(11.31,-2.5,;9.81,-2.18,;8.78,-3.32,;9.33,-.71,;10.23,.53,;9.33,1.78,;7.87,1.3,;6.53,2.07,;5.2,1.3,;5.2,-.24,;6.53,-1.01,;6.53,-2.55,;5.2,-3.32,;5.2,-4.86,;3.86,-5.63,;3.86,-7.17,;5.2,-7.94,;2.53,-7.94,;2.53,-9.48,;4.05,-9.74,;3.06,-10.92,;1.01,-9.74,;.02,-8.56,;.49,-11.19,;2.53,-4.86,;1.2,-5.63,;2.53,-3.32,;1.2,-2.55,;3.86,-2.55,;3.86,-1.01,;7.87,-.24,;3.86,2.07,;3.86,3.61,;2.53,4.38,;1.2,3.61,;1.2,2.07,;2.53,1.3,;-.27,1.6,;-.74,.13,;-.04,-1.24,;-1.42,-1.94,;-1.06,-3.44,;-2.12,-.57,;-2.59,-2.94,;-2.31,-4.45,;-3.48,-5.45,;-4.93,-4.94,;-5.21,-3.43,;-4.04,-2.43,;-1.17,2.84,;-2.71,2.84,;-.27,4.09,;.04,5.6,;-1.4,5.13,)|
CNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2cnc3c(c2)N(C(=O)C3(C)C)C2(C)CC(C2)N2CCCCC2)c(F)c(F)c1Cl
CC(C)n1cnc2cc(nc(Nc3cc(C(=O)NCC(F)F)c(Cl)c(F)c3F)c12)-c1cnc2c(c1)N(C1CC(C)(C1)N1CCCC3(CC3)C1)C(=O)C2(C)C
CCNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2cnc3c(c2)N(C2CC(C)(C2)N2CCCC4(CC4)C2)C(=O)C3(C)C)c(F)c(F)c1Cl
CC(C)n1cnc2cc(nc(Nc3cc(C(=O)NCC(F)F)c(C)c(F)c3F)c12)-c1cnc2c(c1)N(C1CC(C)(C1)N1CCCC3(CC3)C1)C(=O)C2(C)C
CCNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2cnc3c(c2)N(C2CC(C)(C2)N2CCCC4(CC4)C2)C(=O)C3(C)C)c(F)c(F)c1C
CCNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2cnc3c(c2)N(C2CC(C)(C2)N2CCCCC2)C(=O)C3(C)C)c(F)c(F)c1Cl |(-1.47,-5.63,;-.14,-4.86,;-.14,-3.32,;1.2,-2.55,;1.2,-1.01,;2.53,-3.32,;3.86,-2.55,;5.2,-3.32,;6.53,-2.55,;6.53,-1.01,;5.2,-.24,;5.2,1.3,;6.53,2.07,;7.87,1.3,;9.33,1.78,;10.23,.53,;9.33,-.71,;9.81,-2.18,;11.31,-2.5,;8.78,-3.32,;7.87,-.24,;3.86,2.07,;3.86,3.61,;2.53,4.38,;1.2,3.61,;1.2,2.07,;2.53,1.3,;-.27,1.6,;-.74,.13,;-.04,-1.24,;-1.42,-1.94,;-1.06,-3.44,;-2.12,-.57,;-2.59,-2.94,;-2.31,-4.45,;-3.48,-5.45,;-4.93,-4.94,;-5.21,-3.43,;-4.04,-2.43,;-1.17,2.84,;-2.71,2.84,;-.27,4.09,;.04,5.6,;-1.4,5.13,;5.2,-4.86,;6.53,-5.63,;3.86,-5.63,;3.86,-7.17,;2.53,-4.86,;1.2,-5.63,)|
CC(C)n1cnc2cc(nc(Nc3cc(C(=O)NCC(F)F)c(Cl)c(F)c3F)c12)-c1ccc2c(c1)N(C(=O)C2(C)C)C1(C)CC(C1)N1CCCCC1
CCNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N(C2CC(C)(C2)N2CCCCC2)C(=O)C3(C)C)c(F)c(F)c1Cl |(18.26,-.24,;16.93,-1.01,;15.59,-.24,;14.26,-1.01,;14.26,-2.55,;12.93,-.24,;12.93,1.3,;11.59,2.07,;11.59,3.61,;10.26,4.38,;8.93,3.61,;7.59,4.38,;7.59,5.92,;8.93,6.69,;9.25,8.2,;10.78,8.36,;11.4,6.95,;12.91,6.63,;13.94,7.78,;13.39,5.17,;10.26,5.92,;6.26,3.61,;6.26,2.07,;4.92,1.3,;3.59,2.07,;3.59,3.61,;4.92,4.38,;2.13,4.09,;1.65,5.55,;.28,6.25,;.98,7.62,;1.34,9.12,;2.35,6.93,;-.19,8.62,;-1.65,8.11,;-2.82,9.11,;-2.54,10.63,;-1.08,11.14,;.09,10.14,;1.22,2.84,;-.32,2.84,;2.13,1.6,;2.43,.09,;.99,.55,;10.26,1.3,;8.93,2.07,;10.26,-.24,;8.93,-1.01,;11.59,-1.01,;11.59,-2.55,)|
CC(C)n1cnc2cc(nc(Nc3cc(C(=O)NCC(F)F)c(Cl)cc3F)c12)-c1ccc2c(c1)N(C(=O)C2(C)C)C1(C)CC(C1)N1CCCCC1
CCNC(=O)c1cc(Nc2nc(cc3ncn(C(C)C)c23)-c2ccc3c(c2)N(C2CC(C)(C2)N2CCCCC2)C(=O)C3(C)C)c(F)cc1Cl |(18.26,-.24,;16.93,-1.01,;15.59,-.24,;14.26,-1.01,;14.26,-2.55,;12.93,-.24,;12.93,1.3,;11.59,2.07,;11.59,3.61,;10.26,4.38,;8.93,3.61,;7.59,4.38,;7.59,5.92,;8.93,6.69,;9.25,8.2,;10.78,8.36,;11.4,6.95,;12.91,6.63,;13.94,7.78,;13.39,5.17,;10.26,5.92,;6.26,3.61,;6.26,2.07,;4.92,1.3,;3.59,2.07,;3.59,3.61,;4.92,4.38,;2.13,4.09,;1.65,5.55,;.28,6.25,;.98,7.62,;1.34,9.12,;2.35,6.93,;-.19,8.62,;-1.65,8.11,;-2.82,9.11,;-2.54,10.63,;-1.08,11.14,;.09,10.14,;1.22,2.84,;-.32,2.84,;2.13,1.6,;2.43,.09,;.99,.55,;10.26,1.3,;8.93,2.07,;10.26,-.24,;11.59,-1.01,;11.59,-2.55,)|
CC(C)n1cnc2cc(nc(Nc3cc(C(=O)NC4(CC4)C(F)F)c(Cl)c(F)c3F)c12)-c1cc2N(C3CC(C)(C3)N3CCCCC3)C(=O)C(C)(C)c2nc1F |(11.31,-2.5,;9.81,-2.18,;8.78,-3.32,;9.33,-.71,;10.23,.53,;9.33,1.78,;7.87,1.3,;6.53,2.07,;5.2,1.3,;5.2,-.24,;6.53,-1.01,;6.53,-2.55,;5.2,-3.32,;5.2,-4.86,;3.86,-5.63,;3.86,-7.17,;5.2,-7.94,;2.53,-7.94,;2.53,-9.48,;3.06,-10.92,;4.05,-9.74,;1.01,-9.74,;.49,-11.19,;.02,-8.56,;2.53,-4.86,;1.2,-5.63,;2.53,-3.32,;1.2,-2.55,;3.86,-2.55,;3.86,-1.01,;7.87,-.24,;3.86,2.07,;2.53,1.3,;1.2,2.07,;-.27,1.6,;-.74,.13,;-.04,-1.24,;-1.42,-1.94,;-1.06,-3.44,;-2.12,-.57,;-2.59,-2.94,;-2.31,-4.45,;-3.48,-5.45,;-4.93,-4.94,;-5.21,-3.43,;-4.04,-2.43,;-1.17,2.84,;-2.71,2.84,;-.27,4.09,;.04,5.6,;-1.4,5.13,;1.2,3.61,;2.53,4.38,;3.86,3.61,;5.2,4.38,)|
CC(C)n1cnc2cc(nc(Nc3cc(C(=O)NC4(CF)CC4)c(Cl)c(F)c3F)c12)-c1ccc2c(c1)N(C1CC(C)(C1)N1CCCCC1)C(=O)C2(C)C |(13.94,7.78,;12.91,6.63,;13.39,5.17,;11.4,6.95,;10.78,8.36,;9.25,8.2,;8.93,6.69,;7.59,5.92,;7.59,4.38,;8.93,3.61,;10.26,4.38,;11.59,3.61,;11.59,2.07,;12.93,1.3,;12.93,-.24,;14.26,-1.01,;14.26,-2.55,;15.59,-.24,;16.93,-1.01,;17.92,.17,;17.39,1.62,;17.92,-2.19,;16.4,-2.45,;11.59,-1.01,;11.59,-2.55,;10.26,-.24,;8.93,-1.01,;10.26,1.3,;8.93,2.07,;10.26,5.92,;6.26,3.61,;6.26,2.07,;4.92,1.3,;3.59,2.07,;3.59,3.61,;4.92,4.38,;2.13,4.09,;1.65,5.55,;.28,6.25,;.98,7.62,;1.34,9.12,;2.35,6.93,;-.19,8.62,;-1.65,8.11,;-2.82,9.11,;-2.54,10.63,;-1.08,11.14,;.09,10.14,;1.22,2.84,;-.32,2.84,;2.13,1.6,;2.43,.09,;.99,.55,)|
CC(C)n1cnc2cc(nc(Nc3cc(C(=O)NC4(CF)CC4)c(Cl)cc3F)c12)-c1ccc2c(c1)N(C1CC(C)(C1)N1CCCCC1)C(=O)C2(C)C |(13.94,7.78,;12.91,6.63,;13.39,5.17,;11.4,6.95,;10.78,8.36,;9.25,8.2,;8.93,6.69,;7.59,5.92,;7.59,4.38,;8.93,3.61,;10.26,4.38,;11.59,3.61,;11.59,2.07,;12.93,1.3,;12.93,-.24,;14.26,-1.01,;14.26,-2.55,;15.59,-.24,;16.93,-1.01,;17.92,.17,;17.39,1.62,;17.92,-2.19,;16.4,-2.45,;11.59,-1.01,;11.59,-2.55,;10.26,-.24,;10.26,1.3,;8.93,2.07,;10.26,5.92,;6.26,3.61,;6.26,2.07,;4.92,1.3,;3.59,2.07,;3.59,3.61,;4.92,4.38,;2.13,4.09,;1.65,5.55,;.28,6.25,;.98,7.62,;1.34,9.12,;2.35,6.93,;-.19,8.62,;-1.65,8.11,;-2.82,9.11,;-2.54,10.63,;-1.08,11.14,;.09,10.14,;1.22,2.84,;-.32,2.84,;2.13,1.6,;2.43,.09,;.99,.55,)|
CC(C)n1cnc2cc(nc(Nc3cc(C(=O)NC4(CC4)C(F)F)c(Cl)cc3F)c12)-c1ccc2c(c1)N(C1CC(C)(C1)N1CCCCC1)C(=O)C2(C)C |(13.94,7.78,;12.91,6.63,;13.39,5.17,;11.4,6.95,;10.78,8.36,;9.25,8.2,;8.93,6.69,;7.59,5.92,;7.59,4.38,;8.93,3.61,;10.26,4.38,;11.59,3.61,;11.59,2.07,;12.93,1.3,;12.93,-.24,;14.26,-1.01,;14.26,-2.55,;15.59,-.24,;16.93,-1.01,;17.92,-2.19,;16.4,-2.45,;17.92,.17,;17.39,1.62,;19.43,-.09,;11.59,-1.01,;11.59,-2.55,;10.26,-.24,;10.26,1.3,;8.93,2.07,;10.26,5.92,;6.26,3.61,;6.26,2.07,;4.92,1.3,;3.59,2.07,;3.59,3.61,;4.92,4.38,;2.13,4.09,;1.65,5.55,;.28,6.25,;.98,7.62,;1.34,9.12,;2.35,6.93,;-.19,8.62,;-1.65,8.11,;-2.82,9.11,;-2.54,10.63,;-1.08,11.14,;.09,10.14,;1.22,2.84,;-.32,2.84,;2.13,1.6,;2.43,.09,;.99,.55,)|
CC(C)n1cnc2cc(nc(Nc3cc(C(=O)NC4(CC4)C(F)F)c(C)cc3F)c12)-c1ccc2c(c1)N(C(=O)C2(C)C)C1(C)CC(C1)N1CCCCC1
CC(C)n1cnc2cc(nc(Nc3cc(C(=O)NC4(CC4)C(F)F)c(Cl)c(F)c3F)c12)-c1ccc2c(c1)N(C(=O)C2(C)C)C1(C)CC(C1)N1CCCCC1
CC(C)n1cnc2cc(nc(Nc3cc(C(=O)NC4(CC4)C(F)F)c(Cl)c(F)c3F)c12)-c1cnc2c(c1)N(C(=O)C2(C)C)C1(C)CC(C1)N1CCCCC1 |(4.38,3.25,;3.35,2.1,;3.83,.64,;1.85,2.42,;1.22,3.83,;-.31,3.67,;-.63,2.16,;-1.97,1.39,;-1.97,-.15,;-.63,-.92,;.7,-.15,;2.04,-.92,;2.04,-2.46,;3.37,-3.23,;3.37,-4.77,;4.7,-5.54,;4.7,-7.08,;6.04,-4.77,;7.37,-5.54,;8.36,-6.72,;6.84,-6.99,;8.36,-4.36,;7.83,-2.91,;9.88,-4.63,;2.04,-5.54,;2.04,-7.08,;.7,-4.77,;-.63,-5.54,;.7,-3.23,;-.63,-2.46,;.7,1.39,;-3.3,-.92,;-3.3,-2.46,;-4.63,-3.23,;-5.97,-2.46,;-5.97,-.92,;-4.63,-.15,;-7.43,-.44,;-8.34,-1.69,;-9.88,-1.69,;-7.43,-2.93,;-7.13,-4.44,;-8.57,-3.98,;-7.91,1.02,;-9.37,.55,;-8.38,2.49,;-6.92,2.96,;-6.44,1.5,;-6.22,4.33,;-7.06,5.63,;-6.36,7,;-4.82,7.08,;-3.98,5.79,;-4.68,4.42,)|
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2ccc(nc12)-c1ccccc1
COc1ccccc1-c1ccc2[nH]nc(-c3ccc(cc3)N3CCN(C)CC3)c2n1
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2ccc(nc12)-c1ccccc1C
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2ccc(nc12)-c1ccccc1F
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2ccc(nc12)-c1ccccc1C(F)(F)F
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2ccc(nc12)-c1cccc(N)c1C
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2ccc(nc12)-c1c(C)cccc1F
COc1cccc(F)c1-c1ccc2[nH]nc(-c3ccc(cc3)N3CCN(C)CC3)c2n1
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2ccc(nc12)-c1cccc(F)c1F
COc1ccc(F)c(F)c1-c1ccc2[nH]nc(-c3ccc(cc3)N3CCN(C)CC3)c2n1
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2ccc(nc12)-c1c(F)cccc1CO
CCOC(=O)c1cccc(c1F)-c1ccc2[nH]nc(-c3ccc(cc3)N3CCN(C)CC3)c2n1
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2ccc(nc12)-c1cccc(NS(C)(=O)=O)c1F
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2ccc(nc12)-c1ccccc1O
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2ccc(nc12)-c1cccc2CCOc12
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2ccc(nc12)-c1cccc2OCCOc12
CNC(=O)c1cccc(c1)-c1ccc2[nH]nc(-c3ccc(cc3)N3CCN(C)CC3)c2n1
CN(C)c1cccc(c1)-c1ccc2[nH]nc(-c3ccc(cc3)N3CCN(C)CC3)c2n1
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2ccc(nc12)-c1ccccc1C#N
COC(=O)c1ccccc1-c1ccc2[nH]nc(-c3ccc(cc3)N3CCN(C)CC3)c2n1
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2ccc(nc12)-c1ccccc1NC(C)=O
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2ccc(nc12)-c1ccccc1-c1ccccc1
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2ccc(nc12)-c1cccc2[nH]ncc12
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2ccc(nc12)-c1cccnc1
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2ccc(nc12)-c1ccncc1
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2ccc(nc12)-c1cncnc1
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2ccc(nc12)-c1cnc2NC(=O)Cc2c1
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2ccc(nc12)-c1cnc2cnn(C)c2c1
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2ccc(nc12)-c1cncc(c1)-c1ncco1
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2ccc(nc12)-c1ccc(=O)n(C)c1
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2ccc(nc12)-c1cnc2n(C)cnc2c1
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2ccc(nc12)-c1cnc2nccnc2c1
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2ccc(nc12)-c1cncc2oc(nc12)C(C)(C)C
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2ccc(nc12)-c1c[nH]nc1C
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2ccc(nc12)-c1cnn2ccccc12
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2ccc(nc12)-c1cccc2ncccc12
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2ccc(nc12)-c1cncc2ccccc12
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2ccc(nc12)-c1cccc2NC(=O)Cc12
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2ccc(nc12)-c1cccc2n(C)ccc12
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2ccc(nc12)-c1cccc(C(N)=O)c1F
CNC(=O)c1cccc(-c2ccc3[nH]nc(-c4ccc(cc4)N4CCN(C)CC4)c3n2)c1F
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2ccc(nc12)-c1cccc(C(=O)NCc2ccccc2)c1F
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2ccc(nc12)-c1cccc(C(=O)NCc2ccncc2)c1F
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2ccc(nc12)-c1cccn2ccnc12
CCc1cn2cccc(-c3ccc4[nH]nc(-c5ccc(cc5)N5CCN(C)CC5)c4n3)c2n1
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2ccc(nc12)-c1cccc2CNCCc12
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2ccc(nc12)-c1cccc2C(N)CCc12
CNC1CCc2c1cccc2-c1ccc2[nH]nc(-c3ccc(cc3)N3CCN(C)CC3)c2n1
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2ccc(nc12)-c1cccc2C(CCc12)NCCO
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2ccc(nc12)-c1cccc2C(CCc12)NCc1ccccc1
Fc1ccccc1-c1ccc2[nH]nc(-c3ccccc3)c2n1
Fc1ccccc1-c1ccc2[nH]nc(-c3ccncc3)c2n1
CNC(=O)c1ccc(cc1)-c1n[nH]c2ccc(nc12)-c1ccccc1F
Cn1cc(cn1)-c1n[nH]c2ccc(nc12)-c1ccccc1F
CN1CCC(CC1)NC(=O)c1ccc(cc1)-c1n[nH]c2ccc(nc12)-c1ccccc1F
CN1CCN(CC1)C(=O)c1ccc(cc1)-c1n[nH]c2ccc(nc12)-c1ccccc1F
Fc1ccccc1-c1ccc2[nH]nc(-c3ccc(cc3)C(=O)Nc3ccccc3)c2n1
Fc1ccccc1-c1ccc2[nH]nc(-c3cnn(c3)C3CCNCC3)c2n1
CS(=O)(=O)N1CCC(CC1)n1cc(cn1)-c1n[nH]c2ccc(nc12)-c1ccccc1F
CC(=O)N1CCC(CC1)n1cc(cn1)-c1n[nH]c2ccc(nc12)-c1ccccc1F
CNCc1cc(F)c(c(F)c1)-c1ccc2[nH]nc(-c3ccc(cc3)N3CCN(C)CC3)c2n1
CN1CCN(CC1)c1ccc(cn1)-c1n[nH]c2cc(C#N)c(nc12)-c1c(C)cccc1F |(8.46,2.25,;7.09,1.55,;7.01,.01,;5.64,-.69,;4.35,.15,;4.43,1.69,;5.8,2.39,;2.98,-.55,;1.68,.29,;.31,-.41,;.23,-1.94,;1.52,-2.78,;2.89,-2.08,;-1.14,-2.64,;-1.38,-4.16,;-2.9,-4.4,;-3.6,-3.03,;-5.09,-2.63,;-5.49,-1.15,;-6.98,-.75,;-8.46,-.35,;-4.4,-.06,;-2.91,-.46,;-2.51,-1.94,;-4.8,1.43,;-3.71,2.52,;-2.22,2.12,;-4.11,4.01,;-5.6,4.4,;-6.68,3.32,;-6.29,1.83,;-7.37,.74,)|
Cc1cccc(F)c1-c1nc2c(n[nH]c2cc1C#N)-c1cnc(nc1)N1CCOCC1 |(-1.74,2.14,;-3.23,2.52,;-3.64,4.01,;-5.13,4.39,;-6.21,3.29,;-5.8,1.8,;-6.87,.7,;-4.31,1.42,;-3.89,-.06,;-2.4,-.44,;-1.98,-1.92,;-.64,-2.58,;-.82,-4.13,;-2.34,-4.39,;-3.06,-3.03,;-4.55,-2.64,;-4.96,-1.16,;-6.46,-.78,;-7.95,-.4,;.77,-1.97,;1.97,-2.93,;3.41,-2.37,;3.64,-.85,;2.44,.11,;1.01,-.44,;5.08,-.29,;6.28,-1.25,;7.72,-.7,;7.95,.83,;6.75,1.79,;5.31,1.23,)|
CCN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2cc(C#N)c(nc12)-c1c(C)cccc1F |(9.27,.42,;8.07,1.39,;6.63,.83,;6.4,-.7,;4.96,-1.25,;3.76,-.29,;3.99,1.23,;5.43,1.79,;2.33,-.85,;2.09,-2.37,;.66,-2.93,;-.54,-1.97,;-.31,-.44,;1.12,.11,;-1.96,-2.58,;-2.14,-4.13,;-3.66,-4.39,;-4.37,-3.03,;-5.87,-2.64,;-6.28,-1.16,;-7.78,-.78,;-9.27,-.4,;-5.21,-.06,;-3.71,-.44,;-3.3,-1.92,;-5.62,1.42,;-4.55,2.52,;-3.05,2.14,;-4.96,4.01,;-6.45,4.39,;-7.53,3.29,;-7.12,1.8,;-8.19,.7,)|
CNC(=O)c1ccc(cn1)-c1n[nH]c2cc(C#N)c(nc12)-c1c(C)cccc1F |(7.83,-.7,;6.4,-1.25,;5.2,-.29,;5.43,1.23,;3.76,-.85,;2.56,.11,;1.12,-.44,;.89,-1.97,;2.09,-2.93,;3.53,-2.37,;-.52,-2.58,;-.71,-4.13,;-2.22,-4.39,;-2.94,-3.03,;-4.43,-2.64,;-4.85,-1.16,;-6.34,-.78,;-7.83,-.4,;-3.77,-.06,;-2.28,-.44,;-1.86,-1.92,;-4.19,1.42,;-3.11,2.52,;-1.62,2.14,;-3.53,4.01,;-5.02,4.39,;-6.1,3.29,;-5.68,1.8,;-6.76,.7,)|
CNCc1cc(C)c(c(F)c1)-c1nc2c(n[nH]c2cc1C#N)-c1cnn(C)c1 |(-.71,5.3,;-2.21,5.68,;-3.28,4.58,;-2.87,3.1,;-1.38,2.71,;-.96,1.23,;.53,.85,;-2.04,.13,;-3.53,.51,;-4.61,-.59,;-3.95,2,;-1.62,-1.35,;-.13,-1.73,;.29,-3.22,;1.63,-3.87,;1.44,-5.42,;-.07,-5.68,;-.79,-4.32,;-2.28,-3.94,;-2.7,-2.45,;-4.19,-2.07,;-5.68,-1.69,;3.04,-3.26,;4.37,-4.04,;5.52,-3.02,;4.9,-1.6,;5.68,-.28,;3.37,-1.75,)|
CNCc1cc(C)c(c(F)c1)-c1nc2c(n[nH]c2cc1C#N)-c1ccc(nc1)N1CCN(C)CC1 |(-3.7,5.3,;-5.19,5.68,;-6.27,4.58,;-5.85,3.1,;-4.36,2.71,;-3.95,1.23,;-2.45,.85,;-5.02,.13,;-6.51,.51,;-7.59,-.59,;-6.93,2,;-4.61,-1.35,;-3.11,-1.73,;-2.7,-3.22,;-1.36,-3.87,;-1.54,-5.42,;-3.06,-5.68,;-3.77,-4.32,;-5.27,-3.94,;-5.68,-2.45,;-7.17,-2.07,;-8.67,-1.69,;.06,-3.26,;.29,-1.74,;1.72,-1.18,;2.93,-2.14,;2.69,-3.66,;1.26,-4.22,;4.36,-1.58,;5.56,-2.55,;7,-1.99,;7.23,-.46,;8.67,.09,;6.03,.5,;4.59,-.06,)|
CNCc1cc(C)c(c(F)c1)-c1nc2c(n[nH]c2cc1C#N)-c1cnc(nc1)N1CCN(C)CC1 |(-3.7,5.3,;-5.19,5.68,;-6.27,4.58,;-5.85,3.1,;-4.36,2.71,;-3.95,1.23,;-2.45,.85,;-5.02,.13,;-6.51,.51,;-7.59,-.59,;-6.93,2,;-4.61,-1.35,;-3.11,-1.73,;-2.7,-3.22,;-1.36,-3.87,;-1.54,-5.42,;-3.06,-5.68,;-3.77,-4.32,;-5.27,-3.94,;-5.68,-2.45,;-7.17,-2.07,;-8.67,-1.69,;.06,-3.26,;1.26,-4.22,;2.69,-3.66,;2.93,-2.14,;1.72,-1.18,;.29,-1.74,;4.36,-1.58,;5.56,-2.55,;7,-1.99,;7.23,-.46,;8.67,.09,;6.03,.5,;4.59,-.06,)|
CCN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2cc(C#N)c(nc12)-c1c(C)cc(CNC)cc1F |(9.27,-.87,;8.07,.09,;6.63,-.46,;6.4,-1.99,;4.96,-2.55,;3.76,-1.58,;3.99,-.06,;5.43,.5,;2.33,-2.14,;2.09,-3.66,;.66,-4.22,;-.54,-3.26,;-.31,-1.74,;1.12,-1.18,;-1.96,-3.87,;-2.14,-5.42,;-3.66,-5.68,;-4.37,-4.32,;-5.87,-3.94,;-6.28,-2.45,;-7.78,-2.07,;-9.27,-1.69,;-5.21,-1.35,;-3.71,-1.73,;-3.3,-3.22,;-5.62,.13,;-4.55,1.23,;-3.05,.85,;-4.96,2.71,;-6.45,3.1,;-6.87,4.58,;-5.79,5.68,;-4.3,5.3,;-7.53,2,;-7.12,.51,;-8.19,-.59,)|
CNCc1cc(C)c(c(F)c1)-c1nc2c(n[nH]c2cc1C#N)-c1cnc(nc1)N1CCOCC1 |(-2.98,5.3,;-4.47,5.68,;-5.55,4.58,;-5.13,3.1,;-3.64,2.71,;-3.23,1.23,;-1.74,.85,;-4.31,.13,;-5.8,.51,;-6.87,-.59,;-6.21,2,;-3.89,-1.35,;-2.4,-1.73,;-1.98,-3.22,;-.64,-3.87,;-.82,-5.42,;-2.34,-5.68,;-3.06,-4.32,;-4.55,-3.94,;-4.96,-2.45,;-6.46,-2.07,;-7.95,-1.69,;.77,-3.26,;1.97,-4.22,;3.41,-3.66,;3.64,-2.14,;2.44,-1.18,;1.01,-1.74,;5.08,-1.58,;6.28,-2.55,;7.72,-1.99,;7.95,-.46,;6.75,.5,;5.31,-.06,)|
CNCc1cc(C)c(c(F)c1)-c1nc2c(n[nH]c2cc1C#N)-c1ccc(nc1)C(C)(C)O |(-1.89,5.28,;-3.36,5.72,;-4.48,4.66,;-4.12,3.16,;-2.64,2.72,;-2.28,1.23,;-.8,.79,;-3.4,.16,;-4.87,.6,;-5.99,-.46,;-5.23,2.1,;-3.03,-1.33,;-1.56,-1.77,;-1.2,-3.27,;.16,-4,;-.12,-5.51,;-1.65,-5.72,;-2.31,-4.33,;-3.79,-3.89,;-4.15,-2.39,;-5.63,-1.96,;-7.1,-1.52,;1.55,-3.34,;1.67,-1.8,;3.06,-1.14,;4.33,-2.01,;4.21,-3.54,;2.82,-4.21,;5.71,-1.34,;5.83,.19,;6.99,-2.21,;7.1,-.68,)|
CNCc1cc(C)c(c(F)c1)-c1nc2c(n[nH]c2cc1C#N)-c1ccc(nc1)C(=O)NC |(-2.52,5.28,;-4,5.72,;-5.11,4.66,;-4.75,3.16,;-3.28,2.72,;-2.91,1.23,;-1.44,.79,;-4.03,.16,;-5.51,.6,;-6.62,-.46,;-5.87,2.1,;-3.67,-1.33,;-2.19,-1.77,;-1.83,-3.27,;-.48,-4,;-.76,-5.51,;-2.28,-5.72,;-2.95,-4.33,;-4.42,-3.89,;-4.79,-2.39,;-6.26,-1.96,;-7.74,-1.52,;.91,-3.34,;1.03,-1.8,;2.42,-1.14,;3.69,-2.01,;3.57,-3.54,;2.18,-4.21,;5.08,-1.34,;5.2,.19,;6.35,-2.21,;7.74,-1.55,)|
Cn1cc(cn1)-c1n[nH]c2cc(C#N)c(nc12)-c1c(F)ccc2CNCCc12 |(5.6,.7,;4.86,-.65,;3.34,-.85,;3.06,-2.37,;4.41,-3.1,;5.53,-2.04,;1.67,-3.03,;1.39,-4.55,;-.14,-4.75,;-.8,-3.36,;-2.28,-2.92,;-2.64,-1.43,;-4.12,-.99,;-5.6,-.56,;-1.53,-.37,;-.05,-.8,;.31,-2.3,;-1.89,1.13,;-3.36,1.57,;-4.48,.51,;-3.72,3.06,;-2.61,4.12,;-1.13,3.69,;-.02,4.75,;1.46,4.31,;1.82,2.82,;.71,1.76,;-.77,2.19,)|
CCN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2cc(C#N)c(nc12)-c1c(F)ccc2CNCCc12 |(9.13,.75,;7.86,1.62,;6.47,.95,;6.35,-.58,;4.96,-1.25,;3.69,-.38,;3.81,1.16,;5.2,1.82,;2.3,-1.04,;1.03,-.17,;-.36,-.83,;-.48,-2.37,;.79,-3.24,;2.18,-2.58,;-1.87,-3.03,;-2.15,-4.55,;-3.67,-4.75,;-4.34,-3.36,;-5.81,-2.92,;-6.17,-1.43,;-7.65,-.99,;-9.13,-.56,;-5.06,-.37,;-3.58,-.8,;-3.22,-2.3,;-5.42,1.13,;-6.9,1.57,;-8.01,.51,;-7.26,3.06,;-6.14,4.12,;-4.66,3.69,;-3.55,4.75,;-2.07,4.31,;-1.67,2.83,;-2.83,1.76,;-4.3,2.19,)|
CN1CCN(CC1)c1ccc(cn1)-c1n[nH]c2cc(C#N)c(nc12)-c1c(F)ccc2CNCCc12 |(8.49,1.62,;7.1,.95,;6.99,-.58,;5.6,-1.25,;4.33,-.38,;4.45,1.16,;5.83,1.82,;2.94,-1.04,;1.67,-.17,;.28,-.83,;.16,-2.37,;1.43,-3.24,;2.82,-2.58,;-1.23,-3.03,;-1.51,-4.55,;-3.04,-4.75,;-3.7,-3.36,;-5.18,-2.92,;-5.54,-1.43,;-7.02,-.99,;-8.49,-.56,;-4.42,-.37,;-2.95,-.8,;-2.59,-2.3,;-4.78,1.13,;-6.26,1.57,;-7.38,.51,;-6.62,3.06,;-5.51,4.12,;-4.03,3.69,;-2.91,4.75,;-1.44,4.31,;-1.04,2.83,;-2.19,1.76,;-3.67,2.19,)|
Cc1cccc(F)c1-c1nc2c(n[nH]c2cc1C#N)-c1cnn(C)c1 |(.71,2.07,;-.77,2.5,;-1.13,4,;-2.61,4.44,;-3.72,3.38,;-3.36,1.88,;-4.48,.82,;-1.89,1.44,;-1.53,-.05,;-.05,-.49,;.31,-1.99,;1.67,-2.72,;1.39,-4.23,;-.14,-4.44,;-.8,-3.05,;-2.28,-2.61,;-2.64,-1.12,;-4.12,-.68,;-5.6,-.24,;3.06,-2.06,;4.41,-2.79,;5.53,-1.73,;4.86,-.34,;5.6,1.02,;3.34,-.54,)|
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(cc2n1)-c1ccccc1
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(cc2n1)-c1cnccc1C
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(cc2n1)-c1cncc(N)c1C
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(cc2n1)-c1cnc2OCCNc2c1C
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(cc2n1)-c1c(C)cccc1F
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(cc2n1)-c1cccc2CNCCc12
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(cc2n1)-c1cc(F)ccc1CN
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(cc2n1)-c1ccc(F)cc1CN
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(cc2n1)-c1cccc2CCNCc12
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(cc2n1)-c1ccccc1N1CCOC1=O
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(cc2n1)-c1cc(C)ccc1N1CCOC1=O
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(cc2n1)-c1ccc(nc1)C(F)(F)C(N)=O
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(cc2n1)-c1cnn(CCO)c1
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(cc2n1)-c1cncc(c1)C(C)(C)O
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(cc2n1)C1=CN=[c]([s]1)C(C)(C)O |c:30,t:28|
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(cc2n1)-c1ccn2ncnc2c1
COc1cncc(c1)-c1ccc2cnc(Nc3cc4CN(C)CCc4cc3OC)nc2c1
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(cc2n1)-c1ccc(NC(C)=O)nc1
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(cc2n1)-c1cnc(N)nc1C
CCn1cc(cn1)-c1ccc2cnc(Nc3cc4CN(C)CCc4cc3OC)nc2c1
CNC(=O)c1ccc(cn1)-c1ccc2cnc(Nc3cc4CN(C)CCc4cc3OC)nc2c1
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(cc2n1)-c1cnc2c(cnn2c1)C#N
CCNC(=O)c1ccc(cn1)-c1ccc2cnc(Nc3cc4CN(C)CCc4cc3OC)nc2c1
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(cc2n1)-c1cncc2cccnc12
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(cc2n1)-c1cnc2cccnc2c1
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(cc2n1)-c1cnn(c1)C(F)F
COc1cc2CCNCc2cc1Nc1ncc2ccc(cc2n1)-c1ccc(N)nc1
CNC(=O)c1ccc(cn1)-c1ccc2cnc(Nc3cc4CNCCc4cc3OC)nc2c1
COc1cc2CCNCc2cc1Nc1ncc2ccc(cc2n1)-c1cnc2N(C)CCOc2c1
COc1cc2CCNCc2cc1Nc1ncc2ccc(cc2n1)-c1ccc(NC(C)=O)nc1
COc1cc2CCNCc2cc1Nc1ncc2ccc(cc2n1)-c1cccc(N)c1C
COc1cc2CCNCc2cc1Nc1ncc2ccc(cc2n1)-c1ccc(cc1C)S(N)(=O)=O
COc1cc2CCNCc2cc1Nc1ncc2ccc(cc2n1)-c1ccc(cc1C)C#N
COc1cc2CCNCc2cc1Nc1ncc2ccc(cc2n1)-c1cnn(C)c1
COc1cc2CCNCc2cc1Nc1ncc2ccc(cc2n1)-c1cnn2CCCc12
COc1cc2CCNCc2cc1Nc1ncc2ccc(cc2n1)-c1cncc(NS(C)(=O)=O)c1
COc1cc2CCNCc2cc1Nc1ncc2ccc(cc2n1)-c1cnccc1Cl
COc1ccc(cn1)-c1ccc2cnc(Nc3cc4CNCCc4cc3OC)nc2c1
COc1cc2CCNCc2cc1Nc1ncc2ccc(cc2n1)-c1cccnc1
COc1cc2CCNCc2cc1Nc1ncc2ccc(cc2n1)-c1cncc(C)c1
COc1cc2CCNCc2cc1Nc1ncc2ccc(cc2n1)-c1cncc(c1)N1CCOCC1
COc1cc2CCNCc2cc1Nc1ncc2ccc(cc2n1)-c1cncc(c1)S(C)(=O)=O
COc1cncc(c1)-c1ccc2cnc(Nc3cc4CNCCc4cc3OC)nc2c1
COc1cc2CCNCc2cc1Nc1ncc2ccc(cc2n1)-c1cncc2[nH]ccc12
COc1cc2CCNCc2cc1Nc1ncc2ccc(cc2n1)-c1ccncc1
COc1cc2CCNCc2cc1Nc1ncc2ccc(cc2n1)-c1cncc(c1)C(=O)N1CCOCC1
COc1cc2CCNCc2cc1Nc1ncc2ccc(cc2n1)-c1ccc(NCCN2CCOCC2)nc1
COc1cc2CCNCc2cc1Nc1ncc2ccc(cc2n1)-c1cncc(CN)c1
COc1cc2CCNCc2cc1Nc1ncc2ccc(cc2n1)-c1cncc(c1)N1CCNCC1
COc1cc2CCNCc2cc1Nc1ncc2ccc(cc2n1)-c1cncc(NS(=O)(=O)C(C)C)c1
CCCC(=O)Nc1cncc(c1)-c1ccc2cnc(Nc3cc4CNCCc4cc3OC)nc2c1
COc1cc2CCNCc2cc1Nc1ncc2ccc(cc2n1)-c1cncc(CO)c1
COc1cc2CCNCc2cc1Nc1ncc2ccc(cc2n1)-c1cncc(c1)N1CCN(C)CC1
COc1cc2CCNCc2cc1Nc1ncc2ccc(cc2n1)-c1cccc(CC#N)c1
COc1cc2CCNCc2cc1Nc1ncc2ccc(cc2n1)-c1cccc(c1)-c1cn[nH]c1
COc1cc2CCNCc2cc1Nc1ncc2ccc(cc2n1)-c1ccc(CN(C)C)cc1
COc1cc2CCNCc2cc1Nc1ncc2ccc(cc2n1)-c1cccc(N)c1
COc1cc2CCNCc2cc1Nc1ncc2ccc(cc2n1)-c1cccc(O)c1
COc1cc2CCNCc2cc1Nc1ncc2ccc(cc2n1)-c1cccc(CO)c1
COc1cc2CCNCc2cc1Nc1ncc2ccc(cc2n1)-c1cccc(CN)c1
COc1cc2CCNCc2cc1Nc1ncc2ccc(cc2n1)-c1cc(N)cc(c1)C#N
COc1cc2CCNCc2cc1Nc1ncc2ccc(cc2n1)-c1cc(ccc1OC)C#N
COc1cc2CCNCc2cc1Nc1ncc2ccc(cc2n1)-c1ccc(CC#N)cc1
COc1cc2CCNCc2cc1Nc1ncc2ccc(cc2n1)-c1cccc(c1)C#N
COc1cc2CCNCc2cc1Nc1ncc2ccc(cc2n1)-c1cccc(c1)C(C)=O
COc1cc2CCNCc2cc1Nc1ncc2ccc(cc2n1)-c1cccc(c1)C(=O)NC1CC1
COc1cc2CCNCc2cc1Nc1ncc2ccc(cc2n1)-c1ccc2CN(CC3CC3)C(=O)c2c1
COc1cc2CCNCc2cc1Nc1ncc2ccc(cc2n1)-c1cccc(CN2CCCCC2)c1
COc1cc2CCNCc2cc1Nc1ncc2ccc(cc2n1)-c1ccc2OCCOc2c1
COc1cc2CCNCc2cc1Nc1ncc2ccc(cc2n1)-c1ccc2OCOc2c1
COc1cc2CCNCc2cc1Nc1ncc2ccc(cc2n1)-c1ccc2OCCc2c1
COc1cc2CCNCc2cc1Nc1ncc2ccc(cc2n1)-c1cccc2nc(N)[nH]c12
COc1cc2CCNCc2cc1Nc1ncc2ccc(cc2n1)-c1cc(ccc1OC)C1(CO)CC1
COc1cc2CCNCc2cc1Nc1ncc2ccc(cc2n1)-c1ccc2OCCCc2c1
COc1cc2CCNCc2cc1Nc1ncc2ccc(cc2n1)-c1ccc2CCOCc2c1
COc1cc2CCNCc2cc1Nc1ncc2ccc(cc2n1)-c1cccc(c1)S(=O)(=O)N1CCOCC1
COc1cc2CCNCc2cc1Nc1ncc2ccc(cc2n1)-c1cc(ccc1C)S(=O)(=O)N1CCCC1
COc1cc2CCNCc2cc1Nc1ncc2ccc(cc2n1)-c1cc(ccc1C)S(=O)(=O)N(C)C
CCN(CC)S(=O)(=O)c1cccc(c1)-c1ccc2cnc(Nc3cc4CNCCc4cc3OC)nc2c1
COc1cc2CCNCc2cc1Nc1ncc2ccc(cc2n1)-c1ccc(cc1)S(=O)(=O)N1CCCC1
COc1cc2CCNCc2cc1Nc1ncc2ccc(cc2n1)-c1cccc(c1)S(=O)(=O)N1CCCCC1
COc1cc2CCNCc2cc1Nc1ncc2ccc(cc2n1)-c1cccc(c1)C(=O)NCCN1CCCC1
CCNS(=O)(=O)c1cccc(c1)-c1ccc2cnc(Nc3cc4CNCCc4cc3OC)nc2c1
COc1cc2CCNCc2cc1Nc1ncc2ccc(cc2n1)-c1cc(NC(C)=O)ccc1C
COc1cc2CCNCc2cc1Nc1ncc2ccc(cc2n1)-c1cccc(c1)C(=O)N1CCCC1
COc1cc2CCNCc2cc1Nc1ncc2ccc(cc2n1)-c1ccc2NCCc2c1
COc1cc2CCNCc2cc1Nc1ncc2ccc(cc2n1)-c1ccc2NC(=O)CCc2c1
COc1cc2CCNCc2cc1Nc1ncc2ccc(cc2n1)-c1cccc(c1)C(C)(C)N
COc1cc2CCNCc2cc1Nc1ncc2ccc(cc2n1)-c1cc(ccc1F)C#N
COc1cc2CCNCc2cc1Nc1ncc2ccc(cc2n1)-c1cccc(c1)N1CCOCC1
COc1cc2CCNCc2cc1Nc1ncc2ccc(cc2n1)-c1ccccc1C1CC1
COc1cc2CCNCc2cc1Nc1ncc2ccc(cc2n1)-c1cc(N)ccc1C
COc1cc2CCNCc2cc1Nc1ncc2ccc(cc2n1)-c1c(C)cccc1F
COc1cc2CCN(C)Cc2cc1Nc1ncc2cc(F)c(cc2n1)-c1cnc2OCCNc2c1C
COc1cc2CCN(C)Cc2cc1Nc1ncc2cc(Cl)c(cc2n1)-c1cnc2OCCNc2c1C
COc1cc2CCN(C)Cc2cc1Nc1ncc2cc(C#N)c(cc2n1)-c1cnc2OCCNc2c1C
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(cc2n1)-c1cccc(NCC(C)=O)c1
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(cc2n1)-c1cccc(c1)C1CCC(=O)N1
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(cc2n1)-c1cccc(c1)C(C)(C)NC(C)=O
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(cc2n1)-c1cccc(c1)C(N)=O
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(cc2n1)-c1cnn(CC(C)O)c1
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(cc2n1)-c1ccc(nc1)C#N
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(cc2n1)-c1cnc(C#N)c(C)c1
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(cc2n1)-c1c[nH]nc1C
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(cc2n1)-c1cnc2[nH]c(=O)[nH]c2c1
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(cc2n1)-c1ccc(nc1)-n1cccn1
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(cc2n1)-c1ccc(CC#N)nc1
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(cc2n1)-c1ccccc1-c1ccnn1C
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(cc2n1)-c1ccccc1-c1nnc(C)o1
Cc1c2NCCOc2ncc1-c1cc2nc(Nc3ccc4C(=O)N(CC(C)(C)O)Cc4c3)ncc2cc1F
Cc1c2NCCOc2ncc1-c1cc2nc(Nc3ccc4C(=O)OC(C)(C)c4c3)ncc2cc1F
Cc1c2NCCOc2ncc1-c1cc2nc(Nc3ccc(CS(C)(=O)=O)nc3)ncc2cc1F
CN1CCc2ccc(Nc3ncc4cc(F)c(cc4n3)-c3cnc4OCCNc4c3C)cc2C1
Cc1c2NCCOc2ncc1-c1cc2nc(Nc3ccc(CS(C)(=O)=O)cc3)ncc2cc1F
CNC(=O)[C@@H](C)c1ccc(Nc2ncc3cc(F)c(cc3n2)-c2cnc3OCCNc3c2C)cc1 |r|
CNC(=O)[C@H](C)c1ccc(Nc2ncc3cc(F)c(cc3n2)-c2cnc3OCCNc3c2C)cc1 |r|
CNC(=O)[C@@H]1CCc2cc(Nc3ncc4cc(F)c(cc4n3)-c3cnc4OCCNc4c3C)ccc12 |r|
CNC(=O)[C@H]1CCc2cc(Nc3ncc4cc(F)c(cc4n3)-c3cnc4OCCNc4c3C)ccc12 |r|
CNC(=O)C1(CCCC1)c1ccc(Nc2ncc3cc(F)c(cc3n2)-c2cnc3OCCNc3c2C)cc1
CNC(=O)C1(CCC1)c1ccc(Nc2ncc3cc(F)c(cc3n2)-c2cnc3OCCNc3c2C)cc1
CNC(=O)C(F)(F)c1ccc(Nc2ncc3cc(F)c(cc3n2)-c2cnc3OCCNc3c2C)cc1
Cc1c2NCCOc2ncc1-c1ccc2cnc(Nc3ccc(CS(C)(=O)=O)cc3)nc2c1
C[C@@H](c1ccc(Nc2ncc3cc(F)c(cc3n2)-c2cnc3OCCNc3c2C)cc1)S(C)(=O)=O |r|
CN1CC[C@H](C1=O)c1ccc(Nc2ncc3cc(F)c(cc3n2)-c2cnc3OCCNc3c2C)cc1 |r|
C[C@H](c1ccc(Nc2ncc3cc(F)c(cc3n2)-c2cnc3OCCNc3c2C)cc1)S(C)(=O)=O |r|
CN1CC[C@@H](C1=O)c1ccc(Nc2ncc3cc(F)c(cc3n2)-c2cnc3OCCNc3c2C)cc1 |r|
CC(C)S(=O)(=O)Cc1ccc(Nc2ncc3cc(F)c(cc3n2)-c2cnc3OCCNc3c2C)cc1
CC(C)S(=O)(=O)Cc1ccc(Nc2ncc3ccc(cc3n2)-c2cnc3OCCNc3c2C)cc1
CNC(=O)Cc1ccc(Nc2ncc3cc(F)c(cc3n2)-c2cnc3OCCNc3c2C)cc1
Cc1c2NCCOc2ncc1-c1cc2nc(Nc3ccc(CC(N)=O)cc3)ncc2cc1F
CN(C)C(=O)Cc1ccc(Nc2ncc3cc(F)c(cc3n2)-c2cnc3OCCNc3c2C)cc1
Cc1c2NCCOc2ncc1-c1cc2nc(Nc3ccc(CC(=O)N4CCOCC4)cc3)ncc2cc1F
CCS(=O)(=O)Cc1ccc(Nc2ncc3ccc(cc3n2)-c2cnc3OCCNc3c2C)cc1
CN1CCc2ncc(Nc3ncc4cc(F)c(cc4n3)-c3cnc4OCCNc4c3C)cc2C1
COc1cc2CCN(C)Cc2cc1Nc1ncc2c(N)c(F)c(cc2n1)-c1cncc(N)c1C
COc1cc2CCN(C)Cc2cc1Nc1ncc2c(N)c(F)c(cc2n1)-c1cnc2OCCNc2c1C
COC(=O)Cc1ccc(OC)c(Nc2ncc3c(N)c(F)c(cc3n2)-c2cnc3OCCNc3c2C)c1
COc1cc2CCNCc2cc1Nc1ncc2c(N)c(F)c(cc2n1)-c1cnc2OCCNc2c1C
COc1ccc(CC#N)cc1Nc1ncc2c(N)c(F)c(cc2n1)-c1cnc2OCCNc2c1C
COc1cc(ccc1Nc1ncc2c(N)c(F)c(cc2n1)-c1cnc2OCCNc2c1C)S(N)(=O)=O
CC(=O)N1CCCc2cc(Nc3ncc4c(N)c(F)c(cc4n3)-c3cnc4OCCNc4c3C)ccc12
Cc1c2NCCOc2ncc1-c1cc2nc(Nc3ccccc3OC(F)(F)F)ncc2c(N)c1F
Cc1c2NCCOc2ncc1-c1cc2nc(Nc3cccnc3)ncc2c(N)c1F
CC(=O)N[C@@H]1CCc2cc(Nc3ncc4c(N)c(F)c(cc4n3)-c3cnc4OCCNc4c3C)ccc12 |r|
CC(=O)N[C@H]1CCc2cc(Nc3ncc4c(N)c(F)c(cc4n3)-c3cnc4OCCNc4c3C)ccc12 |r|
CC(=O)N1CCc2ccc(Nc3ncc4c(N)c(F)c(cc4n3)-c3cnc4OCCNc4c3C)cc2C1
CNC(=O)Cc1ccc(Nc2ncc3c(N)c(F)c(cc3n2)-c2cnc3OCCNc3c2C)cc1
Cc1c2NCCOc2ncc1-c1cc2nc(Nc3cccc(c3)S(C)(=O)=O)ncc2c(N)c1F
CC(=O)Nc1ccc(Nc2ncc3c(N)c(F)c(cc3n2)-c2cnc3OCCNc3c2C)cc1
Cc1c2NCCOc2ncc1-c1cc2nc(Nc3ccc(NS(C)(=O)=O)cc3)ncc2c(N)c1F
Cc1c2NCCOc2ncc1-c1cc2nc(Nc3ccc(cc3)S(C)(=O)=O)ncc2c(N)c1F
Cc1c2NCCOc2ncc1-c1cc2nc(Nc3ccc(cc3)C3(CC3)C#N)ncc2c(N)c1F
Cc1c2NCCOc2ncc1-c1cc2nc(Nc3cncnc3)ncc2c(N)c1F
COc1ccncc1Nc1ncc2c(N)c(F)c(cc2n1)-c1cnc2OCCNc2c1C
COc1c2CCNC(=O)Cc2ccc1Nc1ncc2c(N)c(F)c(cc2n1)-c1cnc2OCCNc2c1C
Cc1c2NCCOc2ncc1-c1cc2nc(Nc3ccccc3F)ncc2c(N)c1F
CNC(=O)c1ccc(Nc2ncc3c(N)c(F)c(cc3n2)-c2cnc3OCCNc3c2C)cc1
Cc1c2NCCOc2ncc1-c1cc2nc(Nc3ccc(CS(C)(=O)=O)cc3)ncc2c(N)c1F
Cc1c2NCCOc2ncc1-c1cc2nc(Nc3ccccc3)ncc2c(N)c1F
Cc1c2NCCOc2ncc1-c1cc2nc(Nc3ccccc3C3CC3)ncc2c(N)c1F
COc1ncccc1Nc1ncc2c(N)c(F)c(cc2n1)-c1cnc2OCCNc2c1C
CC(=O)N1CCC[C@@H]1c1ccc(Nc2ncc3c(N)c(F)c(cc3n2)-c2cnc3OCCNc3c2C)cc1 |r|
CC(=O)N1CCC[C@H]1c1ccc(Nc2ncc3c(N)c(F)c(cc3n2)-c2cnc3OCCNc3c2C)cc1 |r|
CC(=O)NCc1ccc(Nc2ncc3c(N)c(F)c(cc3n2)-c2cnc3OCCNc3c2C)cc1
Cc1c2NCCOc2ncc1-c1cc2nc(Nc3ccccc3Cl)ncc2c(N)c1F
Cc1ncccc1Nc1ncc2c(N)c(F)c(cc2n1)-c1cnc2OCCNc2c1C
Cc1c2NCCOc2ncc1-c1cc2nc(Nc3cccc(c3)S(=O)(=O)NC(C)(C)C)ncc2c(N)c1F
CNS(=O)(=O)c1cccc(Nc2ncc3c(N)c(F)c(cc3n2)-c2cnc3OCCNc3c2C)c1
COc1cc2CCN(C)[C@H](C)c2cc1Nc1ncc2c(N)c(F)c(cc2n1)-c1cnc2OCCNc2c1C |r|
COc1cc2CCN(C)[C@@H](C)c2cc1Nc1ncc2c(N)c(F)c(cc2n1)-c1cnc2OCCNc2c1C |r|
COc1cc2CCNCc2cc1Nc1ncc2c(N)cc(cc2n1)-c1cnccc1C
COc1cc2CCN(C)Cc2cc1Nc1ncc2c(N)cc(cc2n1)-c1c(C)cccc1F
COc1cc2CCN(C)Cc2cc1Nc1ncc2c(N)cc(cc2n1)-c1cncc(N)c1C
COc1cc2CCN(C)Cc2cc1Nc1ncc2c(N)cc(cc2n1)-c1cnc2OCCNc2c1C
Cc1c2NCCOc2ncc1-c1cc2nc(Nc3ccc4C(=O)OC(C)(C)c4c3)ncc2c(N)c1F
Cc1c2NCCOc2ncc1-c1cc2nc(Nc3ccc4C(=O)N(CC(C)(C)O)Cc4c3)ncc2c(N)c1F
Cc1c2NCCOc2ncc1-c1cc2nc(Nc3ccc4c(CCS4(=O)=O)c3)ncc2c(N)c1F
Cc1ccncc1-c1cc2nc(Nc3ccc(CS(C)(=O)=O)cc3)ncc2c(N)c1F
COc1cc2CCN(C)C(CO)c2cc1Nc1ncc2c(N)c(F)c(cc2n1)-c1cnc2OCCNc2c1C
COc1cc2CCN(C)Cc2cc1Nc1ncc2c(N)c(F)c(cc2n1)-c1cnc2ncsc2c1
COc1cc2CC(C)N(C)C(C)c2cc1Nc1ncc2c(N)c(F)c(cc2n1)-c1cnc2OCCNc2c1C
COc1cc2CCN(C)Cc2cc1Nc1ncc2c(N)c(F)c(cc2n1)-c1cc2oc(=O)[nH]c2cc1C
COc1cc(CS(C)(=O)=O)ccc1Nc1ncc2c(N)c(F)c(cc2n1)-c1cnc2OCCNc2c1C
COc1cc2CCN(C)Cc2cc1Nc1ncc2c(N)c(F)c(cc2n1)-c1cc(ccc1C)C#N
Cc1ccc(cc1-c1cc2nc(Nc3ccc(cc3)S(C)(=O)=O)ncc2c(N)c1F)C#N
Cc1ccc(cc1-c1cc2nc(Nc3ccc(CS(C)(=O)=O)cc3)ncc2c(N)c1F)C#N
COc1cc(ccc1Nc1ncc2c(N)c(F)c(cc2n1)-c1cnc2OCCNc2c1C)[C@@H]1CCN(C)C1=O |r|
COc1cc(ccc1Nc1ncc2c(N)c(F)c(cc2n1)-c1cnc2OCCNc2c1C)[C@H](C)S(C)(=O)=O |r|
COc1cc(ccc1Nc1ncc2c(N)c(F)c(cc2n1)-c1cnc2OCCNc2c1C)[C@@H](C)S(C)(=O)=O |r|
COc1cc(ccc1Nc1ncc2c(N)c(F)c(cc2n1)-c1cnc2OCCNc2c1C)[C@H]1CCN(C)C1=O |r|
COC1CC(C1)NC(=O)c1ccc(Nc2ncc3c(N)c(F)c(cc3n2)-c2cnc3OCCNc3c2C)cc1 |(-12.56,-18.03,;-12.56,-16.49,;-11.22,-15.72,;-10.82,-14.23,;-9.34,-14.63,;-9.73,-16.12,;-8,-13.86,;-8,-12.32,;-9.34,-11.55,;-6.67,-11.55,;-6.67,-10.01,;-5.33,-9.24,;-4,-10.01,;-2.67,-9.24,;-2.67,-7.7,;-4,-6.93,;-4,-5.39,;-2.67,-4.62,;-2.67,-3.08,;-4,-2.31,;-1.33,-2.31,;-1.33,-.77,;,-3.08,;,-4.62,;-1.33,-5.39,;-1.33,-6.93,;1.33,-2.31,;1.33,-.77,;2.67,,;4,-.77,;5.33,,;6.67,-.77,;6.67,-2.31,;5.33,-3.08,;4,-2.31,;2.67,-3.08,;2.67,-4.62,;-4,-11.55,;-5.33,-12.32,)|
CN1CCc2cc(F)c(Nc3ncc4c(N)c(F)c(cc4n3)-c3cnc4OCCNc4c3C)cc2C1
COc1cc2CCN(C)Cc2cc1Nc1ncc2c(N)c(F)c(cc2n1)-c1ccc(cc1C)-c1ncco1
COc1cc2CCN(C)Cc2cc1Nc1ncc2c(N)c(F)c(cc2n1)-c1cnc(cc1C)-c1ncco1
C[C@@H](c1ccc(Nc2ncc3c(N)c(F)c(cc3n2)-c2cnc3OCCNc3c2C)cc1)S(C)(=O)=O |r|
C[C@H](c1ccc(Nc2ncc3c(N)c(F)c(cc3n2)-c2cnc3OCCNc3c2C)cc1)S(C)(=O)=O |r|
CN1CCc2cc(Cl)c(Nc3ncc4c(N)c(F)c(cc4n3)-c3cnc4OCCNc4c3C)cc2C1
COc1cc2CCN(C)Cc2cc1Nc1ncc2c(N)c(F)c(cc2n1)-c1ccccc1-c1ccnn1C
COc1nc(C)ccc1Nc1ncc2c(N)c(F)c(cc2n1)-c1cnc2OCCNc2c1C
Cc1c2NCCOc2ncc1-c1cc2nc(Nc3ccc(cc3)N3CCOC3=O)ncc2c(N)c1F
COc1nc(ccc1Nc1ncc2c(N)c(F)c(cc2n1)-c1cnc2OCCNc2c1C)C1(CC1)C#N
COc1cc(F)ccc1Nc1ncc2c(N)c(F)c(cc2n1)-c1cnc2OCCNc2c1C
CN1CCc2ccc(Nc3ncc4c(N)c(F)c(cc4n3)-c3cnc4OCCNc4c3C)cc2C1
COc1ccccc1Nc1ncc2c(N)c(F)c(cc2n1)-c1cnc2OCCNc2c1C
COc1cc2CCN(Cc2cc1Nc1ncc2c(N)c(F)c(cc2n1)-c1cnc2OCCNc2c1C)C(C)C
CN1Cc2cc(Nc3ncc4c(N)c(F)c(cc4n3)-c3cnc4OCCNc4c3C)ccc2C2(CC2)C1
CNC(=O)c1ccc(Nc2ncc3c(N)c(F)c(cc3n2)-c2cnc3OCCNc3c2C)c(OC)c1
COc1cc2c(CN(C)CC2(C)C)cc1Nc1ncc2c(N)c(F)c(cc2n1)-c1cnc2OCCNc2c1C
CC(C)N1CCc2ccc(Nc3ncc4c(N)c(F)c(cc4n3)-c3cnc4OCCNc4c3C)cc2C1
COc1ccc(Nc2ncc3c(N)c(F)c(cc3n2)-c2cnc3OCCNc3c2C)c(C)n1
CN1Cc2cc(Nc3ncc4c(N)c(F)c(cc4n3)-c3cnc4OCCNc4c3C)ccc2C1=O
CN1CC2CC1c1cc(Nc3ncc4c(N)c(F)c(cc4n3)-c3cnc4OCCNc4c3C)ccc21
CNC(=O)C1(CCCCC1)c1ccc(Nc2ncc3c(N)c(F)c(cc3n2)-c2cnc3OCCNc3c2C)cc1
CNC(=O)C1(CC1)c1ccc(Nc2ncc3c(N)c(F)c(cc3n2)-c2cnc3OCCNc3c2C)cc1
CNC(=O)C1(CCC1)c1ccc(Nc2ncc3c(N)c(F)c(cc3n2)-c2cnc3OCCNc3c2C)cc1
CNC(=O)C1(CCCC1)c1ccc(Nc2ncc3c(N)c(F)c(cc3n2)-c2cnc3OCCNc3c2C)cc1
Cc1c2NCCOc2ncc1-c1cc2nc(Nc3ccc(CS(C)(=O)=O)nc3)ncc2c(N)c1F
C[C@H]1Cc2ccc(Nc3ncc4c(N)c(F)c(cc4n3)-c3cnc4OCCNc4c3C)cc2CN1C |r|
C[C@@H]1Cc2ccc(Nc3ncc4c(N)c(F)c(cc4n3)-c3cnc4OCCNc4c3C)cc2CN1C |r|
CN1CCc2cc(C(N)=O)c(Nc3ncc4c(N)c(F)c(cc4n3)-c3cnc4OCCNc4c3C)cc2C1
COc1cc2CN(C)CCc2cc1Nc1ncc2c(N)c(F)c(cc2n1)-c1cnc2OCCNc2c1C
CCS(=O)(=O)Cc1ccc(Nc2ncc3c(N)c(F)c(cc3n2)-c2cnc3OCCNc3c2C)c(OC)c1
COc1cc2CCN(C)Cc2cc1Nc1ncc2c(N)c(F)c(c(Cl)c2n1)-c1cnc2OCCNc2c1C |(-9,-1.94,;-7.67,-1.17,;-6.33,-1.94,;-6.33,-3.47,;-5,-4.25,;-5,-5.79,;-3.66,-6.56,;-2.33,-5.79,;-1,-6.56,;-2.33,-4.25,;-3.66,-3.48,;-3.66,-1.94,;-5,-1.17,;-5,.37,;-3.66,1.14,;-3.66,2.68,;-2.33,3.45,;-1,2.68,;.33,3.45,;.33,4.99,;1.67,2.68,;3,3.45,;1.67,1.14,;.33,.37,;.33,-1.17,;-1,1.14,;-2.33,.37,;3,.37,;4.33,1.14,;5.67,.37,;5.67,-1.17,;7,-1.94,;7,-3.48,;5.67,-4.25,;4.34,-3.48,;4.33,-1.94,;3,-1.17,;1.67,-1.94,)|
Cc1c2NCCOc2ncc1-c1c(F)c(N)c2cnc(Nc3ccc(CS(C)(=O)=O)cc3)nc2c1Cl |(1.67,-1.94,;3,-1.17,;4.33,-1.94,;4.34,-3.48,;5.67,-4.25,;7,-3.48,;7,-1.94,;5.67,-1.17,;5.67,.37,;4.33,1.14,;3,.37,;1.67,1.14,;1.67,2.68,;3,3.45,;.33,3.45,;.33,4.99,;-1,2.68,;-2.33,3.45,;-3.66,2.68,;-3.66,1.14,;-5,.37,;-5,-1.17,;-6.33,-1.94,;-6.33,-3.47,;-5,-4.25,;-5,-5.79,;-3.66,-6.56,;-2.33,-5.79,;-3.66,-8.1,;-3.66,-5.02,;-3.66,-3.48,;-3.66,-1.94,;-2.33,.37,;-1,1.14,;.33,.37,;.33,-1.17,)|
CN1CCc2ccc(Nc3ncc4c(N)c(F)c(c(Cl)c4n3)-c3cnc4OCCNc4c3C)cc2C1 |(-1,-6.56,;-2.33,-5.79,;-3.66,-6.56,;-5,-5.79,;-5,-4.25,;-6.33,-3.47,;-6.33,-1.94,;-5,-1.17,;-5,.37,;-3.66,1.14,;-3.66,2.68,;-2.33,3.45,;-1,2.68,;.33,3.45,;.33,4.99,;1.67,2.68,;3,3.45,;1.67,1.14,;.33,.37,;.33,-1.17,;-1,1.14,;-2.33,.37,;3,.37,;4.33,1.14,;5.67,.37,;5.67,-1.17,;7,-1.94,;7,-3.48,;5.67,-4.25,;4.34,-3.48,;4.33,-1.94,;3,-1.17,;1.67,-1.94,;-3.66,-1.94,;-3.66,-3.48,;-2.33,-4.25,)|
CC(C)N1CCc2ccc(Nc3ncc4c(N)c(F)c(c(Cl)c4n3)-c3cnc4OCCNc4c3C)cc2C1 |(-1,-8.1,;-1,-6.56,;.34,-5.79,;-2.33,-5.79,;-3.66,-6.56,;-5,-5.79,;-5,-4.25,;-6.33,-3.47,;-6.33,-1.94,;-5,-1.17,;-5,.37,;-3.66,1.14,;-3.66,2.68,;-2.33,3.45,;-1,2.68,;.33,3.45,;.33,4.99,;1.67,2.68,;3,3.45,;1.67,1.14,;.33,.37,;.33,-1.17,;-1,1.14,;-2.33,.37,;3,.37,;4.33,1.14,;5.67,.37,;5.67,-1.17,;7,-1.94,;7,-3.48,;5.67,-4.25,;4.34,-3.48,;4.33,-1.94,;3,-1.17,;1.67,-1.94,;-3.66,-1.94,;-3.66,-3.48,;-2.33,-4.25,)|
CNC(=O)c1ccc(Nc2ncc3c(N)c(F)c(c(Cl)c3n2)-c2cnc3OCCNc3c2C)c(OC)c1 |(-7.67,-5.79,;-6.33,-6.56,;-5,-5.79,;-3.66,-6.56,;-5,-4.25,;-3.66,-3.48,;-3.66,-1.94,;-5,-1.17,;-5,.37,;-3.66,1.14,;-3.66,2.68,;-2.33,3.45,;-1,2.68,;.33,3.45,;.33,4.99,;1.67,2.68,;3,3.45,;1.67,1.14,;.33,.37,;.33,-1.17,;-1,1.14,;-2.33,.37,;3,.37,;4.33,1.14,;5.67,.37,;5.67,-1.17,;7,-1.94,;7,-3.48,;5.67,-4.25,;4.34,-3.48,;4.33,-1.94,;3,-1.17,;1.67,-1.94,;-6.33,-1.94,;-7.67,-1.17,;-9,-1.94,;-6.33,-3.47,)|
COc1cc(CS(C)(=O)=O)ccc1Nc1ncc2c(N)c(F)c(c(Cl)c2n1)-c1cnc2OCCNc2c1C |(-9,-1.94,;-7.67,-1.17,;-6.33,-1.94,;-6.33,-3.47,;-5,-4.25,;-5,-5.79,;-6.33,-6.56,;-7.67,-5.79,;-6.33,-8.1,;-5,-7.33,;-3.66,-3.48,;-3.66,-1.94,;-5,-1.17,;-5,.37,;-3.66,1.14,;-3.66,2.68,;-2.33,3.45,;-1,2.68,;.33,3.45,;.33,4.99,;1.67,2.68,;3,3.45,;1.67,1.14,;.33,.37,;.33,-1.17,;-1,1.14,;-2.33,.37,;3,.37,;4.33,1.14,;5.67,.37,;5.67,-1.17,;7,-1.94,;7,-3.48,;5.67,-4.25,;4.34,-3.48,;4.33,-1.94,;3,-1.17,;1.67,-1.94,)|
CN1Cc2cc(Nc3ncc4c(N)c(F)c(c(Cl)c4n3)-c3cnc4OCCNc4c3C)ccc2C2(CC2)C1 |(-1,-6.56,;-2.33,-5.79,;-2.33,-4.25,;-3.66,-3.48,;-3.66,-1.94,;-5,-1.17,;-5,.37,;-3.66,1.14,;-3.66,2.68,;-2.33,3.45,;-1,2.68,;.33,3.45,;.33,4.99,;1.67,2.68,;3,3.45,;1.67,1.14,;.33,.37,;.33,-1.17,;-1,1.14,;-2.33,.37,;3,.37,;4.33,1.14,;5.67,.37,;5.67,-1.17,;7,-1.94,;7,-3.48,;5.67,-4.25,;4.34,-3.48,;4.33,-1.94,;3,-1.17,;1.67,-1.94,;-6.33,-1.94,;-6.33,-3.47,;-5,-4.25,;-5,-5.79,;-6.53,-5.95,;-5.47,-7.25,;-3.66,-6.56,)|
Cc1c2NCCOc2ncc1-c1c(F)c(N)c2cnc(Nc3ccc(cc3)S(C)(=O)=O)nc2c1Cl |(1.67,-1.94,;3,-1.17,;4.33,-1.94,;4.34,-3.48,;5.67,-4.25,;7,-3.48,;7,-1.94,;5.67,-1.17,;5.67,.37,;4.33,1.14,;3,.37,;1.67,1.14,;1.67,2.68,;3,3.45,;.33,3.45,;.33,4.99,;-1,2.68,;-2.33,3.45,;-3.66,2.68,;-3.66,1.14,;-5,.37,;-5,-1.17,;-6.33,-1.94,;-6.33,-3.47,;-5,-4.25,;-3.66,-3.48,;-3.66,-1.94,;-5,-5.79,;-5,-7.33,;-6.33,-6.56,;-3.66,-6.56,;-2.33,.37,;-1,1.14,;.33,.37,;.33,-1.17,)|
COc1cc2c(CN(C)CC2(C)C)cc1Nc1ncc2c(N)c(F)c(c(Cl)c2n1)-c1cnc2OCCNc2c1C |(-9,-1.94,;-7.67,-1.17,;-6.33,-1.94,;-6.33,-3.47,;-5,-4.25,;-3.66,-3.48,;-2.33,-4.25,;-2.33,-5.79,;-1,-6.56,;-3.66,-6.56,;-5,-5.79,;-6.33,-6.55,;-5,-7.33,;-3.66,-1.94,;-5,-1.17,;-5,.37,;-3.66,1.14,;-3.66,2.68,;-2.33,3.45,;-1,2.68,;.33,3.45,;.33,4.99,;1.67,2.68,;3,3.45,;1.67,1.14,;.33,.37,;.33,-1.17,;-1,1.14,;-2.33,.37,;3,.37,;4.33,1.14,;5.67,.37,;5.67,-1.17,;7,-1.94,;7,-3.48,;5.67,-4.25,;4.34,-3.48,;4.33,-1.94,;3,-1.17,;1.67,-1.94,)|
COc1cc2CCN(Cc2cc1Nc1ncc2c(N)c(F)c(c(Cl)c2n1)-c1cnc2OCCNc2c1C)C(C)C |(-9,-1.94,;-7.67,-1.17,;-6.33,-1.94,;-6.33,-3.47,;-5,-4.25,;-5,-5.79,;-3.66,-6.56,;-2.33,-5.79,;-2.33,-4.25,;-3.66,-3.48,;-3.66,-1.94,;-5,-1.17,;-5,.37,;-3.66,1.14,;-3.66,2.68,;-2.33,3.45,;-1,2.68,;.33,3.45,;.33,4.99,;1.67,2.68,;3,3.45,;1.67,1.14,;.33,.37,;.33,-1.17,;-1,1.14,;-2.33,.37,;3,.37,;4.33,1.14,;5.67,.37,;5.67,-1.17,;7,-1.94,;7,-3.48,;5.67,-4.25,;4.34,-3.48,;4.33,-1.94,;3,-1.17,;1.67,-1.94,;-1,-6.56,;-1,-8.1,;.34,-5.79,)|
CN1CCc2cc(F)c(Nc3ncc4c(N)c(F)c(c(Cl)c4n3)-c3cnc4OCCNc4c3C)cc2C1 |(-1,-6.56,;-2.33,-5.79,;-3.66,-6.56,;-5,-5.79,;-5,-4.25,;-6.33,-3.47,;-6.33,-1.94,;-7.67,-1.17,;-5,-1.17,;-5,.37,;-3.66,1.14,;-3.66,2.68,;-2.33,3.45,;-1,2.68,;.33,3.45,;.33,4.99,;1.67,2.68,;3,3.45,;1.67,1.14,;.33,.37,;.33,-1.17,;-1,1.14,;-2.33,.37,;3,.37,;4.33,1.14,;5.67,.37,;5.67,-1.17,;7,-1.94,;7,-3.48,;5.67,-4.25,;4.34,-3.48,;4.33,-1.94,;3,-1.17,;1.67,-1.94,;-3.66,-1.94,;-3.66,-3.48,;-2.33,-4.25,)|
CN1Cc2cc(Nc3ncc4c(N)c(F)c(c(Cl)c4n3)-c3cnc4OCCNc4c3C)ccc2C2(CC2)C1 |(-1,-6.56,;-2.33,-5.79,;-2.33,-4.25,;-3.66,-3.48,;-3.66,-1.94,;-5,-1.17,;-5,.37,;-3.66,1.14,;-3.66,2.68,;-2.33,3.45,;-1,2.68,;.33,3.45,;.33,4.99,;1.67,2.68,;3,3.45,;1.67,1.14,;.33,.37,;.33,-1.17,;-1,1.14,;-2.33,.37,;3,.37,;4.33,1.14,;5.67,.37,;5.67,-1.17,;7,-1.94,;7,-3.48,;5.67,-4.25,;4.34,-3.48,;4.33,-1.94,;3,-1.17,;1.67,-1.94,;-6.33,-1.94,;-6.33,-3.47,;-5,-4.25,;-5,-5.79,;-6.5,-6.11,;-5.47,-7.25,;-3.66,-6.56,)|
CN1Cc2cc(Nc3ncc4c(N)c(F)c(-c5cnc6OCCNc6c5C)c(C#N)c4n3)ccc2C2(CC2)C1 |(-1,-6.56,;-2.33,-5.79,;-2.33,-4.25,;-3.66,-3.48,;-3.66,-1.94,;-5,-1.17,;-5,.37,;-3.66,1.14,;-3.66,2.68,;-2.33,3.45,;-1,2.68,;.33,3.45,;.33,4.99,;1.67,2.68,;3,3.45,;1.67,1.14,;3,.37,;4.33,1.14,;5.67,.37,;5.67,-1.17,;7,-1.94,;7,-3.48,;5.67,-4.25,;4.34,-3.48,;4.33,-1.94,;3,-1.17,;1.67,-1.94,;.33,.37,;.33,-1.17,;.33,-2.71,;-1,1.14,;-2.33,.37,;-6.33,-1.94,;-6.33,-3.47,;-5,-4.25,;-5,-5.79,;-6.5,-6.11,;-5.47,-7.25,;-3.66,-6.56,)|
CN1Cc2cc(Nc3ncc4c(N)c(F)c(c(C)c4n3)-c3cnc4OCCNc4c3C)ccc2C2(CC2)C1 |(-1,-6.56,;-2.33,-5.79,;-2.33,-4.25,;-3.66,-3.48,;-3.66,-1.94,;-5,-1.17,;-5,.37,;-3.66,1.14,;-3.66,2.68,;-2.33,3.45,;-1,2.68,;.33,3.45,;.33,4.99,;1.67,2.68,;3,3.45,;1.67,1.14,;.33,.37,;.33,-1.17,;-1,1.14,;-2.33,.37,;3,.37,;4.33,1.14,;5.67,.37,;5.67,-1.17,;7,-1.94,;7,-3.48,;5.67,-4.25,;4.34,-3.48,;4.33,-1.94,;3,-1.17,;1.67,-1.94,;-6.33,-1.94,;-6.33,-3.47,;-5,-4.25,;-5,-5.79,;-6.5,-6.11,;-5.47,-7.25,;-3.66,-6.56,)|
CN1Cc2cc(Nc3ncc4c(N)c(F)c(c(Br)c4n3)-c3cnc4OCCNc4c3C)ccc2C2(CC2)C1 |(-1,-6.56,;-2.33,-5.79,;-2.33,-4.25,;-3.66,-3.48,;-3.66,-1.94,;-5,-1.17,;-5,.37,;-3.66,1.14,;-3.66,2.68,;-2.33,3.45,;-1,2.68,;.33,3.45,;.33,4.99,;1.67,2.68,;3,3.45,;1.67,1.14,;.33,.37,;.33,-1.17,;-1,1.14,;-2.33,.37,;3,.37,;4.33,1.14,;5.67,.37,;5.67,-1.17,;7,-1.94,;7,-3.48,;5.67,-4.25,;4.34,-3.48,;4.33,-1.94,;3,-1.17,;1.67,-1.94,;-6.33,-1.94,;-6.33,-3.47,;-5,-4.25,;-5,-5.79,;-6.5,-6.11,;-5.47,-7.25,;-3.66,-6.56,)|
Cc1c2NCCOc2ncc1-c1cc2nc(Nc3ccc(CS(=O)(=O)N4CCCC4)cc3)ncc2c(N)c1F
Cc1c2NCCOc2ncc1-c1cc2nc(Nc3ccc(CCC#N)cc3)ncc2c(N)c1F
CN1CCCc2ccc(Nc3ncc4c(N)c(F)c(cc4n3)-c3cnc4OCCNc4c3C)cc2C1
Cc1c2NCCOc2ncc1-c1cc2nc(Nc3ccc4CCOCc4c3)ncc2c(N)c1F
CN1CCc2ccc(Nc3ncc4c(N)c(F)c(cc4n3)-c3cnc4OCCNc4c3C)cc2CC1
Cc1c2NCCOc2ncc1-c1cc2nc(Nc3ccc4CCCNCc4c3)ncc2c(N)c1F
CN1C2CCC1c1cc(Nc3ncc4c(N)c(F)c(cc4n3)-c3cnc4OCCNc4c3C)ccc21 |TLB:0:1:35.6:3.4|
CN1CCc2ccc(Nc3ncc4c(N)c(F)c(cc4n3)-c3cnccc3C)cc2C1
CN1CCc2ccc(Nc3ncc4c(N)c(F)c(cc4n3)-c3cnc4OCCNc4c3Cl)cc2C1
CCS(=O)(=O)Cc1ccc(Nc2ncc3c(N)c(F)c(cc3n2)-c2cnc3OCCNc3c2C)c(F)c1
CN1Cc2ccc(Nc3ncc4c(N)c(F)c(cc4n3)-c3cnc4OCCNc4c3C)cc2CC1(C)C
CN1Cc2cccc(Nc3ncc4c(N)c(F)c(cc4n3)-c3cnc4OCCNc4c3C)c2CC1(C)C
CN1Cc2cc(Nc3ncc4c(N)c(F)c(cc4n3)-c3cnc4OCCNc4c3C)ccc2CC1(C)C
CN1CCc2ccc(Nc3ncc4c(N)c(F)c(cc4n3)-c3cnc4cc[nH]c4c3C)cc2C1
Cc1c2NCCOc2ncc1-c1c(F)c(N)c2cnc(Nc3ccc(CS(C)(=O)=O)cc3F)nc2c1Cl |(1.67,-1.94,;3,-1.17,;4.33,-1.94,;4.34,-3.48,;5.67,-4.25,;7,-3.48,;7,-1.94,;5.67,-1.17,;5.67,.37,;4.33,1.14,;3,.37,;1.67,1.14,;1.67,2.68,;3,3.45,;.33,3.45,;.33,4.99,;-1,2.68,;-2.33,3.45,;-3.66,2.68,;-3.66,1.14,;-5,.37,;-5,-1.17,;-3.66,-1.94,;-3.66,-3.48,;-5,-4.25,;-5,-5.79,;-3.66,-6.56,;-2.33,-5.79,;-3.66,-8.1,;-2.33,-7.33,;-6.33,-3.47,;-6.33,-1.94,;-7.67,-1.17,;-2.33,.37,;-1,1.14,;.33,.37,;.33,-1.17,)|
Cc1c2NCCOc2ncc1-c1c(F)c(N)c2cnc(Nc3ccc(CS(=O)(=O)C4CC4)cc3)nc2c1Cl |(1.67,-1.94,;3,-1.17,;4.33,-1.94,;4.34,-3.48,;5.67,-4.25,;7,-3.48,;7,-1.94,;5.67,-1.17,;5.67,.37,;4.33,1.14,;3,.37,;1.67,1.14,;1.67,2.68,;3,3.45,;.33,3.45,;.33,4.99,;-1,2.68,;-2.33,3.45,;-3.66,2.68,;-3.66,1.14,;-5,.37,;-5,-1.17,;-6.33,-1.94,;-6.33,-3.47,;-5,-4.25,;-5,-5.79,;-3.66,-6.56,;-3.66,-8.1,;-2.33,-7.33,;-2.33,-5.79,;-1.43,-4.54,;-.79,-5.79,;-3.66,-3.48,;-3.66,-1.94,;-2.33,.37,;-1,1.14,;.33,.37,;.33,-1.17,)|
CC(C)S(=O)(=O)Cc1ccc(Nc2ncc3c(N)c(F)c(c(Cl)c3n2)-c2cnc3OCCNc3c2C)cc1 |(-2.33,-4.25,;-2.33,-5.79,;-1,-6.56,;-3.66,-6.56,;-3.66,-8.1,;-2.33,-7.33,;-5,-5.79,;-5,-4.25,;-6.33,-3.47,;-6.33,-1.94,;-5,-1.17,;-5,.37,;-3.66,1.14,;-3.66,2.68,;-2.33,3.45,;-1,2.68,;.33,3.45,;.33,4.99,;1.67,2.68,;3,3.45,;1.67,1.14,;.33,.37,;.33,-1.17,;-1,1.14,;-2.33,.37,;3,.37,;4.33,1.14,;5.67,.37,;5.67,-1.17,;7,-1.94,;7,-3.48,;5.67,-4.25,;4.34,-3.48,;4.33,-1.94,;3,-1.17,;1.67,-1.94,;-3.66,-1.94,;-3.66,-3.48,)|
CCS(=O)(=O)Cc1ccc(Nc2ncc3c(N)c(F)c(c(Cl)c3n2)-c2cnc3OCCNc3c2C)cc1 |(-2.33,-4.25,;-2.33,-5.79,;-3.66,-6.56,;-3.66,-8.1,;-2.33,-7.33,;-5,-5.79,;-5,-4.25,;-6.33,-3.47,;-6.33,-1.94,;-5,-1.17,;-5,.37,;-3.66,1.14,;-3.66,2.68,;-2.33,3.45,;-1,2.68,;.33,3.45,;.33,4.99,;1.67,2.68,;3,3.45,;1.67,1.14,;.33,.37,;.33,-1.17,;-1,1.14,;-2.33,.37,;3,.37,;4.33,1.14,;5.67,.37,;5.67,-1.17,;7,-1.94,;7,-3.48,;5.67,-4.25,;4.34,-3.48,;4.33,-1.94,;3,-1.17,;1.67,-1.94,;-3.66,-1.94,;-3.66,-3.48,)|
Cc1c2NCCOc2ncc1-c1cc2nc(Nc3ccc(CS(=O)(=O)C4CC4)cc3)ncc2c(N)c1F
Cc1c2NCCOc2ncc1-c1cc2nc(Nc3ccc4CS(=O)(=O)CCc4c3)ncc2c(N)c1F
CN1CCc2ccc(Nc3ncc4c(N)c(F)c(cc4n3)-c3cncc4[nH]ccc34)cc2C1
CC1CNc2c(C)c(cnc2O1)-c1cc2nc(Nc3ccc4CCN(C)Cc4c3)ncc2c(N)c1F
CN1CCc2cnc(Nc3ncc4c(N)c(F)c(cc4n3)-c3cnc4OCCNc4c3C)cc2C1
CCS(=O)(=O)Cc1ccc(Nc2ncc3c(N)c(F)c(cc3n2)-c2cnc3OC(C)(C)CNc3c2C)c(F)c1
CC(C)N1CCc2ccc(Nc3ncc4c(N)c(F)c(cc4n3)-c3cnc4OC(C)CNc4c3C)cc2C1
CN1CC[C@H](C1=O)c1ccc(Nc2ncc3c(N)c(F)c(cc3n2)-c2cnc3OCCNc3c2C)cc1 |r|
CN1CC[C@@H](C1=O)c1ccc(Nc2ncc3c(N)c(F)c(cc3n2)-c2cnc3OCCNc3c2C)cc1 |r|
Cc1c2NCCOc2ncc1-c1cc2nc(Nc3ccc(cc3)C3(CC3)S(C)(=O)=O)ncc2c(N)c1F
Cc1c2NCCOc2ncc1-c1cc2nc(Nc3ccc(CS(=O)(=O)CC(F)(F)F)cc3)ncc2c(N)c1F
CN1Cc2cc(Nc3ncc4c(N)c(F)c(cc4n3)-c3cnc4OCCNc4c3C)ccc2C(C)(C)C1
CN1Cc2cc(Nc3ncc4c(N)c(F)c(cc4n3)-c3cnc4OCCNc4c3Cl)ccc2C2(CC2)C1
CN1Cc2cc(Nc3ncc4c(N)c(F)c(cc4n3)-c3cncc(N)c3C)ccc2C2(CC2)C1
CN1Cc2cc(Nc3ncc4c(N)c(F)c(cc4n3)-c3cnc4OCCNc4c3C)ccc2C(F)(F)C1
Cc1c2NCCOc2ncc1-c1cc2nc(Nc3ccc(CS(C)(=O)=O)cc3F)ncc2c(N)c1F
Cc1c2NCCOc2ncc1-c1c(F)c(N)c2cnc(Nc3ccc(cc3)N3CCOC3=O)nc2c1Cl |(1.67,-1.94,;3,-1.17,;4.33,-1.94,;4.34,-3.48,;5.67,-4.25,;7,-3.48,;7,-1.94,;5.67,-1.17,;5.67,.37,;4.33,1.14,;3,.37,;1.67,1.14,;1.67,2.68,;3,3.45,;.33,3.45,;.33,4.99,;-1,2.68,;-2.33,3.45,;-3.66,2.68,;-3.66,1.14,;-5,.37,;-5,-1.17,;-6.33,-1.94,;-6.33,-3.47,;-5,-4.25,;-3.66,-3.48,;-3.66,-1.94,;-5,-5.79,;-6.24,-6.69,;-5.77,-8.16,;-4.23,-8.16,;-3.75,-6.69,;-2.29,-6.21,;-2.33,.37,;-1,1.14,;.33,.37,;.33,-1.17,)|
CC(C)S(=O)(=O)Cc1ccc(Nc2ncc3c(N)c(F)c(cc3n2)-c2cnc3OCCNc3c2C)cc1
CN1CCc2cc(Nc3ncc4c(N)c(F)c(cc4n3)-c3cnc4OCCNc4c3C)ccc2C1
Cc1c2NCC(C)(C)Oc2ncc1-c1c(F)c(N)c2cnc(Nc3ccc(CS(C)(=O)=O)cc3)nc2c1Cl |(1.67,-1.94,;3,-1.17,;4.33,-1.94,;4.34,-3.48,;5.67,-4.25,;7,-3.48,;8.34,-4.25,;7,-5.02,;7,-1.94,;5.67,-1.17,;5.67,.37,;4.33,1.14,;3,.37,;1.67,1.14,;1.67,2.68,;3,3.45,;.33,3.45,;.33,4.99,;-1,2.68,;-2.33,3.45,;-3.66,2.68,;-3.66,1.14,;-5,.37,;-5,-1.17,;-6.33,-1.94,;-6.33,-3.47,;-5,-4.25,;-5,-5.79,;-3.66,-6.56,;-2.33,-5.79,;-3.66,-8.1,;-3.66,-5.02,;-3.66,-3.48,;-3.66,-1.94,;-2.33,.37,;-1,1.14,;.33,.37,;.33,-1.17,)|
CN1CCc2ccc(Nc3ncc4c(N)c(F)c(cc4n3)-c3cnc4nc[nH]c4c3C)cc2C1
COc1cc2c(CN(C)CC22CC2)cc1Nc1ncc2c(N)c(F)c(c(Cl)c2n1)-c1cnc2OCCNc2c1C |(-9,-1.94,;-7.67,-1.17,;-6.33,-1.94,;-6.33,-3.47,;-5,-4.25,;-3.66,-3.48,;-2.33,-4.25,;-2.33,-5.79,;-1,-6.56,;-3.66,-6.56,;-5,-5.79,;-6.33,-6.56,;-5,-7.33,;-3.66,-1.94,;-5,-1.17,;-5,.37,;-3.66,1.14,;-3.66,2.68,;-2.33,3.45,;-1,2.68,;.33,3.45,;.33,4.99,;1.67,2.68,;3,3.45,;1.67,1.14,;.33,.37,;.33,-1.17,;-1,1.14,;-2.33,.37,;3,.37,;4.33,1.14,;5.67,.37,;5.67,-1.17,;7,-1.94,;7,-3.48,;5.67,-4.25,;4.34,-3.48,;4.33,-1.94,;3,-1.17,;1.67,-1.94,)|
Cc1c2NCCOc2ncc1-c1c(F)c(N)c2cnc(Nc3ccc(CC(C)(C)O)cc3)nc2c1Cl |(1.67,-1.94,;3,-1.17,;4.33,-1.94,;4.34,-3.48,;5.67,-4.25,;7,-3.48,;7,-1.94,;5.67,-1.17,;5.67,.37,;4.33,1.14,;3,.37,;1.67,1.14,;1.67,2.68,;3,3.45,;.33,3.45,;.33,4.99,;-1,2.68,;-2.33,3.45,;-3.66,2.68,;-3.66,1.14,;-5,.37,;-5,-1.17,;-6.33,-1.94,;-6.33,-3.47,;-5,-4.25,;-5,-5.79,;-6.33,-6.56,;-6.33,-8.1,;-5,-7.33,;-7.67,-5.79,;-3.66,-3.48,;-3.66,-1.94,;-2.33,.37,;-1,1.14,;.33,.37,;.33,-1.17,)|
Cc1c2NCC(C)(C)Oc2ncc1-c1cc2nc(Nc3ccc(CS(C)(=O)=O)cc3)ncc2c(N)c1F
CN1CCc2ccc(Nc3ncc4c(N)c(F)c(cc4n3)-c3cnc4OC(C)(C)CNc4c3C)cc2C1
Cc1c2NCCOc2ncc1-c1c(F)c(N)c2cnc(Nc3ccc(CC(C)(C)O)cc3)nc2c1Cl |(1.67,-1.94,;3,-1.17,;4.33,-1.94,;4.34,-3.48,;5.67,-4.25,;7,-3.48,;7,-1.94,;5.67,-1.17,;5.67,.37,;4.33,1.14,;3,.37,;1.67,1.14,;1.67,2.68,;3,3.45,;.33,3.45,;.33,4.99,;-1,2.68,;-2.33,3.45,;-3.66,2.68,;-3.66,1.14,;-5,.37,;-5,-1.17,;-6.33,-1.94,;-6.33,-3.47,;-5,-4.25,;-5,-5.79,;-3.66,-6.56,;-3.66,-8.1,;-3.66,-5.02,;-2.33,-5.79,;-3.66,-3.48,;-3.66,-1.94,;-2.33,.37,;-1,1.14,;.33,.37,;.33,-1.17,)|
COc1cc(CS(=O)(=O)C(C)C)ccc1Nc1ncc2c(N)c(F)c(cc2n1)-c1cnc2OC(C)(C)CNc2c1C
Cc1c2NCCOc2ncc1-c1cc2nc(Nc3ccc(cc3)S(C)=O)ncc2c(N)c1F
CC(C)N1CCc2cc(F)c(Nc3ncc4c(N)c(F)c(cc4n3)-c3cnc4OCCNc4c3C)cc2C1
Cc1ccc(F)cc1-c1cc2nc(Nc3ccc(CS(C)(=O)=O)cc3)ncc2c(N)c1F
CCc1ccc(Nc2ncc3c(N)c(F)c(cc3n2)-c2cnc3OCCNc3c2C)cn1
CN1CCc2ccc(Nc3ncc4c(N)c(F)c(cc4n3)-c3cc(F)ccc3C)cc2C1
CC(C)N1CCc2ncc(Nc3ncc4c(N)c(F)c(cc4n3)-c3cnc4OCCNc4c3C)cc2C1
COc1cc(ccc1Nc1ncc2c(N)c(F)c(cc2n1)-c1cnc2OCCNc2c1C)C1CC1
COc1cc(C)ccc1Nc1ncc2c(N)c(F)c(cc2n1)-c1cnc2OCCNc2c1C
Cc1c2NCCOc2ncc1-c1cc2nc(Nc3ccc(CC(C)(C)O)cc3)ncc2c(N)c1F
COc1nc(ccc1Nc1ncc2c(N)c(F)c(c(Cl)c2n1)-c1cnc2OCCNc2c1C)C1(CC1)C#N |(-9,-1.94,;-7.67,-1.17,;-6.33,-1.94,;-6.33,-3.47,;-5,-4.25,;-3.66,-3.48,;-3.66,-1.94,;-5,-1.17,;-5,.37,;-3.66,1.14,;-3.66,2.68,;-2.33,3.45,;-1,2.68,;.33,3.45,;.33,4.99,;1.67,2.68,;3,3.45,;1.67,1.14,;.33,.37,;.33,-1.17,;-1,1.14,;-2.33,.37,;3,.37,;4.33,1.14,;5.67,.37,;5.67,-1.17,;7,-1.94,;7,-3.48,;5.67,-4.25,;4.34,-3.48,;4.33,-1.94,;3,-1.17,;1.67,-1.94,;-5,-5.79,;-6.46,-6.26,;-5.32,-7.29,;-3.47,-5.95,;-1.93,-6.11,)|
CN1CCc2ncc(Nc3ncc4c(N)c(F)c(cc4n3)-c3cnc4OCCNc4c3C)cc2C1
CNC(=O)C(F)(F)c1ccc(Nc2ncc3c(N)c(F)c(cc3n2)-c2cnc3OCCNc3c2C)cc1
CNC(=O)C(C)(C)c1ccc(Nc2ncc3c(N)c(F)c(cc3n2)-c2cnc3OCCNc3c2C)cc1
CNC(=O)C1CCc2cc(Nc3ncc4c(N)c(F)c(cc4n3)-c3cnc4OCCNc4c3C)ccc12
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(cc2n1)N1CCCC1=O
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(cc2n1)N1[C@@H](C)COC1=O |r|
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(cc2n1)N1CC2(CCOC2)OC1=O
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(cc2n1)N1CC(CO)OC1=O
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(cc2n1)N1CC2(CCCNCC2)OC1=O
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(cc2n1)N1C(=O)OCC1(C)C
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(cc2n1)N1CC(C)(CO)OC1=O
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(cc2n1)N1CC(OC1=O)C(C)(C)O
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(cc2n1)N1[C@@H](COC1=O)C(C)C |r|
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(cc2n1)N1CC(CN)OC1=O
CNCC1CN(C(=O)O1)c1ccc2cnc(Nc3cc4CN(C)CCc4cc3OC)nc2c1
CC[C@@H]1COC(=O)N1c1ccc2cnc(Nc3cc4CN(C)CCc4cc3OC)nc2c1 |r|
CC[C@H]1COC(=O)N1c1ccc2cnc(Nc3cc4CN(C)CCc4cc3OC)nc2c1 |r|
CC[C@@H]1COC(=O)N1c1cc(N)c2cnc(Nc3cc4CN(C)CCc4cc3OC)nc2c1 |r|
CC[C@H]1COC(=O)N1c1cc(N)c2cnc(Nc3cc4CN(C)CCc4cc3OC)nc2c1 |r|
COc1cc2CCN(C)Cc2cc1Nc1ncc2c(N)cc(cc2n1)N1[C@@H](C)COC1=O |r|
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(NCC3=NS(=O)(=O)c4cc(C)ccc4N3)cc2n1 |t:25|
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(cc2n1)-n1nc(C)nc1C1CCCN1
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(cc2n1)N1CCCC(CN2CCCC2=O)C1
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(Nc3ccc4CCNC(=O)c4c3)cc2n1
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(N[C@H]3CCN(C3)C(=O)C3CC3)cc2n1 |r|
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(Nc3ccc4CN(C)C(=O)c4c3)cc2n1
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(Nc3cc(ccc3C)S(C)(=O)=O)cc2n1
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(NCc3ccc4NC(C)=NS(=O)(=O)c4c3)cc2n1 |c:31|
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(NCC3CNC(=O)O3)cc2n1
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(Nc3cccc(n3)C#N)cc2n1
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(NCc3ccc4CNC(=O)c4c3)cc2n1
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(Nc3cccc(CO)n3)cc2n1
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(cc2n1)N(C)CC1CNC(=O)O1
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(Nc3cccc(CO)c3)cc2n1
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(Nc3ccc4CCN(C(C)=O)c4c3)cc2n1
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(Nc3cccc(c3)S(C)(=O)=O)cc2n1
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(Nc3cccc(c3)C(=O)N(C)C)cc2n1
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(Nc3nccc(CO)n3)cc2n1
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(Nc3nc(ccc3F)S(C)(=O)=O)cc2n1
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(NCC3CCS(=O)(=O)C3)cc2n1
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(NC3CCN(CC3)C(C)=O)cc2n1
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(NC3CCCC(O)C3)cc2n1
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(Nc3cc(CO)ccn3)cc2n1
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(Nc3cc(ccn3)C(N)=O)cc2n1
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(Nc3cc(c(C)cc3C)S(C)(=O)=O)cc2n1
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(Nc3cccc(c3)N3CCN(C)C3=O)cc2n1
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(Nc3ccc(C)c(c3)S(N)(=O)=O)cc2n1
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(NCC3CCC(=O)N3)cc2n1
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(N[C@@H]3CC[C@H](O)CC3)cc2n1 |r,wU:22.23,25.27,(-9,-1.94,;-7.67,-1.17,;-6.33,-1.94,;-6.33,-3.47,;-5,-4.25,;-5,-5.79,;-3.66,-6.56,;-2.33,-5.79,;-1,-6.56,;-2.33,-4.25,;-3.66,-3.48,;-3.66,-1.94,;-5,-1.17,;-5,.37,;-3.66,1.14,;-3.66,2.68,;-2.33,3.45,;-1,2.68,;.33,3.45,;1.67,2.68,;1.67,1.14,;3,.37,;4.33,1.14,;5.67,.37,;7,1.14,;7,2.68,;8.33,3.45,;5.67,3.45,;4.33,2.68,;.33,.37,;-1,1.14,;-2.33,.37,)|
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(N[C@H]3CCCOCC3)cc2n1
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(NC[C@@H]3CN(C)C(=O)C3)cc2n1 |r|
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(NC3CCN(C)C3=O)cc2n1
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(cc2n1)N1CCC[C@@H](C1)N1CCOC1=O |r|
COC1CC(C1)Nc1ccc2cnc(Nc3cc4CN(C)CCc4cc3OC)nc2c1 |(-6.67,1.41,;-5.33,.64,;-5.33,-.9,;-4.25,-1.99,;-5.33,-3.08,;-6.42,-1.99,;-5.33,-4.62,;-4,-5.39,;-4,-6.93,;-2.67,-7.7,;-1.33,-6.93,;,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;1.33,-.77,;;,1.54,;-1.33,2.31,;1.33,2.31,;2.67,1.54,;2.67,,;4,-.77,;4,-2.31,;5.33,-3.08,;5.33,-4.62,;,-4.62,;-1.33,-5.39,;-2.67,-4.62,)|
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(NCc3noc(C)n3)cc2n1
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(cc2n1)N1CC(C1)C(N)=O
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(cc2n1)N1CC(O)(C1)C(F)(F)F
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(NC3(C)COC3)cc2n1
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(cc2n1)N1CCn2c(C)nnc2C1
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(N[C@H]3CCC[C@@H]3O)cc2n1 |r|
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(NC[C@H]3CN(C)C(=O)C3)cc2n1 |r|
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(cc2n1)N1CC2CCS(=O)(=O)C2C1
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(NC3(CCC3)C(=O)N(C)C)cc2n1
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(NCC3(C)CCC3)cc2n1
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(NCc3cnsn3)cc2n1
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(NCC(=O)N3CCOCC3)cc2n1
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(NCC(=O)N3CCCC3)cc2n1
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(NC3(CC3)C(=O)N(C)C)cc2n1
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(N[C@@H]3COC[C@@H]3F)cc2n1 |r|
COCC1CN(C1)c1ccc2cnc(Nc3cc4CN(C)CCc4cc3OC)nc2c1
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(NC3CCCOC3)cc2n1
CNC(=O)CNc1ccc2cnc(Nc3cc4CN(C)CCc4cc3OC)nc2c1
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(NCC(=O)N(C)C)cc2n1
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(NCc3cc(C)n(C)n3)cc2n1
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(cc2n1)N1CCN(C2CC2)C(=O)C1
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(NC3C4COCC34)cc2n1
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(NCC3(C)CCOC3)cc2n1
COc1cc(ccc1Nc1ncc2c(N)cc(cc2n1)N1[C@H](C)COC1=O)S(C)(=O)=O |r|
COc1cc(CS(C)(=O)=O)ccc1Nc1ncc2c(N)cc(cc2n1)N1[C@@H](C)COC1=O |r|
CNC(=O)c1ccc(Nc2ncc3c(N)cc(cc3n2)N2[C@@H](C)COC2=O)c(OC)c1 |r|
COc1cc2CCN(C)Cc2cc1Nc1ncc2c(N)cc(Nc3cc(CO)ccn3)cc2n1
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(OCc3ccc(nc3)N3CCNCC3)cc2n1
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(OCc3ccc4CNCc4c3)cc2n1
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(OCC3CCNCC3)cc2n1
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(OCC3CCN(CC3)c3cncc(C)n3)cc2n1
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(Oc3cn[nH]c3)cc2n1
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(Oc3ccc(cc3)C(=O)N3CCN(C)CC3)cc2n1
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(Oc3ccc(cc3)C(=O)N3CCN(CC3)C(C)=O)cc2n1
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(Oc3ccc(cc3)[C@H](C)N)cc2n1 |r|
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(Oc3ccc4CCNCc4c3)cc2n1
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(cc2n1)[C@H]1CC[C@H](N)CC1 |r,wU:24.27,wD:27.31,(-9,-1.94,;-7.67,-1.17,;-6.33,-1.94,;-6.33,-3.47,;-5,-4.25,;-5,-5.79,;-3.66,-6.56,;-2.33,-5.79,;-1,-6.56,;-2.33,-4.25,;-3.66,-3.48,;-3.66,-1.94,;-5,-1.17,;-5,.37,;-3.66,1.14,;-3.66,2.68,;-2.33,3.45,;-1,2.68,;.33,3.45,;1.67,2.68,;1.67,1.14,;.33,.37,;-1,1.14,;-2.33,.37,;3,.37,;4.33,1.14,;5.67,.37,;5.67,-1.17,;7,-1.94,;4.33,-1.94,;3,-1.17,)|
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccc(cc2n1)[C@H]1CC[C@H](CN)CC1 |r,wU:24.27,wD:27.31,(-9,-1.94,;-7.67,-1.17,;-6.33,-1.94,;-6.33,-3.47,;-5,-4.25,;-5,-5.79,;-3.66,-6.56,;-2.33,-5.79,;-1,-6.56,;-2.33,-4.25,;-3.66,-3.48,;-3.66,-1.94,;-5,-1.17,;-5,.37,;-3.66,1.14,;-3.66,2.68,;-2.33,3.45,;-1,2.68,;.33,3.45,;1.67,2.68,;1.67,1.14,;.33,.37,;-1,1.14,;-2.33,.37,;3,.37,;4.33,1.14,;5.67,.37,;5.67,-1.17,;7,-1.94,;7,-3.48,;4.33,-1.94,;3,-1.17,)|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2n(C)c(nc2c1N1C[C@H](N)C[C@H]1CO)-c1ncccc1F |r|
Cn1c(nc2c(N3C[C@H](N)C[C@H]3CO)c(NC(=O)c3ccnc(n3)-c3c(F)cccc3F)ccc12)-c1ncccc1F |r|
COc1cccnc1-c1nc2c(N3C[C@H](N)C[C@H]3CO)c(NC(=O)c3ccnc(n3)-c3c(F)cccc3F)ccc2n1C |r|
Cn1c(nc2c(N3C[C@H](N)C[C@H]3CO)c(NC(=O)c3ccnc(n3)-c3c(F)cccc3F)ccc12)-c1ccccc1C#N |r|
N[C@@H]1C[C@@H](CO)N(C1)c1c(NC(=O)c2ccnc(n2)-c2c(F)cccc2F)ccc2n(C3CC3)c(nc12)-c1ccccc1C#N |r|
CN([C@@H]1CCCNC1)c1c(NC(=O)c2ccnc(n2)-c2c(F)cccc2F)ccc2n(C)c(nc12)-c1c(F)cncc1F |r,wD:2.1,(-.83,.97,;.51,.2,;1.84,.97,;1.84,2.51,;3.17,3.28,;4.51,2.51,;4.51,.97,;3.17,.2,;.51,-1.34,;-.83,-2.11,;-2.16,-1.34,;-3.49,-2.11,;-3.49,-3.65,;-4.83,-1.34,;-6.16,-2.11,;-7.5,-1.34,;-7.5,.2,;-6.16,.97,;-4.83,.2,;-6.16,2.51,;-4.83,3.28,;-3.49,2.51,;-4.83,4.82,;-6.16,5.59,;-7.5,4.82,;-7.5,3.28,;-8.83,2.51,;-.83,-3.65,;.51,-4.42,;1.84,-3.65,;3.3,-4.13,;3.78,-5.59,;4.21,-2.88,;3.3,-1.63,;1.84,-2.11,;5.75,-2.88,;6.52,-1.55,;5.75,-.21,;8.06,-1.55,;8.83,-2.88,;8.06,-4.21,;6.52,-4.21,;5.75,-5.55,)|
Cn1c(nc2c(N3C[C@H](N)C[C@H]3CO)c(NC(=O)c3ccnc(n3)-c3c(F)cccc3F)ccc12)-c1ccncc1F |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2n(C)c(nc2c1N1CCOC[C@@H]1CN)-c1ccncc1F |r|
Cn1c(nc2c(N3CCNC[C@@H]3CO)c(NC(=O)c3ccnc(n3)-c3c(F)cccc3F)ccc12)-c1ccncc1F |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2n(C)c(nc2c1N1C[C@@H]2C[C@H]1CN2)-c1ccncc1F |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2n(C)c(nc2c1N1C[C@@H]2C[C@H]1CO2)-c1ccncc1F |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2n(C)c(C)nc2c1N1CCC[C@H]1CN |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2n(C)c(C)nc2c1N1CCC[C@@H]1CN |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2n(C)c(C)nc2c1N1CCC[C@@H]1CO |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2n(C)c(C)nc2c1N1C[C@H](N)C[C@H]1CO |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2n(C)c(C)nc2c1N1C[C@H]2C[C@@H]1CN2 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2n(C)c(nc2c1N1C[C@@H]2C[C@H]1CN2)C(C)C |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2n(C)c(nc2c1N1CCC[C@H]1CN)-c1ccncc1F |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2n(C)c(nc2c1N1CCC[C@H]1CN)-c1ccnn1C |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2n(C)c(nc2c1N1CCC[C@H]1CN)C1CCOCC1 |r|
COCCn1c(C)nc2c(N3CCC[C@H]3CN)c(NC(=O)c3ccnc(n3)-c3c(F)cccc3OC)ccc12 |r|
COC[C@@H](C)n1c(C)nc2c(N3CCC[C@H]3CN)c(NC(=O)c3ccnc(n3)-c3c(F)cccc3OC)ccc12 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2n(CC(C)(C)OC)c(C)nc2c1N1CCC[C@H]1CN |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2n([C@H]3CCOC3)c(C)nc2c1N1CCC[C@H]1CN |r|
COCc1nc2c(N3CCC[C@H]3CN)c(NC(=O)c3ccnc(n3)-c3c(F)cccc3OC)ccc2n1C |r|
COCCc1nc2c(N3CCC[C@H]3CN)c(NC(=O)c3ccnc(n3)-c3c(F)cccc3OC)ccc2n1C |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2n(cnc2c1N1CCC[C@H]1CN)[C@@H]1CCOC1 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2n(C)cnc2c1N1CCC[C@H]1CN |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2n(Cc3ccncc3)c(C)nc2c1N1CC[C@H](N)C1 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2n(Cc3cnn(C)c3)c(C)nc2c1N1CC[C@H](N)C1 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2n(C)c(C)nc2c1-c1ccccc1N |(-7.96,3.28,;-6.62,2.51,;-5.29,3.28,;-5.29,4.82,;-3.96,5.59,;-2.62,4.82,;-2.62,3.28,;-1.29,2.51,;-3.96,2.51,;-3.96,.97,;-5.29,.2,;-5.29,-1.34,;-3.96,-2.11,;-2.62,-1.34,;-2.62,.2,;-1.29,-2.11,;-1.29,-3.65,;.05,-1.34,;1.38,-2.11,;1.38,-3.65,;2.71,-4.42,;4.05,-3.65,;5.51,-4.13,;5.99,-5.59,;6.42,-2.88,;7.96,-2.88,;5.51,-1.63,;4.05,-2.11,;2.71,-1.34,;2.71,.2,;1.38,.97,;1.38,2.51,;2.71,3.28,;4.05,2.51,;4.05,.97,;5.38,.2,)|
Cc1nc2c(N3CCC[C@H]3CN)c(NC(=O)c3ccnc(n3)-c3c(F)cccc3F)ccc2n1C |r|
Cc1nc2c(N3CCC[C@H]3CN)c(NC(=O)c3ccnc(n3)-c3c(C)cccc3F)ccc2n1C |r|
COc1cccc(F)c1-c1nc(ccc1F)C(=O)Nc1ccc2n(C)c(C)nc2c1N1CCC[C@H]1CN |r,wU:34.39,(-7.96,3.28,;-6.62,2.51,;-5.29,3.28,;-5.29,4.82,;-3.96,5.59,;-2.62,4.82,;-2.62,3.28,;-1.29,2.51,;-3.96,2.51,;-3.96,.97,;-2.62,.2,;-2.62,-1.34,;-3.96,-2.11,;-5.29,-1.34,;-5.29,.2,;-6.62,.97,;-1.29,-2.11,;-1.29,-3.65,;.05,-1.34,;1.38,-2.11,;1.38,-3.65,;2.71,-4.42,;4.05,-3.65,;5.51,-4.13,;5.99,-5.59,;6.42,-2.88,;7.96,-2.88,;5.51,-1.63,;4.05,-2.11,;2.71,-1.34,;2.71,.2,;1.47,1.11,;1.94,2.57,;3.48,2.57,;3.96,1.11,;5.42,.63,;6.57,1.66,)|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2n(C)ccc2c1N1CCC[C@@H]1CN |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2n(C)ccc2c1N1C[C@@H](N)C[C@H]1CO |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2n(C)ccc2c1N1CCNC[C@H]1C |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2n(C)ccc2c1N1C[C@@H]2C[C@H]1CN2 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2n(Cc3ccncc3)ccc2c1N1C[C@@H]2C[C@H]1CN2 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2[nH]ccc2c1N1C[C@@H]2C[C@H]1CN2 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2n(CC3CCCCO3)ccc2c1N1C[C@@H]2C[C@H]1CN2 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2n(Cc3cnc(C)s3)ccc2c1N1C[C@@H]2C[C@H]1CN2 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2n(CCN3CCOCC3)ccc2c1N1C[C@@H]2C[C@H]1CN2 |r|
COc1cc(ccn1)-n1ccc2c(N3C[C@@H]4C[C@H]3CN4)c(NC(=O)c3ccnc(n3)-c3c(F)cccc3OC)ccc12 |r|
COc1ccc(c(F)c1)-n1ccc2c(N3C[C@@H](N)C[C@H]3CO)c(NC(=O)c3ccnc(n3)-c3c(F)cccc3OC)ccc12 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2n(ccc2c1N1C[C@@H](N)C[C@H]1CO)-c1ccnn1C |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2n(ccc2c1N1C[C@@H](N)C[C@H]1CO)-c1cccc(F)c1C#N |r|
Cc1c2NCCOc2ncc1-c1ccc2cnc(Nc3cnn(c3)C3COC3)nc2c1
Cc1c2NCCOc2ncc1-c1ccc2cnc(Nc3cnn(c3)C3CC4(C3)CC(C4)C3(C)COC3)nc2c1 |(9.96,-5.39,;11.29,-4.62,;12.63,-5.39,;12.63,-6.93,;13.96,-7.7,;15.29,-6.93,;15.29,-5.39,;13.96,-4.62,;13.96,-3.08,;12.63,-2.31,;11.29,-3.08,;9.96,-2.31,;9.96,-.77,;8.63,,;7.29,-.77,;5.96,,;4.62,-.77,;4.62,-2.31,;3.29,-3.08,;3.29,-4.62,;2.04,-5.53,;2.52,-6.99,;4.06,-6.99,;4.54,-5.53,;4.97,-8.24,;6.49,-8.48,;6.25,-10,;4.73,-9.76,;7.77,-10.24,;7.53,-11.76,;6.01,-11.52,;8.43,-13.01,;7.19,-13.91,;9.68,-12.1,;10.58,-13.35,;9.34,-14.25,;5.96,-3.08,;7.29,-2.31,;8.63,-3.08,)|
CCC(=O)N1CC(C1)n1cc(Nc2ncc3ccc(cc3n2)-c2cnc3OCCNc3c2C)cn1
CN1CC2(CC2)c2cc(Nc3ncc4ccc(cc4n3)-c3cnc4OCCNc4c3C)nn2CC1=O
Cc1c2NCCOc2ncc1-c1ccc2cnc(Nc3cnn(C)c3)nc2c1
CC(C)N1CCc2cc(Nc3ncc4ccc(cc4n3)-c3cnc4OCCNc4c3C)nn2CC1=O
CC(C)N1CCn2nc(Nc3ncc4ccc(cc4n3)-c3cnc4OCCNc4c3C)cc2CC1=O
Cc1c2NCCOc2ncc1-c1ccc2cnc(Nc3cc4CC(=O)N(CCn4n3)C(C)(C)O)nc2c1
CCC(=O)N1CC(C1)n1cc(Nc2ncc3c(N)c(F)c(cc3n2)-c2cnc3OCCNc3c2C)cn1
Cc1c2NCCOc2ncc1-c1cc2nc(Nc3cnn(c3)C3CC4(C3)CN(C4)C3(C)COC3)ncc2c(N)c1F
Cc1c2NCCOc2ncc1-c1cc2nc(Nc3cnn(c3)C3CCN(CC3)C3(C)COC3)ncc2c(N)c1F
Cc1c2NCCOc2ncc1-c1cc2nc(Nc3cnn(c3)C3CC4(CNC4)C3)ncc2c(N)c1F
Cc1c2NCCOc2ncc1-c1cc2nc(Nc3cnn(c3)C3CNC3)ncc2c(N)c1F
Cc1c2NCCOc2ncc1-c1cc2nc(Nc3cnn(CC4CC4)c3)ncc2c(N)c1F
Cc1c2NCCOc2ncc1-c1cc2nc(Nc3cnn(CC(F)(F)F)c3)ncc2c(N)c1F
Cc1c2NCCOc2ncc1-c1cc2nc(Nc3cnn(c3)C3(C)CC3)ncc2c(N)c1F
Cc1c2NCCOc2ncc1-c1cc2nc(Nc3cnn(c3)C3CC3)ncc2c(N)c1F
Cc1c2NCCOc2ncc1-c1cc2nc(Nc3cnn(C)c3)ncc2c(N)c1F
Cc1c2NCCOc2ncc1-c1cc2nc(Nc3cnn(c3)C3CCNCC3)ncc2c(N)c1F
Cc1c2NCCOc2ncc1-c1cc2nc(Nc3cnn(Cc4ccccc4)c3)ncc2c(N)c1F
CC(C)Cn1cc(Nc2ncc3c(N)c(F)c(cc3n2)-c2cnc3OCCNc3c2C)cn1
CC(C)n1cc(Nc2ncc3c(N)c(F)c(cc3n2)-c2cnc3OCCNc3c2C)cn1
COC(=O)C12CC(C1)(C2)n1cc(Nc2ncc3c(N)c(F)c(cc3n2)-c2cnc3OCCNc3c2C)cn1
CCn1ncc(Nc2ncc3c(N)c(F)c(cc3n2)-c2cnc3OCCNc3c2C)c1C
Cc1cc(Nc2ncc3c(N)c(F)c(cc3n2)-c2cnc3OCCNc3c2C)sn1
Cc1c2NCCOc2ncc1-c1cc2nc(Nc3cnn(CC(C)(C)O)c3Cl)ncc2c(N)c1F
CN1CC[C@H](C1=O)n1cc(Nc2ncc3c(N)c(F)c(cc3n2)-c2cnc3OCCNc3c2C)cn1 |r|
CC(C)N1CCn2nc(Nc3ncc4c(N)c(F)c(cc4n3)-c3cnc4OCCNc4c3C)cc2CC1=O
CN1CC[C@@H](C1=O)n1cc(Nc2ncc3c(N)c(F)c(cc3n2)-c2cnc3OCCNc3c2C)cn1 |r|
CCn1cc(Nc2ncc3c(N)c(F)c(cc3n2)-c2cnc3OCCNc3c2C)cn1
Cc1c2NCCOc2ncc1-c1cc2nc(Nc3cnn(c3)C3CCC3)ncc2c(N)c1F
Cc1c2NCCOc2ncc1-c1cc2nc(Nc3cnn(CC(C)(C)O)c3)ncc2c(N)c1F
Cc1c2NCCOc2ncc1-c1cc2nc(Nc3cnn(C4CC4)c3Cl)ncc2c(N)c1F
Cc1c2NCCOc2ncc1-c1cc2nc(Nc3cnn(c3Cl)C3(C)CC3)ncc2c(N)c1F
CCn1cc(Nc2ncc3c(N)c(F)c(cc3n2)-c2cnc3OCCNc3c2C)c(C)n1
CNC(=O)C12CC(C1)(C2)n1cc(Nc2ncc3c(N)c(F)c(cc3n2)-c2cnc3OCCNc3c2C)cn1
Cc1c(Nc2ncc3c(N)c(F)c(cc3n2)-c2cnc3OCCNc3c2C)cnn1C(F)F
Cc1c(Nc2ncc3c(N)c(F)c(cc3n2)-c2cnc3OCCNc3c2C)cnn1C
Cc1nn(CC(F)F)cc1Nc1ncc2c(N)c(F)c(cc2n1)-c1cnc2OCCNc2c1C
Cc1c2NCCOc2ncc1-c1cc2nc(Nc3cnn(CC(F)F)c3)ncc2c(N)c1F
CC(C)n1cc(Nc2ncc3c(N)c(F)c(cc3n2)-c2cnc3OCCNc3c2C)c(C)n1
Cc1nn(C)cc1Nc1ncc2c(N)c(F)c(cc2n1)-c1cnc2OCCNc2c1C
Cc1c2NCCOc2ncc1-c1cc2nc(Nc3cnn4CCCc34)ncc2c(N)c1F
Cc1nsc(Nc2ncc3c(N)c(F)c(cc3n2)-c2cnc3OCCNc3c2C)c1Cl
Cc1cnsc1Nc1ncc2c(N)c(F)c(cc2n1)-c1cnc2OCCNc2c1C
CCn1ncc(Nc2ncc3c(N)c(F)c(cc3n2)-c2cnc3OCCNc3c2C)c1F
Cc1c2NCCOc2ncc1-c1cc2nc(Nc3cnn(c3)C3COC3)ncc2c(N)c1F
CNC(=O)Cn1cc(Nc2ncc3c(N)c(F)c(cc3n2)-c2cnc3OCCNc3c2C)c(C)n1
CNC(=O)C(C)(C)n1cc(Nc2ncc3c(N)c(F)c(cc3n2)-c2cnc3OCCNc3c2C)cn1
Cc1c2NCCOc2ncc1-c1cc2nc(Nc3cnn(CS(C)(=O)=O)c3)ncc2c(N)c1F
Cc1c2NCCOc2ncc1-c1c(F)c(N)c2cnc(Nc3cnn(c3)C3(C)CC3)nc2c1Cl |(9.96,-5.39,;11.29,-4.62,;12.63,-5.39,;12.63,-6.93,;13.96,-7.7,;15.29,-6.93,;15.29,-5.39,;13.96,-4.62,;13.96,-3.08,;12.63,-2.31,;11.29,-3.08,;9.96,-2.31,;9.96,-.77,;11.29,,;8.63,,;8.63,1.54,;7.29,-.77,;5.96,,;4.62,-.77,;4.62,-2.31,;3.29,-3.08,;3.29,-4.62,;4.54,-5.53,;4.06,-6.99,;2.52,-6.99,;2.04,-5.53,;1.62,-8.24,;.09,-7.99,;2.09,-9.7,;3.14,-8.48,;5.96,-3.08,;7.29,-2.31,;8.63,-3.08,;8.63,-4.62,)|
CN1CCC(CC1)n1cc(Nc2ncc3c(N)c(F)c(c(Cl)c3n2)-c2cnc3OCCNc3c2C)cn1 |(-1.1,-11.97,;-.19,-10.73,;-.82,-9.32,;.08,-8.07,;1.62,-8.24,;2.24,-9.64,;1.34,-10.89,;2.52,-6.99,;2.04,-5.53,;3.29,-4.62,;3.29,-3.08,;4.62,-2.31,;4.62,-.77,;5.96,,;7.29,-.77,;8.63,,;8.63,1.54,;9.96,-.77,;11.29,,;9.96,-2.31,;8.63,-3.08,;8.63,-4.62,;7.29,-2.31,;5.96,-3.08,;11.29,-3.08,;12.63,-2.31,;13.96,-3.08,;13.96,-4.62,;15.29,-5.39,;15.29,-6.93,;13.96,-7.7,;12.63,-6.93,;12.63,-5.39,;11.29,-4.62,;9.96,-5.39,;4.54,-5.53,;4.06,-6.99,)|
Cc1c(Nc2ncc3c(N)c(F)c(c(Cl)c3n2)-c2cnc3OCCNc3c2C)cnn1C1CC1 |(.58,-5.05,;2.04,-5.53,;3.29,-4.62,;3.29,-3.08,;4.62,-2.31,;4.62,-.77,;5.96,,;7.29,-.77,;8.63,,;8.63,1.54,;9.96,-.77,;11.29,,;9.96,-2.31,;8.63,-3.08,;8.63,-4.62,;7.29,-2.31,;5.96,-3.08,;11.29,-3.08,;12.63,-2.31,;13.96,-3.08,;13.96,-4.62,;15.29,-5.39,;15.29,-6.93,;13.96,-7.7,;12.63,-6.93,;12.63,-5.39,;11.29,-4.62,;9.96,-5.39,;4.54,-5.53,;4.06,-6.99,;2.52,-6.99,;1.62,-8.24,;.21,-8.86,;1.54,-9.77,)|
Cc1c2NCCOc2ncc1-c1cc2nc(Nc3cnn(c3)C34CC(C3)(C4)C(C)(C)O)ncc2c(N)c1F
CN1CC[C@@H](C1)n1cc(Nc2ncc3c(N)c(F)c(c(Cl)c3n2)-c2cnc3OCCNc3c2C)cn1 |r,wD:4.6,(.85,-12.15,;.85,-10.61,;-.4,-9.7,;.08,-8.24,;1.62,-8.24,;2.09,-9.7,;2.52,-6.99,;2.04,-5.53,;3.29,-4.62,;3.29,-3.08,;4.62,-2.31,;4.62,-.77,;5.96,,;7.29,-.77,;8.63,,;8.63,1.54,;9.96,-.77,;11.29,,;9.96,-2.31,;8.63,-3.08,;8.63,-4.62,;7.29,-2.31,;5.96,-3.08,;11.29,-3.08,;12.63,-2.31,;13.96,-3.08,;13.96,-4.62,;15.29,-5.39,;15.29,-6.93,;13.96,-7.7,;12.63,-6.93,;12.63,-5.39,;11.29,-4.62,;9.96,-5.39,;4.54,-5.53,;4.06,-6.99,)|
CN1CC[C@H](C1)n1cc(Nc2ncc3c(N)c(F)c(c(Cl)c3n2)-c2cnc3OCCNc3c2C)cn1 |r,wU:4.6,(.85,-12.15,;.85,-10.61,;-.4,-9.7,;.08,-8.24,;1.62,-8.24,;2.09,-9.7,;2.52,-6.99,;2.04,-5.53,;3.29,-4.62,;3.29,-3.08,;4.62,-2.31,;4.62,-.77,;5.96,,;7.29,-.77,;8.63,,;8.63,1.54,;9.96,-.77,;11.29,,;9.96,-2.31,;8.63,-3.08,;8.63,-4.62,;7.29,-2.31,;5.96,-3.08,;11.29,-3.08,;12.63,-2.31,;13.96,-3.08,;13.96,-4.62,;15.29,-5.39,;15.29,-6.93,;13.96,-7.7,;12.63,-6.93,;12.63,-5.39,;11.29,-4.62,;9.96,-5.39,;4.54,-5.53,;4.06,-6.99,)|
COc1cc2CCN(C)Cc2cc1Nc1ncc(C(N)=O)c(Nc2cccc(CO)c2)n1
COc1cc2CCN(C)Cc2cc1Nc1ncc(C(N)=O)c(Nc2cccc(CNC(=O)OC(C)(C)C)c2)n1
COc1cc2CCN(C)Cc2cc1Nc1ncc(C(N)=O)c(Nc2cccc(CN)c2)n1
COc1cc2CCN(C)Cc2cc1Nc1ncc(C(N)=O)c(Nc2ccccc2CN)n1
CNCc1ccccc1Nc1nc(Nc2cc3CN(C)CCc3cc2OC)ncc1C(N)=O
COc1cc2CCN(C)Cc2cc1Nc1ncc(C(N)=O)c(Nc2cccc(c2)C(C)N)n1
CC(N)c1cccc(Nc2nc(Nc3cc4CN(C)CCc4cc3Cl)ncc2C(N)=O)c1
CC(N)c1cccc(Nc2nc(Nc3cc4CN(C)CCc4cc3F)ncc2C(N)=O)c1
COc1cc2CCN(C)Cc2cc1Nc1ncc(C(N)=O)c(Nc2cccc(CNC(=O)C3(F)CC3)c2)n1
COc1cc2CCN(C)Cc2cc1Nc1ncc(C(N)=O)c(Nc2c(F)cccc2F)n1
COc1cc2CCN(C)Cc2cc1Nc1ncc(C(N)=O)c(Nc2c(C)cccc2C)n1
COc1cc2CCN(C)Cc2cc1Nc1ncc(C(N)=O)c(Nc2c(C)cccc2F)n1
COc1cc2CCN(C)Cc2cc1Nc1ncc(C(N)=O)c(Nc2c(F)cccc2Br)n1
CN1CCc2cc(Cl)c(Nc3ncc(C(N)=O)c(Nc4c(C)cccc4F)n3)cc2C1
CN1CCc2cc(F)c(Nc3ncc(C(N)=O)c(Nc4c(C)cccc4F)n3)cc2C1
CN1CCc2cc(c(cc2C1)Nc3ncc(c(n3)Nc4c(cccc4F)C(F)(F)F)C(=O)N)OC
COc1cc2CCN(C)Cc2cc1Nc1ncc(C(N)=O)c(Nc2c(F)cccc2C#N)n1
COc1cc2CCN(C)Cc2cc1Nc1ncc(C(N)=O)c(Nc2ccc(F)cc2F)n1
COc1cc2CCN(C)Cc2cc1Nc1ncc(C(N)=O)c(Nc2cc(F)ccc2F)n1
COc1cc2CCN(C)Cc2cc1Nc1ncc(C(N)=O)c(Nc2cccc(Cl)c2F)n1
COc1cc2CCN(C)Cc2cc1Nc1ncc(C(N)=O)c(Nc2ccc(F)c(F)c2F)n1
COc1cc2CCN(C)Cc2cc1Nc1ncc(C(N)=O)c(Nc2cccc(C)c2F)n1
COc1cc(F)c(Nc2nc(Nc3cc4CN(C)CCc4cc3OC)ncc2C(N)=O)c(F)c1
COc1cc2CCN(C)Cc2cc1Nc1ncc(C(N)=O)c(Nc2c(F)ccc(C)c2Cl)n1
COc1cc2CCN(C)Cc2cc1Nc1ncc(C(N)=O)c(Nc2c(O)cccc2F)n1
COc1cc2CCN(C)Cc2cc1Nc1ncc(C(N)=O)c(Nc2cc(C)ccc2Cl)n1
COc1cc2CCN(C)Cc2cc1Nc1ncc(C(N)=O)c(Nc2ccc(C)cc2Cl)n1
COc1cc2CCN(C)Cc2cc1Nc1ncc(C(N)=O)c(Nc2c(Cl)ccc(C)c2F)n1
COc1cc2CCN(C)Cc2cc1Nc1ncc(C(N)=O)c(Nc2c(F)cc(F)cc2Cl)n1
Cc1cccc(F)c1Nc1nc(Nc2cnn(CC3CC3)c2)ncc1C(N)=O
Cc1cccc(F)c1Nc1nc(Nc2cnn(CC(C)(C)O)c2)ncc1C(N)=O
Cc1cccc(F)c1Nc1nc(Nc2cnn(CC(F)(F)F)c2)ncc1C(N)=O
Cc1cccc(F)c1Nc1nc(Nc2ccc(cc2)S(C)(=O)=O)ncc1C(N)=O
COc1cc2CCN(C)Cc2cc1Nc1ncc(C(N)=O)c(Nc2ccc(C)cc2C2CC2)n1
CCc1cc(C)ccc1Nc1nc(Nc2cc3CN(C)CCc3cc2OC)ncc1C(N)=O
COc1cc2CCN(C)Cc2cc1Nc1ncc(C(N)=O)c(Nc2ccc(C)cc2C(C)(C)C)n1
CN1CCc2cc(F)c(Nc3ncc(C(N)=O)c(Nc4c(F)cc(C)cc4C(F)(F)F)n3)cc2C1
COc1cc2CCN(C)Cc2cc1Nc1ncc(C(N)=O)c(Nc2c(F)cc(Br)cc2F)n1
COc1cc2CCN(C)Cc2cc1Nc1ncc(C(N)=O)c(Nc2c(F)cccc2CC(F)F)n1
CN1CCc2cc(F)c(Nc3ncc(C(N)=O)c(Nc4c5OC(C)(C)Cc5ccc4F)n3)cc2C1
COc1cc2CCN(C)Cc2cc1Nc1ncc(C(N)=O)c(Nc2c(C)cc(cc2F)C#N)n1
Cc1n[nH]c(C)c1Nc1ncc(C(N)=O)c(Nc2c(C)cccc2F)n1
Cc1nn(C)c(C)c1Nc1ncc(C(N)=O)c(Nc2c(C)cccc2F)n1
COc1cc2CCN(CC(C)(C)O)Cc2cc1Nc1ncc(C(N)=O)c(Nc2c(F)cccc2C(F)(F)F)n1
COc1cc2CCN(CC(C)(C)O)Cc2cc1Nc1ncc(C(N)=O)c(Nc2c(C)cccc2F)n1
CN1CCc2cc(c(cc2C1)Nc3ncc(c(n3)Nc4ccccc4)C(=O)N)OC
CS(=O)(=O)c1ccc(Nc2ncc(C(N)=O)c(Nc3cccc4CNCCc34)n2)cc1
Cc1ccncc1-c1cc2c(NC(=O)c3ccc(cc3)N3CCOCC3)n[nH]c2cn1
CN1CCN(CC1)c1ccc(cc1)C(=O)Nc1n[nH]c2cnc(cc12)-c1cnccc1C
CCOC(=O)N1CCN(CC1)c1ccc(cc1)C(=O)Nc1n[nH]c2cnc(cc12)-c1cnccc1C
COC1CCN(CC1)c1ccc(cc1)C(=O)Nc1n[nH]c2cnc(cc12)-c1cnccc1C
Cc1ccncc1-c1cc2c(NC(=O)c3ccc(cc3)N3CCCC(N)C3)n[nH]c2cn1
Cc1c(cnn1C)-c1cc2c(NC(=O)c3ccc(cc3)N3CCOCC3)n[nH]c2cn1
CN1CCN(CC1)c1ccc(cc1)C(=O)Nc1n[nH]c2cnc(cc12)-c1cnn(C)c1C
CCOC(=O)N1CCN(CC1)c1ccc(cc1)C(=O)Nc1n[nH]c2cnc(cc12)-c1cnn(C)c1C
COC1CCN(CC1)c1ccc(cc1)C(=O)Nc1n[nH]c2cnc(cc12)-c1cnn(C)c1C
COC1CCCN(C1)c1ccc(cc1)C(=O)Nc1n[nH]c2cnc(cc12)-c1cnn(C)c1C
CCCNc1ccc(cc1)C(=O)Nc1n[nH]c2cnc(cc12)-c1cnn(C)c1C
COCCNc1ccc(cc1)C(=O)Nc1n[nH]c2cnc(cc12)-c1cnn(C)c1C
Cc1c(cnn1C)-c1cc2c(NC(=O)c3ccc(cc3)N3CCC(F)(F)C3)n[nH]c2cn1
COc1ccncc1-c1cc2c(NC(=O)c3ccc(cc3)N3CCN(C)CC3)n[nH]c2cn1
CN1CCN(CC1)c1ccc(NC(=O)c2n[nH]c3cnc(cc23)-c2cnccc2C)cc1
COc1ccncc1-c1cc2c(n[nH]c2cn1)C(=O)Nc1ccc(cc1)N1CCN(C)CC1
CCN(CC)CCNC(=O)c1c(C)[nH]c(\C=C2/C(=O)Nc3cc(F)c(cc23)-c2cnc3OCCNc3c2C)c1C
Cc1ncc(\C=C2/C(=O)Nc3ccc(cc23)-c2ccc3OCCNc3c2C)[nH]1
Cc1ncc(\C=C2/C(=O)Nc3cc(C)c(cc23)-c2cnc3OCCNc3c2C)[nH]1
Cc1ncc(\C=C2/C(=O)Nc3c2c(C)c(cc3F)-c2cnc3OCCNc3c2C)[nH]1
Cc1ncc(\C=C2/C(=O)Nc3c2c(C)c(cc3F)-c2cnc3OCCNc3c2)[nH]1
CCc1nc(C)c(\C=C2/C(=O)Nc3ccc(cc23)-c2cnc3OCCNc3c2C)[nH]1
Cc1ncc(\C=C2/C(=O)Nc3cc(Cl)c(cc23)-c2cnc3OCCNc3c2C)[nH]1
Cc1ncc(\C=C2/C(=O)Nc3cc(F)c(cc23)-c2cnc3OCCNc3c2C)[nH]1
CCN(CC)CCNC(=O)c1c(C)[nH]c(\C=C2/C(=O)Nc3c2cc(cc3F)-c2cnc3OCCNc3c2C)c1C
Cc1ncc(\C=C2/C(=O)Nc3c2cc(cc3F)-c2cnc3OCCNc3c2C)[nH]1
C\C(=C1\C(=O)Nc2ccc(cc12)-c1cnc2OCCNc2c1C)c1cnc[nH]1
Cc1c2\C(=C\c3cc(c[nH]3)C#N)C(=O)Nc2c(F)cc1-c1cnc2OCCNc2c1C
Cc1c[nH]c(\C=C2/C(=O)Nc3c2c(C)c(cc3F)-c2cnc3OCCNc3c2C)c1
Cc1c2\C(=C\c3ccc[nH]3)C(=O)Nc2c(F)cc1-c1cnc2OCCNc2c1C
Cc1ncc(\C=C2/C(=O)Nc3ccc(cc23)-c2cnc3OCCNc3c2C)[nH]1
CCN(CC)CCNC(=O)c1c(C)[nH]c(\C=C2/C(=O)Nc3ccc(cc23)-c2cnc3OCCNc3c2C)c1C
Cc1ccc(\C=C2/C(=O)Nc3ccc(cc23)-c2cnc3OCCNc3c2C)[nH]1
Cc1c2NCCOc2ncc1-c1ccc2NC(=O)\C(=C/c3ccns3)c2c1
Cc1c2NCCOc2ncc1-c1ccc2NC(=O)C(=Cc3cccs3)c2c1 |w:19.21|
Cc1c2NCCOc2ncc1-c1ccc2NC(=O)\C(=C/c3cc(Br)c[nH]3)c2c1
Cc1c2NCCOc2ncc1-c1ccc2NC(=O)\C(=C/c3cc(c[nH]3)C#N)c2c1
Cc1c[nH]c(\C=C2/C(=O)Nc3c2cc(cc3Cl)-c2cnc3OCCNc3c2C)c1
Cc1c2NCCOc2ncc1-c1cc2\C(=C\c3ccc[nH]3)C(=O)Nc2c(Cl)c1
Cc1c[nH]c(\C=C2/C(=O)Nc3c2cc(cc3C)-c2cnc3OCCNc3c2C)c1
Cc1c[nH]c(\C=C2/C(=O)Nc3c2cc(cc3F)-c2cnc3OCCNc3c2C)c1
Cc1c2NCCOc2ncc1-c1cc2\C(=C\c3ccc[nH]3)C(=O)Nc2c(F)c1
Cc1c2NCCOc2ncc1-c1ccc2NC(=O)\C(=C/c3cnn[nH]3)c2c1
Cc1c[nH]c(\C=C2/C(=O)Nc3ccc(cc23)-c2cnc3OCCNc3c2C)c1
Cc1c2NCCOc2ncc1-c1ccc2NC(=O)\C(=C/c3ccc[nH]3)c2c1
Cc1c2NCCOc2ncc1-c1ccc2NC(=O)\C(=C/c3ccn[nH]3)c2c1
Cc1c2NCCOc2ncc1-c1ccc2NC(=O)\C(=C/c3ncc[nH]3)c2c1
Cc1c2NCCOc2ncc1-c1ccc2NC(=O)\C(=C/c3cnc[nH]3)c2c1
Cc1c2NC(=O)C3(CC3)Oc2ncc1-c1ccc2NC(=O)\C(=C/c3ncc[nH]3)c2c1
Cc1c2NCCOc2ncc1-c1ccc2NC(=O)\C(=C/c3cnc([nH]3)C3CC3)c2c1
Cc1c2NCCOc2ncc1-c1cc2\C(=C\c3cnc([nH]3)C3CC3)C(=O)Nc2c(F)c1
CC\C(=C1\C(=O)Nc2ccc(cc12)-c1cnc2OCCNc2c1C)c1cnc[nH]1
Cc1cc2NC(=O)\C(=C/c3cc4ccncc4[nH]3)c2cc1-c1cnc2OCCNc2c1C
Cc1cc2NC(=O)\C(=C/c3cc4ncccc4[nH]3)c2cc1-c1cnc2OCCNc2c1C
Cc1c2NC(=O)COc2ccc1-c1ccc2NC(=O)\C(=C/c3cc4cnccc4[nH]3)c2c1
Cc1cc2NC(=O)\C(=C/c3cc4cnccc4[nH]3)c2cc1-c1cnc2OCCNc2c1C
Cc1cc2NC(=O)\C(=C/c3cc4cnccc4[nH]3)c2cc1-c1cnc2OCCNc2c1
Cc1c2\C(=C\c3cc4cnccc4[nH]3)C(=O)Nc2c(F)cc1-c1cnc2OCCNc2c1
Cc1c2NCCOc2ncc1-c1cc2\C(=C\c3cc4ccncc4[nH]3)C(=O)Nc2cc1F
Cc1c2NCCOc2ncc1-c1cc2\C(=C\c3cc4ncccc4[nH]3)C(=O)Nc2cc1F
Cc1c2NCCOc2ncc1-c1cc2\C(=C\c3cc4ccncc4[nH]3)C(=O)Nc2c(F)c1
Cc1c2NCCOc2ncc1-c1cc2\C(=C\c3cc4ncccc4[nH]3)C(=O)Nc2c(F)c1
Cc1c2NCCOc2ncc1-c1cnc2NC(=O)\C(=C/c3cc4cnccc4[nH]3)c2c1
Cc1c2NCCOc2ncc1-c1cc2\C(=C\c3cc4cnccc4[nH]3)C(=O)Nc2cc1Cl
Cc1c2NCCOc2ncc1-c1cc2\C(=C\c3cc4cnccc4[nH]3)C(=O)Nc2cc1F
Cc1c2NCCOc2ncc1-c1cc2\C(=C\c3cc4ccccc4[nH]3)C(=O)Nc2cc1Cl
Cc1c2NCCOc2ncc1-c1cc2\C(=C\c3cc4ccccc4[nH]3)C(=O)Nc2cc1F
Cc1c2NCCOc2ncc1-c1cc2\C(=C\c3cc4cnccc4[nH]3)C(=O)Nc2c(F)c1
Cc1c2NCCOc2ncc1-c1cc2\C(=C\c3cc4ccccc4[nH]3)C(=O)Nc2c(F)c1
Cc1c2\C(=C\c3cc4cnccc4[nH]3)C(=O)Nc2c(F)cc1-c1cnc2OCCNc2c1C
Cc1c2NCCOc2ncc1-c1cnc2NC(=O)\C(=C/c3cc4ccccc4[nH]3)c2c1
Cc1c2\C(=C\c3cc4ccccc4[nH]3)C(=O)Nc2c(F)cc1-c1cnc2OCCNc2c1C
Cc1c2NCCOc2ncc1-c1ccc2NC(=O)\C(=C/c3cc4ncccc4[nH]3)c2c1
Cc1c2NCCOc2ncc1-c1ccc2NC(=O)\C(=C/c3cc4ccncc4[nH]3)c2c1
Cc1c2NCCOc2ncc1-c1ccc2NC(=O)\C(=C/c3nc4ccccc4[nH]3)c2c1
Cc1c2NCCOc2ncc1-c1ccc2NC(=O)\C(=C/c3cc4cnccc4[nH]3)c2c1
Cc1c2NCCOc2ncc1-c1ccc2NC(=O)\C(=C/c3cc4cccnc4[nH]3)c2c1
Cc1c2NCCOc2ncc1-c1ccc2NC(=O)\C(=C/c3cc4ccccc4[nH]3)c2c1
Cc1c2\C(=C\c3cc4ccncc4[nH]3)C(=O)Nc2c(F)cc1-c1cnc2OCCNc2c1C
Cc1c2\C(=C\c3cc4ncccc4[nH]3)C(=O)Nc2c(F)cc1-c1cnc2OCCNc2c1C
Cc1c2\C(=C\c3cn[nH]c3)C(=O)Nc2c(F)cc1-c1cnc2OCCNc2c1C
Cc1c2NCCOc2ncc1-c1cc2\C(=C\c3cn[nH]c3)C(=O)Nc2c(Cl)c1
Cc1cc(cc2\C(=C\c3cn[nH]c3)C(=O)Nc12)-c1cnc2OCCNc2c1C
Cc1n[nH]cc1\C=C1/C(=O)Nc2ccc(cc12)-c1cnc2OCCNc2c1C
Cc1c2NCCOc2ncc1-c1ccc2NC(=O)\C(=C/c3cn[nH]c3)c2c1
Cc1c2NCCOc2ncc1-c1ccc2NC(=O)\C(=C/c3c[nH]c4ccccc34)c2c1
O=C1Nc2ccc(cc2\C1=C\c1ncc[nH]1)-c1cnc2OCCNc2c1
Cc1c2NCC3(CC3)Oc2ncc1-c1ccc2NC(=O)\C(=C/c3ncc[nH]3)c2c1
COc1ncc([C@H](C)N)c2cc(Nc3ccnc(n3)C(C)(C)F)ncc12 |r|
CNc1ncc(c2cc(Nc3ccnc(n3)C(C)(C)F)ncc12)C(C)(C)N
COc1ncc(c2cc(Nc3ccnc(n3)C(C)(C)F)ncc12)C(C)(C)N
COc1ncc(c2cc(Nc3ccnc(OC(C)C)n3)ncc12)C(C)(C)N
COc1ccc(c2cc(Nc3ccnc(n3)C(C)(C)F)ncc12)C(C)(C)N
CNc1ncc(c2cc(Nc3cnc(C#N)c(n3)C(C)C)ncc12)C(C)(C)N
CNc1ncc(c2cc(Nc3ccc4C(=O)CCCc4n3)ncc12)C(C)(C)N
COc1ncc(c2cc(Nc3cnc(C#N)c(n3)C(C)C)ncc12)C(C)(C)N
COc1ncc(c2cc(Nc3ccc4C(=O)NCCc4n3)ncc12)C(C)(C)N
COc1ncc(c2cc(Nc3ccc4C(=O)OCCc4n3)ncc12)C(C)(C)N
CNc1ncc(c2cc(Nc3ccnc(n3)N3CC[C@@H]3C)ncc12)C(C)(C)N |r|
CC[C@H](C)n1nc(Nc2cc3c(cnc(OC)c3cn2)C(C)(C)N)ccc1=O |r|
CC[C@@H](C)n1nc(Nc2cc3c(cnc(OC)c3cn2)C(C)(C)N)ccc1=O |r|
CCOc1ncc(c2cc(Nc3ccnc(n3)C(C)(C)F)ncc12)C(C)(C)N
CNC(C)(C)c1cnc(OC)c2cnc(Nc3ccnc(n3)C(C)(C)F)cc12
CC[C@@H](C)c1nc(Nc2cc3c(cnc(OC)c3cn2)C(C)(C)N)ccc1C#N |r|
CC[C@H](C)c1nc(Nc2cc3c(cnc(OC)c3cn2)C(C)(C)N)ccc1C#N |r|
CC[C@H](C)c1nc(Nc2cc3c(cnc(OC)c3cn2)C(C)(C)N)cnc1C#N |r|
CC[C@@H](C)c1nc(Nc2cc3c(cnc(OC)c3cn2)C(C)(C)N)cnc1C#N |r|
COc1ncc(c2cc(Nc3ccc4C(=O)OC[C@H](C)c4n3)ncc12)C(C)(C)N |r|
COc1ncc(c2cc(Nc3ccc4C(=O)O[C@H](C)Cc4n3)ncc12)C(C)(C)N |r|
COc1ncc(c2cc(Nc3ccc4C(=O)O[C@@H](C)Cc4n3)ncc12)C(C)(C)N |r|
COc1ncc(c2cc(Nc3ccc4C(=O)OC(C)(C)c4n3)ncc12)C(C)(C)N
COc1ncc(c2cc(Nc3ccnc(n3)N3CCC[C@@H]3C)ncc12)C(C)(C)N |r|
COc1ncc(c2cc(Nc3ccc(C#N)c(n3)C(C)(C)F)ncc12)C(C)(C)N
COc1ncc(c2cc(Nc3cnc(C#N)c(n3)C(C)(C)F)ncc12)C(C)(C)N
CC[C@H](F)c1nc(Nc2cc3c(cnc(OC)c3cn2)C(C)(C)N)cnc1C#N |r|
CC[C@@H](F)c1nc(Nc2cc3c(cnc(OC)c3cn2)C(C)(C)N)cnc1C#N |r|
CCOc1ccc(c2cc(Nc3ccnc(n3)C(C)(C)F)ncc12)C(C)(C)NC
COc1ncc(c2cc(Nc3ccc4C(=O)OC5(CC5)Cc4n3)ncc12)C(C)(C)N
COc1ncc(c2cc(Nc3ccc4C(=O)CC(C)(C)Cc4n3)ncc12)C(C)(C)N
COc1ncc(c2cc(Nc3ccc4C(=O)OC(C)(C)Cc4n3)ncc12)C(C)(C)N
COc1ncc(c2cc(Nc3ccc4C(=O)O[C@@H](C)[C@H](C)c4n3)ncc12)C(C)(C)N |r|
COc1ncc(c2cc(Nc3ccc4C(=O)O[C@H](C)[C@@H](C)c4n3)ncc12)C(C)(C)N |r|
COc1ncc(c2cc(Nc3ccc4C(=O)O[C@H](C)[C@H](C)c4n3)ncc12)C(C)(C)N |r|
COc1ncc(c2cc(Nc3ccc4C(=O)O[C@@H](C)[C@@H](C)c4n3)ncc12)C(C)(C)N |r|
CCOc1ncc(c2cc(Nc3ccc4C(=O)O[C@@H](C)Cc4n3)ncc12)C(C)(C)N |r|
CCOc1ncc(c2cc(Nc3ccc4C(=O)O[C@H](C)Cc4n3)ncc12)C(C)(C)N |r|
CCOc1ncc(c2cc(Nc3ccc4C(=O)OC[C@H](C)c4n3)ncc12)C(C)(C)N |r|
CCOc1ncc(c2cc(Nc3ccc4C(=O)OC[C@@H](C)c4n3)ncc12)C(C)(C)N |r|
CCOc1ncc(c2cc(Nc3ccc4C(=O)OC(C)(C)c4n3)ncc12)C(C)(C)N
COc1cnc(c2cc(Nc3ccc4C(=O)OC(C)(C)Cc4n3)ncc12)C(C)(C)N
COc1ncc(c2cc(Nc3cnc4C(=O)OC(C)(C)Cc4n3)ncc12)C(C)(C)N
CNc1ncc(c2cc(Nc3cnc(C#N)c(n3)N3CCC[C@@H]3C)ncc12)C(C)(C)N |r|
COc1ncc(c2cc(Nc3cnc(C#N)c(n3)N3CCC[C@@H]3C)ncc12)C(C)(C)N |r|
COc1ncc(C2CCCN2)c2cc(Nc3ccc4C(=O)OC(C)(C)Cc4n3)ncc12
COc1ncc(c2cc(Nc3ccc4C(=O)O[C@@H]5CCC[C@@H]5c4n3)ncc12)C(C)(C)N |r|
COc1ncc(c2cc(Nc3ccc4C(=O)O[C@H]5CCC[C@H]5c4n3)ncc12)C(C)(C)N |r|
CCNc1ncc(c2cc(Nc3ccc4C(=O)OC(C)(C)Cc4n3)ncc12)C(C)(C)N
CCOc1ncc(c2cc(Nc3ccc4C(=O)OC(C)(C)Cc4n3)ncc12)C(C)(C)N
COc1ncc(c2cc(Nc3ccc4C(=O)OC(C)(C)[C@@H](C)c4n3)ncc12)C(C)(C)N |r|
COc1ncc(c2cc(Nc3ccc4C(=O)OC(C)(C)[C@H](C)c4n3)ncc12)C(C)(C)N |r|
CCOc1ncc(c2cc(Nc3ccc4C(=O)O[C@@H](C)[C@H](C)c4n3)ncc12)C(C)(C)N |r|
CCOc1ncc(c2cc(Nc3ccc4C(=O)O[C@H](C)[C@@H](C)c4n3)ncc12)C(C)(C)N |r|
CCOc1ncc(c2cc(Nc3ccc4C(=O)O[C@H](C)[C@H](C)c4n3)ncc12)C(C)(C)N |r|
CCOc1ncc(c2cc(Nc3ccc4C(=O)O[C@@H](C)[C@@H](C)c4n3)ncc12)C(C)(C)N |r|
CC[C@@](C)(N)c1cnc(OC)c2cnc(Nc3ccc4C(=O)OC(C)(C)Cc4n3)cc12 |r|
CC[C@](C)(N)c1cnc(OC)c2cnc(Nc3ccc4C(=O)OC(C)(C)Cc4n3)cc12 |r|
COc1ncc(c2cc(Nc3cnc(C#N)c(n3)C(C)C(F)(F)F)ncc12)C(C)(C)N
CC(C)(N)c1cnc(OC2CC2)c2cnc(Nc3ccc4C(=O)OC(C)(C)Cc4n3)cc12
C[C@H]1OC(=O)c2ccc(Nc3cc4c(cnc(OC5CC5)c4cn3)C(C)(C)N)nc2[C@@H]1C |r|
C[C@@H]1OC(=O)c2ccc(Nc3cc4c(cnc(OC5CC5)c4cn3)C(C)(C)N)nc2[C@H]1C |r|
CCOc1ncc(c2cc(Nc3ccc4C(=O)OC(C)(C)[C@H](C)c4n3)ncc12)C(C)(C)N |r|
CCOc1ncc(c2cc(Nc3ccc4C(=O)OC(C)(C)[C@@H](C)c4n3)ncc12)C(C)(C)N |r|
CC(C)Oc1ncc(c2cc(Nc3ccc4C(=O)OC(C)(C)Cc4n3)ncc12)C(C)(C)N
C[C@H]1c2nc(Nc3cc4c(cnc(OC5CC5)c4cn3)C(C)(C)N)ccc2C(=O)OC1(C)C |r|
C[C@@H]1c2nc(Nc3cc4c(cnc(OC5CC5)c4cn3)C(C)(C)N)ccc2C(=O)OC1(C)C |r|
CC(C)(N)c1cnc(OC2CCC2)c2cnc(Nc3ccc4C(=O)OC(C)(C)Cc4n3)cc12
CC(C)(N)c1cnc(OCC(F)F)c2cnc(Nc3ccc4C(=O)OC(C)(C)Cc4n3)cc12
C[C@@](N)(C1CC1)c1cnc(OC2CC2)c2cnc(Nc3ccc4C(=O)OC(C)(C)Cc4n3)cc12 |r|
C[C@@H]1OC(=O)c2ccc(Nc3cc4c(cnc(OC5CC5)c4cn3)[C@](C)(N)C3CC3)nc2[C@H]1C |r|
C[C@@H]1c2nc(Nc3cc4c(ncc(OC5CC5)c4cn3)[C@](C)(N)C3CC3)ccc2C(=O)OC1(C)C |r|
CC(C)(N)c1cnc(OCC(F)(F)F)c2cnc(Nc3ccc4C(=O)OC(C)(C)Cc4n3)cc12
C[C@@H]1OC(=O)c2ccc(Nc3cc4c(cnc(OCC(F)(F)F)c4cn3)C(C)(C)N)nc2[C@H]1C |r|
C[C@@H]1c2nc(Nc3cc4c(cnc(OCC(F)(F)F)c4cn3)C(C)(C)N)ccc2C(=O)OC1(C)C |r|
CC[C@@](C)(N)c1cnc(OC2CC2)c2cnc(Nc3ccc4C(=O)O[C@@H](C)[C@H](C)c4n3)cc12 |r|
C[C@@H]1OC(=O)c2ccc(Nc3cc4c(cnc(OC5(C)CC5)c4cn3)C(C)(C)N)nc2[C@H]1C |r|
C[C@@H]1c2nc(Nc3cc4c(cnc(OC5(C)CC5)c4cn3)C(C)(C)N)ccc2C(=O)OC1(C)C |r|
CC[C@@](C)(N)c1cnc(OC2(C)CC2)c2cnc(Nc3ccc4C(=O)O[C@@H](C)[C@H](C)c4n3)cc12 |r|
CC[C@](C)(N)c1cnc(OC2(C)CC2)c2cnc(Nc3ccc4C(=O)O[C@@H](C)[C@H](C)c4n3)cc12 |r|
CC[C@@](C)(N)c1cnc(OC2(C)CC2)c2cnc(Nc3ccc4C(=O)OC(C)(C)[C@H](C)c4n3)cc12 |r|
CC[C@](C)(N)c1cnc(OC2(C)CC2)c2cnc(Nc3ccc4C(=O)OC(C)(C)[C@H](C)c4n3)cc12 |r|
C[C@@H]1OC(=O)c2ccc(Nc3cc4c(cnc(OC5(C)CC5)c4cn3)[C@@](C)(N)C3CC3)nc2[C@H]1C |r|
C[C@@H]1OC(=O)c2ccc(Nc3cc4c(cnc(OC5(C)CC5)c4cn3)[C@](C)(N)C3CC3)nc2[C@H]1C |r|
C[C@@H]1c2nc(Nc3cc4c(cnc(OC5(C)CC5)c4cn3)[C@@](C)(N)C3CC3)ccc2C(=O)OC1(C)C |r|
C[C@@H]1c2nc(Nc3cc4c(cnc(OC5(C)CC5)c4cn3)[C@](C)(N)C3CC3)ccc2C(=O)OC1(C)C |r|
CC[C@](C)(N)c1cnc(OC2(C)CC2)c2cnc(Nc3ccc4C(=O)O[C@H](C)[C@H](C)c4n3)cc12 |r|
CC[C@@](C)(N)c1cnc(OC2(C)CC2)c2cnc(Nc3ccc4C(=O)O[C@H](C)[C@H](C)c4n3)cc12 |r|
C[C@H]1OC(=O)c2ccc(Nc3cc4c(cnc(OC5(C)CC5)c4cn3)[C@](C)(N)C3CC3)nc2[C@H]1C |r|
C[C@H]1OC(=O)c2ccc(Nc3cc4c(cnc(OC5(C)CC5)c4cn3)[C@@](C)(N)C3CC3)nc2[C@H]1C |r|
CC[C@@](C)(N)c1cnc(OC2CC2)c2cnc(Nc3ccc4C(=O)O[C@H](C)[C@H](C)c4n3)cc12 |r|
COc1ncc(c2cc(Nc3ccc4C(=O)OC(C)(C)c4n3)ncc12)[C@@](C)(N)C1CC1 |r|
COc1ncc(c2cc(Nc3ccc4CO[C@@H](C)[C@H](C)c4n3)ncc12)[C@@](C)(N)C1CC1 |r|
COc1ncc(c2cc(Nc3ccc4CO[C@@H](C)[C@H](C)c4n3)ncc12)[C@](C)(N)C1CC1 |r|
COc1ncc(c2cc(Nc3ccc4C(=O)OC(C)(C)[C@H](C)c4n3)ncc12)[C@](C)(N)C1CC1 |r|
COc1ncc(c2cc(Nc3ccc4C(=O)OC(C)(C)[C@H](C)c4n3)ncc12)[C@@](C)(N)C1CC1 |r|
COc1ccc(c2cc(Nc3ccc4C(=O)OC(C)(C)Cc4n3)ncc12)C(C)(C)N
CC(C)(N)c1ccc(Cl)c2cnc(Nc3ccc4C(=O)OC(C)(C)Cc4n3)cc12
CC(C)(N)c1cnc(OC2CC2)c2cnc(Nc3ccc4C(=O)OC(C)(C)c4n3)cc12
C[C@@](N)(C1CC1)c1cnc(OC2CC2)c2cnc(Nc3ccc4C(=O)NCCc4n3)cc12 |r|
CC(C)(N)c1cnc(OC2CC2)c2cnc(Nc3ccc4C(=O)OCC5(CC5)c4n3)cc12
C[C@@](N)(C1CC1)c1cnc(OC2CC2)c2cnc(Nc3ccc4C(=O)OCCc4n3)cc12 |r|
C[C@@H]1OC(=O)c2ccc(Nc3cc4c(cnc(NC5CC5)c4cn3)C(C)(C)N)nc2[C@H]1C |r|
CC[C@@](C)(N)c1cnc(OC2CC2)c2cnc(Nc3ccc4C(=O)OC(C)(C)c4n3)cc12 |r|
CC[C@](C)(N)c1cnc(OC2CC2)c2cnc(Nc3ccc4C(=O)OC(C)(C)c4n3)cc12 |r|
CC(C)(N)c1cnc(OC2CC2)c2cnc(Nc3ccc4C(=O)OCC(C)(C)c4n3)cc12
CC[C@]1(C)OC(=O)c2ccc(Nc3cc4c(cnc(OC5CC5)c4cn3)C(C)(C)N)nc12 |r|
CC[C@@]1(C)OC(=O)c2ccc(Nc3cc4c(cnc(OC5CC5)c4cn3)C(C)(C)N)nc12 |r|
CC(C)(N)c1cnc(OCC(F)(F)F)c2cnc(Nc3ccnc(n3)C(C)(C)F)cc12
CC(C)(N)c1cnc(OCC(F)F)c2cnc(Nc3ccc4C(=O)OC(C)(C)c4n3)cc12
C[C@H]1COC(=O)c2ccc(Nc3cc4c(cnc(OC5CC5)c4cn3)[C@](C)(N)C3CC3)nc12 |r|
C[C@@H]1COC(=O)c2ccc(Nc3cc4c(cnc(OC5CC5)c4cn3)[C@](C)(N)C3CC3)nc12 |r|
C[C@H]1OC(=O)c2ccc(Nc3cc4c(cnc(OC5CC5)c4cn3)C(C)(C)N)nc2C11CC1 |r|
C[C@@H]1OC(=O)c2ccc(Nc3cc4c(cnc(OC5CC5)c4cn3)C(C)(C)N)nc2C11CC1 |r|
CC[C@@](C)(N)c1cnc(NC2CC2)c2cnc(Nc3ccc4C(=O)O[C@@H](C)[C@H](C)c4n3)cc12 |r|
CC[C@](C)(N)c1cnc(NC2CC2)c2cnc(Nc3ccc4C(=O)O[C@@H](C)[C@H](C)c4n3)cc12 |r|
C[C@@H]1c2nc(Nc3cc4c(cnc(NC5CC5)c4cn3)C(C)(C)N)ccc2C(=O)OC1(C)C |r|
C[C@@H]1OC(=O)c2ccc(Nc3cc4c(cnc(NC5CCC5)c4cn3)C(C)(C)N)nc2[C@H]1C |r|
CC(C)(N)c1cnc(OC2CC2)c2cnc(Nc3ccc4c(CCC(C)(C)OC4=O)n3)cc12
C[C@H]1OC(=O)c2ccc(Nc3cc4c(cnc(OC5CC5)c4cn3)C(C)(C)N)nc2C1(C)C |r|
CC[C@@H]1[C@H](C)OC(=O)c2ccc(Nc3cc4c(cnc(OC5CC5)c4cn3)C(C)(C)N)nc12 |r|
CC[C@@](C)(N)c1cnc(OC2CC2)c2cnc(Nc3ccc4C(=O)O[C@@](C)(CC)c4n3)cc12 |r|
CC[C@H]1OC(=O)c2ccc(Nc3cc4c(cnc(OC5CC5)c4cn3)C(C)(C)N)nc2[C@@H]1C |r|
CC[C@](C)(N)c1cnc(OC2CC2)c2cnc(Nc3ccc4C(=O)O[C@@H](C)[C@H](C)c4n3)cc12 |r|
CC[C@@](C)(N)c1cnc(OC2CC2)c2cnc(Nc3ccc4C(=O)OC(C)(C)Cc4n3)cc12 |r|
CC[C@](C)(N)c1cnc(OC2CC2)c2cnc(Nc3ccc4C(=O)OC(C)(C)Cc4n3)cc12 |r|
CC[C@@H]1OC(=O)c2ccc(Nc3cc4c(cnc(OC5CC5)c4cn3)C(C)(C)N)nc2[C@H]1C |r|
CC(C)(N)c1cnc(OC2(C)CC2)c2cnc(Nc3ccc4C(=O)OC(C)(C)Cc4n3)cc12
CC[C@@](C)(N)c1cnc(OC2CC2)c2cnc(Nc3ccc4C(=O)OCC(C)(C)c4n3)cc12 |r|
C[C@@H]1OC(=O)c2ccc(Nc3cc4c(cnc(OC5CC5)c4cn3)C(C)(C)N)nc2C1(C)C |r|
C[C@@H]1OC(=O)c2ccc(Nc3cc4c(cnc(OC5CC5)c4cn3)[C@](C)(N)CO)nc2[C@H]1C |r|
C[C@@H]1OC(=O)c2ccc(Nc3cc4c(cnc(OC5COC5)c4cn3)C(C)(C)N)nc2[C@H]1C |r|
CCCOc1ncc(c2cc(Nc3ccc4C(=O)O[C@@H](C)[C@H](C)c4n3)ncc12)[C@](C)(N)CC |r|
CCCOc1ncc(c2cc(Nc3ccc4C(=O)OC(C)(C)Cc4n3)ncc12)[C@](C)(N)CC |r|
CCCOc1ncc(c2cc(Nc3ccc4C(=O)OC(C)(C)Cc4n3)ncc12)[C@@](C)(N)CC |r|
CCCOc1ncc(c2cc(Nc3ccc4C(=O)O[C@@H](C)[C@H](C)c4n3)ncc12)[C@@](C)(N)CC |r|
C[C@@](N)(C1CC1)c1cnc(OC2CC2)c2cnc(Nc3ccc4C(=O)OCC5(CC5)c4n3)cc12 |r|
C[C@@](N)(C1CC1)c1cnc(OC2CC2)c2cnc(Nc3ccc4C(=O)OC5(CC5)Cc4n3)cc12 |r|
C[C@@](N)(C1CC1)c1cnc(OC2CC2)c2cnc(Nc3ccc4C(=O)NC(C)(C)Cc4n3)cc12 |r|
C[C@@H]1OC(=O)c2ccc(Nc3cc4c(cnc(NC5CC5)c4cn3)[C@](C)(N)C3CC3)nc2[C@H]1C |r|
C[C@@H]1OC(=O)c2ccc(Nc3cc4c(cnc(NC5CC5)c4cn3)[C@@](C)(N)C3CC3)nc2[C@H]1C |r|
C[C@@](N)(C1CC1)c1cnc(OC2CC2)c2cnc(Nc3ccc4C(=O)OCC(C)(C)c4n3)cc12 |r|
CC[C@]1(C)OC(=O)c2ccc(Nc3cc4c(cnc(OC5CC5)c4cn3)[C@](C)(N)C3CC3)nc12 |r|
C[C@](N)(C1CC1)c1cnc(OC2CC2)c2cnc(Nc3ccc4C(=O)OC(C)(C)Cc4n3)cc12 |r|
C[C@H]1OC(=O)c2ccc(Nc3cc4c(cnc(OC5CC5)c4cn3)[C@](C)(N)C3CC3)nc2[C@H]1C |r|
C[C@@H]1OC(=O)c2ccc(Nc3cc4c(cnc(OC5CC5)c4cn3)[C@](C)(N)C3CC3)nc2[C@@H]1C |r|
CC[C@@](C)(N)c1cnc(OC2CC2)c2cnc(Nc3ccc4C(=O)OC(C)(C)[C@H](C)c4n3)cc12 |r|
CC[C@](C)(N)c1cnc(OC2CC2)c2cnc(Nc3ccc4C(=O)O[C@H](C)C(C)(C)c4n3)cc12 |r|
COc1ncc(c2cc(Nc3ccc4C(=O)OC(C)(C)Cc4n3)ncc12)C(C)(C)NC1CCC1
C[C@@H]1OC(=O)c2ccc(Nc3cc4c(cnc(O[C@H]5CCOC5)c4cn3)C(C)(C)N)nc2[C@H]1C |r|
C[C@@H]1OC(=O)c2ccc(Nc3cc4c(cnc(O[C@@H]5CCOC5)c4cn3)C(C)(C)N)nc2[C@H]1C |r|
C[C@@H]1OC(=O)c2ccc(Nc3cc4c(cnc(O[C@H]5C[C@H](F)C5)c4cn3)C(C)(C)N)nc2[C@H]1C |r,wU:18.17,1.0,wD:32.37,20.20,(7.34,-2.08,;6,-1.31,;6,.23,;4.67,1,;4.67,2.54,;3.33,.23,;2,1,;.67,.23,;.67,-1.31,;-.67,-2.08,;-2,-1.31,;-3.33,-2.08,;-4.67,-1.31,;-6,-2.08,;-7.34,-1.31,;-7.34,.23,;-6,1,;-6,2.54,;-4.67,3.31,;-4.27,4.79,;-2.78,4.39,;-1.45,5.16,;-3.18,2.91,;-4.67,.23,;-3.33,1,;-2,.23,;-6,-3.62,;-7.34,-4.39,;-4.67,-4.39,;-6,-5.16,;2,-2.08,;3.33,-1.31,;4.67,-2.08,;4.67,-3.62,)|
C[C@@H]1OC(=O)c2ccc(Nc3cc4c(cnc(OCC5(F)CC5)c4cn3)C(C)(C)N)nc2[C@H]1C |r|
C[C@@H]1OC(=O)c2ccc(Nc3cc4c(cnc(O[C@@H]5C[C@H](F)C5)c4cn3)C(C)(C)N)nc2[C@H]1C |r,wU:1.0,wD:18.17,32.37,20.20,(7.34,-2.08,;6,-1.31,;6,.23,;4.67,1,;4.67,2.54,;3.33,.23,;2,1,;.67,.23,;.67,-1.31,;-.67,-2.08,;-2,-1.31,;-3.33,-2.08,;-4.67,-1.31,;-6,-2.08,;-7.34,-1.31,;-7.34,.23,;-6,1,;-6,2.54,;-4.67,3.31,;-4.27,4.79,;-2.78,4.39,;-1.45,5.16,;-3.18,2.91,;-4.67,.23,;-3.33,1,;-2,.23,;-6,-3.62,;-7.34,-4.39,;-4.67,-4.39,;-6,-5.16,;2,-2.08,;3.33,-1.31,;4.67,-2.08,;4.67,-3.62,)|
C[C@H](Oc1ncc(c2cc(Nc3ccc4C(=O)OC(C)(C)Cc4n3)ncc12)C(C)(C)N)C(F)F |r|
C[C@@H](Oc1ncc(c2cc(Nc3ccc4C(=O)OC(C)(C)Cc4n3)ncc12)C(C)(C)N)C(F)F |r|
C[C@@H]1OC(=O)c2ccc(Nc3cc4c(cnc(OCC(C)(F)F)c4cn3)C(C)(C)N)nc2[C@H]1C |r|
C[C@H]1OC(=O)c2ccc(Nc3cc4c(cnc(OC5CC5)c4cn3)[C@](C)(N)C3CC3)nc2C11CC1 |r|
C[C@@](N)(C1CCC1)c1cnc(OC2CC2)c2cnc(Nc3ccc4C(=O)OC(C)(C)Cc4n3)cc12 |r|
C[C@](N)(C1CCC1)c1cnc(OC2CC2)c2cnc(Nc3ccc4C(=O)OC(C)(C)Cc4n3)cc12 |r|
C[C@@H]1OC(=O)c2ccc(Nc3cc4c(cnc(OC5CC5)c4cn3)[C@](C)(N)C3CCC3)nc2[C@H]1C |r|
C[C@H]1OC(=O)c2ccc(Nc3cc4c(cnc(OC5CC5)c4cn3)[C@](C)(N)C3CC3)nc2C1(C)C |r|
CC[C@]1(C)OC(=O)c2ccc(Nc3cc4c(cnc(OCC(F)(F)F)c4cn3)C(C)(C)N)nc12 |r|
CC[C@](C)(N)c1cnc(OCC(F)(F)F)c2cnc(Nc3ccc4C(=O)OC(C)(C)c4n3)cc12 |r|
CC[C@@]1(C)OC(=O)c2ccc(Nc3cc4c(cnc(OCC(F)(F)F)c4cn3)C(C)(C)N)nc12 |r|
CC[C@@](C)(N)c1cnc(OCC(F)(F)F)c2cnc(Nc3ccc4C(=O)OC(C)(C)c4n3)cc12 |r|
CC(C)(N)c1cnc(OCC(F)(F)F)c2cnc(Nc3ccnc(n3)[C@@H]3CCC[C@@H](O)C3)cc12 |r|
CC(C)(NCCO)c1cnc(OC2CC2)c2cnc(Nc3ccc4C(=O)OC(C)(C)Cc4n3)cc12
C[C@@H]1OC(=O)c2ccc(Nc3cc4c(cnc(OC5CC(F)(F)C5)c4cn3)C(C)(C)N)nc2[C@H]1C |r|
C[C@@H](Oc1ncc(c2cc(Nc3ccc4C(=O)OC(C)(C)Cc4n3)ncc12)C(C)(C)N)C(F)(F)F |r|
C[C@H](Oc1ncc(c2cc(Nc3ccc4C(=O)OC(C)(C)Cc4n3)ncc12)C(C)(C)N)C(F)(F)F |r|
CC[C@@](C)(N)c1cnc(OCC(F)(F)F)c2cnc(Nc3ccc4C(=O)O[C@@H](C)[C@H](C)c4n3)cc12 |r|
CC(C)(NC1COC1)c1cnc(OC2CC2)c2cnc(Nc3ccc4C(=O)OC(C)(C)Cc4n3)cc12
COC[C@](C)(N)c1cnc(OC2CC2)c2cnc(Nc3ccc4C(=O)O[C@H](C)[C@@H](C)c4n3)cc12 |r|
C[C@@](N)(C1CC1)c1cnc(OC2(C)CC2)c2cnc(Nc3ccc4C(=O)OCC(C)(C)c4n3)cc12 |r|
C[C@@H]1OC(=O)c2ccc(Nc3cc4c(cnc(OC5(C)CC5)c4cn3)C(C)(C)N)nc2C1(C)C |r|
CC[C@](C)(N)c1cnc(OC2CC2)c2cnc(Nc3ccc4C(=O)O[C@@H](C)C5(CC5)c4n3)cc12 |r|
COC[C@@](C)(N)c1cnc(OC)c2cnc(Nc3ccc4C(=O)O[C@@H](C)[C@H](C)c4n3)cc12 |r|
COC[C@@](C)(N)c1cnc(OC2CC2)c2cnc(Nc3ccc4C(=O)OC(C)(C)[C@H](C)c4n3)cc12 |r|
COC[C@@](C)(N)c1cnc(OC2CC2)c2cnc(Nc3ccc4C(=O)O[C@@H](C)[C@@H](C)c4n3)cc12 |r|
CC[C@@H](N)c1cnc(OC2(C)CC2)c2cnc(Nc3ccc4C(=O)OC(C)(C)[C@H](C)c4n3)cc12 |r|
COC[C@@](C)(N)c1cnc(OC)c2cnc(Nc3ccc4C(=O)OC(C)(C)[C@H](C)c4n3)cc12 |r|
C[C@@H]1OC(=O)c2ccc(Nc3cc4c(cnc(O[C@H]5C[C@H](O)C5)c4cn3)[C@@](C)(N)C3CC3)nc2[C@H]1C |r,wU:26.29,18.17,34.40,wD:26.30,20.20,1.0,(8.16,8.71,;6.82,7.94,;6.82,6.4,;5.49,5.63,;5.49,4.09,;4.15,6.4,;2.82,5.63,;1.49,6.4,;1.49,7.94,;.15,8.71,;-1.18,7.94,;-2.51,8.71,;-3.85,7.94,;-5.18,8.71,;-6.51,7.94,;-6.51,6.4,;-5.18,5.63,;-5.18,4.09,;-3.85,3.32,;-2.36,3.72,;-1.96,2.23,;-.63,1.46,;-3.45,1.83,;-3.85,6.4,;-2.51,5.63,;-1.18,6.4,;-5.18,10.25,;-4.41,11.58,;-3.64,10.25,;-6.67,10.65,;-7.76,11.73,;-8.16,10.25,;2.82,8.71,;4.15,7.94,;5.49,8.71,;5.49,10.25,)|
CC[C@@H](N)c1cnc(OC)c2cnc(Nc3ccc4C(=O)O[C@@H](C)[C@H](C)c4n3)cc12 |r|
CC(C)(N)c1cnc(OC2CC2)c2cnc(Nc3ccc4C(=O)OC(C)(C)C5(CC5)c4n3)cc12
CC[C@](C)(N)c1cnc(OC2CC2)c2cnc(Nc3ccc4C(=O)OC(C)(C)C5(CC5)c4n3)cc12 |r|
C[C@@H]1OC(=O)c2ccc(Nc3cc4c(cnc(OC5(C)COC5)c4cn3)C(C)(C)N)nc2[C@H]1C |r|
CC(C)(N)c1cnc(OC2(C)COC2)c2cnc(Nc3cnc4C(=O)OC(C)(C)C(=O)c4c3)cc12
CC(C)(N)c1cnc(OC2(C)CC2)c2cnc(Nc3ccc4C(=O)OC(C)(C)C5(CC5)c4n3)cc12
COC[C@@](C)(N)c1cnc(OC2CC2)c2cnc(Nc3ccc4C(=O)OC(C)(C)Cc4n3)cc12 |r|
CC[C@@H](N)c1cnc(C)c2cnc(Nc3ccc4C(=O)O[C@@H](C)[C@H](C)c4n3)cc12 |r|
CC[C@@H](N)c1cnc(OC)c2cnc(Nc3ccc4C(=O)OC(C)(C)[C@H](C)c4n3)cc12 |r|
COC[C@@](C)(N)c1cnc(C)c2cnc(Nc3ccc4C(=O)O[C@@H](C)[C@H](C)c4n3)cc12 |r|
COC[C@@](C)(N)c1cnc(C)c2cnc(Nc3ccc4C(=O)OC(C)(C)[C@H](C)c4n3)cc12 |r|
CC[C@@H](N)c1ccc(OC)c2cnc(Nc3ccc4C(=O)OC(C)(C)C5(CC5)c4n3)cc12 |r|
COC[C@@H](N)c1cnc(OC)c2cnc(Nc3ccc4C(=O)OC(C)(C)[C@H](C)c4n3)cc12 |r|
CC[C@@H](N)c1ccc(Cl)c2cnc(Nc3ccc4C(=O)OC(C)(C)[C@H](C)c4n3)cc12 |r|
CC[C@@H](N)c1cnc(C)c2cnc(Nc3ccc4C(=O)OC(C)(C)[C@H](C)c4n3)cc12 |r|
CNCc1cc(F)c(c(F)c1)-c1ncc2[nH]nc(-c3ccc(NC4CCN(CC4)S(C)(=O)=O)cc3)c2n1
CNCc1cc(F)c(-c2ncc3[nH]nc(-c4ccc(nc4)N4CCCCC4)c3n2)c(c1)C(F)(F)F
CN1CCN(CC1)c1ncc(cn1)-c1n[nH]c2cnc(nc12)-c1c(F)cc(CC#N)cc1F
COc1ncc([C@@H](C)O)c2cc(Nc3ccnc(n3)C(C)(C)F)ncc12 |r|
COc1ncc([C@H](C)O)c2cc(Nc3ccnc(n3)C(C)(C)F)ncc12 |r|
CNc1ncc(c2cc(Nc3ccnc(n3)C(C)(C)C)ncc12)C(C)(C)O
COc1ncc(c2cc(Nc3ccnc(n3)C(C)(C)F)ncc12)C(C)(C)O
COc1ncc(c2cc(Nc3cnc(C#N)c(n3)C(C)C)ncc12)C(C)(C)O
COc1ncc(c2cc(Nc3ccc4C(=O)OCCc4n3)ncc12)C(C)(C)O
COc1ncc(c2cc(Nc3ccnc(n3)N3CCCC3)ncc12)C(C)(C)O
COc1ncc(c2cc(Nc3ccnc(n3)N3CCC[C@@H]3C)ncc12)C(C)(C)O |r|
COc1ncc(c2cc(Nc3ccnc(n3)C(C)(C)F)ncc12)[C@@](C)(O)C(F)F |r|
COc1ncc(c2cc(Nc3ccnc(n3)C(C)(C)F)ncc12)[C@](C)(O)C(F)F |r|
COc1ncc(c2cc(Nc3cnc(C#N)c(n3)N3CCC[C@@H]3C)ncc12)C(C)(C)O |r|
CC[C@@H](O)c1cnc(OC)c2cnc(Nc3ccc4C(=O)OC(C)(C)[C@H](C)c4n3)cc12 |r|
CC[C@H](O)c1cnc(OC)c2cnc(Nc3ccc4C(=O)OC(C)(C)[C@H](C)c4n3)cc12 |r|
CC[C@@](C)(O)c1cnc(OC)c2cnc(Nc3ccc4C(=O)OC(C)(C)[C@H](C)c4n3)cc12 |r|
COC[C@@H](O)c1cnc(OC)c2cnc(Nc3ccc4C(=O)OC(C)(C)[C@H](C)c4n3)cc12 |r|
COC[C@H](O)c1cnc(OC)c2cnc(Nc3ccc4C(=O)OC(C)(C)[C@H](C)c4n3)cc12 |r|
CC[C@](C)(O)c1cnc(NC2CC2)c2cnc(Nc3ccc4C(=O)O[C@@H](C)[C@H](C)c4n3)cc12 |r|
CC[C@@](C)(O)c1cnc(NC2CC2)c2cnc(Nc3ccc4C(=O)O[C@@H](C)[C@H](C)c4n3)cc12 |r|
CC(C)(O)c1cnc(OC2CC2)c2cnc(Nc3ccc4c(CCC(C)(C)OC4=O)n3)cc12
CCOc1ncc(c2cc(Nc3ccc4C(=O)OC(C)(C)[C@H](C)c4n3)ncc12)[C@](C)(O)CC |r|
CCOc1ncc(c2cc(Nc3ccc4C(=O)OC(C)(C)[C@H](C)c4n3)ncc12)[C@@](C)(O)CC |r|
C[C@@H]1OC(=O)c2ccc(Nc3cc4c(cnc(OC5CC5)c4cn3)[C@@](C)(O)C3CC3)nc2[C@H]1C |r|
Cn1ccc2c(cccc12)-c1ccc(Nc2ccc(cn2)C2CCNCC2)c2C(=O)NCc12
CC1=CC2N=CC(=C2C=C1)c1ccc(Nc2ccc(cn2)N2CCC(O)CC2)c2C(=O)NCc12 |c:4,6,9,t:1|
COC1CCN(CC1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3c(F)cccn23)nc1
CC(C)(O)[C@H]1CN(CCO1)c1ccc(Nc2cnc(c3CNC(=O)c23)-c2cnc3cnccn23)nc1 |r|
CN(C)Cc1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3ccccn23)ccc1[C@@H]1CCOC1 |r|
CO[C@H]1CC[C@@H](C1)c1ccc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)nc1CN(C)C |r|
CN1CCN(CC1)c1nc(Nc2ccc(c3CNC(=O)c23)-c2cnc3cc(F)ccn23)ccc1C1CCOC1
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(CC(C)C)cccc3n2C(=O)OC(C)(C)C)c1=O
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(CC(C)C)cccc3[nH]2)c1=O
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(CC(C)C)c(F)cc(F)c3[nH]2)c1=O
CC(C)Cc1cccc2[nH]c(Cn3cccc(NC(=O)[C@H](CC\C=C\C(N)=O)NC(=O)OCc4ccccc4)c3=O)nc12 |r|
COC(=O)N[C@@H](CC\C=C\C(N)=O)C(=O)Nc1cccn(Cc2nc3c(CC(C)C)cccc3n2C(=O)OC(C)(C)C)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(N)=O)C(=O)Nc1cccn(Cc2nc3c(CC(C)C)cccc3[nH]2)c1=O |r|
CC(C)Cc1cccc2n(C(=O)OC(C)(C)C)c(Cn3cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)NC(=O)OCc4ccccc4)c3=O)nc12 |r|
CC(C)Cc1cccc2[nH]c(Cn3cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)NC(=O)OCc4ccccc4)c3=O)nc12 |r|
CC(C)Cc1cccc2n(C(=O)OC(C)(C)C)c(Cn3cccc(NC(=O)[C@H](CC\C=C\C(N)=O)NC(=O)OC4CCOC4)c3=O)nc12 |r,w:38.38|
CC(C)Cc1cccc2[nH]c(Cn3cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)NC(=O)OCC4CCOC4)c3=O)nc12 |r,w:34.34|
CC(C)Cc1cccc2[nH]c(Cn3cccc(NC(=O)[C@H](CC\C=C\C(N)=O)NC(=O)OC4CCOC4)c3=O)nc12 |r,w:31.31|
CC(C)Cc1cccc2n(C(=O)OC(C)(C)C)c(Cn3cccc(NC(=O)[C@H](CC\C=C\C(N)=O)NC(=O)OCC4CCOC4)c3=O)nc12 |r,w:39.39|
CC(C)Cc1cccc2[nH]c(Cn3cccc(NC(=O)[C@H](CC\C=C\C(N)=O)NC(=O)OCC4CCOC4)c3=O)nc12 |r,w:32.32|
CC(C)Cc1cccc2[nH]c(Cn3cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)NC(=O)OCCO)c3=O)nc12 |r|
CNC(=O)\C=C\CC[C@H](NC(=O)OC)C(=O)Nc1cccn(Cc2nc3c(CC(C)C)cccc3n2C(=O)OC(C)(C)C)c1=O |r|
CNC(=O)\C=C\CC[C@H](NC(=O)OC)C(=O)Nc1cccn(Cc2nc3c(CC(C)C)cccc3[nH]2)c1=O |r|
CC(C)Cc1cccc2n(C(=O)OC(C)(C)C)c(Cn3cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c3=O)nc12 |r|
CC(C)Cc1cccc2nc(Cn3cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c3=O)[nH]c12 |r|
CC(C)Cc1c(F)c(F)cc2nc(Cn3cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c3=O)[nH]c12 |r|
CC(C)Cc1c(F)c(F)cc2n(C(=O)OC(C)(C)C)c(Cn3cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c3=O)nc12 |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3cc(F)c(F)c(CC(C)C)c3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(CC(C)C)c(F)c(F)cc3n2C(=O)OC(C)(C)C)c1=O |r|
CC(C)Cc1cc(F)cc2nc(Cn3cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c3=O)[nH]c12 |r|
CC(C)Cc1cc(F)cc2n(C(=O)OC(C)(C)C)c(Cn3cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c3=O)nc12 |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(CC(C)C)cc(F)cc3[nH]2)c1=O |r,$;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;NH;;$|
CC(C)Cc1cc(F)cc2nc(Cn3cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)NC(=O)N(C)C)c3=O)[nH]c12 |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(C=C(C)C)ncnc3[nH]2)c1=O |r,wD:5.4,(-4.6,-4.42,;-3.27,-5.19,;-1.94,-4.42,;-1.94,-2.88,;-.6,-5.19,;-.6,-6.73,;-1.94,-7.5,;-3.27,-6.73,;-4.6,-7.5,;-5.94,-6.73,;-7.27,-7.5,;-7.27,-9.04,;-8.6,-6.73,;-8.6,-5.19,;-9.94,-7.5,;.73,-7.5,;.73,-9.04,;2.07,-6.73,;3.4,-7.5,;3.4,-9.04,;4.73,-9.81,;6.07,-9.04,;6.07,-7.5,;7.4,-6.73,;8.73,-7.5,;8.89,-9.04,;10.4,-9.36,;11.17,-10.69,;10.4,-12.02,;11.17,-13.36,;12.71,-13.36,;10.4,-14.69,;12.71,-10.69,;13.48,-9.36,;12.71,-8.02,;11.17,-8.02,;10.14,-6.88,;4.73,-6.73,;4.73,-5.19,)|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(CC(C)C)ncnc3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(CC(C)C)c(F)cc(F)c3n2C(=O)OC(C)(C)C)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(CC(C)C)c(F)cc(F)c3[nH]2)c1=O |r|
CC(C)Cc1cccc2n(C(=O)OC(C)(C)C)c(Cn3cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)NC(=O)OC(C)(C)C)c3=O)nc12 |r|
CC(C)Cc1cccc2[nH]c(Cn3cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)NC(=O)c4cnco4)c3=O)nc12 |r|
CC(C)Cc1cccc2[nH]c(Cn3cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)NC(=O)c4ncccn4)c3=O)nc12 |r|
CC(C)Cc1cccc2[nH]c(Cn3cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)NC(=O)c4ccccc4F)c3=O)nc12 |r|
CC(C)Cc1cccc2[nH]c(Cn3cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)NC(=O)c4ncco4)c3=O)nc12 |r|
CC(C)Cc1cccc2[nH]c(Cn3cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)NC(=O)c4cncn4C)c3=O)nc12 |r|
CC(C)Cc1cccc2[nH]c(Cn3cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)NC(=O)c4nccn4C)c3=O)nc12 |r|
CC(C)Cc1cccc2[nH]c(Cn3cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)NC(=O)c4ccccn4)c3=O)nc12 |r|
COCCC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(CC(C)C)cccc3[nH]2)c1=O |r|
COCC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3cccc(CC(C)C)c3[nH]2)c1=O |r|
CC(C)Cc1cccc2nc(Cn3cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)NC(=O)C4CCCO4)c3=O)[nH]c12 |r,w:31.32|
COCCOC(=O)N[C@@H](CC\C=C\C(N)=O)C(=O)Nc1cccn(Cc2nc3ccccc3n2C(=O)OC(C)(C)C)c1=O |r|
COCCOC(=O)N[C@@H](CC\C=C\C(N)=O)C(=O)Nc1cccn(Cc2nc3ccccc3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(N)=O)C(=O)Nc1cccn(Cc2nc3ccccc3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3ccccc3[nH]2)c1=O |r|
CN(C)C(=O)\C=C\CC[C@H](NC(=O)OCc1ccccc1)C(=O)Nc1cccn(Cc2nc3ccccc3[nH]2)c1=O |r|
CN(C)C(=O)\C=C\CC[C@H](NC(=O)OC(C)(C)C)C(=O)Nc1cccn(Cc2nc3ccccc3n2C(=O)OC(C)(C)C)c1=O |r|
CNC(=O)\C=C\CC[C@H](NC(=O)OC)C(=O)Nc1cccn(Cc2nc3ccccc3n2C(=O)OC(C)(C)C)c1=O |r|
CNC(=O)\C=C\CC[C@H](NC(=O)OC)C(=O)Nc1cccn(Cc2nc3ccccc3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3cc(F)ccc3[nH]2)c1=O |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3cc(F)c(F)cc3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3cc(F)c(F)cc3n2C(=O)OC(C)(C)C)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3cc(F)c(F)cc3[nH]2)c1=O |r|
CN(C)C(=O)OC(CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3cc(F)ccc3[nH]2)c1=O |w:6.5|
CN(C)C(=O)OC(CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3cc(F)ccc3[nH]2)c1=O
NC(=O)\C=C\CC[C@H](NC(=O)OCCO)C(=O)Nc1cccn(Cc2nc3ccccc3[nH]2)c1=O |r|
CC(C)[C@H](N)C(=O)N[C@@H](C(C)C)C(=O)OCCOC(=O)N[C@@H](CC\C=C\C(N)=O)C(=O)Nc1cccn(Cc2nc3ccccc3[nH]2)c1=O |r|
CN(C)C(=O)\C=C\CC[C@H](NC(=O)CO)C(=O)Nc1cccn(Cc2nc3ccccc3[nH]2)c1=O |r|
CN(C)C(=O)\C=C\CC[C@H](NC(=O)CCO)C(=O)Nc1cccn(Cc2nc3ccccc3[nH]2)c1=O |r|
CN(C)C(=O)\C=C\CC[C@H](NC(=O)CCCO)C(=O)Nc1cccn(Cc2nc3ccccc3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)NCCO)C(=O)Nc1cccn(Cc2nc3ccccc3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(CC(C)(C)C)cc(F)cc3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N1CCCC1)C(=O)Nc1cccn(Cc2nc3c(CC(C)(C)C)cc(F)cc3[nH]2)c1=O |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3cc(F)cc(CC(C)(C)C)c3[nH]2)c1=O |r|
COCCOC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(CC(C)(C)C)cc(F)cc3[nH]2)c1=O |r|
COCCN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3cc(F)cc(CC(C)(C)C)c3[nH]2)c1=O |r|
CN(C)C(=O)N[C@@H](CC\C=C\C(=O)N1CCCC1)C(=O)Nc1cccn(Cc2nc3cc(F)cc(CC(C)(C)C)c3[nH]2)c1=O |r|
COc1cc(CC(C)(C)C)c2nc(Cn3cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c3=O)n(C(=O)OC(C)(C)C)c2c1 |r|
COc1cc(CC(C)(C)C)c2nc(Cn3cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c3=O)[nH]c2c1 |r|
COC(=O)N[C@@H](CC\C=C\C(N)=O)C(=O)Nc1cccn(Cc2nc3c(CC(C)(C)C)cccc3n2C(=O)OC(C)(C)C)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(CC(C)(C)C)cccc3n2C(=O)OC(C)(C)C)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(N)=O)C(=O)Nc1cccn(Cc2nc3cccc(CC(C)(C)C)c3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3cccc(CC(C)(C)C)c3[nH]2)c1=O |r|
CN(C)C(=O)\C=C\CC[C@H](NC(=O)OCC1CCOCC1)C(=O)Nc1cccn(Cc2nc3c(CC(C)(C)C)cccc3n2C(=O)OC(C)(C)C)c1=O |r|
CN(C)C(=O)\C=C\CC[C@H](NC(=O)OCC1CCOCC1)C(=O)Nc1cccn(Cc2nc3cccc(CC(C)(C)C)c3[nH]2)c1=O |r|
CN(C)C(=O)\C=C\CC[C@H](NC(=O)OC1CCOC1)C(=O)Nc1cccn(Cc2nc3c(CC(C)(C)C)cccc3[nH]2)c1=O |r,w:13.13|
CC(C)(C)Cc1cccc2n(C(=O)OC(C)(C)C)c(Cn3cccc(NC(=O)[C@H](CC\C=C\C(N)=O)NC(=O)OC4CCOC4)c3=O)nc12 |r,w:39.39|
CC(C)(C)Cc1cccc2[nH]c(Cn3cccc(NC(=O)[C@H](CC\C=C\C(N)=O)NC(=O)OC4CCOC4)c3=O)nc12 |r,w:32.32|
CC(C)(C)Cc1cccc2n(C(=O)OC(C)(C)C)c(Cn3cccc(NC(=O)[C@H](CC\C=C\C(N)=O)NC(=O)OCC4CCOCC4)c3=O)nc12 |r|
CC(C)(C)Cc1cccc2[nH]c(Cn3cccc(NC(=O)[C@H](CC\C=C\C(N)=O)NC(=O)OCC4CCOCC4)c3=O)nc12 |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(CC(C)(C)C)cc(F)cc3n2C)c1=O |r|
COCCOC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(CC(C)(C)C)cc(F)cc3n2C)c1=O |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1ccnn(Cc2nc3c(CC(C)(C)C)cc(F)cc3n2C(=O)OC(C)(C)C)c1=O |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1ccnn(Cc2nc3c(CC(C)(C)C)cc(F)cc3n2C)c1=O |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1nccn(Cc2nc3c(CC(C)(C)C)cc(F)cc3n2C(=O)OC(C)(C)C)c1=O |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1nccn(Cc2nc3cc(F)cc(CC(C)(C)C)c3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(CCC(F)(F)F)cc(F)cc3n2C(=O)OC(C)(C)C)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3cc(F)cc(CCC(F)(F)F)c3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(N)=O)C(=O)Nc1cccn(Cc2nc3c(CCC(F)(F)F)cccc3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(CCC(F)(F)F)cccc3[nH]2)c1=O |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3cc(F)cc(CCC(F)(F)F)c3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N1CCCC1)C(=O)Nc1cccn(Cc2nc3c(CCC(F)(F)F)cc(F)cc3n2C(=O)OC(C)(C)C)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N1CCCC1)C(=O)Nc1nccn(Cc2nc3c(CCC(F)(F)F)cc(F)cc3[nH]2)c1=O |r|
CNC(=O)\C=C\CC[C@H](OC(=O)N(C)C)C(=O)Nc1nccn(Cc2nc3cc(F)cc(CCC(F)(F)F)c3n2C(=O)OC(C)(C)C)c1=O |r|
CNC(=O)\C=C\CC[C@H](OC(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3cc(F)cc(CCC(F)(F)F)c3[nH]2)c1=O |r|
COC(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(F)cc(F)c(CCC(F)(F)F)c3[nH]2)c1=O |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(CCC(F)(F)F)c(F)cc(F)c3n2C(=O)OC(C)(C)C)c1=O |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(F)cc(F)c(CCC(F)(F)F)c3[nH]2)c1=O |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(CCC(F)(F)F)cc(F)cc3n2C)c1=O |r|
COCCOC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(CCC(F)(F)F)cc(F)cc3n2C)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(CCC(F)(F)F)cc(F)cc3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(CC4CC4)cc(F)cc3n2C(=O)OC(C)(C)C)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(CC4CC4)cc(F)cc3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(CC4CC4)cccc3n2C(=O)OC(C)(C)C)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(CC4CC4)cccc3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(N)=O)C(=O)Nc1cccn(Cc2nc3c(CC4CC4)cccc3n2C(=O)OC(C)(C)C)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(N)=O)C(=O)Nc1cccn(Cc2nc3c(CC4CC4)cccc3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(Oc4ccc(F)cc4F)cccc3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(Oc4ccccc4)cccc3n2C(=O)OC(C)(C)C)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3cccc(Oc4ccccc4)c3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(N)=O)C(=O)Nc1cccn(Cc2nc3c(Oc4ccccc4)cccc3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3ccc(Oc4ccc(F)cc4F)cc3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(OCc4ccc(F)cc4F)cccc3[nH]2)c1=O |r|
CC(C)Oc1cccc2[nH]c(Cn3cccc(NC(=O)[C@H](CC\C=C\C(N)=O)NC(=O)OCc4ccccc4)c3=O)nc12 |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3cccc(OCc4ccccc4)c3[nH]2)c1=O |r|
CC(C)COc1cccc2nc(Cn3cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)NC(=O)OCc4ccccc4)c3=O)n(C)c12 |r|
COC(=O)N[C@@H](CC\C=C\C(N)=O)C(=O)Nc1cccn(Cc2nc3cccc(OCC(C)C)c3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(N)=O)C(=O)Nc1cccn(Cc2nc3cccc(OCc4ccccc4)c3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(N)=O)C(=O)Nc1cccn(Cc2nc3c(OC(C)C)cccc3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(N)=O)C(=O)Nc1cccn(Cc2nc3cccc(OCC4CC4)c3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3ccc(OCc4ccc(F)cc4F)cc3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(OCC(F)F)cc(F)cc3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(N)=O)C(=O)Nc1cccn(Cc2nc3c(OCC(F)F)cc(F)cc3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(OCC(F)(F)F)cc(F)cc3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(N)=O)C(=O)Nc1cccn(Cc2nc3c(OCC(F)(F)F)cc(F)cc3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3cc(F)cc(OCc4ccc(F)cc4F)c3[nH]2)c1=O |r|
CNC(=O)\C=C\CC[C@H](NC(=O)OC)C(=O)Nc1cccn(Cc2nc3c(OCc4ccc(F)cc4F)cc(F)cc3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(N)=O)C(=O)Nc1cccn(Cc2nc3cc(F)cc(OCc4ccc(F)cc4F)c3[nH]2)c1=O |r|
COCCOC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3cc(F)cc(OCc4ccc(F)cc4F)c3[nH]2)c1=O |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3cc(F)cc(OCc4ccc(F)cc4F)c3[nH]2)c1=O |r|
COCCN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3cc(F)cc(OCc4ccc(F)cc4F)c3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3cc(F)cc(OC(F)(F)C(F)F)c3[nH]2)c1=O |r|
CN(C)C(=O)\C=C\CC[C@H](NC(=O)c1ncco1)C(=O)Nc1cccn(Cc2nc3cccc(Oc4ccc(F)cc4F)c3[nH]2)c1=O |r|
COCC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3cccc(Oc4ccc(F)cc4F)c3[nH]2)c1=O |r|
CN(C)C(=O)\C=C\CC[C@H](NC(=O)c1cncn1C)C(=O)Nc1cccn(Cc2nc3cccc(Oc4ccc(F)cc4F)c3[nH]2)c1=O |r|
CN(C)C(=O)\C=C\CC[C@H](NC(=O)c1ncco1)C(=O)Nc1cccn(Cc2nc3c(OCc4ccc(F)cc4F)cccc3[nH]2)c1=O |r|
COCC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3cccc(OCc4ccc(F)cc4F)c3[nH]2)c1=O |r|
CN(C)C(=O)\C=C\CC[C@H](NC(=O)c1nccn1C)C(=O)Nc1cccn(Cc2nc3c(OCc4ccc(F)cc4F)cccc3[nH]2)c1=O |r|
CN(C)C(=O)\C=C\CC[C@H](NC(=O)C1CCC(F)(F)CC1)C(=O)Nc1cccn(Cc2nc3cccc(OCc4ccc(F)cc4F)c3[nH]2)c1=O |r|
COCC(=O)N[C@@H](CC\C=C\C(N)=O)C(=O)Nc1cccn(Cc2nc3cc(F)cc(OCc4ccc(F)cc4F)c3[nH]2)c1=O |r|
NC(=O)\C=C\CC[C@H](NC(=O)c1ccc(F)cn1)C(=O)Nc1cccn(Cc2nc3cc(F)cc(OCc4ccc(F)cc4F)c3[nH]2)c1=O |r|
COCC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(OCc4ccc(F)cc4F)cc(F)cc3[nH]2)c1=O |r|
CN(C)C(=O)\C=C\CC[C@H](NC(=O)c1ccc(F)cn1)C(=O)Nc1cccn(Cc2nc3c(OCc4ccc(F)cc4F)cc(F)cc3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(COc4ccc(F)cc4F)cccc3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(COC(C)C)cccc3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(CC(C(F)(F)F)C(F)(F)F)cccc3n2COCC[Si](C)(C)C)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(CC(C(F)(F)F)C(F)(F)F)cccc3[nH]2)c1=O |r,$;;;;;;;;;;;;;;;;;N;;;;;;;;;;;;;;;;;;;;;;;;;N;;$|
COC(=O)N[C@@H](CC\C=C\C(N)=O)C(=O)Nc1cccn(Cc2nc3c(CC(C(F)(F)F)C(F)(F)F)cccc3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(cccc3[nH]2)C(O)C(C)C)c1=O |r,w:33.35,$;;;;;;;;;;;;;;;;;N;;;;;;;;;;;;;;;N;;;;;;;$|
COC(=O)N[C@@H](CC\C=C\C(N)=O)C(=O)Nc1cccn(Cc2nc3c(cccc3[nH]2)C(O)C(C)C)c1=O |r,w:31.33|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3cccc(C(O)C(C)C)c3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3cccc(C(F)C(C)C)c3[nH]2)c1=O |r,w:31.31|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3cccc(C(O)C(C)(C)C)c3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(N)=O)C(=O)Nc1cccn(Cc2nc3cccc(C(O)C(C)(C)C)c3[nH]2)c1=O |r|
CC(C)C(O)c1cccc2nc(Cn3cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)NC(=O)OC(C)(C)C)c3=O)[nH]c12 |r,w:3.3|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(CC(C)(C)C)ccc(F)c3[nH]2)c1=O |r|
CN(C)C(=O)\C=C\CC[C@H](NC(=O)c1ncco1)C(=O)Nc1cccn(Cc2nc3cccc(C(O)C(C)(C)C)c3[nH]2)c1=O |r,w:34.35|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3cccc(C(=O)C(C)(C)C)c3[nH]2)c1=O |r,$;;;;;;;;;;;;;;;;;N;;;;;;;;;;;;;;;;;;;;;;;$|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3cccc(C(F)C(C)(C)C)c3[nH]2)c1=O |r,w:31.31,$;;;;;;;;;;;;;;;;;N;;;;;;;;;;;;;;;;;;;;;;;$|
COC(=O)N[C@@H](CC\C=C\C(N)=O)C(=O)Nc1cccn(Cc2nc3c(cccc3[nH]2)C(F)C(C)(C)C)c1=O |r,w:31.33|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(cccc3[nH]2)C(F)(F)C(C)(C)O)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(cccc3[nH]2)C(F)(F)C(C)C)c1=O |r,$;;;;;;;;;;;;;;;;;N;;;;;;;;;;;;;;;N;;;;;;;;$|
COC(=O)N[C@@H](CC\C=C\C(N)=O)C(=O)Nc1cccn(Cc2nc3c(cccc3[nH]2)C(F)(F)C(C)C)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(cccc3[nH]2)C(F)(F)C(C)=C)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(N)=O)C(=O)Nc1cccn(Cc2nc3c(cccc3[nH]2)C(F)(F)C(C)=C)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3cc(F)cc(OC(C)(C)C)c3[nH]2)c1=O
COC(=O)N[C@@H](CC\C=C\C(N)=O)C(=O)Nc1cccn(Cc2nc3cc(F)cc(OC(C)(C)C)c3[nH]2)c1=O |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3cc(F)ccc3n2C)c1=O
CN(C)C(=O)\C=C\CC[C@H](NC([O-])=O)C(=O)Nc1cncn(Cc2nc3cc(F)ccc3n2C)c1=O
CC(C)CCn1c(Cn2cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c2=O)nc2cc(F)c(F)cc12 |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3cc(F)ccc3n2CC2CC2)c1=O |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3cc(F)ccc3n2CC(C)(C)C)c1=O |r|
CCn1c(Cn2cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c2=O)nc2cc(F)ccc12 |r|
CC(C)Cn1c(Cn2cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c2=O)nc2cc(F)ccc12 |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3cc(F)ccc3n2CCC(F)(F)F)c1=O |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3cc(F)c(F)cc3n2CCC2CC2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3cc(F)c(F)cc3n2CCC2CC2)c1=O |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cncn(Cc2nc3cc(F)ccc3n2CCC(F)(F)F)c1=O |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cncn(Cc2nc3cc(F)ccc3n2Cc2ccccc2)c1=O |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3cc(F)ccc3n2Cc2ccc(F)cc2F)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cncn(Cc2nc3cc(F)ccc3n2Cc2ccc(F)cc2F)c1=O |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cncn(Cc2nc3cc(F)ccc3n2CC(C)(C)C)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)NC1=CB=CN(Cc2nc3cc(F)ccc3n2Cc2ccc(F)cc2)C1=O |r,c:20,t:18|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cncn(Cc2nc3cc(F)ccc3n2CC2CC2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cncn(Cc2nc3cc(F)ccc3n2CC(C)C)c1=O |r|
CCn1c(Cn2cncc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c2=O)nc2cc(F)ccc12 |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cncn(Cc2nc3cc(F)ccc3n2C)c1=O |r|
CCOC(=O)n1c(Cn2cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c2=O)nc2cc(F)ccc12
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3cc(F)ccc3n2C(=O)OCC2CC2)c1=O
COC(=O)n1c(Cn2cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c2=O)nc2cc(F)ccc12 |r|
CCOC(=O)n1c(Cn2cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c2=O)nc2cc(F)c(F)cc12 |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3cc(F)c(F)cc3n2C(=O)OCC2CC2)c1=O |r|
CCOC(=O)n1c(Cn2cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)NC(=O)OC)c2=O)nc2cc(F)c(F)cc12 |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3cc(F)ccc3n2C(=O)OCC2CC2)c1=O |r|
CCOC(=O)n1c(Cn2cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)NC(=O)OC)c2=O)nc2cc(F)ccc12 |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cncn(Cc2nc3cc(F)ccc3n2C(=O)OC)c1=O
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3cc(F)ccc3n2-c2ccccc2)c1=O |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3cc(F)ccc3n2Cc2ccc(F)cc2)c1=O |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3ccc(F)cc3n2Cc2ccc(F)cc2)c1=O |r|
COC(=O)N[C@@H](CC/C=C/C(=O)N(C)C)C(=O)Nc3cccn(Cc2cc1cc(F)ccc1[nH]2)c3=O
COC(=O)N[C@@H](CC\C=C\C(=O)N1CCCC1)C(=O)Nc1cccn(Cc2cc3cc(F)ccc3n2C(=O)OC(C)(C)C)c1=O |r|
CC(C)(C)OC(=O)n1c(Cn2cccc(NC(=O)[C@H](CC\C=C\C(=O)N3CCCC3)NC(=O)OCCO)c2=O)cc2cc(F)ccc12 |r|
OCCOC(=O)N[C@@H](CC\C=C\C(=O)N1CCCC1)C(=O)Nc1cccn(Cc2cc3cc(F)ccc3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(N)=O)C(=O)Nc1cccn(Cc2cc3cc(F)ccc3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N1CCCC1)C(=O)Nc1cccn(Cc2cc3cc(F)ccc3[nH]2)c1=O |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3cc(F)ccc3[nH]2)c1=O |r|
COCCN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3cc(F)ccc3[nH]2)c1=O |r|
CN(C)C(=O)\C=C\CC[C@H](OC(=O)N1CCCC1)C(=O)Nc1cccn(Cc2cc3cc(F)ccc3[nH]2)c1=O |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(N)=O)C(=O)Nc1cccn(Cc2cc3cc(F)ccc3n2C(=O)OC(C)(C)C)c1=O |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(N)=O)C(=O)Nc1cccn(Cc2cc3cc(F)ccc3[nH]2)c1=O |r|
COCCN(CCOC)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3cc(F)ccc3n2C(=O)OC(C)(C)C)c1=O |r|
COCCN(CCOC)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3cc(F)ccc3[nH]2)c1=O |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3cc(F)ccc3n2C(=O)OCc2ccccc2)c1=O |r|
CN(C)C(=O)OC(CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3cc(F)ccc3[nH]2)c1=O |w:6.5|
CN(C)C(=O)OC(CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3cc(F)ccc3n2C(=O)OC(C)(C)C)c1=O |w:6.5|
CN(C)C(=O)OC(CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3cc(F)ccc3[nH]2)c1=O
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1nccn(Cc2cc3cc(F)ccc3n2C(=O)OC(C)(C)C)c1=O
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1nccn(Cc2cc3cc(F)ccc3[nH]2)c1=O
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cncn(Cc2cc3cc(F)ccc3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3c(CC(C)C)cccc3n2C(=O)OC(C)(C)C)c1=O
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3c(CC(C)C)cccc3[nH]2)c1=O
COC(=O)N[C@@H](CC\C=C\C(N)=O)C(=O)Nc1cccn(Cc2cc3c(CC(C)C)cccc3n2C(=O)OC(C)(C)C)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(N)=O)C(=O)Nc1cccn(Cc2cc3c(CC(C)C)cccc3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(N)=O)C(=O)Nc1cccn(Cc2cc3cccc(CC(C)C)c3n2C(=O)OC(C)(C)C)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3cccc(CC(C)C)c3n2C(=O)OC(C)(C)C)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(N)=O)C(=O)Nc1cccn(Cc2cc3cccc(CC(C)C)c3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3cccc(CC(C)C)c3[nH]2)c1=O |r|
CC(C)Cc1cccc2cc(Cn3cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c3=O)[nH]c12 |r|
CNC(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3cccc(CC(C)C)c3n2C(=O)OC(C)(C)C)c1=O |r|
CNC(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3cccc(CC(C)C)c3[nH]2)c1=O |r|
CNC(=O)\C=C\CC[C@H](OC(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3cccc(CC(C)C)c3[nH]2)c1=O |r|
CC(C)Cc1cccc2cc(Cn3cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N4CCCC4)c3=O)n(C(=O)OC(C)(C)C)c12 |r|
CC(C)Cc1cccc2cc(Cn3cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N4CCCC4)c3=O)[nH]c12 |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N1CCCC1)C(=O)Nc1cccn(Cc2cc3cccc(CC(C)C)c3n2C(=O)OC(C)(C)C)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N1CCCC1)C(=O)Nc1cccn(Cc2cc3cccc(CC(C)C)c3[nH]2)c1=O |r|
CC(C)Cc1cccc2cc(Cn3cccc(NC(=O)C(CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c3=O)[nH]c12 |w:20.29|
CC(C)Cc1cccc2cc(Cn3cccc(NC(=O)C(CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c3=O)n(C(=O)OC(C)(C)C)c12 |w:20.29|
CC(C)Cc1cccc2cc(Cn3cccc(NC(=O)C(CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c3=O)[nH]c12
CC(C)Cc1cccc2cc(Cn3cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)NC(=O)OCCOC(C)=O)c3=O)[nH]c12
CC(C)Cc1cccc2cc(Cn3cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)NC(=O)OCCO)c3=O)n(C(=O)OC(C)(C)C)c12
CC(C)Cc1cccc2cc(Cn3cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)NC(=O)OCCO)c3=O)[nH]c12
CC(C)Cc1cccc2cc(Cn3cccc(NC(=O)[C@H](CC\C=C\C(=O)N4CCCC4)NC(=O)OCCO)c3=O)n(C(=O)OC(C)(C)C)c12 |r|
CC(C)Cc1cccc2cc(Cn3cccc(NC(=O)[C@H](CC\C=C\C(=O)N4CCCC4)NC(=O)OCCO)c3=O)[nH]c12 |r|
CN(C)C(=O)\C=C\CC[C@H](NC(=O)C1CCC(F)(F)CC1)C(=O)Nc1cccn(Cc2cc3cccc(OCc4ccc(F)cc4F)c3[nH]2)c1=O
CN(C)C(=O)\C=C\CC[C@H](NC(=O)OC(C)(C)C)C(=O)Nc1cccn(Cc2cc3cccc(OCc4ccc(F)cc4F)c3[nH]2)c1=O |r|
CN(C)C(=O)\C=C\CC[C@H](NC(=O)c1ncco1)C(=O)Nc1cccn(Cc2cc3cccc(OCc4ccc(F)cc4F)c3[nH]2)c1=O |r|
COCC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3cccc(OCc4ccc(F)cc4F)c3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3cccc(OCC4CC4)c3[nH]2)c1=O |r|
CN(C)C(=O)\C=C\CC[C@H](NC(=O)CC(F)(F)F)C(=O)Nc1cccn(Cc2cc3cccc(OCc4ccc(F)cc4F)c3[nH]2)c1=O |r|
CN(C)C(=O)\C=C\CC[C@H](NC(=O)c1ccccc1F)C(=O)Nc1cccn(Cc2cc3cccc(OCc4ccc(F)cc4F)c3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3cccc(OCc4ccc(F)cc4F)c3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3cccc(OCc4ccc(F)cc4F)c3n2C(=O)OC(C)(C)C)c1=O |r|
CC(C)(C)OC(=O)N[C@@H](CC\C=C\C(N)=O)C(=O)Nc1cccn(Cc2cc3cccc(OCc4ccc(F)cc4F)c3n2C(=O)OC(C)(C)C)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(N)=O)C(=O)Nc1cccn(Cc2cc3cccc(OCc4ccc(F)cc4F)c3n2C(=O)OC(C)(C)C)c1=O |r|
NC(=O)\C=C\CC[C@H](NC(=O)c1ccccc1F)C(=O)Nc1cccn(Cc2cc3cccc(OCc4ccc(F)cc4F)c3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(N)=O)C(=O)Nc1cccn(Cc2cc3cccc(OCC(F)F)c3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3cccc(OCC(F)F)c3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3cccc(OCC(F)F)c3n2C(=O)OC(C)(C)C)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(N)=O)C(=O)Nc1cccn(Cc2cc3cccc(OCc4ccc(F)cc4F)c3[nH]2)c1=O |r|
COCC(=O)N[C@@H](CC\C=C\C(N)=O)C(=O)Nc1cccn(Cc2cc3cccc(OCc4ccc(F)cc4F)c3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3cc(F)cc(OCc4ccc(F)cc4F)c3n2C(=O)OC(C)(C)C)c1=O
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3cc(F)cc(OCc4ccc(F)cc4F)c3[nH]2)c1=O
COC(=O)N[C@@H](CC\C=C\C(N)=O)C(=O)Nc1cccn(Cc2cc3cc(F)cc(OCc4ccc(F)cc4F)c3n2C(=O)OC(C)(C)C)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(N)=O)C(=O)Nc1cccn(Cc2cc3cc(F)cc(OCc4ccc(F)cc4F)c3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3cc(F)cc(OCC(F)F)c3n2C(=O)OC(C)(C)C)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3cc(F)cc(OCC(F)F)c3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(N)=O)C(=O)Nc1cccn(Cc2cc3cc(F)cc(OCC(F)F)c3n2C(=O)OC(C)(C)C)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(N)=O)C(=O)Nc1cccn(Cc2cc3cc(F)cc(OCC(F)F)c3[nH]2)c1=O |r|
CNC(=O)\C=C\CC[C@H](NC(=O)OC)C(=O)Nc1cccn(Cc2cc3cc(F)cc(OCc4ccc(F)cc4F)c3n2C(=O)OC(C)(C)C)c1=O |r|
CNC(=O)\C=C\CC[C@H](NC(=O)OC)C(=O)Nc1cccn(Cc2cc3cc(F)cc(OCc4ccc(F)cc4F)c3[nH]2)c1=O |r|
COCCOC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3cc(F)cc(OCc4ccc(F)cc4F)c3n2C(=O)OC(C)(C)C)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N1CCCC1)C(=O)Nc1cccn(Cc2cc3cc(F)cc(OCc4ccc(F)cc4F)c3n2C(=O)OC(C)(C)C)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N1CCCC1)C(=O)Nc1cccn(Cc2cc3cc(F)cc(OCc4ccc(F)cc4F)c3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3cc(F)cc(CC(C)C)c3n2C(=O)OC(C)(C)C)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3cc(F)cc(CC(C)C)c3[nH]2)c1=O |r|
OCCOC(=O)N[C@@H](CC\C=C\C(=O)N1CCCC1)C(=O)Nc1cccn(Cc2cc3cc(F)cc(OCc4ccc(F)cc4F)c3[nH]2)c1=O |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3cc(F)cc(OCc4ccc(F)cc4F)c3[nH]2)c1=O |r|
COCCN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3cc(F)cc(OCc4ccc(F)cc4F)c3n2C(=O)OC(C)(C)C)c1=O |r|
COCCN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3cc(F)cc(OCc4ccc(F)cc4F)c3[nH]2)c1=O |r|
CN(C)C(=O)\C=C\CC[C@H](OC(=O)N1CCCC1)C(=O)Nc1cccn(Cc2cc3cc(F)cc(OCc4ccc(F)cc4F)c3n2C(=O)OC(C)(C)C)c1=O |r|
CN(C)C(=O)\C=C\CC[C@H](OC(=O)N1CCCC1)C(=O)Nc1cccn(Cc2cc3cc(F)cc(OCc4ccc(F)cc4F)c3[nH]2)c1=O |r|
COCCOC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3cc(F)cc(OCc4ccc(F)cc4F)c3[nH]2)c1=O |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N1CCCC1)C(=O)Nc1cccn(Cc2cc3cc(F)cc(OCc4ccc(F)cc4F)c3n2C(=O)OC(C)(C)C)c1=O |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N1CCCC1)C(=O)Nc1cccn(Cc2cc3cc(F)cc(OCc4ccc(F)cc4F)c3[nH]2)c1=O |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(N)=O)C(=O)Nc1cccn(Cc2cc3cc(F)cc(OCc4ccc(F)cc4F)c3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N1CCCC1)C(=O)Nc1cccn(Cc2cc3cc(F)cc(CC(C)C)c3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N1CCCC1)C(=O)Nc1cccn(Cc2cc3cc(F)cc(CC(C)C)c3n2C(=O)OC(C)(C)C)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3cc(F)cc(OCc4ccc(F)cc4F)c3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3cc(F)cc(OCc4ccc(F)cc4F)c3n2C(=O)OC(C)(C)C)c1=O |r|
CN(C)C(=O)OC(CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3cc(F)cc(OCc4ccc(F)cc4F)c3n2C(=O)OC(C)(C)C)c1=O |w:6.5|
CN(C)C(=O)OC(CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3cc(F)cc(OCc4ccc(F)cc4F)c3[nH]2)c1=O |w:6.5|
CN(C)C(=O)OC(CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3cc(F)cc(OCc4ccc(F)cc4F)c3[nH]2)c1=O
CC(C)Cc1cc(F)cc2cc(Cn3cccc(NC(=O)C(CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c3=O)n(C(=O)OC(C)(C)C)c12 |w:21.30|
CC(C)Cc1cc(F)cc2cc(Cn3cccc(NC(=O)C(CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c3=O)[nH]c12 |w:21.30|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3cc(F)cc(CCC(F)(F)F)c3[nH]2)c1=O
COC(=O)N[C@@H](CC\C=C\C(=O)N1CCCC1)C(=O)Nc1cccn(Cc2cc3cc(F)cc(CCC(F)(F)F)c3n2C(=O)OC(C)(C)C)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N1CCCC1)C(=O)Nc1cccn(Cc2cc3cc(F)cc(CCC(F)(F)F)c3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3cc(F)cc(CCC(F)(F)F)c3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3cc(F)cc(CCC(F)(F)F)c3n2C(=O)OC(C)(C)C)c1=O |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3cc(F)cc(c3[nH]2)C(F)(F)F)c1=O |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3cc(F)cc(c3n2C(=O)OC(C)(C)C)C(F)(F)F)c1=O |r|
CNC(=O)\C=C\CC[C@H](OC(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3cc(F)cc(CCC(F)(F)F)c3n2C(=O)OC(C)(C)C)c1=O |r|
CNC(=O)\C=C\CC[C@H](OC(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3cc(F)cc(CCC(F)(F)F)c3[nH]2)c1=O |r|
CN(C)C(=O)\C=C\CC[C@H](OC(=O)N1CCCC1)C(=O)Nc1cccn(Cc2cc3cc(F)cc(CC(C)(C)C)c3n2C(=O)OC(C)(C)C)c1=O
CN(C)C(=O)\C=C\CC[C@H](OC(=O)N1CCCC1)C(=O)Nc1cccn(Cc2cc3cc(F)cc(CC(C)(C)C)c3[nH]2)c1=O
COCCOC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3cc(F)cc(CC(C)(C)C)c3[nH]2)c1=O |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3cc(F)cc(CC(C)(C)C)c3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N1CCCC1)C(=O)Nc1cccn(Cc2cc3cc(F)cc(CC(C)(C)C)c3[nH]2)c1=O |r|
COCCN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3cc(F)cc(CC(C)(C)C)c3[nH]2)c1=O |r|
CC(C)(C)Cc1cc(F)cc2cc(Cn3cccc(NC(=O)[C@H](CC\C=C\C(=O)N4CCCC4)OC(=O)N4CCCC4)c3=O)[nH]c12 |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3cc(F)cc(CC(C)(C)C)c3[nH]2)c1=O |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1nccn(Cc2cc3cc(F)cc(CC(C)(C)C)c3n2C(=O)OC(C)(C)C)c1=O
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1nccn(Cc2cc3cc(F)cc(CC(C)(C)C)c3[nH]2)c1=O
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cncn(Cc2cc3cc(F)cc(CC(C)(C)C)c3n2C(=O)OC(C)(C)C)c1=O |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cncn(Cc2cc3cc(F)cc(CC(C)(C)C)c3[nH]2)c1=O |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cncn(Cc2cc3cc(F)cc(CCC(F)(F)F)c3n2C(=O)OC(C)(C)C)c1=O |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cncn(Cc2cc3cc(F)cc(CCC(F)(F)F)c3[nH]2)c1=O |r|
CNC(=O)\C=C\CC[C@H](OC(=O)N(C)C)C(=O)Nc1cncn(Cc2cc3cc(F)cc(CCC(F)(F)F)c3n2C(=O)OC(C)(C)C)c1=O |r|
CC(C)Cn1c(Cn2cncc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c2=O)cc2cc(F)ccc12
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3cc(F)ccc3n2Cc2ccccc2)c1=O |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3cc(F)ccc3n2CC2CC2)c1=O |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3cc(F)ccc3n2C)c1=O |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3cc(F)ccc3n2Cc2ccc(F)cc2)c1=O |r|
CCn1c(Cn2cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c2=O)cc2cc(F)ccc12 |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3cc(F)ccc3n2Cc2ccc(F)cc2F)c1=O |r|
COC(=O)n1c(Cn2cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c2=O)cc2cc(F)ccc12
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3cc(F)ccc3n2C(=O)OCc2ccc(F)cc2F)c1=O |r|
CC(C)Cn1c(Cn2cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c2=O)cc2cc(F)ccc12 |r|
CCn1c(Cn2ccnc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c2=O)cc2cc(F)ccc12 |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1nccn(Cc2cc3cc(F)ccc3n2Cc2ccccc2)c1=O |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1nccn(Cc2cc3cc(F)ccc3n2CC2CC2)c1=O |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1nccn(Cc2cc3cc(F)ccc3n2Cc2ccc(F)cc2)c1=O |r|
CC(C)Cn1c(Cn2cncc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c2=O)cc2cc(F)ccc12 |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1nccn(Cc2cc3cc(F)ccc3n2Cc2ccc(F)cc2F)c1=O |r|
CN(C)C(=O)\C=C\CC[C@H](OC(=O)N(C)CCN(C)C(=O)OC(C)(C)C)C(=O)Nc1cccn(Cc2cc3cc(F)ccc3n2C)c1=O
CN(C)CCN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3cc(F)ccc3n2C)c1=O
COC(=O)N[C@@H](CC\C=C\C(N)=O)C(=O)Nc1cccn(Cc2cccc3ccn(C(=O)OC(C)(C)C)c23)c1=O
COC(=O)N[C@@H](CC\C=C\C(N)=O)C(=O)Nc1cccn(Cc2nc3cc(F)cc(OCc4ccc(F)cc4F)c3s2)c1=O
CN(C)C(=O)\C=C\CC[C@H](NC(=O)OCCO)C(=O)Nc1cccn(Cc2cc3ccccc3n2C(=O)OC(C)(C)C)c1=O |r|
CNC(=O)\C=C\CC[C@H](NC(=O)OC)C(=O)Nc1cccn(Cc2nc3cc(F)cc(OCc4ccc(F)cc4F)c3s2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3cccc(CC(C)C)c3o2)c1=O
CNC(=O)\C=C\CC[C@H](OC(=O)N(C)C)C(=O)Nc1cncn(Cc2cc3cc(F)cc(CCC(F)(F)F)c3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(N)=O)C(=O)Nc1cccn(Cc2nc3cccc(CC(C)C)c3o2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(CC(C)C)cccc3o2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(N)=O)C(=O)Nc1cccn(Cc2nc3c(CC(C)C)cccc3o2)c1=O |r|
CC(C)Cc1cccc2nc(Cn3cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)NC(=O)OCCO)c3=O)oc12 |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3cccc(CC(C)C)c3s2)c1=O
COC(=O)N[C@@H](CC\C=C\C(N)=O)C(=O)Nc1cccn(Cc2nc3cccc(CC(C)C)c3s2)c1=O |r|
CC(C)Cc1cccc2nc(Cn3cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)NC(=O)OCCO)c3=O)sc12 |r|
CN(C)C(=O)\C=C\CC[C@H](NC(=O)OC(C)(C)C)C(=O)Nc1cccn(Cc2nc3cccc(OCc4ccc(F)cc4F)c3s2)c1=O
CN(C)C(=O)\C=C\CC[C@H](NC(=O)c1ncco1)C(=O)Nc1cccn(Cc2nc3cccc(OCc4ccc(F)cc4F)c3s2)c1=O
CN(C)C(=O)\C=C\CC[C@H](NC(=O)C1CCC(F)(F)CC1)C(=O)Nc1cccn(Cc2nc3cccc(OCc4ccc(F)cc4F)c3s2)c1=O |r|
CN(C)C(=O)\C=C\CC[C@H](NC(=O)c1ccccc1F)C(=O)Nc1cccn(Cc2nc3cccc(OCc4ccc(F)cc4F)c3s2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(N)=O)C(=O)Nc1cccn(Cc2nc3cccc(OCc4ccc(F)cc4F)c3s2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3cccc(OCc4ccc(F)cc4F)c3s2)c1=O |r|
COCC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3cccc(OCc4ccc(F)cc4F)c3s2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(N)=O)C(=O)Nc1cccn(Cc2nc3cccc(OCC(F)F)c3s2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3cccc(OCC(F)F)c3s2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(N)=O)C(=O)Nc1cccn(Cc2nc3cccc(OC(F)(F)C(F)F)c3s2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3cccc(OC(F)(F)C(F)F)c3s2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3cccc(OCC(F)(F)F)c3s2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(N)=O)C(=O)Nc1cccn(Cc2nc3cccc(OCC(F)(F)F)c3s2)c1=O |r|
CC(C)(C)OC(=O)N[C@@H](CC\C=C\C(N)=O)C(=O)Nc1cccn(Cc2nc3cccc(OCc4ccc(F)cc4F)c3s2)c1=O |r|
COCC(=O)N[C@@H](CC\C=C\C(N)=O)C(=O)Nc1cccn(Cc2nc3cccc(OCc4ccc(F)cc4F)c3s2)c1=O |r|
NC(=O)\C=C\CC[C@H](NC(=O)c1ccccc1F)C(=O)Nc1cccn(Cc2nc3cccc(OCc4ccc(F)cc4F)c3s2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3cc(F)ccc3s2)c1=O
COC(=O)N[C@@H](CC\C=C\C(N)=O)C(=O)Nc1cccn(Cc2nc3cc(F)ccc3s2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N1CCCC1)C(=O)Nc1cccn(Cc2nc3cc(F)ccc3s2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3cccc(COc4ccc(F)cc4F)c3s2)c1=O |r|
CN(C)C(=O)\C=C\CC[C@H](NC(=O)OCCO)C(=O)Nc1cccn(Cc2nc3ccccc3s2)c1=O
NC(=O)\C=C\CC[C@H](NC(=O)OCCO)C(=O)Nc1cccn(Cc2nc3ccccc3o2)c1=O |r|
NC(=O)\C=C\CC[C@H](NC(=O)OCCO)C(=O)Nc1cccn(Cc2nc3ccccc3s2)c1=O |r|
NC(=O)\C=C\CC[C@H](NC(=O)OCCO)C(=O)Nc1cccn(Cc2cc3ccccc3[nH]2)c1=O |r|
CC(C)(C)OC(=O)n1c(Cn2cccc(NC(=O)[C@H](CC\C=C\C(N)=O)NC(=O)OCCO)c2=O)cc2ccccc12 |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3cc(F)c(F)cc3n2CCOC(C)C)c1=O |r|
COC(=O)NC(CC\C=C\C(=O)N(C)C)CNc1cccn(Cc2nc3c(CC(C)C)c(F)cc(F)c3[nH]2)c1=O
COC(=O)N[C@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(CC(C)C)cccc3[nH]2)c1=O |r|
CNC(=O)\C=C\CC[C@H](NC(=O)OC)C(=O)Nc1cncn(Cc2nc3c(CCC(F)(F)F)cc(F)cc3n2C(=O)OC(C)(C)C)c1=O |r|
CC(C)Cc1cccc2n(C(=O)OC(C)(C)C)c(Cn3cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)NC(=O)N(C)C)c3=O)nc12 |r|
CC(C)Cc1cccc2[nH]c(Cn3cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)NC(=O)N(C)C)c3=O)nc12 |r|
CNC(=O)\C=C\CC[C@H](NC(=O)OC)C(=O)Nc1cncn(Cc2nc3cc(F)cc(CCC(F)(F)F)c3[nH]2)c1=O |r|
COCCN(C)C(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(CC(C)C)cc(F)cc3n2C(=O)OC(C)(C)C)c1=O |r|
COCCN(C)C(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3cc(F)cc(CC(C)C)c3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(CC(C)(C)C)c(F)cc(F)c3n2C(=O)OC(C)(C)C)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(CC(C)(C)C)c(F)cc(F)c3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(CCC(F)(F)F)c(F)c(F)cc3n2C(=O)OC(C)(C)C)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(CCC(F)(F)F)c(F)c(F)cc3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(Oc4ccc(F)cc4F)c(F)cc(F)c3n2C(=O)OC(C)(C)C)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(OC(C)C)c(F)c(F)cc3n2C(=O)OC(C)(C)C)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3cc(F)c(F)c(OC(C)C)c3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(Oc4ccc(F)cc4F)c(F)c(F)cc3n2C(=O)OC(C)(C)C)c1=O
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(Oc4ccc(F)cc4F)c(F)c(F)cc3[nH]2)c1=O
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(OCc4ccccc4)c(F)c(F)cc3n2C(=O)OC(C)(C)C)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(Oc4ccccc4)c(F)cc(F)c3n2C(=O)OC(C)(C)C)c1=O
CC(C)Cc1cc(F)cc2n(C(=O)OC(C)(C)C)c(Cn3cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)NC(=O)N(C)C)c3=O)nc12 |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3cc(F)c(F)c(OCc4ccccc4)c3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3cc(F)c(F)c(OCc4ccc(F)cc4F)c3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(OCc4ccc(F)cc4F)c(F)c(F)cc3n2C(=O)OC(C)(C)C)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(CC(C)C)nccc3n2C(=O)OC(C)(C)C)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(CC(C)C)ccnc3n2C(=O)OC(C)(C)C)c1=O |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(C=C(C)C)ncnc3[nH]2)c1=O |r,wD:6.5,(-5.04,6.29,;-3.71,5.52,;-2.37,6.29,;-3.71,3.98,;-5.04,3.21,;-2.37,3.21,;-2.37,1.67,;-3.71,.9,;-5.04,1.67,;-6.37,.9,;-7.71,1.67,;-9.04,.9,;-9.04,-.64,;-10.38,1.67,;-11.71,.9,;-10.38,3.21,;-1.04,.9,;-1.04,-.64,;.29,1.67,;1.63,.9,;1.63,-.64,;2.96,-1.41,;4.29,-.64,;4.29,.9,;5.63,1.67,;6.96,.9,;7.12,-.63,;8.63,-.95,;9.4,-2.29,;8.63,-3.62,;9.4,-4.95,;8.63,-6.29,;10.94,-4.95,;10.94,-2.29,;11.71,-.95,;10.94,.38,;9.4,.38,;8.37,1.52,;2.96,1.67,;2.96,3.21,)|
CC(C)Cc1ncnc2[nH]c(Cn3cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c3=O)nc12 |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(CC(C)C)ccnc3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(C=C(C)C)ccnc3[nH]2)c1=O |r,wD:5.4,(-5.04,6.29,;-3.71,5.52,;-3.71,3.98,;-5.04,3.21,;-2.37,3.21,;-2.37,1.67,;-3.71,.9,;-5.04,1.67,;-6.37,.9,;-7.71,1.67,;-9.04,.9,;-9.04,-.64,;-10.38,1.67,;-11.71,.9,;-10.38,3.21,;-1.04,.9,;-1.04,-.64,;.29,1.67,;1.63,.9,;1.63,-.64,;2.96,-1.41,;4.29,-.64,;4.29,.9,;5.63,1.67,;6.96,.9,;7.12,-.63,;8.63,-.95,;9.4,-2.29,;8.63,-3.62,;9.4,-4.95,;8.63,-6.29,;10.94,-4.95,;10.94,-2.29,;11.71,-.95,;10.94,.38,;9.4,.38,;8.37,1.52,;2.96,1.67,;2.96,3.21,)|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(C=C(C)C)nccc3[nH]2)c1=O |r,wD:5.4,(-5.04,6.29,;-3.71,5.52,;-3.71,3.98,;-5.04,3.21,;-2.37,3.21,;-2.37,1.67,;-3.71,.9,;-5.04,1.67,;-6.37,.9,;-7.71,1.67,;-9.04,.9,;-9.04,-.64,;-10.38,1.67,;-11.71,.9,;-10.38,3.21,;-1.04,.9,;-1.04,-.64,;.29,1.67,;1.63,.9,;1.63,-.64,;2.96,-1.41,;4.29,-.64,;4.29,.9,;5.63,1.67,;6.96,.9,;7.12,-.63,;8.63,-.95,;9.4,-2.29,;8.63,-3.62,;9.4,-4.95,;8.63,-6.29,;10.94,-4.95,;10.94,-2.29,;11.71,-.95,;10.94,.38,;9.4,.38,;8.37,1.52,;2.96,1.67,;2.96,3.21,)|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(ncnc3[nH]2)C2CCCCC2)c1=O |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(ncnc3[nH]2)C2CCCCC2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(Oc4ccccc4)c(F)c(F)cc3n2C(=O)OC(C)(C)C)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3ncnc(Oc4ccccc4)c3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(CC(C)C)nccc3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(OC(C)C)c(F)cc(F)c3n2C(=O)OC(C)(C)C)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(OCc4ccccc4)c(F)cc(F)c3n2C(=O)OC(C)(C)C)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(Oc4ccccc4)c(F)cc(F)c3[nH]2)c1=O
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(Oc4ccc(F)cc4F)ncnc3n2C(=O)OC(C)(C)C)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(Oc4ccc(F)cc4F)ncnc3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(Oc4ccc(F)cc4F)c(F)cc(F)c3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(OCc4ccccc4)c(F)cc(F)c3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(OCc4ccc(F)cc4F)c(F)cc(F)c3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(OC(C)C)ncnc3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(CC(C)C)ncc(F)c3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(CC(C)C)nc(C)nc3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(CC(C)C)nc(C)nc3n2C(=O)OC(C)(C)C)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(\C=C\C4CC4)ncnc3[nH]2)c1=O |r|
CC(C)Oc1c(F)c(F)cc2nc(Cn3cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c3=O)[nH]c12 |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(CCC4CC4)ncnc3[nH]2)c1=O |r|
CCCCCc1ncnc2[nH]c(Cn3cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)NC(=O)OC)c3=O)nc12 |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(C=C(C)C)nc(C)nc3[nH]2)c1=O |r,wD:5.4,(-5.81,6.29,;-4.48,5.52,;-4.48,3.98,;-5.81,3.21,;-3.14,3.21,;-3.14,1.67,;-4.48,.9,;-5.81,1.67,;-7.14,.9,;-8.48,1.67,;-9.81,.9,;-9.81,-.64,;-11.15,1.67,;-12.48,.9,;-11.15,3.21,;-1.81,.9,;-1.81,-.64,;-.48,1.67,;.86,.9,;.86,-.64,;2.19,-1.41,;3.52,-.64,;3.52,.9,;4.86,1.67,;6.19,.9,;6.35,-.63,;7.86,-.95,;8.63,-2.29,;7.86,-3.62,;8.63,-4.95,;7.86,-6.29,;10.17,-4.95,;10.17,-2.29,;10.94,-.95,;12.48,-.95,;10.17,.38,;8.63,.38,;7.6,1.52,;2.19,1.67,;2.19,3.21,)|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(Oc4ccc(F)cc4F)c(F)c(F)cc3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(C=C(C)C)cncc3[nH]2)c1=O |r,wD:5.4,(-5.04,6.29,;-3.71,5.52,;-3.71,3.98,;-5.04,3.21,;-2.37,3.21,;-2.37,1.67,;-3.71,.9,;-5.04,1.67,;-6.37,.9,;-7.71,1.67,;-9.04,.9,;-9.04,-.64,;-10.38,1.67,;-11.71,.9,;-10.38,3.21,;-1.04,.9,;-1.04,-.64,;.29,1.67,;1.63,.9,;1.63,-.64,;2.96,-1.41,;4.29,-.64,;4.29,.9,;5.63,1.67,;6.96,.9,;7.12,-.63,;8.63,-.95,;9.4,-2.29,;8.63,-3.62,;9.4,-4.95,;8.63,-6.29,;10.94,-4.95,;10.94,-2.29,;11.71,-.95,;10.94,.38,;9.4,.38,;8.37,1.52,;2.96,1.67,;2.96,3.21,)|
CC(C)Cc1ncc(F)c2[nH]c(Cn3cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c3=O)nc12 |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(OCC(C)C)ncnc3[nH]2)c1=O |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(F)cc(F)c(OCc4ccc(F)cc4F)c3[nH]2)c1=O |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(OCc4ccc(F)cc4F)c(F)c(F)cc3n2C(=O)OC(C)(C)C)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(C=C(C)C)ncc(F)c3[nH]2)c1=O |r,wD:5.4,(-5.04,6.29,;-3.71,5.52,;-3.71,3.98,;-5.04,3.21,;-2.37,3.21,;-2.37,1.67,;-3.71,.9,;-5.04,1.67,;-6.37,.9,;-7.71,1.67,;-9.04,.9,;-9.04,-.64,;-10.38,1.67,;-11.71,.9,;-10.38,3.21,;-1.04,.9,;-1.04,-.64,;.29,1.67,;1.63,.9,;1.63,-.64,;2.96,-1.41,;4.29,-.64,;4.29,.9,;5.63,1.67,;6.96,.9,;7.12,-.63,;8.63,-.95,;9.4,-2.29,;8.63,-3.62,;9.4,-4.95,;10.94,-4.95,;8.63,-6.29,;10.94,-2.29,;11.71,-.95,;10.94,.38,;11.71,1.71,;9.4,.38,;8.37,1.52,;2.96,1.67,;2.96,3.21,)|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3ncnc(CCC4CCCCC4)c3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(\C=C\c4ccccc4)ncnc3[nH]2)c1=O |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(OCc4ccc(F)cc4F)c(F)c(F)cc3[nH]2)c1=O |r|
CC(C)Cc1ncnc2cc(Cn3cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)NC([O-])=O)c3=O)[nH]c12
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(CC(C)C)cncc3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(CC(C)(C)C)c(F)c(F)cc3n2C(=O)OC(C)(C)C)c1=O
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(OCc4ccccc4)ncnc3[nH]2)c1=O
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(CC(C)C)nc(C)cc3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(C=C(C)C)nc(C)cc3[nH]2)c1=O |r,wD:5.4,(-5.81,6.29,;-4.48,5.52,;-4.48,3.98,;-5.81,3.21,;-3.14,3.21,;-3.14,1.67,;-4.48,.9,;-5.81,1.67,;-7.14,.9,;-8.48,1.67,;-9.81,.9,;-9.81,-.64,;-11.15,1.67,;-12.48,.9,;-11.15,3.21,;-1.81,.9,;-1.81,-.64,;-.48,1.67,;.86,.9,;.86,-.64,;2.19,-1.41,;3.52,-.64,;3.52,.9,;4.86,1.67,;6.19,.9,;6.35,-.63,;7.86,-.95,;8.63,-2.29,;7.86,-3.62,;8.63,-4.95,;10.17,-4.95,;7.86,-6.29,;10.17,-2.29,;10.94,-.95,;12.48,-.95,;10.17,.38,;8.63,.38,;7.6,1.52,;2.19,1.67,;2.19,3.21,)|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(CC(C)(C)C)c(F)c(F)cc3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(Cc4ccccc4)ncnc3[nH]2)c1=O
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(CC(C)(C)C)c(F)c(F)cc3[nH]2)c1=O
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(CC(C)(C)C)ncnc3[nH]2)c1=O
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(CC(C)(C)C)ncnc3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(CCC(F)(F)F)ncnc3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(CCC(C)C)ncnc3[nH]2)c1=O
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(CCC(C)(C)C)ncnc3[nH]2)c1=O |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(CCC(C)(C)C)ncnc3[nH]2)c1=O |r|
CC(C)Cc1ncnc2cc(Cn3cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c3=O)[nH]c12 |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(CCC(C)(C)C)ncnc3n2C2CCCCO2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(OCc4ccc(F)cc4F)ncnc3[nH]2)c1=O |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(OCc4ccc(F)cc4F)ncnc3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(CC4CC4)ncnc3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3ncnc(CCc4ccccc4)c3[nH]2)c1=O |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(CCc4ccccc4)ncnc3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(CCC(C)(C)C)ncnc3n2C2CCCCO2)c1=O |r|
CC(C)CCc1ncnc2n(C3CCCCO3)c(Cn3cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c3=O)nc12 |r|
CC(C)CCc1ncnc2nc(Cn3cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c3=O)[nH]c12 |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(CCC(F)(F)F)ncnc3n2C2CCCCO2)c1=O |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(CCC(F)(F)F)ncnc3n2C2CCCCO2)c1=O |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(CCC(F)(F)F)ncnc3[nH]2)c1=O |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(C=C(C)C)cncc3[nH]2)c1=O |r,wD:6.5,(-5.04,6.29,;-3.71,5.52,;-2.37,6.29,;-3.71,3.98,;-5.04,3.21,;-2.37,3.21,;-2.37,1.67,;-3.71,.9,;-5.04,1.67,;-6.37,.9,;-7.71,1.67,;-9.04,.9,;-9.04,-.64,;-10.38,1.67,;-11.71,.9,;-10.38,3.21,;-1.04,.9,;-1.04,-.64,;.29,1.67,;1.63,.9,;1.63,-.64,;2.96,-1.41,;4.29,-.64,;4.29,.9,;5.63,1.67,;6.96,.9,;7.12,-.63,;8.63,-.95,;9.4,-2.29,;8.63,-3.62,;9.4,-4.95,;8.63,-6.29,;10.94,-4.95,;10.94,-2.29,;11.71,-.95,;10.94,.38,;9.4,.38,;8.37,1.52,;2.96,1.67,;2.96,3.21,)|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(CC(C)(C)C)c(F)c(F)cc3n2C(=O)OC(C)(C)C)c1=O |r|
CC(C)Cc1cncc2[nH]c(Cn3cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c3=O)nc12 |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3ncnc(CCC(F)(F)F)c3[nH]2)c1=O |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3ncnc(CCC(F)(F)F)c3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(CC(C)(C)C)nc(C)nc3n2C2CCCCO2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(CC(C)(C)C)nc(C)nc3[nH]2)c1=O |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(CC(C)(C)C)nc(C)nc3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(CC4CCCCC4)ncnc3[nH]2)c1=O |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(CC4CCCCC4)ncnc3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3nc(C)nc(CC(C)C)c3[nH]2)c1=O |r|
CC(C)Cc1nc(C)nc2cc(Cn3cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c3=O)[nH]c12 |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(CC(C(F)(F)F)C(F)(F)F)ncnc3[nH]2)c1=O |r|
CC(C)Cc1c(F)cnc2cc(Cn3cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c3=O)[nH]c12 |r|
CC(C)(C)OC(=O)n1c(Cn2cccc(N)c2=O)cc2ccccc12
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3c(F)cnc(C=C(C)C)c3[nH]2)c1=O |r,wD:6.5,(-5.04,6.29,;-3.71,5.52,;-2.38,6.29,;-3.71,3.98,;-5.04,3.21,;-2.38,3.21,;-2.38,1.67,;-3.71,.9,;-5.04,1.67,;-6.38,.9,;-7.71,1.67,;-9.04,.9,;-9.04,-.64,;-10.38,1.67,;-11.71,.9,;-10.38,3.21,;-1.04,.9,;-1.04,-.64,;.29,1.67,;1.63,.9,;1.63,-.64,;2.96,-1.41,;4.29,-.64,;4.29,.9,;5.63,1.67,;6.96,.9,;8.37,1.52,;9.4,.37,;10.94,.37,;11.71,1.7,;11.7,-.97,;10.92,-2.3,;9.38,-2.29,;8.61,-3.62,;9.37,-4.96,;8.6,-6.29,;10.91,-4.97,;8.62,-.96,;7.11,-.63,;2.96,1.67,;2.96,3.21,)|
CC(C)Cc1ccnc2cc(Cn3cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c3=O)[nH]c12 |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3nc(C)nc(N(C)C)c3[nH]2)c1=O |r|
CC(C)Cc1cncc2cc(Cn3cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c3=O)[nH]c12 |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3nccc(CC(C)C)c3[nH]2)c1=O |r|
CC(C)Cc1ncc(F)c2cc(Cn3cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c3=O)[nH]c12 |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3c(F)cnc(CC(C)C)c3[nH]2)c1=O |r|
COC(=O)NC(CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3cncc(CC(C)C)c3[nH]2)c1=O |w:5.4|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1ccc(C)n(Cc2nc3c(CC(C)C)cccc3[nH]2)c1=O
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3cncc(C=C(C)C)c3[nH]2)c1=O |r,wD:6.5,(-5.04,6.29,;-3.71,5.52,;-2.37,6.29,;-3.71,3.98,;-5.04,3.21,;-2.37,3.21,;-2.37,1.67,;-3.71,.9,;-5.04,1.67,;-6.37,.9,;-7.71,1.67,;-9.04,.9,;-9.04,-.64,;-10.38,1.67,;-11.71,.9,;-10.38,3.21,;-1.04,.9,;-1.04,-.64,;.29,1.67,;1.63,.9,;1.63,-.64,;2.96,-1.41,;4.29,-.64,;4.29,.9,;5.63,1.67,;6.96,.9,;8.37,1.52,;9.4,.38,;10.94,.38,;11.71,-.95,;10.94,-2.29,;9.4,-2.29,;8.63,-3.62,;9.4,-4.95,;10.94,-4.95,;8.63,-6.29,;8.63,-.95,;7.12,-.63,;2.96,1.67,;2.96,3.21,)|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3ccnc(CC(C)C)c3[nH]2)c1=O
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3nccc(C=C(C)C)c3[nH]2)c1=O |r,wD:5.4,(-5.04,6.29,;-3.71,5.52,;-3.71,3.98,;-5.04,3.21,;-2.37,3.21,;-2.37,1.67,;-3.71,.9,;-5.04,1.67,;-6.37,.9,;-7.71,1.67,;-9.04,.9,;-9.04,-.64,;-10.38,1.67,;-11.71,.9,;-10.38,3.21,;-1.04,.9,;-1.04,-.64,;.29,1.67,;1.63,.9,;1.63,-.64,;2.96,-1.41,;4.29,-.64,;4.29,.9,;5.63,1.67,;6.96,.9,;8.37,1.52,;9.4,.38,;10.94,.38,;11.71,-.95,;10.94,-2.29,;9.4,-2.29,;8.63,-3.62,;9.4,-4.95,;10.94,-4.95,;8.63,-6.29,;8.63,-.95,;7.12,-.63,;2.96,1.67,;2.96,3.21,)|
CC(C)Cc1cccc2[nH]c(Cn3c(C)ccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c3=O)nc12
CC(C)Cc1nccc2cc(Cn3cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c3=O)[nH]c12 |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1ccc(C)n(Cc2nc3c(CC(C)C)ncc(F)c3[nH]2)c1=O
CC(C)Cc1ncc(F)c2[nH]c(Cn3c(C)ccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c3=O)nc12
CC(C)Cc1ncc(F)c2cc(Cn3c(C)ccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c3=O)[nH]c12 |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1ccc(C)n(Cc2cc3c(F)cnc(CC(C)C)c3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3ncc(F)c(CC(C)C)c3[nH]2)c1=O |r|
CC(C)Cc1c(F)cnc2cc(Cn3cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)NC(=O)N(C)C)c3=O)[nH]c12 |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1ccc(Cl)n(Cc2nc3cccc(CC(C)C)c3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1ccc(Cl)n(Cc2nc3c(CC(C)C)ncc(F)c3[nH]2)c1=O
CC(C)Cc1ncc(F)c2[nH]c(Cn3c(Cl)ccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c3=O)nc12
CC(C)Cc1c(F)cnc2nc(Cn3cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c3=O)[nH]c12
CC(C)Cc1cccc2nc(Cn3c(Cl)ccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c3=O)[nH]c12 |r|
COCCOC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3ncc(F)c(CC(C)C)c3[nH]2)c1=O
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1ccc(C)n(Cc2nc3c(CC(C)C)c(F)cnc3[nH]2)c1=O |r|
CC(C)Cc1c(F)cnc2nc(Cn3c(C)ccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c3=O)[nH]c12 |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3ncc(c(C=C(C)C)c3[nH]2)C(F)(F)F)c1=O |r,wD:5.4,(-5.71,6.29,;-4.37,5.52,;-4.37,3.98,;-5.71,3.21,;-3.04,3.21,;-3.04,1.67,;-4.37,.9,;-5.71,1.67,;-7.04,.9,;-8.38,1.67,;-9.71,.9,;-9.71,-.64,;-11.04,1.67,;-12.38,.9,;-11.04,3.21,;-1.71,.9,;-1.71,-.64,;-.37,1.67,;.96,.9,;.96,-.64,;2.29,-1.41,;3.63,-.64,;3.63,.9,;4.96,1.67,;6.3,.9,;7.7,1.52,;8.73,.38,;10.27,.38,;11.04,-.95,;10.27,-2.29,;8.73,-2.29,;7.96,-3.62,;8.73,-4.95,;10.27,-4.95,;7.96,-6.29,;7.96,-.95,;6.46,-.63,;11.04,-3.62,;11.81,-4.95,;12.38,-2.85,;9.71,-4.39,;2.29,1.67,;2.29,3.21,)|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2[nH]c3c(CC(C)C)c(F)cnc3c2C)c1=O
CC(C)Cc1c(F)cnc2c(C)c(Cn3cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c3=O)[nH]c12
CC(C)Cc1ncc(F)c2cc(Cn3c(Cl)ccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c3=O)[nH]c12
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1ccc(Cl)n(Cc2cc3c(F)cnc(CC(C)C)c3[nH]2)c1=O |r|
CC(C)Cc1c(F)cnc2nc(Cn3cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c3=O)[nH]c12 |r|
COC(=O)NC(CC\C=C\C(=O)N(C)C)CNc1cccn(Cc2nc3c(CC(C)C)c(F)cc(F)c3n2C(=O)OC(C)(C)C)c1=O
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3ncc(F)c(CC4CC4)c3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3ncc(F)c(OCC(C)C)c3[nH]2)c1=O |r|
CC(C)Cc1c(Cl)cnc2cc(Cn3cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c3=O)[nH]c12 |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3ncc(F)c(CCC(F)(F)F)c3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3nc(C)c(F)c(CC(C)C)c3[nH]2)c1=O |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3ncc(F)c(CCC(F)(F)F)c3[nH]2)c1=O |r|
CC(C)Cc1c(F)cnc2cc(Cn3cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)CCN(C)C)c3=O)[nH]c12
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3ncc(F)c(OC(C)C)c3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1ccc(Cl)n(Cc2nc3ncc(F)c(CC(C)C)c3[nH]2)c1=O |r|
CC(C)Cc1c(F)c(C)nc2cc(Cn3cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c3=O)[nH]c12 |r|
CC(C)Cc1c(F)cnc2cc(Cn3cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)NC(=O)OCCN(C)C)c3=O)[nH]c12
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3ncc(F)c(OCc4ccccc4)c3[nH]2)c1=O |r|
CC(C)Oc1c(F)cnc2cc(Cn3cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c3=O)[nH]c12 |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3ncc(F)c(OCc4ccccc4)c3[nH]2)c1=O |r|
CC(C)COc1c(F)cnc2cc(Cn3cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c3=O)[nH]c12 |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(F)cnc(CCC(F)(F)F)c3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1ccc(C)n(Cc2cc3ncc(F)c(CC(C)C)c3[nH]2)c1=O
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1ccc(Cl)n(Cc2cc3ncc(F)c(CC(C)C)c3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1ccc(Cl)n(Cc2nc3c(F)cnc(CCC(F)(F)F)c3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1ccc(C)n(Cc2nc3c(F)cnc(CCC(F)(F)F)c3[nH]2)c1=O |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1ccc(C)n(Cc2nc3c(F)cnc(CCC(F)(F)F)c3[nH]2)c1=O |r|
CC(C)Cc1ncc(F)c2nc(Cn3cc(C)cc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c3=O)[nH]c12 |r|
CC(C)Cc1c(F)cnc2nc(Cn3c(Cl)ccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c3=O)[nH]c12 |r|
COC(=O)N[C@@H](CC\C=C\S(C)(=O)=O)C(=O)Nc1ccc(C)n(Cc2nc3c(F)cnc(CC(C)C)c3[nH]2)c1=O |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1ccc(Cl)n(Cc2nc3c(F)cnc(CCC(F)(F)F)c3[nH]2)c1=O |r|
CC(C)Cc1c(F)cnc2cc(Cn3c(Cl)ccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c3=O)[nH]c12 |r|
CC(C)Cc1c(F)cnc2cc(Cn3c(C)ccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c3=O)[nH]c12 |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1ccc(CC(C)C)n(Cc2nc3c(F)cnc(CC(C)C)c3[nH]2)c1=O |r|
CC(C)Cc1ccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c(=O)n1Cc1nc2c(F)cnc(CC(C)C)c2[nH]1 |r|
CC(C)Cc1ncc(F)c2nc(Cn3c(C)c(C)cc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c3=O)[nH]c12 |r|
CC(C)Cc1ncc(F)c2nc(Cn3c(ccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c3=O)C(C)C)[nH]c12 |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cc(C)c(C)n(Cc2nc3c(F)cnc(CC(C)C)c3[nH]2)c1=O |r|
CCc1ccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)NC(=O)OC)c(=O)n1Cc1nc2c(F)cnc(CC(C)C)c2[nH]1 |r|
CCc1ccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c(=O)n1Cc1nc2c(F)cnc(CC(C)C)c2[nH]1 |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1ccc(C(C)C)n(Cc2nc3c(F)cnc(CC(C)C)c3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cc(Cl)cn(Cc2nc3c(F)cnc(CC(C)C)c3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cc(F)cn(Cc2nc3c(F)cnc(CC(C)C)c3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1ccc(n(Cc2nc3c(F)cnc(CC(C)C)c3[nH]2)c1=O)C(F)(F)F |r|
CC(C)Cc1ncc(F)c2nc(Cn3c(ccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c3=O)C(F)(F)F)[nH]c12 |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(F)cnc(CC4CC4)c3[nH]2)c1=O |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(F)cnc(CC4CC4)c3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1ccc(CO)n(Cc2nc3c(F)cnc(CC(C)C)c3[nH]2)c1=O |r|
CC(C)Oc1c(cnc2cc(Cn3cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c3=O)[nH]c12)C(F)(F)F |r|
CCCc1ccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)NC(=O)OC)c(=O)n1Cc1nc2c(F)cnc(CC(C)C)c2[nH]1 |r|
CC(C)Cc1ncc(F)c2nc(Cn3c(C)c(F)cc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c3=O)[nH]c12 |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3ncc(F)c(CC4CCC4)c3[nH]2)c1=O |r|
CC(C)Cc1ncc(F)c2nc(Cn3cc(Cl)cc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c3=O)[nH]c12 |r|
CC(C)Cc1ncc(F)c2nc(Cn3cc(F)cc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c3=O)[nH]c12 |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2cc3ncc(F)c(CC4CCC4)c3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1ccc(F)n(Cc2nc3c(F)cnc(CC(C)C)c3[nH]2)c1=O |r|
CC(C)Cc1ncc(F)c2nc(Cn3c(F)ccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c3=O)[nH]c12 |r|
CC(C)Cc1ncc(F)c2nc(Cn3c(CO)ccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c3=O)[nH]c12 |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1ccc(C)n(Cc2[nH]c3c(CC(C)C)c(F)cnc3c2C)c1=O |r|
CC(C)Cc1c(F)cnc2c(C)c(Cn3c(C)ccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c3=O)[nH]c12 |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1ccc(Cl)n(Cc2nc3c(F)cnc(CC4CC4)c3[nH]2)c1=O |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1ccc(Cl)n(Cc2nc3c(F)cnc(CC4CC4)c3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1ccc(C)n(Cc2nc3c(F)cnc(CC4CC4)c3[nH]2)c1=O |r|
CN(C)C(=O)O[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1ccc(C)n(Cc2nc3c(F)cnc(CC4CC4)c3[nH]2)c1=O |r|
CCCc1ccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c(=O)n1Cc1nc2c(F)cnc(CC(C)C)c2[nH]1 |r|
COCc1ccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c(=O)n1Cc1nc2c(F)cnc(CC(C)C)c2[nH]1 |r|
CC(C)Cc1c(F)cnc2c(C)c(Cn3cccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c3=O)[nH]c12 |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1cccn(Cc2nc3c(F)cnc(CCC(F)(F)F)c3[nH]2)c1=O |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1ccc(Cl)n(Cc2nc3c(F)cnc(CC(C)C)c3[nH]2)c1=O |r|
CC(C)Cc1ncc(F)c2nc(Cn3c(Cl)ccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c3=O)[nH]c12 |r|
CC(C)Cc1ncc(F)c2nc(Cn3c(C)ccc(NC(=O)[C@H](CC\C=C\C(=O)N(C)C)OC(=O)N(C)C)c3=O)[nH]c12 |r|
COC(=O)N[C@@H](CC\C=C\C(=O)N(C)C)C(=O)Nc1ccc(C)n(Cc2nc3c(F)cnc(CC(C)C)c3[nH]2)c1=O |r|
Cc1cc(ccc1-c1cc(N)c2cnc(NC(=O)[C@H]3CC3C#N)cc2c1)C#N |r|
Cc1ccncc1-c1cc(N)c2cnc(NC(=O)C3CC3)cc2c1
Nc1cc(cc2cc(NC(=O)[C@@H]3C[C@@H]3F)ncc12)-c1cnccc1CO |r|
Cc1ccncc1-c1cc2cc(NC(=O)C3CC3)ncc2c(N)c1F
Cc1ccncc1-c1cc2cc(NC(=O)C3CC3)ncc2c(N)c1C#N
Cn1cc(cn1)-c1cc2cc(NC(=O)C3CC3)ncc2c(N)c1C#N
Nc1c(Cl)ccc2cc(NC(=O)C3CC3)ncc12
Nc1c(ccc2cc(NC(=O)C3CC3)ncc12)C#N
CNC(=O)c1ncc(c(C)n1)-c1cc(N)c2cnc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1 |r|
Cc1cc2[nH]cnc2cc1-c1cc(N)c2cnc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1 |r|
Nc1cc(cc2cc(NC(=O)[C@@H]3C[C@@H]3F)ncc12)-c1cnncc1C1CC1 |r|
Cc1c(cnc2[nH]cnc12)-c1cc(N)c2cnc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1 |r|
CC(C)c1[nH]ncc1-c1cc(N)c2cnc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1 |r|
CCn1cc(C)c(cc1=O)-c1cc(N)c2cnc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1 |r|
Cc1c[nH]c(=O)cc1-c1cc(N)c2cnc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1 |r|
CC(C)NC(=O)Nc1cc2cc(cc(N)c2cn1)-c1cnn(C)c1
Cn1ccc2c(ccnc12)-c1cc(N)c2cnc(NC(=O)[C@H]3C[C@@H]3C#N)cc2c1 |r|
Nc1cc(cc2cc(NC(=O)[C@H]3C[C@@H]3C#N)ncc12)-c1ccnc2[nH]ccc12 |r|
CCc1ccc(=O)n(C)c1-c1cc(N)c2cnc(NC(=O)[C@@H]3C[C@H]3C#N)cc2c1 |r|
Cc1ccn(C)c(=O)c1-c1cc(N)c2cnc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1 |r|
Cc1ccn(C)c(=O)c1-c1cc(N)c2cnc(NC(=O)[C@@H]3C[C@H]3F)cc2c1 |r|
COc1ccc(c(C)n1)-c1cc(N)c2cnc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1 |r|
Cc1[nH]c(=O)ccc1-c1cc(N)c2cnc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1 |r|
Cc1[nH]ncc1-c1cc(N)c2cnc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1 |r|
Nc1cc(cc2cc(NC(=O)[C@@H]3C[C@@H]3F)ncc12)C1CNC(=O)C1 |r|
CCc1cc(CO)ncc1-c1cc(N)c2cnc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1 |r|
Cc1ccncc1-c1cc(N)c2cnc(NC(=O)[C@H]3C[C@@H]3C#N)cc2c1 |r|
CC1COC(=O)N1c1cc(N)c2cnc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1 |r|
Nc1cc(cc2cc(NC(=O)[C@@H]3C[C@H]3C#N)ncc12)-c1ccnc2ccccc12 |r|
CCc1c(N)cncc1-c1cc(N)c2cnc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1 |r|
Cc1ccncc1-c1cc(N)c2cnc(NC(=O)CCN)cc2c1
CC(C)c1[nH]ncc1-c1cc(N)c2cnc(NC(=O)[C@@H]3C[C@H]3F)cc2c1 |r|
Cn1c(cccc1=O)-c1cc(N)c2cnc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1 |r|
Cc1cc2[nH]ncc2cc1-c1cc(N)c2cnc(NC(=O)[C@@H]3C[C@H]3C#N)cc2c1 |r|
Cc1cc2[nH]ncc2cc1-c1cc(N)c2cnc(NC(=O)[C@@H]3C[C@H]3C(N)=O)cc2c1 |r|
COc1ccncc1-c1cc(N)c2cnc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1 |r|
COc1ccncc1-c1cc(N)c2cnc(NC(=O)[C@H]3C[C@@H]3F)cc2c1 |r|
Cc1cc[nH]c(=O)c1-c1cc(N)c2cnc(NC(=O)[C@H]3C[C@H]3F)cc2c1 |r|
Cc1c(F)cncc1-c1cc(N)c2cnc(NC(=O)[C@H]3C[C@H]3F)cc2c1 |r|
Nc1cc(cc2cc(NC(=O)[C@H]3C[C@H]3F)ncc12)-c1cccnc1 |r|
Cc1cnccc1-c1cc(N)c2cnc(NC(=O)[C@@H]3C[C@H]3C#N)cc2c1 |r|
Cc1ccncc1-c1cc2cc(NC(=O)[C@H]3C[C@@H]3C#N)ncc2c(N)c1F |r|
Cc1cc2[nH]c(=O)oc2cc1-c1cc(N)c2cnc(NC(=O)[C@H]3C[C@@H]3C#N)cc2c1 |r|
CCC1CCC(=O)N1c1cc(N)c2cnc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1 |r|
CCOc1cc(CC)c(cn1)-c1cc(N)c2cnc(NC(=O)[C@H]3C[C@@H]3C#N)cc2c1 |r|
Cc1ncc(-c2cc(N)c3cnc(NC(=O)[C@H]4C[C@@H]4C#N)cc3c2)n1C |r|
Cc1cnccc1-c1cc(N)c2cnc(NC(=O)[C@H]3C[C@H]3F)cc2c1 |r|
CC(F)(F)c1ccncc1-c1cc(N)c2cnc(NC(=O)[C@H]3C[C@@H]3C#N)cc2c1 |r|
Cc1ccncc1-c1cc(N)c2cnc(NC(=O)CC3COCCN3)cc2c1
Cc1cnsc1-c1cc(N)c2cnc(NC(=O)C3CC3C#N)cc2c1
CCc1cc(OC(F)F)ncc1-c1cc(N)c2cnc(NC(=O)[C@H]3C[C@@H]3C#N)cc2c1 |r|
Nc1cc(cc2cc(NC(=O)[C@H]3C[C@@H]3C#N)ncc12)-c1cnccc1CCO |r|
CCc1ccncc1-c1cc(N)c2cnc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1 |r|
CCc1ccncc1-c1cc(N)c2cnc(NC(=O)[C@H]3C[C@@H]3C#N)cc2c1 |r|
CCc1ccncc1-c1cc(N)c2cnc(NC(=O)[C@H]3C[C@H]3C#N)cc2c1 |r|
Cc1cc(ncc1-c1cc(N)c2cnc(NC(=O)[C@@H]3C[C@H]3C#N)cc2c1)C#N |r|
Cc1c(cnc2nccnc12)-c1cc(N)c2cnc(NC(=O)[C@@H]3C[C@H]3C#N)cc2c1 |r|
CCc1ccncc1-c1cc(N)c2cnc(NC(=O)C3CC3C#N)cc2c1
Cc1ccncc1-c1cc(N)c2cnc(NC(=O)C3CC3C#N)cc2c1
Cn1ccc2c(cncc12)-c1cc(N)c2cnc(NC(=O)C3CC3C#N)cc2c1
Cn1ncc2c(cncc12)-c1cc(N)c2cnc(NC(=O)C3CC3C#N)cc2c1
CCc1ccncc1-c1cc(N)c2cnc(NC(=O)Cc3ccn[nH]3)cc2c1
Cc1cn2ccnc2cc1-c1cc(N)c2cnc(NC(=O)C3CC3C#N)cc2c1
CNC(=O)c1cc(-c2cc(N)c3cnc(NC(=O)C4CC4C#N)cc3c2)n(C)n1
Cc1ccncc1-c1cc2cc(NC(=O)C3CC3C#N)ncc2c(N)c1C#N
Nc1cc(cc2cc(NC(=O)C3CC3C#N)ncc12)-c1c[nH]nc1C(F)(F)F
Nc1cc(cc2cc(NC(=O)C3CC3C#N)ncc12)-c1cn[nH]c1
Cc1ccncc1-c1cc(N)c2cnc(NC(=O)C3CC3CO)cc2c1
Cn1cc2c(cncc2n1)-c1cc(N)c2cnc(NC(=O)C3CC3C#N)cc2c1
Cn1ccc(=O)cc1-c1cc(N)c2cnc(NC(=O)C3CC3C#N)cc2c1
CC1C=CNC=C1c1cc2cc(NC(=O)C3CC3C#N)ncc2c(N)c1C |c:2,5|
CN1C=CNC=C1c1cc2cc(NC(=O)C3CC3C#N)ncc2c(N)c1Cl |c:2,5|
CN(C)c1ccncc1-c1cc(N)c2cnc(NC(=O)C3CC3C#N)cc2c1
Cc1cc(ccc1-c1cc(N)c2cnc(NC(=O)C3CC3C#N)cc2c1)C(=O)NCC(F)(F)F
Cc1cc2[nH]c(=O)oc2cc1-c1cc(N)c2cnc(NC(=O)C3CC3C#N)cc2c1
Cc1cc2[nH]c(=O)oc2cc1-c1cc(N)c2cnc(NC(=O)[C@@H]3C[C@H]3C#N)cc2c1 |r|
Nc1cc(cc2cc(NC(=O)C3CC3C#N)ncc12)-c1cnccc1CCO
Nc1cc(cc2cc(NC(=O)[C@@H]3CC3C#N)ncc12)-c1cnccc1CCO |r|
Cc1csnc1-c1cc(N)c2cnc(NC(=O)C3CC3C#N)cc2c1
CNC(=O)c1ccc(C)c(c1)-c1cc(N)c2cnc(NC(=O)C3CC3C#N)cc2c1
CC1(C)CN(C(=O)O1)c1cc(N)c2cnc(NC(=O)C3CC3C#N)cc2c1
CC(C)C1COC(=O)N1c1cc(N)c2cnc(NC(=O)C3CC3C#N)cc2c1
Cc1ccncc1-c1cc2cc(NC(=O)C3CC3C#N)ncc2c(N)c1F
CC1COC(=O)N1c1cc(N)c2cnc(NC(=O)C3CC3C#N)cc2c1
Cc1c(N)cncc1-c1cc(N)c2cnc(NC(=O)C3CC3C#N)cc2c1
Cc1[nH]nc(CO)c1-c1cc(N)c2cnc(NC(=O)C3CC3C#N)cc2c1
Cc1ccncc1-c1c(F)c(N)c2cnc(NC(=O)C3CC3C#N)cc2c1F |(3.48,-2.47,;4.8,-1.71,;6.16,-2.49,;7.47,-1.73,;7.47,-.19,;6.13,.62,;4.82,-.14,;3.43,.67,;3.46,2.21,;4.8,2.94,;2.1,2.99,;2.1,4.48,;.78,2.21,;-.58,2.96,;-1.94,2.16,;-1.94,.64,;-3.28,-.19,;-4.62,.59,;-4.62,2.16,;-5.98,-.17,;-7.47,-.17,;-6.73,1.18,;-6.73,2.72,;-6.73,4.26,;-.56,-.14,;.73,.64,;2.12,-.14,;2.12,-1.67,)|
Cc1c(cnc2nccnc12)-c1cc(N)c2cnc(NC(=O)C3CC3C#N)cc2c1
CC1COC(=O)N1c1cc(N)c2cnc(NC(=O)C3CC3F)cc2c1
Cc1cn2ccnc2cc1-c1cc(N)c2cnc(NC(=O)[C@H]3C[C@@H]3C#N)cc2c1 |r|
CNC(=O)c1cc(-c2cc(N)c3cnc(NC(=O)[C@@H]4C[C@H]4C#N)cc3c2)n(C)n1 |r|
Cc1ccncc1-c1cc2cc(NC(=O)[C@H]3C[C@@H]3C#N)ncc2c(N)c1C#N |r|
Cc1ccncc1-c1cc2cc(NC(=O)[C@@H]3C[C@H]3C#N)ncc2c(N)c1C#N |r|
Cc1ccncc1-c1cc2cc(NC(=O)[C@@H]3C[C@H]3C#N)ncc2c(N)c1C |r|
CN(C)c1ccncc1-c1cc(N)c2cnc(NC(=O)[C@@H]3C[C@H]3C#N)cc2c1 |r|
Cn1ccc(=O)cc1-c1cc(N)c2cnc(NC(=O)[C@H]3C[C@@H]3C#N)cc2c1 |r|
Cc1[nH]nc(CO)c1-c1cc(N)c2cnc(NC(=O)[C@H]3C[C@@H]3C#N)cc2c1 |r|
Cc1ccncc1-c1cc(N)c2cnc(NC(=O)[C@H]3C[C@@H]3CO)cc2c1 |r|
Cc1ccncc1-c1cc(N)c2cnc(NC(=O)[C@@H]3C[C@H]3CO)cc2c1 |r|
Nc1cc(cc2cc(NC(=O)[C@@H]3C[C@H]3C#N)ncc12)-c1c[nH]nc1C(F)(F)F |r|
C[C@@H]1COC(=O)N1c1cc(N)c2cnc(NC(=O)[C@@H]3C[C@H]3C#N)cc2c1 |r|
CC1CCC(=O)N1c1cc(N)c2cnc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1 |r|
C[C@@H]1COC(=O)N1c1cc2cc(NC(=O)[C@@H]3C[C@H]3C#N)ncc2c(N)c1F |r|
C[C@H]1COC(=O)N1c1cc(N)c2cnc(NC(=O)[C@@H]3C[C@H]3C#N)cc2c1 |r|
C[C@H]1COC(=O)N1c1cc(N)c2cnc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1 |r|
Cc1csnc1-c1cc(N)c2cnc(NC(=O)[C@@H]3C[C@H]3C#N)cc2c1 |r|
Nc1cc(cc2cc(NC(=O)[C@H]3C[C@@H]3C#N)ncc12)N1CC[C@@H](O)C1=O |r|
Nc1cc(cc2cc(NC(=O)[C@H]3C[C@@H]3C#N)ncc12)N1CC[C@H](O)C1=O |r|
CC(C)c1c(cnn1C)-c1cc(N)c2cnc(NC(=O)[C@@H]3C[C@H]3C#N)cc2c1 |r|
Nc1cc(cc2cc(NC(=O)[C@@H]3C[C@H]3C#N)ncc12)-n1c2ccccc2oc1=O |r|
CNC(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnccc1C
CNC(=O)c1ccc(C)c(c1)-c1cc(N)c2cnc(NC(=O)[C@H]3C[C@@H]3C#N)cc2c1 |r|
Cn1c2ccccc2n(-c2cc(N)c3cnc(NC(=O)[C@H]4C[C@@H]4C#N)cc3c2)c1=O |r|
Nc1cc(cc2cc(NC(=O)[C@H]3C[C@@H]3C#N)ncc12)-c1cn[nH]c1 |r|
Nc1cc(cc2cc(NC(=O)[C@H]3C[C@@H]3C#N)ncc12)-n1c2ccccc2[nH]c1=O |r|
Cc1ccncc1-c1cc2cc(NC(=O)[C@H]3C[C@@H]3C#N)ncc2c(N)c1C(F)(F)F |r|
CC1CNC(=O)N1c1cc(N)c2cnc(NC(=O)[C@@H]3C[C@H]3C#N)cc2c1 |r|
Cc1ccncc1-c1c(F)c(N)c2cnc(NC(=O)[C@H]3C[C@@H]3C#N)cc2c1F |r,wU:21.23,wD:19.19,(2.77,-1.26,;4.1,-.49,;5.44,-1.26,;6.77,-.49,;6.77,1.05,;5.44,1.82,;4.1,1.05,;2.77,1.82,;2.77,3.36,;4.1,4.13,;1.44,4.13,;1.44,5.67,;.1,3.36,;-1.23,4.13,;-2.56,3.36,;-2.56,1.82,;-3.9,1.05,;-3.9,-.49,;-2.56,-1.26,;-5.23,-1.26,;-6.77,-1.26,;-6,-2.59,;-6,-4.13,;-6,-5.67,;-1.23,1.05,;.1,1.82,;1.44,1.05,;1.44,-.49,)|
Cc1ccncc1-c1cc2cc(NC(=O)[C@H]3C[C@@H]3C#N)ncc2c(N)c1Cl |r|
CNC(=O)Nc1cc2cc(c(Cl)c(N)c2cn1)-c1cnccc1C
CNC(=O)Nc1cc2c(Cl)c(cc(N)c2cn1)-c1cnccc1C
CNC(=O)Nc1cc2c(C#N)c(cc(N)c2cn1)-c1cnccc1C
CNC(=O)Nc1cc2cc(-c3cnccc3C)c(C#N)c(N)c2cn1
Nc1cc(cc2cc(NC(=O)[C@H]3C[C@@H]3C#N)ncc12)C1CNC(=O)O1 |r|
Cc1ccncc1-c1cc2cc(NC(=O)[C@@H]3C[C@H]3C#N)ncc2c(N)c1CO |r|
CC(C)NC(=O)Nc1cc2cc(cc(N)c2cn1)N1C(C)COC1=O
Cc1cc(ccc1-c1cc(N)c2cnc(NC(=O)[C@H]3C[C@@H]3C#N)cc2c1)C(=O)NCC(F)(F)F |r|
Cc1coc(=O)n1-c1cc(N)c2cnc(NC(=O)[C@@H]3C[C@H]3C#N)cc2c1 |r|
CC1CNCC(=O)N1c1cc(N)c2cnc(NC(=O)[C@H]3C[C@@H]3C#N)cc2c1 |r|
C[C@H]1COC(=O)N1c1cc2cc(NC(=O)[C@@H]3C[C@H]3C#N)ncc2c(N)c1F |r|
C[C@@H]1COC(=O)N1c1cc(N)c2cnc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1 |r|
C[C@@H]1COC(=O)N1c1cc(N)c2cnc(NC(=O)[C@@H]3C[C@H]3F)cc2c1 |r|
Cc1c(N)cncc1-c1cc(N)c2cnc(NC(=O)[C@H]3C[C@@H]3C#N)cc2c1 |r|
Cc1c(N)cncc1-c1cc(N)c2cnc(NC(=O)[C@@H]3C[C@H]3C#N)cc2c1 |r|
Cc1cnsc1-c1cc(N)c2cnc(NC(=O)[C@H]3C[C@@H]3C#N)cc2c1 |r|
Cn1ccc2c(cncc12)-c1cc(N)c2cnc(NC(=O)[C@H]3C[C@@H]3C#N)cc2c1 |r|
Cn1ncc2c(cncc12)-c1cc(N)c2cnc(NC(=O)[C@H]3C[C@@H]3C#N)cc2c1 |r|
Cn1cc2c(cncc2n1)-c1cc(N)c2cnc(NC(=O)[C@H]3C[C@@H]3C#N)cc2c1 |r|
CC1(C)CN(C(=O)O1)c1cc(N)c2cnc(NC(=O)[C@H]3C[C@@H]3C#N)cc2c1 |r|
CC(C)C1COC(=O)N1c1cc(N)c2cnc(NC(=O)[C@H]3C[C@@H]3C#N)cc2c1 |r|
CC(C)[C@@H]1COC(=O)N1c1cc(N)c2cnc(NC(=O)[C@H]3C[C@@H]3C#N)cc2c1 |r|
Nc1cc(cc2cc(NC(=O)[C@H]3C[C@@H]3C#N)ncc12)N1CCOC1=O |r|
Nc1cc(cc2cc(NC(=O)[C@H]3C[C@@H]3C#N)ncc12)N1C2CCCC2OC1=O |r|
CN(C)S(=O)(=O)c1cc(N)c2cnc(NC(=O)[C@H]3C[C@@H]3C(N)=O)cc2c1 |r|
CN(C)S(=O)(=O)c1cc(N)c2cnc(NC(=O)[C@H]3C[C@@H]3C#N)cc2c1 |r|
Cc1ccnc(-c2ccnn2C)c1-c1cc(N)c2cnc(NC(=O)[C@H]3C[C@@H]3c3cnn(C)c3)cc2c1 |r|
Cc1ccnc(-c2ccnn2C)c1-c1cc(N)c2cnc(NC(=O)[C@@H]3C[C@H]3c3cnn(C)c3)cc2c1 |r|
Cc1ccnc(-c2ccccc2)c1-c1cc(N)c2cnc(NC(=O)[C@@H]3C[C@H]3c3cnn(C)c3)cc2c1 |r|
Cc1ccnc(-c2ccccc2)c1-c1cc(N)c2cnc(NC(=O)[C@H]3C[C@@H]3c3cnn(C)c3)cc2c1 |r|
Cc1ccnc(N2CCCCC2)c1-c1cc(N)c2cnc(NC(=O)[C@H]3C[C@@H]3c3cnn(C)c3)cc2c1 |r|
Cc1c(N)nccc1-c1cc(N)c2cnc(NC(=O)[C@H]3C[C@@H]3c3cnn(C)c3)cc2c1 |r|
CC(C)Nc1nccc(c1C)-c1cc(N)c2cnc(NC(=O)[C@@H]3C[C@H]3C#N)cc2c1 |r|
Cc1ccnc(-c2cnn(C)c2)c1-c1cc(N)c2cnc(NC(=O)[C@H]3C[C@@H]3CC#N)cc2c1 |r|
Nc1cc(cc2cc(NC(=O)C3CC3)ncc12)-c1cncc2NCCc12
COC[C@H]1C(C)[C@@H]1C(=O)Nc1cc2cc(cc(NC(=O)OC(C)(C)C)c2cn1)-c1cnccc1C |r|
C[C@@H]1Cc2c(N1)cncc2-c1cc(N)c2cnc(NC(=O)C3CC3)cc2c1 |r|
C[C@H]1[C@@H](CC#N)[C@H]1C(=O)Nc1cc2cc(cc(N)c2cn1)-c1cnccc1C |r|
C[C@H]1[C@H](CC#N)[C@H]1C(=O)Nc1cc2cc(cc(N)c2cn1)-c1cnccc1C |r|
C[C@@H](C#N)n1cc(Nc2cc3cc(c(F)c(N)c3cn2)-c2cnccc2C)cn1 |r|
C[C@H](C#N)n1cc(Nc2cc3cc(c(F)c(N)c3cn2)-c2cnccc2C)cn1 |r|
C[C@H]1[C@@H]([C@H]1c1cnn(C)c1)C(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnccc1C |r|
C[C@@H]1[C@H]([C@@H]1c1cnn(C)c1)C(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnccc1C |r|
C[C@H]1[C@H]([C@@H]1c1cnn(C)c1)C(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnccc1C |r|
C[C@@H](C#N)n1ccc(Nc2cc3cc(cc(N)c3cn2)-c2cnccc2C)n1 |r|
C[C@H](C#N)n1ccc(Nc2cc3cc(cc(N)c3cn2)-c2cnccc2C)n1 |r|
C[C@@H](C#N)n1cc(Nc2cc3cc(cc(N)c3cn2)-c2cnccc2C)cn1 |r|
C[C@H](C#N)n1cc(Nc2cc3cc(cc(N)c3cn2)-c2cnccc2C)cn1 |r|
CC(C#N)n1cc(Nc2cc3c(Cl)c(cc(N)c3cn2)-c2cnccc2C)cn1
CC(C#N)n1cc(Nc2cc3c(Cl)c(c(Cl)c(N)c3cn2)-c2cnccc2C)cn1 |(-1.37,4.48,;-2.85,4.08,;-3.25,2.59,;-3.65,1.1,;-3.94,5.17,;-3.47,6.63,;-4.71,7.54,;-4.71,9.08,;-3.38,9.85,;-2.04,9.08,;-.71,9.85,;.62,9.08,;.62,7.54,;1.96,9.85,;1.96,11.39,;3.29,12.16,;.62,12.16,;.62,13.7,;-.71,11.39,;-2.04,12.16,;-3.38,11.39,;3.29,9.08,;4.62,9.85,;5.96,9.08,;5.96,7.54,;4.62,6.77,;3.29,7.54,;1.96,6.77,;-5.96,6.63,;-5.48,5.17,)|
C[C@@H](C#N)n1cc(Nc2cc3cc(c(Cl)c(N)c3cn2)-c2cnccc2C)cn1 |r|
C[C@H](C#N)n1cc(Nc2cc3cc(c(Cl)c(N)c3cn2)-c2cnccc2C)cn1 |r|
Cc1ccnc(N2CCCC2)c1-c1cc(N)c2cnc(NC(=O)[C@@H]3C[C@H]3c3cnn(C)c3)cc2c1 |r|
Cc1ccnc(N2CCCC2)c1-c1cc(N)c2cnc(NC(=O)[C@H]3C[C@@H]3c3cnn(C)c3)cc2c1 |r|
Cc1c(N)cncc1-c1cc2cc(NC(=O)[C@H]3C[C@@H]3CC#N)ncc2c(N)c1Cl |r|
Cc1ccnc(-c2cnn(C)c2)c1-c1cc(N)c2cnc(NC(=O)[C@@H]3C[C@H]3c3cnn(C)c3)cc2c1 |r|
Cc1ccnc(-c2cnn(C)c2)c1-c1cc(N)c2cnc(NC(=O)[C@H]3C[C@@H]3c3cnn(C)c3)cc2c1 |r|
C[C@@H]1[C@@H]([C@H]1c1cnn(C)c1)C(=O)Nc1cc2cc(cc(N)c2cn1)-c1cnccc1C |r|
C[C@H]1[C@@H]([C@H]1c1cnn(C)c1)C(=O)Nc1cc2cc(cc(N)c2cn1)-c1cnccc1C |r|
C[C@@H]1[C@H]([C@@H]1c1cnn(C)c1)C(=O)Nc1cc2cc(cc(N)c2cn1)-c1cnccc1C |r|
C[C@H]1[C@H]([C@@H]1c1cnn(C)c1)C(=O)Nc1cc2cc(cc(N)c2cn1)-c1cnccc1C |r|
Cn1cc(cn1)[C@@H]1C[C@H]1C(=O)Nc1cc2cc(cc(N)c2cn1)-c1c(Cl)cccc1Cl |r|
Cn1cc(cn1)[C@H]1C[C@@H]1C(=O)Nc1cc2cc(cc(N)c2cn1)-c1c(Cl)cccc1Cl |r|
Cn1cc(cn1)[C@H]1C[C@@H]1C(=O)Nc1cc2cc(cc(N)c2cn1)-c1c(F)cccc1F |r|
Cn1cc(cn1)[C@@H]1C[C@H]1C(=O)Nc1cc2cc(cc(N)c2cn1)-c1c(F)cccc1F |r|
Cc1cccc(C#N)c1-c1cc(N)c2cnc(NC(=O)[C@H]3C[C@@H]3C#N)cc2c1 |r|
Cc1ccnc(-c2ccn(C)n2)c1-c1cc(N)c2cnc(NC(=O)[C@H]3C[C@@H]3c3cnn(C)c3)cc2c1 |r|
Cc1ccncc1-c1cc2cc(NC(=O)[C@@H]3[C@H]4CC(O)C[C@@H]34)ncc2c(N)c1Cl |r,w:18.19|
Cc1ccncc1-c1cc(N)c2cnc(NC(=O)[C@@H]3[C@H]4CC(O)C[C@@H]34)cc2c1Cl |r,w:21.22|
Cc1ccncc1-c1c(Cl)c(N)c2cnc(NC(=O)[C@@H]3[C@H]4CC(O)C[C@@H]34)cc2c1Cl |r,w:22.23,wU:19.19,wD:20.21,25.25,(4.94,-3.31,;6.27,-2.54,;7.61,-3.31,;8.94,-2.54,;8.94,-1,;7.61,-.23,;6.27,-1,;4.94,-.23,;4.94,1.31,;6.27,2.08,;3.6,2.08,;3.6,3.62,;2.27,1.31,;.94,2.08,;-.4,1.31,;-.4,-.23,;-1.73,-1,;-3.06,-.23,;-3.06,1.31,;-4.4,-1,;-5.94,-1,;-7.44,-1.32,;-7.61,-2.85,;-8.94,-3.62,;-6.2,-3.48,;-5.17,-2.33,;.94,-1,;2.27,-.23,;3.6,-1,;3.6,-2.54,)|
CC1CN(C)C(=O)Cn2nc(Nc3cc4cc(c(F)c(N)c4cn3)-c3cnccc3C)cc12
CN1CC2(CC2)c2cc(Nc3cc4cc(c(F)c(N)c4cn3)-c3cnccc3C)nn2CC1=O
CN1CCc2cc(Nc3cc4cc(c(F)c(N)c4cn3)-c3cncc(N)c3C)nn2CC1=O
CN1CCc2cc(Nc3cc4cc(c(F)c(N)c4cn3)-c3cnccc3C)nn2CC1=O
CC[C@@H]1[C@H]([C@@H]1c1cnn(C)c1)C(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnc2OCCNc2c1C |r|
CC[C@H]1[C@@H]([C@H]1c1cnn(C)c1)C(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnc2OCCNc2c1C |r|
CC[C@@H]1[C@@H]([C@H]1c1cnn(C)c1)C(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnc2OCCNc2c1C |r|
CC[C@H]1[C@H]([C@@H]1c1cnn(C)c1)C(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnc2OCCNc2c1C |r|
Cc1c2NCCOc2ncc1-c1cc2cc(NC(=O)NCC3CC3)ncc2c(N)c1F
C[C@@H]1[C@@H]([C@H]1c1cnn(C)c1)C(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnc2OCCNc2c1C |r|
C[C@H]1[C@H]([C@@H]1c1cnn(C)c1)C(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnc2OCCNc2c1C |r|
C[C@H]1[C@@H]([C@H]1c1cnn(C)c1)C(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnc2OCCNc2c1C |r|
C[C@@H]1[C@H]([C@@H]1c1cnn(C)c1)C(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnc2OCCNc2c1C |r|
Cc1c(N)cncc1-c1cc2cc(NC(=O)OC3CCOCC3)ncc2c(N)c1F
COCCOC(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cncc(N)c1C
Cc1c(N)cncc1-c1cc2cc(NC(=O)C3CC3)ncc2c(N)c1F
Cc1c(N)cncc1-c1cc2cc(NC(=O)[C@@H]3C[C@H]3C#N)ncc2c(N)c1F |r|
Cc1c(N)cncc1-c1cc2cc(NC(=O)[C@H]3C[C@@H]3C#N)ncc2c(N)c1F |r|
Cc1c2NCCOc2ncc1-c1cc2cc(N)ncc2c(N)c1F
Cc1ccncc1-c1cc2cc(N)ncc2c(N)c1C#N
C[C@@H](NC(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnc2OCCNc2c1C)c1cnn(C)c1 |r|
C[C@H](NC(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnc2OCCNc2c1C)c1cnn(C)c1 |r|
Cc1c(N)cncc1-c1cc2cc(NC(=O)OCC3CC3)ncc2c(N)c1F
Cc1c(N)cncc1-c1cc2cc(NC(=O)[C@H]3[C@H](c4cnn(C)c4)C3(C)C)ncc2c(N)c1F |r|
Cc1c(N)cncc1-c1cc2cc(NC(=O)[C@@H]3[C@@H](c4cnn(C)c4)C3(C)C)ncc2c(N)c1F |r|
CC(C)OC(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cncc(N)c1C
Cc1ccncc1-c1cc2cc(Nc3cccc(c3)C3COCCN3)ncc2c(N)c1F
Cc1ccncc1-c1cc2cc(Nc3cccc(c3)[C@H]3COCCN3)ncc2c(N)c1F |r|
Nc1c(F)c(cc2cc(NC(=O)[C@@H]3C[C@@H]3F)ncc12)-c1c(Cl)cccc1Cl |r,wU:12.11,14.15,(2.1,3.75,;2.1,2.21,;3.44,1.44,;4.77,2.21,;3.44,-.1,;2.1,-.87,;.77,-.1,;-.56,-.87,;-1.9,-.1,;-3.23,-.87,;-4.56,-.1,;-4.56,1.44,;-5.9,-.87,;-7.44,-.87,;-6.67,-2.21,;-6.67,-3.75,;-1.9,1.44,;-.56,2.21,;.77,1.44,;4.77,-.87,;4.77,-2.41,;3.44,-3.18,;6.1,-3.18,;7.44,-2.41,;7.44,-.87,;6.1,-.1,;6.1,1.44,)|
Cc1c(N)cncc1-c1cc2cc(NC(=O)[C@@H]3[C@H]4COC[C@@H]34)ncc2c(N)c1F |r|
CC(C)N1CCc2cc(Nc3cc4cc(C5=CCN(CC5)C(C)=O)c(F)c(N)c4cn3)nn2CC1=O |t:15|
CC(C)N1CCc2cc(Nc3cc4cc(c(F)c(N)c4cn3)-c3cnc4OCCNc4c3C)nn2CC1=O
Cc1c(N)cncc1-c1cc2cc(Nc3cc4CC(C)(C)NC(=O)Cn4n3)ncc2c(N)c1F
CN1C(=O)Cn2nc(Nc3cc4cc(c(F)c(N)c4cn3)-c3cncc(N)c3C)cc2CC1(C)C
C[C@H]1[C@H](CC#N)[C@H]1C(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cncc(N)c1C |r|
C[C@@H]1[C@@H](CC#N)[C@@H]1C(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cncc(N)c1C |r|
C[C@H]1[C@@H](CC#N)[C@@H]1C(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cncc(N)c1C |r|
C[C@@H]1[C@H](CC#N)[C@H]1C(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cncc(N)c1C |r|
CC(C)N1CCc2cc(Nc3cc4cc(Cc5ccc[nH]c5=O)c(F)c(N)c4cn3)nn2CC1=O
CCS(=O)(=O)Nc1cc(N)c2cnc(Nc3cc4CCN(C(C)C)C(=O)Cn4n3)cc2c1
CCc1[nH]c(=O)oc1-c1cc2cc(Nc3cc4CCN(C(C)C)C(=O)Cn4n3)ncc2c(N)c1F
CC(C)N1CCc2cc(Nc3cc4cc(c(F)c(N)c4cn3)-c3cncc(N)c3Cl)nn2CC1=O
CC(C)N1CCc2cc(Nc3cc4cc(CN5CCN(C)CC5=O)c(F)c(N)c4cn3)nn2CC1=O
CC(C)N1CCc2cc(Nc3cc4cc(c(F)c(N)c4cn3)-c3cnc(nc3C)C(=O)N(C)C)nn2CC1=O
COc1c(N)cncc1-c1cc2cc(Nc3cc4CCN(C(C)C)C(=O)Cn4n3)ncc2c(N)c1F
Cc1c(N)cncc1-c1cc2cc(Nc3cc4CCn5ccnc5Cn4n3)ncc2c(N)c1F
[#6]-[#6](-[#6])-[#7]-1-[#6]-[#6]-c2cc(-[#7]-c3cc4cc(\[#6]=[#6](\[#6])-[#6])c(F)c(-[#7])c4cn3)nn2-[#6]-[#6]-1=O
CC(C)N1CCc2cc(Nc3cc4cc(Cn5ccc6ccncc56)c(F)c(N)c4cn3)nn2CC1=O
CN1CCn2cc(Nc3cc4cc(c(F)c(N)c4cn3)-c3cnccc3C)nc2CC1=O
CC(C)N1CCc2cc(Nc3cc4cc(-c5c(C)c(N)nn5C)c(F)c(N)c4cn3)nn2CC1=O |(-2.99,-7.11,;-4.32,-6.34,;-5.65,-7.11,;-4.32,-4.8,;-5.71,-4.13,;-6.05,-2.63,;-5.09,-1.42,;-5.57,.04,;-4.32,.95,;-4.32,2.49,;-2.99,3.26,;-1.65,2.49,;-.32,3.26,;1.01,2.49,;2.35,3.26,;3.68,2.49,;3.68,.95,;2.35,.18,;5.15,.47,;5.92,-.86,;6.05,1.72,;5.15,2.96,;5.92,4.3,;2.35,4.8,;3.68,5.57,;1.01,5.57,;1.01,7.11,;-.32,4.8,;-1.65,5.57,;-2.99,4.8,;-3.07,.04,;-3.55,-1.42,;-2.59,-2.63,;-2.93,-4.13,;-1.84,-5.22,)|
Cc1c(N)cncc1-c1cc2cc(Nc3cc4CCS(=O)(=O)Cn4n3)ncc2c(N)c1F
CC(C)N1CCc2cc(Nc3cc4cc(C5CC5)c(F)c(N)c4cn3)nn2CC1=O
CC(C)N1CCc2cc(Nc3cc4ccc(F)c(N)c4cn3)nn2CC1=O
CC(C)Oc1ncc(c(C)n1)-c1cc2cc(Nc3cc4CCN(C(C)C)C(=O)Cn4n3)ncc2c(N)c1F
CC(C)N1Cc2cc(Nc3cc4cc(c(F)c(N)c4cn3)-c3cncc(N)c3C)nn2CS1(=O)=O
CC(C)N1CCc2cc(Nc3cc4cc(OCc5ccccc5)c(F)c(N)c4cn3)nn2CC1=O
CC(C)N1CCc2cc(Nc3cc4cc(C)c(F)c(N)c4cn3)nn2CC1=O
COc1cc2cc(Nc3cc4CCN(C(C)C)C(=O)Cn4n3)ncc2c(N)c1F
CC(C)N1CCc2cc(Nc3cc4cc(COc5ccccn5)c(F)c(N)c4cn3)nn2CC1=O
CC(C)N1CCc2cc(Nc3cc4cc(Cn5ccccc5=O)c(F)c(N)c4cn3)nn2CC1=O
CC1CCC(F)(F)Cn2nc(Nc3cc4cc(c(F)c(N)c4cn3)-c3cncc(N)c3C)cc12
CN1c2ccc(Nc3cc4cc(c(F)c(N)c4cn3)-c3cncc(N)c3C)nc2CS1(=O)=O
CN1CCc2cc(Nc3cc4cc(cc(N)c4cn3)C3CC3C#N)nn2CC1=O
CO[C@H]1CC[C@H](C)c2cc(Nc3cc4cc(c(F)c(N)c4cn3)-c3cncc(N)c3C)nn2C1 |r|
CO[C@@H]1CC[C@@H](C)c2cc(Nc3cc4cc(c(F)c(N)c4cn3)-c3cncc(N)c3C)nn2C1 |r|
CO[C@@H]1CC[C@H](C)c2cc(Nc3cc4cc(c(F)c(N)c4cn3)-c3cncc(N)c3C)nn2C1 |r|
CO[C@H]1CC[C@@H](C)c2cc(Nc3cc4cc(c(F)c(N)c4cn3)-c3cncc(N)c3C)nn2C1 |r|
CCn1nc(cc1-c1cc2cc(Nc3cc4CCN(C(C)C)C(=O)Cn4n3)ncc2c(N)c1F)C#N
CC(C)N1CCc2cc(Nc3cc4cc(-c5cnc6CNCCn56)c(F)c(N)c4cn3)nn2CC1=O
Cc1c(N)cncc1-c1cc2cc(Nc3cc4CCCS(=O)(=O)Cn4n3)ncc2c(N)c1F
CC(C)N1CCc2cc(Nc3cc4cc(c(F)c(N)c4cn3)-c3cc(=O)[nH]cc3C)nn2CC1=O
Cc1ccncc1-c1cc2cc(Nc3cc4CCN(CC(C)(C)O)C(=O)Cn4n3)ncc2c(N)c1F
CC(C)N1CCc2cc(Nc3cc4cc(c(F)c(N)c4cn3)-c3cncc4[C@H](O)CCc34)nn2CC1=O |r|
CC(C)N1CCc2cc(Nc3cc4cc(c(F)c(N)c4cn3)-c3cncc4[C@@H](O)CCc34)nn2CC1=O |r|
CN1Cc2cc(Nc3cc4cc(c(F)c(N)c4cn3)-c3cncc(N)c3C)nn2CS1(=O)=O
Cc1c(N)cncc1-c1cc2cc(Nc3cc4CCN(CC5COC5)C(=O)Cn4n3)ncc2c(N)c1F
COc1ncc(c(C)c1N)-c1cc2cc(Nc3cc4CCN(CC(F)F)C(=O)Cn4n3)ncc2c(N)c1F
CC[C@H]1[C@H]([C@@H]1c1cnn(C)c1)C(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cncc(N)c1C |r|
CC[C@@H]1[C@@H]([C@H]1c1cnn(C)c1)C(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cncc(N)c1C |r|
CC[C@@H]1[C@H]([C@@H]1c1cnn(C)c1)C(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cncc(N)c1C |r|
CC[C@H]1[C@@H]([C@H]1c1cnn(C)c1)C(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cncc(N)c1C |r|
Cc1c(N)cncc1-c1cc2cc(Nc3cc4CCN(C5CC5)C(=O)Cn4n3)ncc2c(N)c1F
CC(C)N1CCc2cc(Nc3cc4cc(c(F)c(N)c4cn3)-c3cncc4NCCOc34)nn2CC1=O
CC1COC(=O)N1c1cc(N)c2cnc(Nc3cc4CCN(C)C(=O)Cn4n3)cc2c1
CCc1c(N)cncc1-c1cc2cc(Nc3cc4CCN(C(C)C)C(=O)Cn4n3)ncc2c(N)c1F
CCC1c2cc(Nc3cc4cc(c(F)c(N)c4cn3)-c3cncc(N)c3C)nn2CS1(=O)=O
Cc1c(N)cncc1-c1cc2cc(Nc3cc4CCN(CC5CC5)C(=O)Cn4n3)ncc2c(N)c1F
CN1CCc2cc(Nc3cc4cc(c(F)c(N)c4cn3)-c3cncc(O)c3C)nn2CC1=O
CC(C)N1CCc2cc(Nc3cc4cc(c(F)c(N)c4cn3)-c3cncc(CO)c3C)nn2CC1=O
COCCN1CCc2cc(Nc3cc4cc(c(F)c(N)c4cn3)-c3cncc(N)c3C)nn2CC1=O
CN1CCc2cc(Nc3cc4cc(-c5cnn6CCNCc56)c(F)c(N)c4cn3)nn2CC1=O
CC1CN(C)S(=O)(=O)Cn2nc(Nc3cc4cc(c(F)c(N)c4cn3)-c3cncc(N)c3C)cc12
COc1ncc(c(C)c1N)-c1cc2cc(NC(=O)[C@H]3[C@@H](C)[C@@H]3c3cnn(C)c3)ncc2c(N)c1F |r|
COc1ncc(c(C)c1N)-c1cc2cc(NC(=O)[C@H]3[C@H](C)[C@@H]3c3cnn(C)c3)ncc2c(N)c1F |r|
COc1ncc(c(C)c1N)-c1cc2cc(NC(=O)[C@@H]3[C@@H](C)[C@H]3c3cnn(C)c3)ncc2c(N)c1F |r|
COc1ncc(c(C)c1N)-c1cc2cc(NC(=O)[C@@H]3[C@H](C)[C@H]3c3cnn(C)c3)ncc2c(N)c1F |r|
CCN1CCc2cc(Nc3cc4cc(c(F)c(N)c4cn3)-c3cncc(N)c3C)nn2CC1=O
CN1CCc2cc(Nc3cc4cc(c(F)c(N)c4cn3)-c3cnc(C)c(N)c3C)nn2CC1=O
Cc1c(N)nccc1-c1cc2cc(Nc3cc4CCN(CC(F)F)C(=O)Cn4n3)ncc2c(N)c1F
CN1CCc2cc(Nc3cc4cc(-c5cn[nH]c5C)c(F)c(N)c4cn3)nn2CC1=O
CN1Cc2cc(Nc3cc4cc(c(F)c(N)c4cn3)-c3cncc(N)c3C)nn2CC1=O
CN1C\C(=C/c2cnn(C)c2)c2cc(Nc3cc4cc(c(F)c(N)c4cn3)-c3cnccc3C)nn2CC1=O
CN1CCc2cc(Nc3cc4cc(-c5c(C)n[nH]c5C)c(F)c(N)c4cn3)nn2CC1=O |(-4.32,-6.72,;-4.32,-5.18,;-5.71,-4.51,;-6.05,-3.01,;-5.09,-1.81,;-5.57,-.34,;-4.32,.56,;-4.32,2.1,;-2.99,2.87,;-1.65,2.1,;-.32,2.87,;1.01,2.1,;2.35,2.87,;3.68,2.1,;5.15,2.58,;5.54,4.07,;6.05,1.33,;5.15,.09,;3.68,.56,;2.35,-.21,;2.35,4.41,;3.68,5.18,;1.01,5.18,;1.01,6.72,;-.32,4.41,;-1.65,5.18,;-2.99,4.41,;-3.07,-.34,;-3.55,-1.81,;-2.59,-3.01,;-2.93,-4.51,;-1.84,-5.6,)|
Cc1c(N)cncc1-c1cc2cc(Nc3cc4CCN(CC(F)(F)F)C(=O)Cn4n3)ncc2c(N)c1F
CN1CCc2cc(Nc3cc4cc(c(F)c(N)c4cn3)-c3cncc(N)c3Cl)nn2CC1=O
CN1CCc2cc(Nc3cc4cc(c(F)c(N)c4cn3)-c3ccc4OCCNc4c3C)nn2CC1=O
CN1CC(F)c2cc(Nc3cc4cc(c(F)c(N)c4cn3)-c3cncc(N)c3C)nn2CC1=O
CN1C[C@@H](F)c2cc(Nc3cc4cc(c(F)c(N)c4cn3)-c3cncc(N)c3C)nn2CC1=O |r|
CN1C[C@H](F)c2cc(Nc3cc4cc(c(F)c(N)c4cn3)-c3cncc(N)c3C)nn2CC1=O |r|
CN1CC(C)(O)c2cc(Nc3cc4cc(c(F)c(N)c4cn3)-c3cnccc3C)nn2CC1=O
Cc1c(N)cncc1-c1cc2cc(Nc3cc4CCN(CC(F)F)C(=O)Cn4n3)ncc2c(N)c1F
COCC1(O)CN(C)C(=O)Cn2nc(Nc3cc4cc(c(F)c(N)c4cn3)-c3cnccc3C)cc12
CN1CC2(CC2)c2cc(Nc3cc4cc(-c5c(C)nn(C)c5C)c(F)c(N)c4cn3)nn2CC1=O |(-3.59,-6.72,;-3.59,-5.18,;-4.97,-4.51,;-5.32,-3.01,;-6.44,-1.96,;-6.79,-3.47,;-4.36,-1.81,;-4.83,-.34,;-3.59,.56,;-3.59,2.1,;-2.25,2.87,;-.92,2.1,;.42,2.87,;1.75,2.1,;3.08,2.87,;4.42,2.1,;5.88,2.58,;6.28,4.07,;6.79,1.33,;5.88,.09,;6.28,-1.4,;4.42,.56,;3.08,-.21,;3.08,4.41,;4.42,5.18,;1.75,5.18,;1.75,6.72,;.42,4.41,;-.92,5.18,;-2.25,4.41,;-2.34,-.34,;-2.82,-1.81,;-1.85,-3.01,;-2.2,-4.51,;-1.11,-5.6,)|
CC(C)N1CCc2cc(Nc3cc4cc(c(F)c(N)c4cn3)-c3cncc(N)c3C)nn2CC1=O
CN1CC2(CC2)c2cc(Nc3cc4cc(c(F)c(N)c4cn3)-c3cncc(N)c3C)nn2CC1=O
CN1CC(=C)c2cc(Nc3cc4cc(c(F)c(N)c4cn3)-c3cnccc3C)nn2CC1=O
CC1CN(C)C(=O)Cn2nc(Nc3cc4cc(c(F)c(N)c4cn3)-c3cnc(cc3C)-c3ncco3)cc12
C[C@H]1[C@H]([C@@H]1c1cnc[nH]1)C(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnccc1C |r|
C[C@@H]1[C@H]([C@@H]1c1cnc[nH]1)C(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnccc1C |r|
C[C@H]1[C@@H]([C@H]1c1cnc[nH]1)C(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnccc1C |r|
C[C@@H]1[C@@H]([C@H]1c1cnc[nH]1)C(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnccc1C |r|
Cc1ccncc1-c1cc2cc(NC(=O)[C@@H]3[C@@H](CC#N)[C@@H]3c3c[nH]cn3)ncc2c(N)c1F |r|
Cc1ccncc1-c1cc2cc(NC(=O)[C@H]3[C@H](CC#N)[C@H]3c3c[nH]cn3)ncc2c(N)c1F |r|
Cc1ccncc1-c1cc2cc(NC(=O)[C@@H]3C[C@@H]3CO)ncc2c(N)c1F |r|
Cc1ccncc1-c1cc2cc(NC(=O)[C@@H]3[C@H](CO)[C@H]3c3cnn(C)c3)ncc2c(N)c1F |r|
C[C@@H]1[C@H]([C@@H]1c1ccn[nH]1)C(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnccc1C |r|
C[C@@H]1[C@@H]([C@H]1c1ccn[nH]1)C(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnccc1C |r|
C[C@H]1[C@@H]([C@H]1c1ccn[nH]1)C(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnccc1C |r|
C[C@H]1[C@H]([C@@H]1c1ccn[nH]1)C(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnccc1C |r|
Cc1ccncc1-c1cc2cc(NC(=O)C3CC3c3cnc[nH]3)ncc2c(N)c1F
Cc1ccncc1-c1cc2cc(NC(=O)[C@@H]3C[C@H]3c3cnc[nH]3)ncc2c(N)c1F |r|
Cc1ccncc1-c1cc2cc(NC(=O)[C@H]3C[C@@H]3c3cnc[nH]3)ncc2c(N)c1F |r|
Cc1ccncc1-c1cc2cc(NC(=O)N3CC4CC3C4)ncc2c(N)c1F |(3.85,-3.47,;5.19,-2.69,;6.52,-3.47,;7.85,-2.69,;7.85,-1.15,;6.52,-.38,;5.19,-1.15,;3.85,-.38,;2.52,-1.15,;1.18,-.38,;-.15,-1.15,;-1.48,-.38,;-2.82,-1.15,;-4.15,-.38,;-4.15,1.15,;-5.48,-1.15,;-5.48,-2.69,;-6.95,-3.17,;-7.85,-1.93,;-6.95,-.68,;-6.18,-2.01,;-1.48,1.15,;-.15,1.93,;1.18,1.15,;2.52,1.93,;2.52,3.47,;3.85,1.15,;5.19,1.93,)|
C[C@H]1[C@H]([C@@H]1c1cnn(CC(F)F)c1)C(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnccc1C |r|
C[C@@H]1[C@H]([C@@H]1c1cnn(CC(F)F)c1)C(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnccc1C |r|
C[C@H]1[C@@H]([C@H]1c1cnn(CC(F)F)c1)C(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnccc1C |r|
C[C@@H]1[C@@H]([C@H]1c1cnn(CC(F)F)c1)C(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnccc1C |r|
CN(C)C[C@@H]1C[C@@H]1C(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnccc1C |r|
CN(C)C[C@H]1C[C@H]1C(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnccc1C |r|
CN(C)C[C@H]1[C@H](CC#N)[C@H]1C(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnccc1C |r|
CN(C)C[C@@H]1[C@@H](CC#N)[C@@H]1C(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnccc1C |r|
C[C@@H]1[C@H]([C@@H]1c1cnn(CCN2CCOCC2)c1)C(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnccc1C |r|
C[C@H]1[C@H]([C@@H]1c1cnn(CCN2CCOCC2)c1)C(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnccc1C |r|
C[C@H]1[C@@H]([C@H]1c1cnn(CCN2CCOCC2)c1)C(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnccc1C |r|
C[C@@H]1[C@@H]([C@H]1c1cnn(CCN2CCOCC2)c1)C(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnccc1C |r|
C[C@@H]1[C@H]([C@@H]1c1cnn(C)c1)C(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnc(cc1C)-c1ncco1 |r|
C[C@H]1[C@@H]([C@H]1c1cnn(C)c1)C(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnc(cc1C)-c1ncco1 |r|
C[C@@H]1[C@@H]([C@H]1c1cnn(C)c1)C(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnc(cc1C)-c1ncco1 |r|
C[C@H]1[C@H]([C@@H]1c1cnn(C)c1)C(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnc(cc1C)-c1ncco1 |r|
Cc1ccncc1-c1cc2cc(NC(=O)C3CC3c3cn(C)nn3)ncc2c(N)c1F
Cc1ccncc1-c1cc2cc(NC(=O)[C@H]3C[C@@H]3c3cn(C)nn3)ncc2c(N)c1F |r|
Cc1ccncc1-c1cc2cc(NC(=O)[C@@H]3C[C@H]3c3cn(C)nn3)ncc2c(N)c1F |r|
C[C@H]1[C@H]([C@@H]1c1cnn(C)c1)C(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cncc(N)c1C |r|
C[C@@H]1[C@@H]([C@H]1c1cnn(C)c1)C(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cncc(N)c1C |r|
C[C@H]1[C@@H]([C@H]1c1cnn(C)c1)C(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cncc(N)c1C |r|
C[C@@H]1[C@H]([C@@H]1c1cnn(C)c1)C(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cncc(N)c1C |r|
C[C@H]1CN(C)C(=O)Cn2nc(Nc3cc4cc(c(F)c(N)c4cn3)-c3cnccc3C)cc12 |r|
C[C@@H]1CN(C)C(=O)Cn2nc(Nc3cc4cc(c(F)c(N)c4cn3)-c3cnccc3C)cc12 |r|
Cc1ccncc1-c1cc2cc(NC(=O)[C@H]3C[C@@H]3c3ccn[nH]3)ncc2c(N)c1F |r|
Cc1ccncc1-c1cc2cc(NC(=O)[C@@H]3C[C@H]3c3ccn[nH]3)ncc2c(N)c1F |r|
C[C@@H]1[C@H]([C@@H]1c1cnn(CCO)c1)C(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnccc1C |r|
C[C@H]1[C@H]([C@@H]1c1cnn(CCO)c1)C(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnccc1C |r|
C[C@H]1[C@@H]([C@H]1c1cnn(CCO)c1)C(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnccc1C |r|
C[C@@H]1[C@@H]([C@H]1c1cnn(CCO)c1)C(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnccc1C |r|
Cc1ccncc1-c1cc2cc(NC(=O)[C@H]3[C@@H](C3c3c[nH]cn3)c3cnn(C)c3)ncc2c(N)c1F |r|
Cc1ccncc1-c1cc2cc(NC(=O)[C@H]3[C@@H]4CCC[C@@H](O)[C@H]34)ncc2c(N)c1F |r|
Cc1ccncc1-c1cc2cc(NC(=O)[C@@H]3[C@H]4CCC[C@@H](O)[C@@H]34)ncc2c(N)c1F |r|
Cc1ccncc1-c1cc2cc(NC(=O)[C@@H]3[C@H]4CCC[C@H](O)[C@@H]34)ncc2c(N)c1F |r|
CC[C@@H]1[C@H]([C@@H]1c1cncn1C)C(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cncc(N)c1C |r|
CC[C@H]1[C@@H]([C@H]1c1cncn1C)C(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cncc(N)c1C |r|
CC[C@H]1[C@H]([C@@H]1c1cncn1C)C(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cncc(N)c1C |r|
CC[C@@H]1[C@@H]([C@H]1c1cncn1C)C(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cncc(N)c1C |r|
C[C@H]1[C@@H]([C@H]1c1cnn(CCN2CC(O)C2)c1)C(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnccc1C |r|
C[C@H]1[C@H]([C@@H]1c1cnn(CCN2CC(O)C2)c1)C(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnccc1C |r|
C[C@@H]1[C@@H]([C@H]1c1cnn(CCN2CC(O)C2)c1)C(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnccc1C |r|
C[C@@H]1[C@H]([C@@H]1c1cnn(CCN2CC(O)C2)c1)C(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnccc1C |r|
C[C@@H]1[C@H](CC#N)[C@H]1C(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnccc1C |r|
C[C@H]1[C@@H](CC#N)[C@@H]1C(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnccc1C |r|
C[C@H]1[C@H](CC#N)[C@H]1C(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnccc1C |r|
C[C@@H]1[C@@H](CC#N)[C@@H]1C(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnccc1C |r|
Cc1ccncc1-c1cc2cc(Nc3cc4CCN(CC(F)(F)F)C(=O)Cn4n3)ncc2c(N)c1F
CN1CCc2cc(Nc3cc4cc(c(F)c(N)c4cn3)-c3cccc(N)c3C)nn2CC1=O
CN1CCc2cc(Nc3cc4cc(c(F)c(N)c4cn3)-c3cc4oc(=O)[nH]c4cc3C)nn2CC1=O
CN1CC(O)c2cc(Nc3cc4cc(c(F)c(N)c4cn3)-c3cccc(N)c3C)nn2CC1=O
Cc1c2NCCOc2ncc1-c1cc2cc(NC(=O)OC3CCOCC3)ncc2c(N)c1F
CN1CC(C1)OC(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnc2OCCNc2c1C
Cc1c2NCCOc2ncc1-c1cc2cc(NC(=O)OC3CCOC3)ncc2c(N)c1F
Cc1c2NCCOc2ncc1-c1cc2cc(NC(=O)O[C@@H]3CCOC3)ncc2c(N)c1F |r|
Cc1c2NCCOc2ncc1-c1cc2cc(NC(=O)O[C@H]3CCOC3)ncc2c(N)c1F |r|
Cc1c2NCCOc2ncc1-c1cc2cc(NC(=O)OC3CCNCC3)ncc2c(N)c1F
Cc1c2NCCOc2ncc1-c1cc2cc(NC(=O)O[C@@H]3CCNC3)ncc2c(N)c1F |r|
Cc1c2NCCOc2ncc1-c1cc2cc(NC(=O)O[C@H]3CCNC3)ncc2c(N)c1F |r|
CN1C2COCC1CC(C2)OC(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnc2OCCNc2c1C |THB:0:1:8.9.7:3.4.5|
CN1CCC(CC1)OC(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnc2OCCNc2c1C
Cc1c2NCCOc2ncc1-c1cc2cc(NC(=O)O[C@@H]3CCCNC3)ncc2c(N)c1F |r|
Cc1c2NCCOc2ncc1-c1cc2cc(NC(=O)O[C@H]3CCCNC3)ncc2c(N)c1F |r|
CN1C[C@@H](CCC1=O)OC(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnc2OCCNc2c1C |r|
CN1C[C@H](CCC1=O)OC(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnc2OCCNc2c1C |r|
CN1C[C@@H](CC1=O)OC(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnc2OCCNc2c1C |r|
CN1C[C@H](CC1=O)OC(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnc2OCCNc2c1C |r|
CN1CC[C@H](C1)OC(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnc2OCCNc2c1C |r|
CN1CC[C@@H](C1)OC(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnc2OCCNc2c1C |r|
Cc1c(cnc2OCC[C@H](O)c12)-c1cc2cc(NC(=O)OC3CCOCC3)ncc2c(N)c1F |r|
Cc1c(cnc2OCC[C@@H](O)c12)-c1cc2cc(NC(=O)OC3CCOCC3)ncc2c(N)c1F |r|
Cc1c2NCCC(O)c2ncc1-c1cc2cc(NC(=O)OC3CCOCC3)ncc2c(N)c1F
CC(=O)NC1CCCC[C@@H]1OC(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnc2OCCNc2c1C |r|
CC(=O)NC1CCCC[C@H]1OC(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnc2OCCNc2c1C |r|
CNC1CCCC[C@@H]1OC(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnc2OCCNc2c1C |r|
CNC1CCCC[C@H]1OC(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnc2OCCNc2c1C |r|
CN1CCC[C@H](C1)OC(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnc2OCCNc2c1C |r|
CN1CCC[C@@H](C1)OC(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnc2OCCNc2c1C |r|
CN1CC2(CC(C2)OC(=O)Nc2cc3cc(c(F)c(N)c3cn2)-c2cnc3OCCNc3c2C)C1
CC(=O)N1CC[C@H](C1)OC(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnc2OCCNc2c1C |r|
CC(C)N1CC(C1)OC(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnc2OCCNc2c1C
Cc1c2NCCOc2ncc1-c1cc2cc(NC(=O)OC3CN(CC(F)(F)F)C3)ncc2c(N)c1F
Cc1c2NCCOc2ncc1-c1cc2cc(NC(=O)OC3CCN(CC3)C3COC3)ncc2c(N)c1F
Cc1c2NCCOc2ncc1-c1cc2cc(NC(=O)OC3CCN(CC(F)(F)F)CC3)ncc2c(N)c1F
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Cc1c2NCCCc2ncc1-c1cc2cc(NC(=O)OC3CC4(C3)CCN(CC4)C3COC3)ncc2c(N)c1F
CN1CC2CC(C1)C2OC(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnc2OCCNc2c1C
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Cc1c2NCCOc2ncc1-c1cc2cc(NC(=O)OC3CN(CC(F)F)C3)ncc2c(N)c1F
CN1CCC(OC(=O)Nc2cc3cc(c(F)c(N)c3cn2)-c2cnc3OCCNc3c2C)C(C)(C)C1
CC(C)OC(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnc2OCCNc2c1C
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Cc1c2NCCOc2ncc1-c1cc2cc(NC(=O)OC3CCC3)ncc2c(N)c1F
CCC(=O)N1CC(C1)OC(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnc2CCCNc2c1C
Cc1c2NCCCc2ncc1-c1cc2cc(NC(=O)OC3CN(C3)S(C)(=O)=O)ncc2c(N)c1F
Cc1c2NCCOc2ncc1-c1cc2cc(NC(=O)OC3CC4(C3)CN(CC(F)F)C4)ncc2c(N)c1F
CC(C)N1C[C@H]2[C@@H](C1)[C@@H]2OC(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnc2OCCNc2c1C |r|
Cc1c2NCCOc2ncc1-c1cc2cc(NC(=O)O[C@@H]3[C@H]4CN(C[C@@H]34)C3COC3)ncc2c(N)c1F |r|
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Cc1c2NCCOc2ncc1-c1cc2cc(NC(=O)OC3C4COCC3CN(CC(F)F)C4)ncc2c(N)c1F |THB:28:27:20:22.24.23,19:20:22.24.23:26.32.27|
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CO[C@@H]1CC[C@@H](C1)NC(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnc2OCCNc2c1C |r|
Cc1c2NCCCc2ncc1-c1cc2cc(NC(=O)N[C@H]3C[C@H](F)C3)ncc2c(N)c1F |r,wU:20.21,wD:22.24,(1.88,-.84,;3.21,-.07,;4.55,-.84,;4.55,-2.38,;5.88,-3.15,;7.21,-2.38,;7.21,-.84,;5.88,-.07,;5.88,1.47,;4.55,2.24,;3.21,1.47,;1.88,2.24,;.54,1.47,;-.79,2.24,;-2.12,1.47,;-3.46,2.24,;-4.79,1.47,;-4.79,-.07,;-3.46,-.84,;-6.12,-.84,;-6.12,-2.38,;-5.03,-3.47,;-6.12,-4.55,;-6.12,-6.09,;-7.21,-3.47,;-3.46,3.78,;-2.12,4.55,;-.79,3.78,;.54,4.55,;.54,6.09,;1.88,3.78,;3.21,4.55,)|
CO[C@H]1C[C@@H](C1)NC(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnc2OCCNc2c1C |r,wU:4.6,wD:2.1,(-4.79,-6.48,;-6.12,-5.71,;-6.12,-4.17,;-5.03,-3.08,;-6.12,-1.99,;-7.21,-3.08,;-6.12,-.45,;-4.79,.32,;-3.46,-.45,;-4.79,1.86,;-3.46,2.63,;-2.12,1.86,;-.79,2.63,;.54,1.86,;1.88,2.63,;1.88,4.17,;3.21,4.94,;.54,4.94,;.54,6.48,;-.79,4.17,;-2.12,4.94,;-3.46,4.17,;3.21,1.86,;4.55,2.63,;5.88,1.86,;5.88,.32,;7.21,-.45,;7.21,-1.99,;5.88,-2.76,;4.55,-1.99,;4.55,-.45,;3.21,.32,;1.88,-.45,)|
Cc1c2NCCOc2ncc1-c1cc2cc(NC(=O)N[C@H]3C[C@H]3F)ncc2c(N)c1F |r|
CC1CC1NC(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnc2OCCNc2c1C
C[C@@H]1C[C@@H]1NC(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnc2OCCNc2c1C |r|
Cc1c2NCCCc2ncc1-c1cc2cc(NC(=O)NC3CC4(C3)CN(CC(F)F)C4)ncc2c(N)c1F
Cc1c2NCCCc2ncc1-c1cc2cc(NC(=O)N[C@H]3C[C@@]4(C3)CCOC4)ncc2c(N)c1F |r,wD:20.21,22.23,(1.96,-.42,;3.29,.35,;4.62,-.42,;4.62,-1.96,;5.96,-2.73,;7.29,-1.96,;7.29,-.42,;5.96,.35,;5.96,1.89,;4.62,2.66,;3.29,1.89,;1.96,2.66,;.62,1.89,;-.71,2.66,;-2.04,1.89,;-3.38,2.66,;-4.71,1.89,;-4.71,.35,;-3.38,-.42,;-6.05,-.42,;-6.05,-1.96,;-7.13,-3.05,;-6.05,-4.14,;-4.96,-3.05,;-7.29,-5.04,;-6.82,-6.51,;-5.28,-6.51,;-4.8,-5.04,;-3.38,4.2,;-2.04,4.97,;-.71,4.2,;.62,4.97,;.62,6.51,;1.96,4.2,;3.29,4.97,)|
Cc1c2NCCCc2ncc1-c1cc2cc(NC(=O)N[C@H]3C[C@@]4(C3)CCOC4)ncc2c(N)c1F |r,wU:20.21,22.24,(1.96,-.42,;3.29,.35,;4.62,-.42,;4.62,-1.96,;5.96,-2.73,;7.29,-1.96,;7.29,-.42,;5.96,.35,;5.96,1.89,;4.62,2.66,;3.29,1.89,;1.96,2.66,;.62,1.89,;-.71,2.66,;-2.04,1.89,;-3.38,2.66,;-4.71,1.89,;-4.71,.35,;-3.38,-.42,;-6.05,-.42,;-6.05,-1.96,;-4.96,-3.05,;-6.05,-4.14,;-7.13,-3.05,;-7.29,-5.04,;-6.82,-6.51,;-5.28,-6.51,;-4.8,-5.04,;-3.38,4.2,;-2.04,4.97,;-.71,4.2,;.62,4.97,;.62,6.51,;1.96,4.2,;3.29,4.97,)|
CN(C)C(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnc2OCCNc2c1C
Cc1c2NCCOc2ncc1-c1cc2cc(NC(=O)N3CCCC3)ncc2c(N)c1F
CC(C)NC(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnc2OCCNc2c1C
Cc1c2NCCOc2ncc1-c1cc2cc(NC(=O)N[C@H]3CCOC[C@H]3F)ncc2c(N)c1F |r|
Cc1c2NCCOc2ncc1-c1cc2cc(NC(=O)N[C@@H]3C[C@H](F)C3)ncc2c(N)c1F |r,wU:20.21,22.24,(1.88,-.84,;3.21,-.07,;4.55,-.84,;4.55,-2.38,;5.88,-3.15,;7.21,-2.38,;7.21,-.84,;5.88,-.07,;5.88,1.47,;4.55,2.24,;3.21,1.47,;1.88,2.24,;.54,1.47,;-.79,2.24,;-2.12,1.47,;-3.46,2.24,;-4.79,1.47,;-4.79,-.07,;-3.46,-.84,;-6.12,-.84,;-6.12,-2.38,;-7.21,-3.47,;-6.12,-4.55,;-6.12,-6.09,;-5.03,-3.47,;-3.46,3.78,;-2.12,4.55,;-.79,3.78,;.54,4.55,;.54,6.09,;1.88,3.78,;3.21,4.55,)|
Cc1c2NCCOc2ncc1-c1cc2cc(NC(=O)N[C@H]3C[C@H](F)C3)ncc2c(N)c1F |r,wU:20.21,wD:22.24,(1.88,-.84,;3.21,-.07,;4.55,-.84,;4.55,-2.38,;5.88,-3.15,;7.21,-2.38,;7.21,-.84,;5.88,-.07,;5.88,1.47,;4.55,2.24,;3.21,1.47,;1.88,2.24,;.54,1.47,;-.79,2.24,;-2.12,1.47,;-3.46,2.24,;-4.79,1.47,;-4.79,-.07,;-3.46,-.84,;-6.12,-.84,;-6.12,-2.38,;-5.03,-3.47,;-6.12,-4.55,;-6.12,-6.09,;-7.21,-3.47,;-3.46,3.78,;-2.12,4.55,;-.79,3.78,;.54,4.55,;.54,6.09,;1.88,3.78,;3.21,4.55,)|
Cc1c(N)cncc1-c1cc2cc(NC(=O)NC3CCCC3)ncc2c(N)c1F
CO[C@H]1COCC[C@H]1NC(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnc2OCCNc2c1C |r|
CO[C@@H]1COCC[C@@H]1NC(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnc2OCCNc2c1C |r|
CC1CN(C1)C(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnc2OCCNc2c1C
CN(C1CCC1)C(=O)Nc1cc2cc(c(F)c(N)c2cn1)-c1cnc2OCCNc2c1C
Cc1c2NCCOc2ncc1-c1cc2cc(NC(=O)N3CC4(C3)CCOCC4)ncc2c(N)c1F
Cc1c2NCCOc2ncc1-c1cc2cc(NC(=O)N3CC(C)(O)C3)ncc2c(N)c1F
Cc1c2NCCOc2ncc1-c1cc2cc(NC(=O)N3CC(C)(F)C3)ncc2c(N)c1F
Cc1c2NCCOc2ncc1-c1cc2cc(NC(=O)N3CCC3)ncc2c(N)c1F
CC(=O)Nc1nc2ccc(cc2s1)-c1c(C)ccc2[nH]ncc12
Cc1ccc2[nH]ncc2c1-c1ccc2nc(NC(=O)C3C[C@@H]3F)sc2c1 |r|
Cc1ccc2[nH]ncc2c1-c1ccc2nc(NC(=O)OC(C)(C)C)sc2c1
Cc1ccc2[nH]ncc2c1-c1ccc2nc(NC(=O)C3CCC3)sc2c1
Cc1ccc2[nH]ncc2c1-c1ccc2nc(NC(=O)C3CC3(F)F)sc2c1
Cc1ccc2[nH]ncc2c1-c1ccc2nc(NC(=O)C3C[C@H](F)C3)sc2c1 |r,wU:21.23,(5.21,-.81,;5.98,.52,;7.52,.52,;8.29,1.86,;7.52,3.19,;8,4.66,;6.75,5.56,;5.51,4.66,;5.98,3.19,;5.21,1.86,;3.67,1.86,;2.9,3.19,;1.36,3.19,;.59,1.86,;-.91,1.54,;-1.07,.01,;-2.41,-.76,;-3.74,.01,;-3.74,1.55,;-5.07,-.76,;-6.56,-.37,;-6.96,-1.85,;-8.29,-2.62,;-5.47,-2.25,;.33,-.62,;1.36,.52,;2.9,.52,)|
Cc1ccc2[nH]ncc2c1-c1ccc2nc(NC(=O)C3C[C@H](F)C3)sc2c1 |r,wD:21.23,(5.21,-.81,;5.98,.52,;7.52,.52,;8.29,1.86,;7.52,3.19,;8,4.66,;6.75,5.56,;5.51,4.66,;5.98,3.19,;5.21,1.86,;3.67,1.86,;2.9,3.19,;1.36,3.19,;.59,1.86,;-.91,1.54,;-1.07,.01,;-2.41,-.76,;-3.74,.01,;-3.74,1.55,;-5.07,-.76,;-5.47,-2.25,;-6.96,-1.85,;-8.29,-2.62,;-6.56,-.37,;.33,-.62,;1.36,.52,;2.9,.52,)|
Cc1ccc2[nH]ncc2c1-c1ccc2nc(NC(=O)c3ccccc3)sc2c1
CCCCC(=O)Nc1nc2ccc(cc2s1)-c1c(C)ccc2[nH]ncc12
Cc1ccc2[nH]ncc2c1-c1ccc2nc(NC(=O)C3CCCC3)sc2c1
Cc1ccc2[nH]ncc2c1-c1ccc2nc(NC(=O)C3CC(F)(F)C3)sc2c1
Cc1ccc2[nH]ncc2c1-c1ccc2nc(NC(=O)c3ccccn3)sc2c1
O=C(Nc1nc2ccc(cc2s1)-c1c(ccc2[nH]ncc12)-c1cccs1)C1CC1
O=C(Nc1nc2ccc(cc2s1)-c1cccc2[nH]ncc12)C1CC1
Fc1ccc2[nH]ncc2c1-c1ccc2nc(NC(=O)C3CC3)sc2c1
Clc1ccc2[nH]ncc2c1-c1ccc2nc(NC(=O)C3CC3)sc2c1
FC(F)(F)c1ccc2[nH]ncc2c1-c1ccc2nc(NC(=O)C3CC3)sc2c1
O=C(Nc1nc2ccc(cc2s1)-c1c(ccc2[nH]ncc12)-c1ccsc1)C1CC1
Clc1ccc(-c2ccc3nc(NC(=O)C4CC4)sc3c2)c2cn[nH]c12
Clc1cc(-c2ccc3nc(NC(=O)C4CC4)sc3c2)c2cn[nH]c2c1
CC(C)(C)OC(=O)c1ccc2[nH]ncc2c1-c1ccc2nc(NC(=O)C3CC3)sc2c1
O=C(Nc1nc2ccc(cc2s1)-c1cc(cc2[nH]ncc12)-c1cccs1)C1CC1
O=C(Nc1nc2ccc(cc2s1)-c1c(ccc2[nH]ncc12)C(=O)NCc1ccsc1)C1CC1
COc1ccc2[nH]ncc2c1-c1ccc2nc(NC(=O)C3CC3)sc2c1
OCc1ccc2[nH]ncc2c1-c1ccc2nc(NC(=O)C3CC3)sc2c1
Cc1ccc2[nH]nc(N)c2c1-c1ccc2nc(NC(=O)C3CC3)sc2c1
Oc1ccc2[nH]ncc2c1-c1ccc2nc(NC(=O)C3CC3)sc2c1
CCc1ccc2[nH]ncc2c1-c1ccc2nc(NC(=O)C3CC3)sc2c1
O=C(Nc1nc2ccc(cc2s1)-c1c(ccc2[nH]ncc12)C#N)C1CC1
F[C@H]1CC1C(=O)Nc1nc2ccc(cc2s1)-c1c(Cl)ccc2[nH]ncc12 |r|
CN(C)CCOc1ccc2[nH]ncc2c1-c1ccc2nc(NC(=O)C3C[C@@H]3F)sc2c1 |r|
Cc1ccc2[nH]ncc2c1-c1ccc2nc(NC(=S)C3CC3)sc2c1
FC(F)c1ccc2[nH]ncc2c1-c1ccc2nc(NC(=O)C3C[C@@H]3F)sc2c1 |r|
COCCOc1ccc2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)sc2c1 |r|
F[C@H]1CC1C(=O)Nc1nc2ccc(cc2s1)-c1c(C=C)ccc2[nH]ncc12 |r|
FCc1ccc2[nH]ncc2c1-c1ccc2nc(NC(=O)C3C[C@@H]3F)sc2c1 |r|
F[C@H]1C[C@H]1C(=O)Nc1nc2ccc(cc2s1)-c1c(ccc2[nH]ncc12)C1CC1 |r|
F[C@H]1CC1C(=O)Nc1nc2ccc(cc2s1)-c1c(Cn2cccn2)ccc2[nH]ncc12 |r|
F[C@H]1CC1C(=O)Nc1nc2ccc(cc2s1)-c1c(ccc2[nH]ncc12)C#C |r|
Cc1c(F)cc2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)sc2c1 |r|
F[C@H]1C[C@H]1C(=O)Nc1nc2ccc(cc2s1)-c1c(Cl)c(F)cc2[nH]ncc12 |r|
F[C@H]1C[C@H]1C(=O)Nc1nc2ccc(cc2s1)-c1c(Br)c(F)cc2[nH]ncc12 |r|
F[C@H]1C[C@H]1C(=O)Nc1nc2ccc(cc2s1)-c1c(C=C)c(F)cc2[nH]ncc12 |r|
Cc1c(F)cc2[nH]nc(Cl)c2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)sc2c1 |r|
Cc1c(F)cc2[nH]nc(I)c2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)sc2c1 |r|
CCc1c(F)cc2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)sc2c1 |r|
F[C@H]1CC1C(=O)Nc1nc2ccc(cc2s1)-c1c(C#C)c(F)cc2[nH]ncc12 |r|
F[C@H]1CC1C(=O)Nc1nc2ccc(cc2s1)-c1c(I)c(F)cc2[nH]ncc12 |r|
Cc1c(F)cc2[nH]nc(Br)c2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)sc2c1 |r|
F[C@H]1CC1C(=O)Nc1nc2ccc(cc2s1)-c1c(c(F)cc2[nH]ncc12)C(F)(F)F |r|
Cc1c(F)c(Cl)c2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)sc2c1 |r|
Cc1c(F)cc2[nH]nc(C=C)c2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)sc2c1 |r|
Cc1c(F)c(Cl)c2[nH]nc(Cl)c2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)sc2c1 |r|
Cc1c(F)c(Cl)c2[nH]nc(Cl)c2c1-c1cc(Cl)c2nc(NC(=O)[C@@H]3C[C@@H]3F)sc2c1 |r|
Cc1c(F)c(F)c2[nH]nc(F)c2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)sc2c1 |r|
Cc1c(F)c(F)c2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)sc2c1 |r|
Cc1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3c2)c2cn[nH]c12 |r|
CSc1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3c2)c2cn[nH]c12 |r|
Cc1c(F)c(C)c2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)sc2c1 |r|
CP(C)(=O)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3c2)c2cn[nH]c12 |r|
F[C@H]1C[C@H]1C(=O)Nc1nc2ccc(cc2s1)-c1c(Cl)c(F)c(C=C)c2[nH]ncc12 |r|
Cc1c(F)c(C=C)c2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)sc2c1 |r|
CS(=O)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3c2)c2cn[nH]c12 |r|
CSc1c(F)c(C)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3c2)c2cn[nH]c12 |r|
Cc1c(F)cc2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)sc2c1CCc1ccncc1 |r,wD:20.21,22.25,(4.42,-.02,;5.45,1.12,;6.96,.8,;7.43,-.66,;7.99,1.95,;7.51,3.41,;8.28,4.75,;7.25,5.89,;5.85,5.26,;6.01,3.73,;4.98,2.59,;3.47,2.91,;2.99,4.37,;1.49,4.69,;.46,3.55,;-1.08,3.55,;-1.56,2.08,;-3.02,1.61,;-4.17,2.64,;-3.85,4.14,;-5.63,2.16,;-6.66,1.02,;-7.14,2.48,;-8.28,3.51,;-.31,1.18,;.93,2.08,;2.44,1.76,;2.92,.3,;1.88,-.85,;2.36,-2.31,;1.33,-3.46,;1.81,-4.92,;3.31,-5.24,;4.34,-4.1,;3.87,-2.63,)|
Cc1c(F)c(S(C)=O)c2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)sc2c1 |r|
Cc1c(F)c(I)c2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)sc2c1 |r|
Nc1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3c2)c2cn[nH]c12 |r|
CN(C)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3c2)c2cn[nH]c12 |r|
NCCSc1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3c2)c2cn[nH]c12 |r|
COCCSc1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3c2)c2cn[nH]c12 |r|
F[C@H]1C[C@H]1C(=O)Nc1nc2ccc(cc2s1)-c1c(Cl)c(F)c(NC(=O)C=C)c2[nH]ncc12 |r|
CC(=O)NCCSc1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3c2)c2cn[nH]c12 |r|
F[C@H]1C[C@H]1C(=O)Nc1nc2ccc(cc2s1)-c1c(Cl)c(F)c(N2CCOCC2)c2[nH]ncc12 |r|
CN1CCN(CC1)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3c2)c2cn[nH]c12 |r|
F[C@H]1C[C@H]1C(=O)Nc1nc2ccc(cc2s1)-c1c(Cl)c(F)c(N2CCNCC2)c2[nH]ncc12 |r|
F[C@H]1C[C@H]1C(=O)Nc1nc2ccc(cc2s1)-c1c(Cl)c(F)c(N2CCCC2)c2[nH]ncc12 |r|
OC1CCN(C1)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3c2)c2cn[nH]c12 |r|
OCCSc1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3c2)c2cn[nH]c12 |r|
COc1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3c2)c2cn[nH]c12 |r|
CCOc1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3c2)c2cn[nH]c12 |r|
CN(CCN)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3c2)c2cn[nH]c12 |r|
NC1CCN(CC1)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3c2)c2cn[nH]c12 |r|
NC1CCCN(C1)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3c2)c2cn[nH]c12 |r|
CN(C)CCN(C)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3c2)c2cn[nH]c12 |r|
OCCCSc1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3c2)c2cn[nH]c12 |r|
CNC(=O)CSc1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3c2)c2cn[nH]c12 |r|
OC(=O)NC1CN(C1)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3c2)c2cn[nH]c12 |r|
CN(C1CN(C1)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3c2)c2cn[nH]c12)C(O)=O |r|
OC(=O)NCC1CN(C1)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3c2)c2cn[nH]c12 |r|
NCC1CCN(C1)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3c2)c2cn[nH]c12 |r|
CNCCN(C)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3c2)c2cn[nH]c12 |r|
CN(CCO)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3c2)c2cn[nH]c12 |r|
CN(CC1CNC1)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3c2)c2cn[nH]c12 |r|
F[C@H]1C[C@H]1C(=O)Nc1nc2ccc(cc2s1)-c1c(Cl)c(F)c(NCC2CNC2)c2[nH]ncc12 |r|
COc1cc(C)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3c2)c2cn[nH]c12 |r|
COc1c(F)c(C)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3c2)c2cn[nH]c12 |r|
CCOc1c(F)c(C)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3c2)c2cn[nH]c12 |r|
CN(C)C(=O)CSc1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3c2)c2cn[nH]c12 |r|
CN(C)C(=O)CN(C)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3c2)c2cn[nH]c12 |r|
CCOc1cc(C)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3c2)c2cn[nH]c12 |r|
CCc1c(F)c(N(C)C)c2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)sc2c1 |r|
CCc1c(F)c(SC)c2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)sc2c1 |r|
CN(C)c1c(F)c(C)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3c2)c2cn[nH]c12 |r|
CSc1c(F)cc2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)sc2c1 |r|
CCc1c(F)c(F)c2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)sc2c1 |r|
CCOc1c(F)c(CC)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3c2)c2cn[nH]c12 |r|
CC(=O)Nc1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3c2)c2cn[nH]c12 |r|
CSc1c(F)c(N(C)C)c2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)sc2c1 |r|
CSc1c(F)c(SC)c2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)sc2c1 |r|
Cc1c(F)c(c2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)sc2c1)S(C)(=O)=O |r|
CC(=O)Nc1c(F)c(C)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3c2)c2cn[nH]c12 |r|
CN(Nc1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3c2)c2cn[nH]c12)C(=O)OC(C)(C)C |r|
CNNc1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3c2)c2cn[nH]c12 |r|
COC(=O)c1c(F)c(C)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3c2)c2cn[nH]c12 |r|
CSc1c(F)c(F)c2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)sc2c1 |r|
CCOc1c(F)c(SC)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3c2)c2cn[nH]c12 |r|
CS(=O)(=O)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3c2)c2cn[nH]c12 |r|
CN(C(C)=O)c1c(F)c(C)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3c2)c2cn[nH]c12 |r|
OC(=O)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3c2)c2cn[nH]c12 |r|
COC(=O)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3c2)c2cn[nH]c12 |r|
CN(C(C)=O)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3c2)c2cn[nH]c12 |r|
Cc1c(F)c(C(O)=O)c2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)sc2c1 |r|
CN(C)C(=O)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3c2)c2cn[nH]c12 |r|
F[C@H]1C[C@H]1C(=O)Nc1nc2ccc(cc2s1)-c1c(Cl)c(F)c(F)c2[nH]ncc12 |r|
CNC(=O)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3c2)c2cn[nH]c12 |r|
CC(=O)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3c2)c2cn[nH]c12 |r|
CN(C1CNC1)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3c2)c2cn[nH]c12 |r|
CN(C)c1c(F)c(c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3c2)c2cn[nH]c12)C(F)(F)F |r|
CC(=O)c1c(F)c(C)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3c2)c2cn[nH]c12 |r|
CNC(=O)c1c(F)c(C)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3c2)c2cn[nH]c12 |r|
CCN(C)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3c2)c2cn[nH]c12 |r|
CN(C)C(=O)c1c(F)c(C)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3c2)c2cn[nH]c12 |r|
NC(=O)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3c2)c2cn[nH]c12 |r|
CCN(C)c1c(F)c(CC)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3c2)c2cn[nH]c12 |r|
CCN(C)c1c(F)c(C)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3c2)c2cn[nH]c12 |r|
CCN(C)c1c(F)c(SC)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3c2)c2cn[nH]c12 |r|
CN(C)c1c(F)cc(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3c2)c2cn[nH]c12 |r|
F[C@H]1C[C@H]1C(=O)Nc1nc2ccc(cc2s1)-c1cc(F)c(OC(F)(F)F)c2[nH]ncc12 |r|
CSc1c(F)cc(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3c2)c2cn[nH]c12 |r|
CSc1ccc(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3c2)c2cn[nH]c12 |r|
F[C@H]1C[C@H]1C(=O)Nc1nc2ccc(cc2s1)-c1c(Cl)c(F)c(C#N)c2[nH]ncc12 |r|
CN(C)C(=O)c1c(F)cc(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3c2)c2cn[nH]c12 |r|
CN(C)C(=O)c1c(F)cc2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)sc2c1 |r|
Cc1ccc2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)sc2n1 |r|
Cc1c(F)cc2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)sc2n1 |r|
CSc1n[nH]c2cc(F)c(C)c(-c3ccc4nc(NC(=O)[C@@H]5C[C@@H]5F)sc4n3)c12 |r|
CCOc1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3n2)c2cn[nH]c12 |r|
CC(C)c1c(F)cc2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)sc2n1 |r|
Nc1c(F)cc2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)sc2n1 |r|
CCc1c(F)cc2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)sc2n1 |r|
F[C@H]1C[C@H]1C(=O)Nc1nc2ccc(nc2s1)-c1c(Cl)c(F)cc2[nH]ncc12 |r|
CCN(CC)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3n2)c2cn[nH]c12 |r|
COc1c(F)cc2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)sc2n1 |r|
CSc1c(F)cc2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)sc2n1 |r|
F[C@H]1C[C@H]1C(=O)Nc1nc2ccc(nc2s1)-c1c(C#N)c(F)cc2[nH]ncc12 |r|
F[C@H]1C[C@H]1C(=O)Nc1nc2ccc(nc2s1)-c1c(C2CC2)c(F)cc2[nH]ncc12 |r|
CCNc1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3n2)c2cn[nH]c12 |r|
F[C@H]1C[C@H]1C(=O)Nc1nc2ccc(nc2s1)-c1c(Br)c(F)cc2[nH]ncc12 |r|
CCc1c(F)c(N(C)C)c2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)sc2n1 |r|
CCc1c(F)c(SC)c2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)sc2n1 |r|
Cc1c(F)c(SCCO)c2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)sc2n1 |r|
CS(=O)c1c(F)cc2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)sc2n1 |r|
CCOC(=O)CSc1c(F)c(CC)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3n2)c2cn[nH]c12 |r|
CCc1c(F)c(SCC(=O)N(C)C)c2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)sc2n1 |r|
CCc1c(F)c(SCC(=O)NC)c2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)sc2n1 |r|
CCc1c(F)c(SCC(O)=O)c2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)sc2n1 |r|
CN(C)c1c(F)c(C)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3n2)c2cn[nH]c12 |r|
CSc1c(F)c(SC)c2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)sc2n1 |r|
F[C@H]1C[C@H]1C(=O)Nc1nc2ccc(nc2s1)-c1c(F)c(cc2[nH]ncc12)C(F)(F)F |r|
CN(C)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3n2)c2cn[nH]c12 |r|
CSc1c(F)c(C)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3n2)c2cn[nH]c12 |r|
CSc1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3n2)c2cn[nH]c12 |r|
CCOc1c(F)c(C)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3n2)c2cn[nH]c12 |r|
CCc1c(F)c(F)c2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)sc2n1 |r|
Cc1c(F)c(S(C)=O)c2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)sc2n1 |r|
CCOc1c(F)c(CC)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3n2)c2cn[nH]c12 |r|
CC(=O)Nc1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3n2)c2cn[nH]c12 |r|
CS(=O)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3n2)c2cn[nH]c12 |r|
CC(=O)Nc1c(F)c(C)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3n2)c2cn[nH]c12 |r|
Cc1c(F)c(c2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)sc2n1)S(C)(=O)=O |r|
COC(=O)c1c(F)c(C)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3n2)c2cn[nH]c12 |r|
CCOc1c(F)c(SC)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3n2)c2cn[nH]c12 |r|
CS(=O)(=O)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3n2)c2cn[nH]c12 |r|
Cc1c(F)c(F)c2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)sc2n1 |r|
CSc1c(F)c(F)c2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)sc2n1 |r|
Cc1c(F)c(C(O)=O)c2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)sc2n1 |r|
CN(C(C)=O)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3n2)c2cn[nH]c12 |r|
CN(C(C)=O)c1c(F)c(C)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3n2)c2cn[nH]c12 |r|
CNNc1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3n2)c2cn[nH]c12 |r|
CN(Nc1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3n2)c2cn[nH]c12)C(=O)OC(C)(C)C |r|
CN(C)C(=O)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3n2)c2cn[nH]c12 |r|
CSc1c(F)c(N(C)C)c2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)sc2n1 |r|
CNC(=O)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3n2)c2cn[nH]c12 |r|
CCN(C)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3n2)c2cn[nH]c12 |r|
CN(C)C(=O)c1c(F)c(C)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3n2)c2cn[nH]c12 |r|
F[C@H]1C[C@H]1C(=O)Nc1nc2ccc(nc2s1)-c1c(c(F)c(Cl)c2[nH]ncc12)C(F)(F)F |r|
Cc1c(F)c(C)c2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)sc2n1 |r|
CCN(C)c1c(F)c(CC)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3n2)c2cn[nH]c12 |r|
CCOc1c(F)cc2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)sc2n1 |r|
CNC(=O)OCCN(C)c1c(F)c(C)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3n2)c2cn[nH]c12 |r|
CCN(C)c1c(F)c(C)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3n2)c2cn[nH]c12 |r|
CN(CCO)c1c(F)c(C)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3n2)c2cn[nH]c12 |r|
Cc1c(F)c(c2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)sc2n1)C(F)(F)F |r|
CNC(=O)c1c(F)c(C)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3n2)c2cn[nH]c12 |r|
CN(C)c1c(F)c(c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3n2)c2cn[nH]c12)C(F)(F)F |r|
F[C@H]1C[C@H]1C(=O)Nc1nc2ccc(nc2s1)-c1c(Cl)c(F)c(F)c2[nH]ncc12 |r|
FC(F)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3n2)c2cn[nH]c12 |r|
CCc1c(F)c(c2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)sc2n1)C(F)(F)F |r|
Cc1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3n2)c2cn[nH]c12 |r|
CSc1ccc(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3n2)c2cn[nH]c12 |r|
Cc1c(F)c(OC(F)(F)F)c2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)sc2n1 |r|
CN(C)c1c(F)cc(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3n2)c2cn[nH]c12 |r|
F[C@H]1C[C@H]1C(=O)Nc1nc2ccc(nc2s1)-c1cc(F)c(OC(F)(F)F)c2[nH]ncc12 |r|
CN(C)c1ccc(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3n2)c2cn[nH]c12 |r|
Cc1c(F)c(C(F)F)c2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)sc2n1 |r|
CCN(C)c1c(F)c(SC)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)sc3n2)c2cn[nH]c12 |r|
CSc1c(F)cc2[nH]ncc2c1-c1cc2sc(NC(=O)[C@@H]3C[C@@H]3F)nc2cn1 |r|
CS(=O)c1c(F)cc2[nH]ncc2c1-c1cc2sc(NC(=O)[C@@H]3C[C@@H]3F)nc2cn1 |r|
Cc1ccc2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)cn2c1 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ccc2n1)-c1cccc2[nH]ncc12 |r|
Clc1ccc2[nH]ncc2c1-c1ccc2nc(NC(=O)C3CC3)cn2c1
COc1ccc2[nH]ncc2c1-c1ccc2nc(NC(=O)C3CC3)cn2c1
Nc1ccc2[nH]ncc2c1-c1ccc2nc(NC(=O)C3CC3)cn2c1
FC(F)(F)c1ccc2[nH]ncc2c1-c1ccc2nc(NC(=O)C3CC3)cn2c1
Nc1c(F)cc2[nH]ncc2c1-c1ccc2nc(NC(=O)C3CC3)cn2c1
Brc1ccc2[nH]ncc2c1-c1ccc2nc(NC(=O)C3CC3)cn2c1
CNc1ccc2[nH]ncc2c1-c1ccc2nc(NC(=O)C3CC3)cn2c1
CN(C)c1ccc2[nH]ncc2c1-c1ccc2nc(NC(=O)C3CC3)cn2c1
Fc1cc2[nH]ncc2c(-c2ccc3nc(NC(=O)C4CC4)cn3c2)c1Br
O=C(Nc1cn2cc(ccc2n1)-c1c(ccc2[nH]ncc12)C#N)C1CC1
OCc1ccc2[nH]ncc2c1-c1ccc2nc(NC(=O)C3CC3)cn2c1
CCc1ccc2[nH]ncc2c1-c1ccc2nc(NC(=O)C3CC3)cn2c1
Fc1cc2[nH]ncc2c(-c2ccc3nc(NC(=O)C4CC4)cn3c2)c1C=C
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ccc2n1)-c1c(ccc2[nH]ncc12)C(F)(F)F |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ccc2n1)-c1c(Cl)ccc2[nH]ncc12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ccc2n1)-c1c(Br)ccc2[nH]ncc12 |r|
CC(=O)c1ccc2[nH]ncc2c1-c1ccc2nc(NC(=O)C3CC3)cn2c1
Nc1c(Cl)cc2[nH]ncc2c1-c1ccc2nc(NC(=O)C3CC3)cn2c1
Fc1cc2[nH]ncc2c(-c2ccc3nc(NC(=O)C4CC4)cn3c2)c1C1CC1
Fc1cc2[nH]ncc2c(-c2ccc3nc(NC(=O)C4CC4)cn3c2)c1Cl
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ccc2n1)-c1c(Cl)c(F)cc2[nH]ncc12 |r|
O=C(Nc1cn2cc(ccc2n1)-c1c(ccc2[nH]ncc12)C1CC1)C1CC1
Cc1c(F)cc2[nH]ncc2c1-c1ccc2nc(NC(=O)C3CC3)cn2c1
CC(C)c1c(F)cc2[nH]ncc2c1-c1ccc2nc(NC(=O)C3CC3)cn2c1
CSc1ccc2[nH]ncc2c1-c1ccc2nc(NC(=O)C3CC3)cn2c1
CCc1c(F)cc2[nH]ncc2c1-c1ccc2nc(NC(=O)C3CC3)cn2c1
FC(F)c1ccc2[nH]ncc2c1-c1ccc2nc(NC(=O)C3CC3)cn2c1
Cc1c(F)cc2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)cn2c1 |r|
OCc1c(F)cc2[nH]ncc2c1-c1ccc2nc(NC(=O)C3CC3)cn2c1
COc1c(F)cc2[nH]ncc2c1-c1ccc2nc(NC(=O)C3CC3)cn2c1
FC(F)c1c(F)cc2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)cn2c1 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ccc2n1)-c1c(Br)c(F)cc2[nH]ncc12 |r|
FC(F)c1c(F)cc2[nH]ncc2c1-c1ccc2nc(NC(=O)C3CC3)cn2c1
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ccc2n1)-c1c(Cl)c(F)c(Cl)c2[nH]ncc12 |r|
Cc1c(F)c(C)c2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)cn2c1 |r|
CN(C)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
CP(C)(=O)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
Cc1c(F)c(Cl)c2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)cn2c1 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ccc2n1)-c1c(Cl)c(F)c(Br)c2[nH]ncc12 |r|
Cc1c(F)c(F)c2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)cn2c1 |r|
Cc1c(F)c(c2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)cn2c1)C(F)(F)F |r|
Cc1cc(C=C)c2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)cn2c1 |r|
CNc1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
CSc1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
CS(=O)(=O)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
Cc1c(F)c(Br)c2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)cn2c1 |r|
CSc1c(F)c(C)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
Cc1c(F)c(c2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)cn2c1)S(C)(=O)=O |r|
COc1c(F)c(C)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
COc1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
CN(C)c1c(F)c(C)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
Cc1cc(NC(=O)C=C)c2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)cn2c1 |r|
CCOc1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ccc2n1)-c1c(Cl)cc(NC(=O)C=C)c2[nH]ncc12 |r|
CN1CCN(CC1)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
Cc1ccc2[nH]ncc2c1-c1ccc2nc(NC(=O)C3CC3CO)cn2c1 |w:17.20|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ccc2n1)-c1c(Cl)c(F)c(N2CCOCC2)c2[nH]ncc12 |r|
CCNc1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
CCN(CC)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ccc2n1)-c1c(Cl)c(F)c(N2CCCC2)c2[nH]ncc12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ccc2n1)-c1c(Cl)c(F)c(N2CCC2)c2[nH]ncc12 |r|
Nc1cc2[nH]ncc2c(c1Cl)-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)cn2c1 |r|
COc1cc(C)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ccc2n1)-c1c(Cl)c(NC(=O)C=C)cc2[nH]ncc12 |r|
CCOc1cc(C)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
CCOc1c(F)c(C)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
Cc1c(NC(=O)C=C)cc2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)cn2c1 |r|
OCCSc1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
CCc1c(F)c(N(C)C)c2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)cn2c1 |r|
Cc1c(F)c(SCCO)c2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)cn2c1 |r|
CCc1c(F)c(SC)c2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)cn2c1 |r|
CCc1c(F)cc2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)cn2c1 |r|
Oc1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
CSc1c(F)cc2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)cn2c1 |r|
CSc1c(F)c(SC)c2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)cn2c1 |r|
CCc1c(F)c(F)c2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)cn2c1 |r|
Cc1c(F)c(S(C)=O)c2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)cn2c1 |r|
CSc1c(F)c(N(C)C)c2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)cn2c1 |r|
CC(=O)Nc1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
CS(=O)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
CSc1c(F)c(F)c2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)cn2c1 |r|
COC(=O)c1c(F)c(C)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
CCN(C)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
CN(C)c1c(F)c(c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12)C(F)(F)F |r|
CC(=O)Nc1c(F)c(C)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
CN(Nc1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12)C(=O)OC(C)(C)C |r|
CCOc1c(F)c(SC)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
CN(C(C)=O)c1c(F)c(C)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
CNC(=O)OCCSc1c(F)c(C)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
Cc1c(F)c(C(O)=O)c2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)cn2c1 |r|
OC(=O)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
COC(=O)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
CN(C(C)=O)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
CNNc1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
CCOc1c(F)c(CC)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
CC(=O)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
CN(C)C(=O)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
CNC(=O)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
CC(=O)c1c(F)c(C)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ccc2n1)-c1c(Cl)c(F)c(F)c2[nH]ncc12 |r|
CCN(C)c1c(F)c(SC)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
NC(=O)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
CCN(C)c1c(F)c(CC)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
CN(C)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)C4CC4)cn3c2)c2cn[nH]c12
CCOc1c(F)cc2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)cn2c1 |r|
CN(C)C(=O)c1c(F)c(C)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
CCN(C)c1c(F)c(C)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
FC(F)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
CN(C)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
CN(C)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@H]4F)cn3c2)c2cn[nH]c12 |r|
CN(C)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@H]4C[C@H]4F)cn3c2)c2cn[nH]c12 |r|
CN(C)c1c(F)cc(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ccc2n1)-c1c(Cl)c(F)c(N2CCCC2=O)c2[nH]ncc12 |r|
CN(c1ccccn1)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
CNC(=O)c1c(F)c(C)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
CCc1c(F)c(c2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)cn2c1)C(F)(F)F |r|
CSc1ccc(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
CCN(C)C(=O)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
CSc1c(F)cc(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
Cc1c(F)c(C(F)F)c2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)cn2c1 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ccc2n1)-c1cc(F)c(OC(F)(F)F)c2[nH]ncc12 |r|
Cc1c(F)c(OC(F)(F)F)c2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)cn2c1 |r|
CN(c1ncccn1)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
CN(CC(F)(F)F)C(=O)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
CN(c1ccncn1)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
CN(Cc1cccnc1)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
Cn1nnnc1-c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r,wD:21.21,23.25,(8.14,-2.58,;8.61,-1.12,;10.08,-.64,;10.08,.9,;8.61,1.37,;7.71,.13,;6.17,.13,;5.4,-1.21,;6.17,-2.54,;3.86,-1.21,;3.09,-2.54,;3.09,.13,;1.55,.13,;.78,1.46,;-.76,1.46,;-1.53,.13,;-3.04,-.19,;-3.2,-1.73,;-4.53,-2.5,;-5.87,-1.73,;-5.87,-.19,;-7.2,-2.5,;-7.97,-3.83,;-8.74,-2.5,;-10.08,-1.73,;-1.79,-2.35,;-.76,-1.21,;.78,-1.21,;3.86,1.46,;3.38,2.92,;4.63,3.83,;5.87,2.92,;5.4,1.46,)|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ccc2n1)-c1c(Cl)c(F)c(C#N)c2[nH]ncc12 |r|
CN(C)c1ccc(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
CN(Cc1ccncc1)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
CN(C)C(=O)c1c(F)cc(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
CN(C)C(=O)c1c(F)cc2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)cn2c1 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ccc2n1)-c1c(Cl)c(F)c(OC(F)(F)F)c2[nH]ncc12 |r|
CCOc1c(F)c(F)c2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)cn2c1 |r|
CN1CCN(C1=O)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
CC(C)Nc1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
CC(C)N(C)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
CN(C1CC1)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
OCc1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
FCc1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
Cc1noc(n1)-c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ccc2n1)-c1c(Cl)c(F)c(-n2cccc2)c2[nH]ncc12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ccc2n1)-c1c(Cl)c(F)c(NCC#N)c2[nH]ncc12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ccc2n1)-c1c(Cl)c(F)c(NC2CC2)c2[nH]ncc12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ccc2n1)-c1c(Cl)c(F)c(N(C2CC2)C(=O)C(F)(F)F)c2[nH]ncc12 |r|
OCCC(=O)Nc1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
CCC(C)Nc1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
CC(Nc1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12)C#N |r|
CC(O)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
COC(C)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
CC(F)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ccc2n1)-c1c(Cl)c(F)c(-c2cc[nH]c2)c2[nH]ncc12 |r|
Cn1ccc(c1)-c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
Cn1cccc1-c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r,wD:21.21,23.25,(8.67,-.59,;8.35,-2.09,;9.38,-3.24,;8.61,-4.57,;7.11,-4.25,;6.94,-2.72,;5.61,-1.95,;4.28,-2.72,;4.28,-4.26,;2.94,-1.95,;1.61,-2.72,;2.94,-.41,;1.61,.36,;1.61,1.9,;.28,2.67,;-1.06,1.9,;-2.52,2.38,;-3.43,1.13,;-4.97,1.13,;-5.74,2.47,;-4.97,3.8,;-7.28,2.47,;-8.61,1.7,;-8.61,3.24,;-9.38,4.57,;-2.52,-.11,;-1.06,.36,;.28,-.41,;4.28,.36,;4.6,1.87,;6.13,2.03,;6.75,.62,;5.61,-.41,)|
Cn1nccc1-c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r,wD:21.21,23.25,(8.67,-.59,;8.35,-2.09,;9.38,-3.24,;8.61,-4.57,;7.11,-4.25,;6.94,-2.72,;5.61,-1.95,;4.28,-2.72,;4.28,-4.26,;2.94,-1.95,;1.61,-2.72,;2.94,-.41,;1.61,.36,;1.61,1.9,;.28,2.67,;-1.06,1.9,;-2.52,2.38,;-3.43,1.13,;-4.97,1.13,;-5.74,2.47,;-4.97,3.8,;-7.28,2.47,;-8.61,1.7,;-8.61,3.24,;-9.38,4.57,;-2.52,-.11,;-1.06,.36,;.28,-.41,;4.28,.36,;4.6,1.87,;6.13,2.03,;6.75,.62,;5.61,-.41,)|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ccc2n1)-c1c(Cl)c(F)c(Cn2ncnn2)c2[nH]ncc12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ccc2n1)-c1c(Cl)c(F)c(CN2CCC2)c2[nH]ncc12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ccc2n1)-c1c(Cl)c(F)c(CN2CCCC2)c2[nH]ncc12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ccc2n1)-c1c(Cl)c(F)c(CN2CCCCC2)c2[nH]ncc12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ccc2n1)-c1c(Cl)c(F)c(Cn2nccn2)c2[nH]ncc12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ccc2n1)-c1c(Cl)c(F)c(Cn2ccnn2)c2[nH]ncc12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ccc2n1)-c1c(Cl)c(F)c(Cn2cncn2)c2[nH]ncc12 |r|
Cn1ccnc1Sc1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
CN(C)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)NC4CC4)cn3c2)c2cn[nH]c12
Cc1cccn1-c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r,wD:21.21,23.25,(8.67,-.59,;8.35,-2.09,;9.38,-3.24,;8.61,-4.57,;7.11,-4.25,;6.94,-2.72,;5.61,-1.95,;4.28,-2.72,;4.28,-4.26,;2.94,-1.95,;1.61,-2.72,;2.94,-.41,;1.61,.36,;1.61,1.9,;.28,2.67,;-1.06,1.9,;-2.52,2.38,;-3.43,1.13,;-4.97,1.13,;-5.74,2.47,;-4.97,3.8,;-7.28,2.47,;-8.61,1.7,;-8.61,3.24,;-9.38,4.57,;-2.52,-.11,;-1.06,.36,;.28,-.41,;4.28,.36,;4.6,1.87,;6.13,2.03,;6.75,.62,;5.61,-.41,)|
CC(C)(O)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
COCc1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
CCOCc1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ccc2n1)-c1c(Cl)c(F)c(Cn2cnnn2)c2[nH]ncc12 |r|
CC(c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12)n1ncnn1 |r|
CC(Nc1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12)C(=O)N(C)C |r|
COC(C)(C)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
CC(N(C)C)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
CN(C)C(=O)CNc1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12
CC(c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12)n1cnnn1 |r|
CC(N)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
CN(C)C(=O)c1ccn(c1)-c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ccc2n1)-c1c(Cl)c(F)c(OC2CC2)c2[nH]ncc12 |r|
CNC(C)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
CC(C)Nc1c(F)c(Cl)c(-c2cc(N)c3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
CC(C)Oc1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
CC(C)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ccc2n1)-c1c(Cl)c(F)c(C2CCCC2)c2[nH]ncc12 |r|
C[C@H](c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12)n1ncnn1
C[C@@H](c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12)n1ncnn1 |r|
OC(c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12)C(F)(F)F |r|
OC1CCCC1c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
CC(=S)Nc1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
CC(N(C)C(C)=O)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
C[C@H](c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12)n1cnnn1 |r|
C[C@@H](c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12)n1cnnn1 |r|
COC(c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12)C(F)(F)F |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ccc2n1)-c1c(Cl)c(F)c(NC2CCOC2)c2[nH]ncc12 |r|
CC(NC(C)=O)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
CCOC(c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12)C(F)(F)F
FC(c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12)C(F)(F)F |r|
CC(Nc1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12)C1CC1 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ccc2n1)-c1c(Cl)c(F)c(NCC2CC2)c2[nH]ncc12 |r|
COC[C@H](C)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
COC[C@@H](C)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
CCC(=O)NC(C)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
CC(Nc1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12)C(F)F |r|
CC(NC=O)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
CC(NC1COC1)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
CC(NC(=O)C(F)(F)F)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12
CC(NC1(CC1)C#N)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
CC(NC(=O)C1CCC1)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ccc2n1)-c1c(Cl)c(F)c(-c2cnc[nH]2)c2[nH]ncc12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ccc2n1)-c1c(Cl)c(F)c(NC2=NCCN2)c2[nH]ncc12 |r,t:26|
CNC(=O)C(C)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
CSCc1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
CNC(=O)N(C)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
CSC(C)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
CS(=O)Cc1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
CS(=O)(=O)Cc1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ccc2n1)-c1c(Cl)c(F)c(C(NC=O)C#N)c2[nH]ncc12 |r|
CO[C@H](C)[C@@H](OC)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
CC(NC(=O)C(F)F)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
Cc1ncc([nH]1)-c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
CC(c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12)S(C)=O |r|
CC(c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12)S(C)(=O)=O |r|
CCNC(=O)C(C)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3c2)c2cn[nH]c12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cc2cc(ccn2n1)-c1c(C=C)c(F)cc2[nH]ncc12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cc2cc(ccn2n1)-c1c(Cl)ccc2[nH]ncc12 |r|
COc1ccc2[nH]ncc2c1-c1ccn2nc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1 |r|
CN(C)c1ccc2[nH]ncc2c1-c1ccn2nc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1 |r|
F[C@H]1C[C@H]1C(=O)Nc1cc2cc(ccn2n1)-c1c(ccc2[nH]ncc12)C(F)(F)F |r|
CCc1ccc2[nH]ncc2c1-c1ccn2nc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1 |r|
CC(=O)c1ccc2[nH]ncc2c1-c1ccn2nc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1 |r|
CN(C)c1c(F)cc2[nH]ncc2c1-c1ccn2nc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1 |r|
F[C@H]1C[C@H]1C(=O)Nc1cc2cc(ccn2n1)-c1c(Br)ccc2[nH]ncc12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cc2cc(ccn2n1)-c1c(ccc2[nH]ncc12)C#N
F[C@H]1C[C@H]1C(=O)Nc1cc2cc(ccn2n1)-c1c(C2CC2)c(F)cc2[nH]ncc12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cc2cc(ccn2n1)-c1c(Cl)c(F)cc2[nH]ncc12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cc2cc(ccn2n1)-c1c(ccc2[nH]ncc12)C1CC1 |r|
Cc1c(F)cc2[nH]ncc2c1-c1ccn2nc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1 |r|
OCc1ccc2[nH]ncc2c1-c1ccn2nc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1 |r|
CC(C)c1c(F)cc2[nH]ncc2c1-c1ccn2nc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1 |r|
CSc1ccc2[nH]ncc2c1-c1ccn2nc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1 |r|
F[C@H]1C[C@H]1C(=O)Nc1cc2cc(ccn2n1)-c1c(Br)c(F)cc2[nH]ncc12 |r|
FC(F)c1ccc2[nH]ncc2c1-c1ccn2nc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1 |r|
CCc1c(F)cc2[nH]ncc2c1-c1ccn2nc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1
COc1c(F)cc2[nH]ncc2c1-c1ccn2nc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1 |r|
FC(F)c1c(F)cc2[nH]ncc2c1-c1ccn2nc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1 |r|
Cc1c(F)cc2[nH]nc(Cl)c2c1-c1ccn2nc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1 |r|
Cc1n[nH]c2cc(F)c(C)c(-c3ccn4nc(NC(=O)[C@@H]5C[C@@H]5F)cc4c3)c12 |r|
CSc1n[nH]c2cc(F)c(C)c(-c3ccn4nc(NC(=O)[C@@H]5C[C@@H]5F)cc4c3)c12 |r|
Cc1c(F)cc2[nH]nc(C#C)c2c1-c1ccn2nc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1 |r|
Cc1c(F)cc2[nH]nc(C3CC3)c2c1-c1ccn2nc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1 |r|
Cc1c(F)cc2[nH]nc(C=C)c2c1-c1ccn2nc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1 |r|
CCc1n[nH]c2cc(F)c(C)c(-c3ccn4nc(NC(=O)[C@@H]5C[C@@H]5F)cc4c3)c12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cc2cc(ccn2n1)-c1c(Cl)c(F)c(Cl)c2[nH]ncc12 |r|
Cc1c(F)c(C)c2[nH]ncc2c1-c1ccn2nc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1 |r|
CP(C)(=O)c1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
Cc1c(F)c(Cl)c2[nH]ncc2c1-c1ccn2nc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1 |r|
F[C@H]1C[C@H]1C(=O)Nc1cc2cc(ccn2n1)-c1c(Cl)c(F)c(Br)c2[nH]ncc12 |r|
Cc1c(F)c(F)c2[nH]ncc2c1-c1ccn2nc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1 |r|
Cc1c(F)c(c2[nH]ncc2c1-c1ccn2nc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1)C(F)(F)F |r|
Cc1cc(C=C)c2[nH]ncc2c1-c1ccn2nc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1 |r|
CN(C)c1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
CSc1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
CS(=O)(=O)c1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
Cc1c(F)c(Br)c2[nH]ncc2c1-c1ccn2nc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1 |r|
CSc1c(F)c(C)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
Cc1c(F)c(c2[nH]ncc2c1-c1ccn2nc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1)S(C)(=O)=O |r|
CN(C)c1c(F)c(C)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
COc1c(F)c(C)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
COc1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
CCOc1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
CNc1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
CN1CCN(CC1)c1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
CCNc1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
CCN(CC)c1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cc2cc(ccn2n1)-c1c(Cl)c(F)c(N2CCOCC2)c2[nH]ncc12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cc2cc(ccn2n1)-c1c(Cl)c(F)c(N2CCCC2)c2[nH]ncc12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cc2cc(ccn2n1)-c1c(Cl)c(F)c(N2CCNCC2)c2[nH]ncc12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cc2cc(ccn2n1)-c1c(Cl)c(F)c(N2CCC2)c2[nH]ncc12 |r|
CN(C)C1CCC(CC1)N(C)c1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r,wD:26.26,28.30,(7.6,-5.75,;8.73,-4.7,;10.2,-5.15,;8.38,-3.2,;6.91,-2.75,;6.56,-1.25,;7.69,-.2,;9.16,-.65,;9.51,-2.15,;7.34,1.31,;8.47,2.36,;5.87,1.76,;4.75,.71,;5.09,-.8,;3.27,1.16,;2.15,.11,;2.93,2.66,;1.45,3.11,;1.11,4.61,;-.37,5.06,;-1.49,4.01,;-3.03,4.14,;-3.63,2.72,;-5.13,2.38,;-6.18,3.5,;-5.73,4.98,;-7.68,3.16,;-8.81,2.11,;-9.15,3.61,;-10.2,4.73,;-2.47,1.71,;-1.15,2.51,;.33,2.06,;4.05,3.71,;4.03,5.25,;5.48,5.75,;6.41,4.52,;5.52,3.26,)|
CN(C1CCC(O)CC1)c1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r,wD:24.24,26.28,(8.82,2.27,;7.69,1.22,;8.04,-.28,;6.91,-1.33,;7.26,-2.83,;8.73,-3.28,;9.08,-4.78,;9.86,-2.23,;9.51,-.73,;6.22,1.67,;5.09,.62,;5.44,-.88,;3.62,1.07,;2.49,.02,;3.27,2.57,;1.8,3.02,;1.45,4.52,;-.02,4.97,;-1.15,3.92,;-2.68,4.05,;-3.28,2.64,;-4.78,2.29,;-5.83,3.42,;-5.38,4.89,;-7.33,3.07,;-8.46,2.02,;-8.81,3.52,;-9.86,4.65,;-2.12,1.63,;-.8,2.42,;.67,1.97,;4.4,3.62,;4.37,5.16,;5.83,5.66,;6.75,4.43,;5.87,3.17,)|
CN[C@H]1CCC(CC1)N(C)c1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r,wD:25.25,27.29,2.1,(9.66,-4.68,;10.43,-3.34,;9.66,-2.01,;10.43,-.68,;9.66,.66,;8.12,.66,;7.35,-.68,;8.12,-2.01,;7.35,1.99,;8.12,3.33,;5.81,1.99,;5.04,.66,;5.81,-.68,;3.5,.66,;2.73,-.68,;2.73,1.99,;1.19,1.99,;.42,3.33,;-1.12,3.33,;-1.89,1.99,;-3.4,1.67,;-3.56,.14,;-4.89,-.63,;-6.22,.14,;-6.22,1.68,;-7.56,-.63,;-8.33,-1.96,;-9.1,-.63,;-10.43,.14,;-2.15,-.49,;-1.12,.66,;.42,.66,;3.5,3.33,;3.03,4.79,;4.27,5.7,;5.52,4.79,;5.04,3.33,)|
CN[C@H]1CCC(CC1)N(C)c1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r,wU:2.1,wD:25.25,27.29,(9.66,-4.37,;10.43,-3.04,;9.66,-1.7,;8.12,-1.7,;7.35,-.37,;8.12,.96,;9.66,.96,;10.43,-.37,;7.35,2.3,;8.12,3.63,;5.81,2.3,;5.04,.96,;5.81,-.37,;3.5,.96,;2.73,-.37,;2.73,2.3,;1.19,2.3,;.42,3.63,;-1.12,3.63,;-1.89,2.3,;-3.4,1.98,;-3.56,.45,;-4.89,-.32,;-6.22,.45,;-6.22,1.99,;-7.56,-.32,;-8.33,-1.66,;-9.1,-.32,;-10.43,.45,;-2.15,-.18,;-1.12,.96,;.42,.96,;3.5,3.63,;3.03,5.1,;4.27,6,;5.52,5.1,;5.04,3.63,)|
COc1cc(C)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cc2cc(ccn2n1)-c1c(Cl)c(F)c(OCC2CCCO2)c2[nH]ncc12 |r|
CNC1CCC(CC1)Nc1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r,wD:24.24,26.28,(7.95,-5.75,;9.08,-4.7,;8.73,-3.2,;7.26,-2.75,;6.91,-1.25,;8.04,-.2,;9.51,-.65,;9.86,-2.15,;7.69,1.31,;6.22,1.76,;5.09,.71,;5.44,-.8,;3.62,1.16,;2.49,.11,;3.27,2.66,;1.8,3.11,;1.45,4.61,;-.02,5.06,;-1.15,4.01,;-2.68,4.14,;-3.28,2.72,;-4.78,2.38,;-5.83,3.5,;-5.38,4.98,;-7.33,3.16,;-8.46,2.11,;-8.81,3.61,;-9.86,4.73,;-2.12,1.71,;-.8,2.51,;.67,2.06,;4.4,3.71,;4.37,5.25,;5.83,5.75,;6.75,4.52,;5.87,3.26,)|
CCOc1c(F)c(C)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
Nc1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
CCOc1cc(C)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
CN(C)C1CCC(CC1)Nc1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r,wD:25.25,27.29,(7.6,-4.98,;8.73,-3.93,;10.2,-4.38,;8.38,-2.43,;6.91,-1.98,;6.56,-.48,;7.69,.57,;9.16,.12,;9.51,-1.38,;7.34,2.07,;5.87,2.53,;4.75,1.48,;5.09,-.03,;3.27,1.93,;2.15,.87,;2.93,3.43,;1.45,3.88,;1.11,5.38,;-.37,5.83,;-1.49,4.78,;-3.03,4.91,;-3.63,3.49,;-5.13,3.15,;-6.18,4.27,;-5.73,5.75,;-7.68,3.93,;-8.81,2.88,;-9.15,4.38,;-10.2,5.5,;-2.47,2.48,;-1.15,3.28,;.33,2.83,;4.05,4.48,;4.03,6.02,;5.48,6.52,;6.41,5.29,;5.52,4.03,)|
CCc1c(F)c(SC)c2[nH]ncc2c1-c1ccn2nc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1 |r|
CN(C1CCC(N)CC1)c1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r,wD:24.24,26.28,(8.82,2.79,;7.69,1.74,;8.04,.24,;6.91,-.81,;7.26,-2.31,;8.73,-2.76,;9.08,-4.26,;9.86,-1.71,;9.51,-.21,;6.22,2.2,;5.09,1.14,;5.44,-.36,;3.62,1.59,;2.49,.54,;3.27,3.1,;1.8,3.55,;1.45,5.05,;-.02,5.5,;-1.15,4.45,;-2.68,4.58,;-3.28,3.16,;-4.78,2.82,;-5.83,3.94,;-5.38,5.42,;-7.33,3.6,;-8.46,2.55,;-8.81,4.05,;-9.86,5.17,;-2.12,2.15,;-.8,2.95,;.67,2.5,;4.4,4.15,;4.37,5.69,;5.83,6.19,;6.75,4.96,;5.87,3.7,)|
NC1CCC(CC1)Nc1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r,wD:23.23,25.27,(9.08,-4.12,;8.73,-2.61,;7.26,-2.16,;6.91,-.66,;8.04,.39,;9.51,-.06,;9.86,-1.56,;7.69,1.89,;6.22,2.34,;5.09,1.29,;5.44,-.21,;3.62,1.74,;2.49,.69,;3.27,3.24,;1.8,3.69,;1.45,5.19,;-.02,5.64,;-1.15,4.59,;-2.68,4.72,;-3.28,3.3,;-4.78,2.96,;-5.83,4.08,;-5.38,5.56,;-7.33,3.74,;-8.46,2.69,;-8.81,4.19,;-9.86,5.31,;-2.12,2.29,;-.8,3.09,;.67,2.64,;4.4,4.29,;4.37,5.83,;5.83,6.33,;6.75,5.1,;5.87,3.84,)|
CC(C)(C)OC(=O)NC1CCC(CC1)Nc1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r,wD:30.30,32.34,(11.89,-3.05,;10.77,-4.1,;11.11,-5.6,;12.24,-4.55,;9.29,-3.65,;8.17,-4.7,;8.51,-6.2,;6.69,-4.25,;6.35,-2.75,;4.87,-2.3,;4.53,-.8,;5.65,.25,;7.13,-.2,;7.47,-1.7,;5.31,1.76,;3.84,2.21,;2.71,1.16,;3.06,-.35,;1.24,1.61,;.11,.56,;.89,3.11,;-.58,3.56,;-.93,5.06,;-2.4,5.51,;-3.53,4.46,;-5.06,4.59,;-5.66,3.17,;-7.16,2.83,;-8.21,3.95,;-7.76,5.43,;-9.72,3.61,;-10.84,2.56,;-11.19,4.06,;-12.24,5.18,;-4.5,2.16,;-3.18,2.96,;-1.71,2.51,;2.02,4.16,;1.99,5.7,;3.45,6.2,;4.37,4.97,;3.49,3.71,)|
OC1CCC(CC1)Nc1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r,wD:23.23,25.27,(9.08,-4.97,;8.73,-3.47,;7.26,-3.02,;6.91,-1.52,;8.04,-.47,;9.51,-.92,;9.86,-2.42,;7.69,1.03,;6.22,1.48,;5.09,.43,;5.44,-1.07,;3.62,.88,;2.49,-.17,;3.27,2.38,;1.8,2.83,;1.45,4.33,;-.02,4.78,;-1.15,3.73,;-2.68,3.87,;-3.28,2.45,;-4.78,2.1,;-5.83,3.23,;-5.38,4.7,;-7.33,2.88,;-8.46,1.83,;-8.81,3.33,;-9.86,4.46,;-2.12,1.44,;-.8,2.23,;.67,1.78,;4.4,3.43,;4.37,4.97,;5.83,5.47,;6.75,4.24,;5.87,2.98,)|
CCN(CC)c1c(F)c(CC)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
CCc1c(F)c(N(C)C)c2[nH]ncc2c1-c1ccn2nc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1 |r|
OCCSc1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
CCc1c(F)c(SCC(=O)NC)c2[nH]ncc2c1-c1ccn2nc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1 |r|
CCc1c(F)c(SCC(=O)N(C)C)c2[nH]ncc2c1-c1ccn2nc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1 |r|
Cc1c(F)c(SCCO)c2[nH]ncc2c1-c1ccn2nc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1 |r|
CCNc1c(F)c(CC)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
CCN(C)c1c(F)c(CC)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
CCc1c(F)c(SCC(O)=O)c2[nH]ncc2c1-c1ccn2nc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1 |r|
CN(C1CCC(N)C1)c1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
Oc1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
CSc1c(F)c(SC)c2[nH]ncc2c1-c1ccn2nc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1 |r|
CSc1c(F)cc2[nH]ncc2c1-c1ccn2nc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1 |r|
CCOc1c(F)c(CC)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
CCc1c(F)c(F)c2[nH]ncc2c1-c1ccn2nc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1 |r|
Cc1c(F)c(S(C)=O)c2[nH]ncc2c1-c1ccn2nc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1 |r|
Cc1c(F)c(OCCO)c2[nH]ncc2c1-c1ccn2nc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1 |r|
Cc1c(F)c(OCCOC(N)=O)c2[nH]ncc2c1-c1ccn2nc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1 |r|
F[C@H]1C[C@H]1C(=O)Nc1cc2cc(ccn2n1)-c1c(Cl)c(F)c(F)c2[nH]ncc12 |r|
CC(=O)Nc1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
CS(=O)c1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
CN(CCOc1c(F)c(C)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12)C(N)=O |r|
CC(=O)Nc1c(F)c(C)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
CSc1c(F)c(F)c2[nH]ncc2c1-c1ccn2nc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1
CN(Nc1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12)C(=O)OC(C)(C)C |r|
CCOc1c(F)c(SC)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
Cc1c(F)c(OCCNC(N)=O)c2[nH]ncc2c1-c1ccn2nc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1 |r|
CNC(=O)NCCOc1c(F)c(C)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
CNC(=O)OCCSc1c(F)c(C)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
Cc1c(F)c(OCCNC(=O)C(F)(F)F)c2[nH]ncc2c1-c1ccn2nc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1 |r|
COC(=O)c1c(F)c(C)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
Cc1c(F)c(C(O)=O)c2[nH]ncc2c1-c1ccn2nc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1 |r|
CN(C(C)=O)c1c(F)c(C)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
OC(=O)c1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
CN(C(C)=O)c1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12
CNNc1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
COC(=O)c1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
CN(C1CCC(O)C1)c1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
CN(C)C(=O)c1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
CN(CCO)c1c(F)c(C)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
CSc1c(F)c(N(C)C)c2[nH]ncc2c1-c1ccn2nc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1 |r|
OC1CCC(C1)Nc1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
CNC(=O)c1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
CN(C1CC(O)C1)c1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r,wD:22.22,24.26,(9.07,1.39,;7.95,.34,;8.29,-1.16,;7.48,-2.47,;8.78,-3.28,;9.13,-4.78,;9.6,-1.98,;6.47,.79,;5.35,-.26,;5.69,-1.76,;3.88,.19,;2.75,-.86,;3.53,1.69,;2.06,2.14,;1.71,3.64,;.24,4.09,;-.89,3.04,;-2.42,3.18,;-3.03,1.76,;-4.53,1.41,;-5.58,2.54,;-5.13,4.01,;-7.08,2.19,;-8.2,1.14,;-8.55,2.64,;-9.6,3.77,;-1.86,.75,;-.54,1.54,;.93,1.09,;4.66,2.74,;4.63,4.28,;6.08,4.78,;7.01,3.55,;6.13,2.29,)|
CSc1c(F)c(C)c(-c2ccn3nc(NC(=O)C4CC4)cc3c2)c2cn[nH]c12
CCN(C)c1c(F)c(C)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
CCN(C)c1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
CN(C)c1c(F)c(c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12)C(F)(F)F |r|
CC(=O)c1c(F)c(C)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
CSc1c(F)c(C)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@H]4F)cc3c2)c2cn[nH]c12 |r|
CSc1c(F)c(C)c(-c2ccn3nc(NC(=O)[C@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
CSc1c(F)cc2[nH]ncc2c1-c1ccn2nc(NC(=O)C3CC3)cc2c1
CN(C)C(=O)c1c(F)c(C)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
CSc1c(F)cc2[nH]ncc2c1-c1ccn2nc(NC(=O)[C@H]3C[C@@H]3F)cc2c1 |r|
CSc1c(F)cc2[nH]ncc2c1-c1ccn2nc(NC(=O)[C@@H]3C[C@H]3F)cc2c1 |r|
CSc1c(F)cc2[nH]ncc2c1-c1ccn2nc(NC(=O)[C@H]3C[C@H]3F)cc2c1
CSc1c(F)c(C)c(-c2ccn3nc(NC(=O)[C@H]4C[C@H]4F)cc3c2)c2cn[nH]c12 |r|
CC(=O)c1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
NC(=O)c1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
CCN(C)c1c(F)c(SC)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
CCOc1c(F)cc2[nH]ncc2c1-c1ccn2nc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1 |r|
Cc1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
CNC(=O)OCCN(C)c1c(F)c(C)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
FC(F)c1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
Cc1c(F)c(C#N)c2[nH]ncc2c1-c1ccn2nc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1 |r|
CN(C)c1c(F)cc(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
CNC(=O)c1c(F)c(C)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12
CCc1c(F)c(c2[nH]ncc2c1-c1ccn2nc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1)C(F)(F)F |r|
F[C@H]1C[C@H]1C(=O)Nc1cc2cc(ccn2n1)-c1c(Cl)c(F)c(C#N)c2[nH]ncc12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cc2cc(ccn2n1)-c1cc(F)c(OC(F)(F)F)c2[nH]ncc12 |r|
CCc1c(F)c(SCC#N)c2[nH]ncc2c1-c1ccn2nc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1 |r|
CSc1c(F)cc(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cc2cc(ccn2n1)-c1c(c(F)cc2[nH]ncc12)C(F)(F)F |r|
Cc1c(F)c(C(F)F)c2[nH]ncc2c1-c1ccn2nc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1 |r|
Cc1c(F)c(OC(F)(F)F)c2[nH]ncc2c1-c1ccn2nc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1 |r|
CSc1ccc(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
Cn1nnnc1-c1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r,wD:21.21,23.25,(8.14,-2.58,;8.61,-1.12,;10.08,-.64,;10.08,.9,;8.61,1.37,;7.71,.13,;6.17,.13,;5.4,-1.21,;6.17,-2.54,;3.86,-1.21,;3.09,-2.54,;3.09,.13,;1.55,.13,;.78,1.46,;-.76,1.46,;-1.53,.13,;-3.04,-.19,;-3.2,-1.73,;-4.53,-2.5,;-5.87,-1.73,;-5.87,-.19,;-7.2,-2.5,;-7.97,-3.83,;-8.74,-2.5,;-10.08,-1.73,;-1.79,-2.35,;-.76,-1.21,;.78,-1.21,;3.86,1.46,;3.38,2.92,;4.63,3.83,;5.87,2.92,;5.4,1.46,)|
CN(C)c1ccc(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12
CN(c1ncccn1)c1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cc2cc(ccn2n1)-c1c(Cl)c(F)c(SCC#N)c2[nH]ncc12 |r|
CSc1c(F)c(F)c2[nH]ncc2c1-c1ccn2nc(NC(=O)[C@H]3C[C@H]3F)cc2c1 |r|
CSc1c(F)c(F)c2[nH]ncc2c1-c1ccn2nc(NC(=O)[C@@H]3C[C@H]3F)cc2c1 |r|
CSc1c(F)c(F)c2[nH]ncc2c1-c1ccn2nc(NC(=O)[C@H]3C[C@@H]3F)cc2c1 |r|
F[C@H]1C[C@H]1C(=O)Nc1cc2cc(ccn2n1)-c1c(Cl)c(F)c(Nc2ncccn2)c2[nH]ncc12 |r|
CCc1c(F)c(SC(C)C#N)c2[nH]ncc2c1-c1ccn2nc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1 |r|
CCc1c(F)c(SC(C)(C)C#N)c2[nH]ncc2c1-c1ccn2nc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1 |r|
CN(C)C(=O)c1c(F)cc(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
CN(C)C(=O)c1c(F)cc2[nH]ncc2c1-c1ccn2nc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1 |r|
CCOc1c(F)c(SC)c2[nH]ncc2c1-c1ccn2nc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1 |r|
F[C@H]1C[C@H]1C(=O)Nc1cc2cc(ccn2n1)-c1c(Cl)c(F)c(OC(F)(F)F)c2[nH]ncc12
CCc1c(F)c(SC2(CC2)C#N)c2[nH]ncc2c1-c1ccn2nc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1 |r|
F[C@H]1C[C@H]1C(=O)Nc1cc2cc(ccn2n1)-c1c(Cl)c(F)c(Nc2ccncc2)c2[nH]ncc12 |r|
CCOc1c(F)c(N(C)C)c2[nH]ncc2c1-c1ccn2nc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1 |r|
CCOc1c(F)c(F)c2[nH]ncc2c1-c1ccn2nc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1 |r|
CN(CC#N)C(=O)c1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
CN(c1ncc(F)cn1)c1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
CN(c1ccncc1)c1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
CC(=O)N(CC#N)c1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
CN(CCc1ccncc1)c1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
CN(c1ncncn1)c1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12
CN(c1nccnn1)c1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
CC(C)Nc1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
CN(C1CCC1)c1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
CCSc1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
CC(C)N(C)c1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
CN1CCN(C1=O)c1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
COC1CN(C1)c1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
CN(C1CC1)c1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cc2cc(ccn2n1)-c1c(Cl)c(F)c(C=O)c2[nH]ncc12 |r|
COCC1CN(C1)c1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cc2cc(ccn2n1)-c1c(Cl)c(F)c(N2CCS(=O)(=O)CC2)c2[nH]ncc12
OCc1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
CC1CN(C1)c1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cc2cc(ccn2n1)-c1c(Cl)c(F)c(N2CCSCC2)c2[nH]ncc12 |r|
CC1(F)CN(C1)c1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cc2cc(ccn2n1)-c1c(Cl)c(F)c(\C=C\C#N)c2[nH]ncc12 |r|
FCc1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cc2cc(ccn2n1)-c1c(Cl)c(F)c(N2CCS(=O)CC2)c2[nH]ncc12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cc2cc(ccn2n1)-c1c(Cl)c(F)c(NCC#N)c2[nH]ncc12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cc2cc(ccn2n1)-c1c(Cl)c(F)c(-n2cccc2)c2[nH]ncc12 |r|
CC(C)(Nc1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12)C#N |r|
CC(=C)c1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12
CC(C)c1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
CC(Nc1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12)C#N |r|
F[C@H]1C[C@H]1C(=O)Nc1cc2cc(ccn2n1)-c1c(Cl)c(F)c(N2CCC(F)C2)c2[nH]ncc12 |r,w:25.28|
CC(C#N)N(C(=O)OCc1ccccc1)c1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
Cc1cccn1-c1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r,wD:21.21,23.25,(8.67,-.59,;8.35,-2.09,;9.38,-3.24,;8.61,-4.57,;7.11,-4.25,;6.94,-2.72,;5.61,-1.95,;4.28,-2.72,;4.28,-4.26,;2.94,-1.95,;1.61,-2.72,;2.94,-.41,;1.61,.36,;1.61,1.9,;.28,2.67,;-1.06,1.9,;-2.52,2.38,;-3.43,1.13,;-4.97,1.13,;-5.74,2.47,;-4.97,3.8,;-7.28,2.47,;-8.61,1.7,;-8.61,3.24,;-9.38,4.57,;-2.52,-.11,;-1.06,.36,;.28,-.41,;4.28,.36,;4.6,1.87,;6.13,2.03,;6.75,.62,;5.61,-.41,)|
CSc1c(F)c(Cl)c(-c2ccn3nc(NC(=O)O[C@@H]4COC[C@H]4C)cc3c2)c2cn[nH]c12 |r|
C[C@H]1[C@@H]([C@H]1c1cnn(C)c1)C(=O)Nc1cc2cc(ccn2n1)-c1c(Cl)c(F)c(N(C)C)c2[nH]ncc12 |r|
CN(C)c1c(F)c(Cl)c(-c2ccn3nc(NC(=O)NC4CC4)cc3c2)c2cn[nH]c12
C[C@@H]1[C@@H]([C@H]1c1cnn(C)c1)C(=O)Nc1cc2cc(ccn2n1)-c1c(Cl)c(F)c(N(C)C)c2[nH]ncc12 |r|
CN(C)C(=O)c1ccn(c1)-c1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
CC(C)Oc1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12
F[C@H]1C[C@H]1C(=O)Nc1cc2cc(ccn2n1)-c1c(Cl)c(F)c(C2CCCC2)c2[nH]ncc12 |r|
OC(c1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12)C(F)(F)F |r|
CC(Nc1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12)C1CC1 |r|
F[C@H]1C[C@H]1C(=O)Nc1cc2cc(ccn2n1)-c1c(Cl)c(F)c(NCC2CC2)c2[nH]ncc12 |r|
COC[C@H](C)c1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
COC[C@@H](C)c1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
CC(Nc1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12)C(F)F |r|
OC1COC(C1)c1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
CC(NC=O)c1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
CCC(=O)NC(C)c1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
CC(NC(=O)C1CCC1)c1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12
CC(NC(=O)C(F)(F)F)c1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
CC(NC(C)=O)c1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
CNC(=O)N(C)c1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
CC(NC(=O)C(F)F)c1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
CO[C@H](C)[C@@H](OC)c1c(F)c(Cl)c(-c2ccn3nc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)c2cn[nH]c12 |r|
CC[C@@H](N)c1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nnc2CC[C@H](C)n12)N1CCC[C@H]1C |r|
CC[C@H]1CCc2nnc(-c3cccc(n3)N3Cc4c(cc(nc4[C@@H](C)N)N4CCC[C@H]4C)C3=O)n12 |r|
CC[C@H]1CCc2nnc(-c3cccc(n3)N3Cc4c(cc(nc4[C@H](C)N)N4CCC[C@H]4C)C3=O)n12 |r|
CC[C@H]1CCc2nnc(-c3cccc(n3)N3Cc4c(cc(nc4[C@@H](C)N)N(C)C(C)C)C3=O)n12 |r|
CC[C@@H](N)c1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nnc2CC[C@H](C)n12)N(C)C(C)C |r|
COC[C@@H](N)c1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nnc2CC[C@H](C)n12)C1(C)CC1 |r|
CC[C@@H]1CCc2nnc(-c3cccc(n3)N3Cc4c(cc(nc4[C@@H](C)N)N4CCC[C@H]4C)C3=O)n12 |r|
CC[C@@H]1CCc2nnc(-c3cccc(n3)N3Cc4c(cc(nc4[C@H](C)N)N4CCC[C@H]4C)C3=O)n12 |r|
CC[C@@H](N)c1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nnc2CC[C@@H](C)n12)N1CCC[C@H]1C |r|
CC[C@H](N)c1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nnc2CC[C@H](C)n12)N1CCC[C@H]1C |r|
CC[C@H](N)c1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nnc2CC[C@@H](C)n12)N1CCC[C@H]1C |r|
CC[C@@H]1CCc2nnc(-c3cccc(n3)N3Cc4c(cc(nc4[C@@H](C)N)N(C)C(C)C)C3=O)n12 |r|
CC[C@@H](N)c1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nnc2CC[C@@H](CC)n12)N1CCC[C@H]1C |r|
CC[C@@H](N)c1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nnc2CC[C@H](CC)n12)N1CCC[C@H]1C |r|
CC[C@H](N)c1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nnc2CC[C@H](CC)n12)N1CCC[C@H]1C |r|
CC[C@H](N)c1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nnc2CC[C@@H](CC)n12)N1CCC[C@H]1C |r|
C[C@@H]1CCCN1c1cc2C(=O)N(Cc2c(n1)C(C)(C)N)c1cccc(n1)-c1nnc2CC[C@H](C)n12 |r|
C[C@H](N)c1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nnc2CC[C@H](CF)n12)N1CCC[C@H]1C |r|
CC[C@@H](N)c1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nnc2CC[C@H](CO)n12)N(C)C(C)C |r|
CC(C)N(C)c1cc2C(=O)N(Cc2c(n1)[C@@H](C)N)c1cccc(n1)-c1nnc2CC[C@H](C)n12 |r|
C[C@H]1CCc2nnc(-c3cccc(n3)N3Cc4c(cc(nc4C(C)(C)N)N(C)C)C3=O)n12 |r|
C[C@@H]1CCc2nnc(-c3cccc(n3)N3Cc4c(cc(nc4C(C)(C)N)N(C)C)C3=O)n12 |r|
C[C@@H](N)c1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nnc2CC[C@H](C)n12)N1CCC[C@H]1C |r|
C[C@@H](N)c1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nnc2CC[C@@H](C)n12)N1CCC[C@H]1C |r|
C[C@H](N)c1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nnc2CC[C@H](C)n12)N1CCC[C@H]1C |r|
C[C@H](N)c1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nnc2CC[C@@H](C)n12)N1CCC[C@H]1C |r|
CC[C@@H](N)c1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nnc2CC[C@H](C)n12)N(C)C |r|
CC[C@@H](N)c1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nnc2CC[C@H](CF)n12)N(C)C(C)C |r|
C[C@@H](N)c1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nnc2CC[C@H](CO)n12)N1CCC[C@H]1C |r|
CC[C@@H](N)c1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nnc2CC[C@H](CO)n12)N1CCC[C@H]1C |r|
CC[C@@H](N)c1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nnc2CC[C@H](CF)n12)N1CCC[C@H]1C |r|
CC[C@@H](N)c1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nnc2CC[C@H](CF)n12)N(C)C |r|
COC[C@@H](N)c1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nnc2CC[C@H](CF)n12)C1(C)CC1 |r|
CC[C@@H](N)c1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nnc2CC[C@H](CO)n12)C1(C)CC1 |r|
CC[C@@H](N)c1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nnc2CC[C@H](C)n12)C1(C)CC1 |r|
COC[C@@H](N)c1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nnc2CC[C@H](CO)n12)C1(C)CC1 |r|
CCn1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2C(C)(C)N)N2CCC[C@H]2C)C1=O |r|
CCCn1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2[C@@H](C)N)N2CCC[C@H]2C)C1=O |r|
CCCn1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2[C@H](C)N)N2CCC[C@H]2C)C1=O |r|
C[C@@H](N)c1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nncn1C1CCC1)C1(C)CC1 |r|
C[C@H](N)c1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nncn1C1CCC1)C1(C)CC1 |r|
CC[C@@H](N)c1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nncn1C1CCC1)C1(C)CC1 |r|
CC[C@H](N)c1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nncn1C1CCC1)C1(C)CC1 |r|
CCn1c(C)nnc1-c1cccc(n1)N1Cc2c(cc(nc2[C@@H](C)NC)N2CCC[C@H]2C)C1=O |r|
CCn1c(C)nnc1-c1cccc(n1)N1Cc2c(cc(nc2[C@H](C)NC)N2CCC[C@H]2C)C1=O |r|
CCn1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2[C@H](C)NC)N2CCC[C@H]2C)C1=O |r|
CCn1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2[C@@H](C)NC)N2CCC[C@H]2C)C1=O |r|
CCn1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2[C@@H](C)NC)C2(C)CC2)C1=O |r|
CCn1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2[C@H](C)NC)C2(C)CC2)C1=O |r|
CCCn1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2[C@H](C)NC)C2(C)CC2)C1=O |r|
CCn1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2C(C)(C)N)C2(C)CC2)C1=O
CCn1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2[C@@H](C)N)C2(C)CC2)C1=O |r|
CCn1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2[C@H](C)N)C2(C)CC2)C1=O |r|
CCCn1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2[C@@H](C)N)C2(C)CC2)C1=O |r|
CCCn1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2[C@H](C)N)C2(C)CC2)C1=O |r|
CC[C@@H](N)c1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nncn1CC)C1(C)CC1 |r|
CC[C@H](N)c1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nncn1CC)C1(C)CC1 |r|
CCCn1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2[C@H](N)CC)C2(C)CC2)C1=O |r|
CCCn1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2[C@@H](N)CC)C2(C)CC2)C1=O |r|
CCN(C)c1cc2C(=O)N(Cc2c(n1)C(C)(C)N)c1cccc(n1)-c1nnc(C)n1CC
CCN(C)c1cc2C(=O)N(Cc2c(n1)C(C)(C)N)c1cccc(n1)-c1nncn1CC
CCC(CC)n1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2[C@H](C)N)C2(C)CC2)C1=O |r|
CCC(CC)n1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2[C@@H](C)N)C2(C)CC2)C1=O |r|
CCN(C)c1cc2C(=O)N(Cc2c(n1)[C@@H](C)N)c1cccc(n1)-c1nnc(C)n1CC |r|
CCN(C)c1cc2C(=O)N(Cc2c(n1)[C@H](C)N)c1cccc(n1)-c1nnc(C)n1CC |r|
CCN(C)c1cc2C(=O)N(Cc2c(n1)[C@@H](C)N)c1cccc(n1)-c1nncn1CC |r|
CCN(C)c1cc2C(=O)N(Cc2c(n1)[C@H](C)N)c1cccc(n1)-c1nncn1CC |r|
CCCn1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2C(C)(C)N)N(C)C)C1=O
CCn1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2C(C)(C)N)N(C)C)C1=O
CCCn1c(C)nnc1-c1cccc(n1)N1Cc2c(cc(nc2C(C)(C)N)N2CCC[C@H]2C)C1=O |r|
CCn1c(C)nnc1-c1cccc(n1)N1Cc2c(cc(nc2C(C)(C)N)N2CCC[C@H]2C)C1=O |r|
CCCn1c(C)nnc1-c1cccc(n1)N1Cc2c(cc(nc2[C@@H](C)N)N2CCC[C@H]2C)C1=O |r|
CCCn1c(C)nnc1-c1cccc(n1)N1Cc2c(cc(nc2[C@H](C)N)N2CCC[C@H]2C)C1=O |r|
CCCn1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2[C@H](C)N)N(C)C)C1=O |r|
CCCn1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2[C@@H](C)N)N(C)C)C1=O |r|
CCCn1c(C)nnc1-c1cccc(n1)N1Cc2c(cc(nc2C(C)(C)N)N(C)C(C)C)C1=O
CC[C@@H](N)c1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nncn1CC)N1CCC[C@H]1C |r|
CC[C@H](N)c1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nncn1CC)N1CCC[C@H]1C |r|
CCCn1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2[C@H](N)CC)N(C)C)C1=O |r|
CCCn1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2[C@@H](N)CC)N(C)C)C1=O |r|
CCCn1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2[C@H](N)CC)N2CCC[C@H]2C)C1=O |r|
CCCn1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2[C@@H](N)CC)N2CCC[C@H]2C)C1=O |r|
CC[C@@H](N)c1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nncn1CC)N(C)C |r|
CC[C@H](N)c1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nncn1CC)N(C)C |r|
CCCn1c(C)nnc1-c1cccc(n1)N1Cc2c(cc(nc2[C@@H](C)N)N(C)C(C)C)C1=O |r|
CCCn1c(C)nnc1-c1cccc(n1)N1Cc2c(cc(nc2[C@H](C)N)N(C)C(C)C)C1=O |r|
CCn1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2[C@H](C)N)N2CCC[C@H]2C)C1=O |r|
CCn1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2[C@@H](C)N)N2CCC[C@H]2C)C1=O |r|
CCn1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2[C@H](C)N)N(C)C)C1=O |r|
CCn1cnnc1-c1cccc(n1)N1Cc2c(cc(nc2[C@@H](C)N)N(C)C)C1=O |r|
CCn1c(C)nnc1-c1cccc(n1)N1Cc2c(cc(nc2[C@@H](C)N)N2CCC[C@H]2C)C1=O |r|
CCn1c(C)nnc1-c1cccc(n1)N1Cc2c(cc(nc2[C@H](C)N)N2CCC[C@H]2C)C1=O |r|
CC[C@H]1CCc2nnc(-c3cccc(n3)N3Cc4c(cc(nc4CNC)N4CCC[C@H]4C)C3=O)n12 |r|
CC[C@H]1CCc2nnc(-c3cccc(n3)N3Cc4c(cc(nc4CNC)N(C)C(C)C)C3=O)n12 |r|
CNCc1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nnc2CC[C@H](CF)n12)N1CCC[C@H]1C |r|
CC[C@@H]1CCc2nnc(-c3cccc(n3)N3Cc4c(cc(nc4CNC)N4CCC[C@H]4C)C3=O)n12 |r|
CC[C@@H]1CCc2nnc(-c3cccc(n3)N3Cc4c(cc(nc4CNC)N(C)C(C)C)C3=O)n12 |r|
CNCc1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nnc2CC[C@H](CF)n12)N(C)C(C)C |r|
CC[C@H]1CCc2nnc(-c3cccc(n3)N3Cc4c(cc(nc4CNC)N(C)C)C3=O)n12 |r|
CC[C@@H]1CCc2nnc(-c3cccc(n3)N3Cc4c(cc(nc4CNC)N(C)C)C3=O)n12 |r|
CNCc1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nnc2CC[C@H](C)n12)N(C)C |r|
CNCc1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nnc2CC[C@@H](C)n12)N(C)C |r|
CNCc1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nnc2CC[C@H](C)n12)N(C)C(C)C |r|
CNCc1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nnc2[C@@H](C)C[C@H](C)n12)N(C)C(C)C |r|
CNCc1nc(cc2C(=O)N(Cc12)c1cccc(n1)-c1nnc2[C@H](C)C[C@H](C)n12)N(C)C(C)C |r|
CNC(=O)c1ccc(cn1)-c1cc(N)c(NC(=O)c2ccnc(n2)-c2c(F)cccc2OC)cc1F
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c(cc1N)-c1ccc(=O)n(C)c1
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc(cc1N)-c1cccnc1C
COc1ccncc1-c1ccc(NC(=O)c2ccnc(n2)-c2c(F)cccc2OC)c(N)c1
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc(cc1N)-c1cnccc1C#N
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc(cc1N)-c1c(C)nn(C)c1C
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c(cc1N)N1CCOCC1
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c(cc1N)N1CCC1
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c(CN2CCOCC2)cc1N
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc(cc1[C@@H]1CC[C@H](N)CC1)-c1cnccc1C#N |r,wU:24.26,27.30,(-8,11.78,;-6.67,11.01,;-5.33,11.78,;-5.33,13.32,;-4,14.09,;-2.67,13.32,;-2.67,11.78,;-1.33,11.01,;-4,11.01,;-4,9.47,;-5.33,8.7,;-5.33,7.16,;-4,6.39,;-2.67,7.16,;-2.67,8.7,;-1.33,6.39,;-1.33,4.85,;,7.16,;1.33,6.39,;1.33,4.85,;2.67,4.08,;4,4.85,;4,6.39,;2.67,7.16,;2.67,8.7,;4,9.47,;4,11.01,;2.67,11.78,;2.67,13.32,;1.33,11.01,;1.33,9.47,;5.33,4.08,;6.67,4.85,;8,4.08,;8,2.54,;6.67,1.77,;5.29,2.51,;3.95,1.74,;2.62,.97,)|
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2cc(=O)n(nc12)-c1c(C)cccc1F |(-7.26,-4.89,;-6.17,-3.8,;-6.57,-2.31,;-5.48,-1.22,;-3.99,-1.62,;-3.59,-3.11,;-4.68,-4.2,;-2.9,-.53,;-3.3,.95,;-2.21,2.04,;-.73,1.64,;-.33,.16,;-1.42,-.93,;.36,2.73,;.2,4.26,;1.61,4.89,;2.64,3.75,;4.18,3.75,;4.95,2.41,;6.49,2.41,;4.18,1.08,;2.64,1.08,;1.87,2.41,;4.95,-.26,;6.49,-.26,;7.26,1.08,;7.26,-1.59,;6.49,-2.92,;4.95,-2.92,;4.18,-1.59,;2.64,-1.59,)|
COc1cccc(C)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc(cc1)N1CCN(C)CC1 |(1.87,-2.92,;2.64,-1.59,;4.18,-1.59,;4.95,-2.92,;6.49,-2.92,;7.26,-1.59,;6.49,-.26,;7.26,1.08,;4.95,-.26,;4.18,1.08,;2.64,1.08,;1.87,2.41,;.36,2.73,;.2,4.26,;1.61,4.89,;2.64,3.75,;4.18,3.75,;4.95,2.41,;6.49,2.41,;-.73,1.64,;-2.21,2.04,;-3.3,.95,;-2.9,-.53,;-1.42,-.93,;-.33,.16,;-3.99,-1.62,;-5.48,-1.22,;-6.57,-2.31,;-6.17,-3.8,;-7.26,-4.89,;-4.68,-4.2,;-3.59,-3.11,)|
COc1ccccc1-n1nc2c(n[nH]c2cc1=O)-c1ccc(cc1)N1CCN(C)CC1
COc1ccc(c(OC)c1)-n1nc2c(n[nH]c2cc1=O)-c1ccc(cc1)C1=CCN(C)CC1 |t:30|
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2cc(=O)n(nc12)-c1ccccc1C
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2cc(=O)n(nc12)-c1ccccc1F
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2cc(=O)n(nc12)-c1ccccc1Cl
CCc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc(cc1)N1CCN(C)CC1 |(1.87,-2.92,;2.64,-1.59,;4.18,-1.59,;4.95,-2.92,;6.49,-2.92,;7.26,-1.59,;6.49,-.26,;7.26,1.08,;4.95,-.26,;4.18,1.08,;2.64,1.08,;1.87,2.41,;.36,2.73,;.2,4.26,;1.61,4.89,;2.64,3.75,;4.18,3.75,;4.95,2.41,;6.49,2.41,;-.73,1.64,;-2.21,2.04,;-3.3,.95,;-2.9,-.53,;-1.42,-.93,;-.33,.16,;-3.99,-1.62,;-5.48,-1.22,;-6.57,-2.31,;-6.17,-3.8,;-7.26,-4.89,;-4.68,-4.2,;-3.59,-3.11,)|
COc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc(cc1)N1CCN(C)CC1 |(1.87,-2.92,;2.64,-1.59,;4.18,-1.59,;4.95,-2.92,;6.49,-2.92,;7.26,-1.59,;6.49,-.26,;7.26,1.08,;4.95,-.26,;4.18,1.08,;2.64,1.08,;1.87,2.41,;.36,2.73,;.2,4.26,;1.61,4.89,;2.64,3.75,;4.18,3.75,;4.95,2.41,;6.49,2.41,;-.73,1.64,;-2.21,2.04,;-3.3,.95,;-2.9,-.53,;-1.42,-.93,;-.33,.16,;-3.99,-1.62,;-5.48,-1.22,;-6.57,-2.31,;-6.17,-3.8,;-7.26,-4.89,;-4.68,-4.2,;-3.59,-3.11,)|
COc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc(nc1)N1CCN(C)CC1 |(1.87,-2.92,;2.64,-1.59,;4.18,-1.59,;4.95,-2.92,;6.49,-2.92,;7.26,-1.59,;6.49,-.26,;7.26,1.08,;4.95,-.26,;4.18,1.08,;2.64,1.08,;1.87,2.41,;.36,2.73,;.2,4.26,;1.61,4.89,;2.64,3.75,;4.18,3.75,;4.95,2.41,;6.49,2.41,;-.73,1.64,;-.33,.16,;-1.42,-.93,;-2.9,-.53,;-3.3,.95,;-2.21,2.04,;-3.99,-1.62,;-5.48,-1.22,;-6.57,-2.31,;-6.17,-3.8,;-7.26,-4.89,;-4.68,-4.2,;-3.59,-3.11,)|
CN1CCN(CC1)c1ccc(cn1)-c1n[nH]c2cc(=O)n(nc12)-c1c(C)cccc1F |(-7.26,-4.89,;-6.17,-3.8,;-6.57,-2.31,;-5.48,-1.22,;-3.99,-1.62,;-3.59,-3.11,;-4.68,-4.2,;-2.9,-.53,;-1.42,-.93,;-.33,.16,;-.73,1.64,;-2.21,2.04,;-3.3,.95,;.36,2.73,;.2,4.26,;1.61,4.89,;2.64,3.75,;4.18,3.75,;4.95,2.41,;6.49,2.41,;4.18,1.08,;2.64,1.08,;1.87,2.41,;4.95,-.26,;4.18,-1.59,;2.64,-1.59,;4.95,-2.92,;6.49,-2.92,;7.26,-1.59,;6.49,-.26,;7.26,1.08,)|
CN1CCN(C(=O)C1)c1ccc(cc1)-c1n[nH]c2cc(=O)n(nc12)-c1c(C)cccc1F |(-7.26,-4.89,;-6.17,-3.8,;-4.68,-4.2,;-3.59,-3.11,;-3.99,-1.62,;-5.48,-1.22,;-5.88,.26,;-6.57,-2.31,;-2.9,-.53,;-3.3,.95,;-2.21,2.04,;-.73,1.64,;-.33,.16,;-1.42,-.93,;.36,2.73,;.2,4.26,;1.61,4.89,;2.64,3.75,;4.18,3.75,;4.95,2.41,;6.49,2.41,;4.18,1.08,;2.64,1.08,;1.87,2.41,;4.95,-.26,;4.18,-1.59,;2.64,-1.59,;4.95,-2.92,;6.49,-2.92,;7.26,-1.59,;6.49,-.26,;7.26,1.08,)|
CN1CCN(CC1)c1c(C)cc(cc1C)-c1n[nH]c2cc(=O)n(nc12)-c1c(C)cccc1F |(-7.26,-4.89,;-6.17,-3.8,;-6.57,-2.31,;-5.48,-1.22,;-3.99,-1.62,;-3.59,-3.11,;-4.68,-4.2,;-2.9,-.53,;-3.3,.95,;-4.79,1.35,;-2.21,2.04,;-.73,1.64,;-.33,.16,;-1.42,-.93,;-1.02,-2.42,;.36,2.73,;.2,4.26,;1.61,4.89,;2.64,3.75,;4.18,3.75,;4.95,2.41,;6.49,2.41,;4.18,1.08,;2.64,1.08,;1.87,2.41,;4.95,-.26,;4.18,-1.59,;2.64,-1.59,;4.95,-2.92,;6.49,-2.92,;7.26,-1.59,;6.49,-.26,;7.26,1.08,)|
COc1cc(ccc1N1CCN(C)CC1)-c1n[nH]c2cc(=O)n(nc12)-c1c(C)cccc1F |(-5.19,2.84,;-4.79,1.35,;-3.3,.95,;-2.21,2.04,;-.73,1.64,;-.33,.16,;-1.42,-.93,;-2.9,-.53,;-3.99,-1.62,;-5.48,-1.22,;-6.57,-2.31,;-6.17,-3.8,;-7.26,-4.89,;-4.68,-4.2,;-3.59,-3.11,;.36,2.73,;.2,4.26,;1.61,4.89,;2.64,3.75,;4.18,3.75,;4.95,2.41,;6.49,2.41,;4.18,1.08,;2.64,1.08,;1.87,2.41,;4.95,-.26,;4.18,-1.59,;2.64,-1.59,;4.95,-2.92,;6.49,-2.92,;7.26,-1.59,;6.49,-.26,;7.26,1.08,)|
CN1CCN(Cc2ccc(cc2)-c2n[nH]c3cc(=O)n(nc23)-c2c(C)cccc2F)C(=O)C1 |(-2.94,-6.23,;-3.34,-4.74,;-2.25,-3.66,;-2.65,-2.17,;-4.14,-1.77,;-4.54,-.28,;-3.45,.81,;-3.85,2.29,;-2.76,3.38,;-1.27,2.98,;-.87,1.5,;-1.96,.41,;-.18,4.07,;-.34,5.61,;1.06,6.23,;2.09,5.09,;3.63,5.09,;4.4,3.75,;5.94,3.75,;3.63,2.42,;2.09,2.42,;1.32,3.75,;4.4,1.09,;3.63,-.25,;2.09,-.25,;4.4,-1.58,;5.94,-1.58,;6.71,-.25,;5.94,1.09,;6.71,2.42,;-5.23,-2.86,;-6.71,-2.46,;-4.83,-4.35,)|
COc1cc(ccc1-c1n[nH]c2cc(=O)n(nc12)-c1c(C)cccc1F)N1CCN(C)CC1 |(-4.1,3.93,;-2.61,3.53,;-2.21,2.04,;-3.3,.95,;-2.9,-.53,;-1.42,-.93,;-.33,.16,;-.73,1.64,;.36,2.73,;.2,4.26,;1.61,4.89,;2.64,3.75,;4.18,3.75,;4.95,2.41,;6.49,2.41,;4.18,1.08,;2.64,1.08,;1.87,2.41,;4.95,-.26,;4.18,-1.59,;2.64,-1.59,;4.95,-2.92,;6.49,-2.92,;7.26,-1.59,;6.49,-.26,;7.26,1.08,;-3.99,-1.62,;-5.48,-1.22,;-6.57,-2.31,;-6.17,-3.8,;-7.26,-4.89,;-4.68,-4.2,;-3.59,-3.11,)|
Cc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1cnn(C)c1 |(1.66,-1.8,;2.99,-1.03,;4.33,-1.8,;5.66,-1.03,;5.66,.51,;4.33,1.28,;4.33,2.82,;2.99,.51,;1.66,1.28,;.32,.51,;-1.01,1.28,;-2.47,.8,;-3.38,2.05,;-2.47,3.29,;-1.01,2.82,;.32,3.59,;1.66,2.82,;2.99,3.59,;-2.95,-.66,;-2.04,-1.91,;-2.95,-3.16,;-4.41,-2.68,;-5.66,-3.59,;-4.41,-1.14,)|
CN1CCC(CC1)n1cc(cn1)-c1n[nH]c2cc(=O)n(nc12)-c1c(C)cccc1F |(-4.56,-5.78,;-4.32,-4.25,;-5.52,-3.29,;-5.28,-1.76,;-3.84,-1.21,;-2.64,-2.18,;-2.88,-3.7,;-3.6,.31,;-2.23,1.01,;-2.47,2.53,;-3.99,2.77,;-4.69,1.4,;-1.38,3.62,;-1.54,5.15,;-.13,5.78,;.9,4.63,;2.44,4.63,;3.21,3.3,;4.75,3.3,;2.44,1.96,;.9,1.96,;.13,3.3,;3.21,.63,;2.44,-.7,;.9,-.7,;3.21,-2.04,;4.75,-2.04,;5.52,-.7,;4.75,.63,;5.52,1.96,)|
COc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1cnn(c1)C1CCN(C)CC1 |(.13,-2.04,;.9,-.7,;2.44,-.7,;3.21,-2.04,;4.75,-2.04,;5.52,-.7,;4.75,.63,;5.52,1.96,;3.21,.63,;2.44,1.96,;.9,1.96,;.13,3.3,;-1.38,3.62,;-1.54,5.15,;-.13,5.78,;.9,4.63,;2.44,4.63,;3.21,3.3,;4.75,3.3,;-2.47,2.53,;-3.99,2.77,;-4.69,1.4,;-3.6,.31,;-2.23,1.01,;-3.84,-1.21,;-5.28,-1.76,;-5.52,-3.29,;-4.32,-4.25,;-4.56,-5.78,;-2.88,-3.7,;-2.64,-2.18,)|
COc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1cnn(C)c1 |(1.66,-3.34,;1.66,-1.8,;2.99,-1.03,;4.33,-1.8,;5.66,-1.03,;5.66,.51,;4.33,1.28,;4.33,2.82,;2.99,.51,;1.66,1.28,;.32,.51,;-1.01,1.28,;-2.47,.8,;-3.38,2.05,;-2.47,3.29,;-1.01,2.82,;.32,3.59,;1.66,2.82,;2.99,3.59,;-2.95,-.66,;-2.04,-1.91,;-2.95,-3.16,;-4.41,-2.68,;-5.66,-3.59,;-4.41,-1.14,)|
COc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc(cc1)C1=CCN(C)CC1 |t:29,(1.87,-2.92,;2.64,-1.59,;4.18,-1.59,;4.95,-2.92,;6.49,-2.92,;7.26,-1.59,;6.49,-.26,;7.26,1.08,;4.95,-.26,;4.18,1.08,;2.64,1.08,;1.87,2.41,;.36,2.73,;.2,4.26,;1.61,4.89,;2.64,3.75,;4.18,3.75,;4.95,2.41,;6.49,2.41,;-.73,1.64,;-2.21,2.04,;-3.3,.95,;-2.9,-.53,;-1.42,-.93,;-.33,.16,;-3.99,-1.62,;-5.48,-1.22,;-6.57,-2.31,;-6.17,-3.8,;-7.26,-4.89,;-4.68,-4.2,;-3.59,-3.11,)|
COc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc(cc1)C1CCN(C)CC1 |(1.87,-2.92,;2.64,-1.59,;4.18,-1.59,;4.95,-2.92,;6.49,-2.92,;7.26,-1.59,;6.49,-.26,;7.26,1.08,;4.95,-.26,;4.18,1.08,;2.64,1.08,;1.87,2.41,;.36,2.73,;.2,4.26,;1.61,4.89,;2.64,3.75,;4.18,3.75,;4.95,2.41,;6.49,2.41,;-.73,1.64,;-2.21,2.04,;-3.3,.95,;-2.9,-.53,;-1.42,-.93,;-.33,.16,;-3.99,-1.62,;-5.48,-1.22,;-6.57,-2.31,;-6.17,-3.8,;-7.26,-4.89,;-4.68,-4.2,;-3.59,-3.11,)|
COc1ccc(c(OC)c1)-n1nc2c(n[nH]c2cc1=O)-c1ccc(cc1)N1CCN(C)CC1
COc1ccc(c(OC)c1)-n1nc2c(n[nH]c2cc1=O)-c1ccc(cc1)C1CCN(C)CC1
COc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc(nc1)N1CCOCC1 |(1.52,-3.27,;2.29,-1.93,;3.83,-1.93,;4.6,-3.27,;6.14,-3.27,;6.91,-1.93,;6.14,-.6,;6.91,.73,;4.6,-.6,;3.83,.73,;2.29,.73,;1.52,2.07,;.02,2.39,;-.14,3.92,;1.26,4.55,;2.29,3.4,;3.83,3.4,;4.6,2.07,;6.14,2.07,;-1.07,1.3,;-2.56,1.7,;-3.65,.61,;-3.25,-.88,;-1.76,-1.28,;-.67,-.19,;-4.34,-1.97,;-5.83,-1.57,;-6.91,-2.66,;-6.52,-4.15,;-5.03,-4.55,;-3.94,-3.46,)|
COc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1cnc(nc1)N1CCN(C)CC1 |(1.87,-2.92,;2.64,-1.59,;4.18,-1.59,;4.95,-2.92,;6.49,-2.92,;7.26,-1.59,;6.49,-.26,;7.26,1.08,;4.95,-.26,;4.18,1.08,;2.64,1.08,;1.87,2.41,;.36,2.73,;.2,4.26,;1.61,4.89,;2.64,3.75,;4.18,3.75,;4.95,2.41,;6.49,2.41,;-.73,1.64,;-2.21,2.04,;-3.3,.95,;-2.9,-.53,;-1.42,-.93,;-.33,.16,;-3.99,-1.62,;-5.48,-1.22,;-6.57,-2.31,;-6.17,-3.8,;-7.26,-4.89,;-4.68,-4.2,;-3.59,-3.11,)|
CC(C)c1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc(cc1)N1CCN(C)CC1 |(1.87,-2.92,;2.64,-1.59,;1.87,-.26,;4.18,-1.59,;4.95,-2.92,;6.49,-2.92,;7.26,-1.59,;6.49,-.26,;7.26,1.08,;4.95,-.26,;4.18,1.08,;2.64,1.08,;1.87,2.41,;.36,2.73,;.2,4.26,;1.61,4.89,;2.64,3.75,;4.18,3.75,;4.95,2.41,;6.49,2.41,;-.73,1.64,;-2.21,2.04,;-3.3,.95,;-2.9,-.53,;-1.42,-.93,;-.33,.16,;-3.99,-1.62,;-5.48,-1.22,;-6.57,-2.31,;-6.17,-3.8,;-7.26,-4.89,;-4.68,-4.2,;-3.59,-3.11,)|
Cc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1cnc(nc1)N1CCOCC1 |(2.29,-1.93,;3.83,-1.93,;4.6,-3.27,;6.14,-3.27,;6.91,-1.93,;6.14,-.6,;6.91,.73,;4.6,-.6,;3.83,.73,;2.29,.73,;1.52,2.07,;.02,2.39,;-.14,3.92,;1.26,4.55,;2.29,3.4,;3.83,3.4,;4.6,2.07,;6.14,2.07,;-1.07,1.3,;-2.56,1.7,;-3.65,.61,;-3.25,-.88,;-1.76,-1.28,;-.67,-.19,;-4.34,-1.97,;-5.83,-1.57,;-6.91,-2.66,;-6.52,-4.15,;-5.03,-4.55,;-3.94,-3.46,)|
COc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc(cc1)N1CCN(C)C(=O)C1 |(2.27,-2.92,;3.04,-1.59,;4.58,-1.59,;5.35,-2.92,;6.89,-2.92,;7.66,-1.59,;6.89,-.26,;7.66,1.08,;5.35,-.26,;4.58,1.08,;3.04,1.08,;2.27,2.41,;.76,2.73,;.6,4.26,;2.01,4.89,;3.04,3.75,;4.58,3.75,;5.35,2.41,;6.89,2.41,;-.33,1.64,;-1.81,2.04,;-2.9,.95,;-2.51,-.53,;-1.02,-.93,;.07,.16,;-3.59,-1.62,;-3.2,-3.11,;-4.28,-4.2,;-5.77,-3.8,;-6.86,-4.89,;-6.17,-2.31,;-7.66,-1.92,;-5.08,-1.22,)|
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2cc(=O)n(nc12)-c1c(F)cccc1C1CC1 |(-7.26,-4.89,;-6.17,-3.8,;-6.57,-2.31,;-5.48,-1.22,;-3.99,-1.62,;-3.59,-3.11,;-4.68,-4.2,;-2.9,-.53,;-3.3,.95,;-2.21,2.04,;-.73,1.64,;-.33,.16,;-1.42,-.93,;.36,2.73,;.2,4.26,;1.61,4.89,;2.64,3.75,;4.18,3.75,;4.95,2.41,;6.49,2.41,;4.18,1.08,;2.64,1.08,;1.87,2.41,;4.95,-.26,;6.49,-.26,;7.26,1.08,;7.26,-1.59,;6.49,-2.92,;4.95,-2.92,;4.18,-1.59,;2.64,-1.59,;1.31,-.82,;1.31,-2.36,)|
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2cc(=O)n(nc12)-c1c(C)cc(cc1F)C#N |(-7.64,-4.54,;-6.56,-3.45,;-6.95,-1.96,;-5.87,-.88,;-4.38,-1.27,;-3.98,-2.76,;-5.07,-3.85,;-3.29,-.18,;-3.69,1.3,;-2.6,2.39,;-1.11,1.99,;-.71,.51,;-1.8,-.58,;-.02,3.08,;-.18,4.61,;1.22,5.24,;2.25,4.1,;3.79,4.1,;4.56,2.76,;6.1,2.76,;3.79,1.43,;2.25,1.43,;1.48,2.76,;4.56,.09,;3.79,-1.24,;2.25,-1.24,;4.56,-2.57,;6.13,-2.62,;6.87,-1.24,;6.1,.09,;6.87,1.43,;6.9,-3.95,;7.67,-5.29,)|
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2cc(=O)n(nc12)-c1cnccc1C
COc1ccncc1-n1nc2c(n[nH]c2cc1=O)-c1ccc(cc1)N1CCN(C)CC1
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2c(C)c(=O)n(nc12)-c1c(C)cccc1F |(-7.26,-4.98,;-6.17,-3.9,;-6.57,-2.41,;-5.48,-1.32,;-3.99,-1.72,;-3.59,-3.21,;-4.68,-4.29,;-2.9,-.63,;-3.3,.86,;-2.21,1.95,;-.73,1.55,;-.33,.06,;-1.42,-1.03,;.36,2.64,;.2,4.17,;1.61,4.8,;2.64,3.65,;4.18,3.65,;4.95,4.98,;4.95,2.32,;6.49,2.32,;4.18,.98,;2.64,.98,;1.87,2.32,;4.95,-.35,;4.18,-1.68,;2.64,-1.68,;4.95,-3.02,;6.49,-3.02,;7.26,-1.68,;6.49,-.35,;7.26,.98,)|
Cc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc(cc1)N1CCN(CC1)C1CC1 |(3.19,-1.6,;4.52,-2.37,;4.52,-3.91,;5.86,-4.68,;7.19,-3.91,;7.19,-2.37,;8.52,-1.6,;5.86,-1.6,;5.86,-.06,;4.52,.71,;4.52,2.25,;3.38,3.28,;4,4.68,;5.54,4.52,;5.86,3.02,;7.19,2.25,;7.19,.71,;8.52,-.06,;1.89,2.88,;.8,3.97,;-.69,3.57,;-1.09,2.08,;0,.99,;1.49,1.39,;-2.57,1.68,;-3.66,2.77,;-5.15,2.37,;-5.55,.89,;-4.46,-.2,;-2.97,.19,;-7.04,.49,;-8.52,.89,;-8.12,-.6,)|
CN1C2CCC1CN(C2)c1ccc(cc1)-c1n[nH]c2cc(=O)n(nc12)-c1c(C)cccc1F |(-7.26,-4.89,;-6.17,-3.8,;-6.57,-2.31,;-5.39,-2,;-4.37,-3.04,;-4.68,-4.2,;-3.59,-3.11,;-3.99,-1.62,;-5.48,-1.22,;-2.9,-.53,;-3.3,.95,;-2.21,2.04,;-.73,1.64,;-.33,.16,;-1.42,-.93,;.36,2.73,;.2,4.26,;1.61,4.89,;2.64,3.75,;4.18,3.75,;4.95,2.41,;6.49,2.41,;4.18,1.08,;2.64,1.08,;1.87,2.41,;4.95,-.26,;4.18,-1.59,;2.64,-1.59,;4.95,-2.92,;6.49,-2.92,;7.26,-1.59,;6.49,-.26,;7.26,1.08,)|
COc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc2CN(C)CCc2c1 |(.58,-3.27,;1.35,-1.93,;2.89,-1.93,;3.66,-3.27,;5.2,-3.27,;5.97,-1.93,;5.2,-.6,;5.97,.73,;3.66,-.6,;2.89,.73,;1.35,.73,;.58,2.07,;-.93,2.39,;-1.09,3.92,;.32,4.55,;1.35,3.4,;2.89,3.4,;3.66,2.07,;5.2,2.07,;-2.01,1.3,;-3.5,1.7,;-4.59,.61,;-4.19,-.88,;-5.28,-1.97,;-4.88,-3.46,;-5.97,-4.55,;-3.39,-3.85,;-2.31,-2.77,;-2.7,-1.28,;-1.62,-.19,)|
COc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc2CCN(C)Cc2c1 |(.24,-2.87,;1.01,-1.54,;2.55,-1.54,;3.32,-2.87,;4.86,-2.87,;5.63,-1.54,;4.86,-.2,;5.63,1.13,;3.32,-.2,;2.55,1.13,;1.01,1.13,;.24,2.47,;-1.27,2.79,;-1.43,4.32,;-.02,4.94,;1.01,3.8,;2.55,3.8,;3.32,2.47,;4.86,2.47,;-2.36,1.7,;-3.85,2.1,;-4.94,1.01,;-4.54,-.48,;-5.63,-1.57,;-5.23,-3.06,;-3.74,-3.46,;-3.34,-4.94,;-2.65,-2.37,;-3.05,-.88,;-1.96,.21,)|
COc1cc(cc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc(cc1)N1CCN(C)CC1)C#N |(1.48,-2.57,;2.25,-1.24,;3.79,-1.24,;4.56,-2.57,;6.13,-2.62,;6.87,-1.24,;6.1,.09,;6.87,1.43,;4.56,.09,;3.79,1.43,;2.25,1.43,;1.48,2.76,;-.02,3.08,;-.18,4.61,;1.22,5.24,;2.25,4.1,;3.79,4.1,;4.56,2.76,;6.1,2.76,;-1.11,1.99,;-2.6,2.39,;-3.69,1.3,;-3.29,-.18,;-1.8,-.58,;-.71,.51,;-4.38,-1.27,;-5.87,-.88,;-6.95,-1.96,;-6.56,-3.45,;-7.64,-4.54,;-5.07,-3.85,;-3.98,-2.76,;6.9,-3.95,;7.67,-5.29,)|
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2cc(=O)n(nc12)-c1cccc2COCc12
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2cc(=O)n(nc12)-c1cccc2OCOc12
COc1cc(F)cc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc(cc1)N1CCN(C)CC1 |(1.87,-2.92,;2.64,-1.59,;4.18,-1.59,;4.95,-2.92,;6.49,-2.92,;7.26,-4.26,;7.26,-1.59,;6.49,-.26,;7.26,1.08,;4.95,-.26,;4.18,1.08,;2.64,1.08,;1.87,2.41,;.36,2.73,;.2,4.26,;1.61,4.89,;2.64,3.75,;4.18,3.75,;4.95,2.41,;6.49,2.41,;-.73,1.64,;-2.21,2.04,;-3.3,.95,;-2.9,-.53,;-1.42,-.93,;-.33,.16,;-3.99,-1.62,;-5.48,-1.22,;-6.57,-2.31,;-6.17,-3.8,;-7.26,-4.89,;-4.68,-4.2,;-3.59,-3.11,)|
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2cc(=O)n(nc12)-c1c(C)cc(Cl)cc1F |(-7.26,-4.89,;-6.17,-3.8,;-6.57,-2.31,;-5.48,-1.22,;-3.99,-1.62,;-3.59,-3.11,;-4.68,-4.2,;-2.9,-.53,;-3.3,.95,;-2.21,2.04,;-.73,1.64,;-.33,.16,;-1.42,-.93,;.36,2.73,;.2,4.26,;1.61,4.89,;2.64,3.75,;4.18,3.75,;4.95,2.41,;6.49,2.41,;4.18,1.08,;2.64,1.08,;1.87,2.41,;4.95,-.26,;4.18,-1.59,;2.64,-1.59,;4.95,-2.92,;6.49,-2.92,;7.26,-4.26,;7.26,-1.59,;6.49,-.26,;7.26,1.08,)|
CNC(=O)c1cc(F)c(c(OC)c1)-n1nc2c(n[nH]c2cc1=O)-c1ccc(cc1)N1CCN(C)CC1 |(8.41,-5.24,;7.64,-3.91,;6.1,-3.91,;5.33,-5.24,;5.33,-2.57,;6.1,-1.24,;5.33,.09,;6.1,1.43,;3.79,.09,;3.02,-1.24,;1.48,-1.24,;.71,-2.57,;3.79,-2.57,;3.02,1.43,;1.48,1.43,;.71,2.76,;-.79,3.08,;-.95,4.61,;.45,5.24,;1.48,4.1,;3.02,4.1,;3.79,2.76,;5.33,2.76,;-1.88,1.99,;-3.37,2.39,;-4.46,1.3,;-4.06,-.18,;-2.57,-.58,;-1.48,.51,;-5.15,-1.27,;-6.64,-.88,;-7.72,-1.96,;-7.33,-3.45,;-8.41,-4.54,;-5.84,-3.85,;-4.75,-2.76,)|
COc1cc(cc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc(cc1)N1CCN(C)CC1)C(=O)N(C)C |(.71,-2.57,;1.48,-1.24,;3.02,-1.24,;3.79,-2.57,;5.33,-2.57,;6.1,-1.24,;5.33,.09,;6.1,1.43,;3.79,.09,;3.02,1.43,;1.48,1.43,;.71,2.76,;-.79,3.08,;-.95,4.61,;.45,5.24,;1.48,4.1,;3.02,4.1,;3.79,2.76,;5.33,2.76,;-1.88,1.99,;-3.37,2.39,;-4.46,1.3,;-4.06,-.18,;-2.57,-.58,;-1.48,.51,;-5.15,-1.27,;-6.64,-.88,;-7.72,-1.96,;-7.33,-3.45,;-8.41,-4.54,;-5.84,-3.85,;-4.75,-2.76,;6.1,-3.91,;5.33,-5.24,;7.64,-3.91,;8.41,-5.24,;8.41,-2.57,)|
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2cc(=O)n(nc12)-c1c(C)cccc1F |(-6.52,-4.15,;-5.43,-3.06,;-5.83,-1.57,;-4.74,-.48,;-3.25,-.88,;-2.85,-2.37,;-3.94,-3.46,;-2.16,.21,;-2.56,1.7,;-1.47,2.79,;.02,2.39,;.42,.9,;-.67,-.19,;1.11,3.48,;.95,5.01,;2.35,5.63,;3.38,4.49,;4.92,4.49,;5.69,3.16,;7.23,3.16,;4.92,1.82,;3.38,1.82,;2.61,3.16,;5.69,.49,;4.92,-.85,;3.38,-.85,;5.69,-2.18,;7.23,-2.18,;8,-.85,;7.23,.49,;8,1.82,)|
C[C@H](N)C(=O)N1CCN(CC1)c1ccc(cc1)-c1n[nH]c2cc(=O)n(nc12)-c1c(C)cc(cc1F)C#C |r,wD:1.1,(-5.01,-5.49,;-6.5,-5.09,;-7.59,-6.18,;-6.9,-3.6,;-8.39,-3.2,;-5.81,-2.51,;-6.21,-1.03,;-5.12,.06,;-3.63,-.34,;-3.24,-1.82,;-4.32,-2.91,;-2.55,.75,;-2.94,2.24,;-1.85,3.33,;-.37,2.93,;.03,1.44,;-1.06,.36,;.72,4.02,;.56,5.55,;1.97,6.18,;3,5.03,;4.54,5.03,;5.31,3.7,;6.85,3.7,;4.54,2.37,;3,2.37,;2.23,3.7,;5.31,1.03,;4.54,-.3,;3,-.3,;5.31,-1.63,;6.85,-1.63,;7.62,-.3,;6.85,1.03,;7.62,2.37,;7.62,-2.97,;8.39,-4.3,)|
CC(O)C(=O)N1CCN(CC1)c1ccc(cc1)-c1n[nH]c2cc(=O)n(nc12)-c1c(C)cc(cc1F)C#C |w:1.0,(-5.01,-5.49,;-6.5,-5.09,;-7.59,-6.18,;-6.9,-3.6,;-8.39,-3.2,;-5.81,-2.51,;-6.21,-1.03,;-5.12,.06,;-3.63,-.34,;-3.24,-1.82,;-4.32,-2.91,;-2.54,.75,;-2.94,2.24,;-1.85,3.33,;-.37,2.93,;.03,1.44,;-1.06,.36,;.72,4.02,;.56,5.55,;1.97,6.18,;3,5.03,;4.54,5.03,;5.31,3.7,;6.85,3.7,;4.54,2.37,;3,2.37,;2.23,3.7,;5.31,1.03,;4.54,-.3,;3,-.3,;5.31,-1.63,;6.85,-1.63,;7.62,-.3,;6.85,1.03,;7.62,2.37,;7.62,-2.97,;8.39,-4.3,)|
Cc1cccc(C)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc(cc1)N1CCN(CC(F)F)CC1 |(8.72,-1.6,;7.39,-2.37,;7.39,-3.91,;6.05,-4.68,;4.72,-3.91,;4.72,-2.37,;3.39,-1.6,;6.05,-1.6,;6.05,-.06,;4.72,.71,;4.72,2.25,;3.58,3.28,;4.2,4.68,;5.73,4.52,;6.05,3.02,;7.39,2.25,;7.39,.71,;8.72,-.06,;2.09,2.88,;1,3.97,;-.49,3.57,;-.89,2.08,;.2,.99,;1.69,1.39,;-2.37,1.68,;-3.46,2.77,;-4.95,2.37,;-5.35,.89,;-6.84,.49,;-7.23,-1,;-6.15,-2.09,;-8.72,-1.4,;-4.26,-.2,;-2.77,.2,)|
Cc1cc(cc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc(cc1)N1CCN(CC1)C1CCOC1)C#N |(3.36,-.48,;4.9,-.48,;5.67,-1.81,;7.21,-1.81,;7.98,-.48,;7.21,.85,;7.98,2.19,;5.67,.85,;4.9,2.19,;3.36,2.19,;2.59,3.52,;1.09,3.84,;.93,5.37,;2.33,6,;3.36,4.86,;4.9,4.86,;5.67,3.52,;7.21,3.52,;-0,2.75,;-1.49,3.15,;-2.58,2.06,;-2.18,.58,;-.69,.18,;.4,1.27,;-3.27,-.51,;-4.75,-.11,;-5.84,-1.2,;-5.45,-2.69,;-3.96,-3.09,;-2.87,-2,;-6.53,-3.78,;-8.06,-3.54,;-8.75,-4.91,;-7.67,-6,;-6.29,-5.3,;7.98,-3.15,;8.75,-4.48,)|
COc1cc(cc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc(cc1)N1CCN(CC1)C1COC1)C#N |(2.25,-2.15,;3.02,-.82,;4.56,-.82,;5.33,-2.15,;6.9,-2.2,;7.64,-.82,;6.87,.51,;7.64,1.85,;5.33,.51,;4.56,1.85,;3.02,1.85,;2.25,3.18,;.75,3.5,;.59,5.03,;1.99,5.66,;3.02,4.52,;4.56,4.52,;5.33,3.18,;6.87,3.18,;-.34,2.41,;-1.83,2.81,;-2.92,1.72,;-2.52,.24,;-1.03,-.16,;.06,.93,;-3.61,-.85,;-5.1,-.45,;-6.18,-1.54,;-5.79,-3.03,;-4.3,-3.43,;-3.21,-2.34,;-6.87,-4.12,;-8.41,-4.12,;-8.41,-5.66,;-6.87,-5.66,;7.67,-3.53,;8.44,-4.87,)|
CN1C[C@@H]2C[C@H]1CN2c1ccc(cc1)-c1n[nH]c2cc(=O)n(nc12)-c1c(C)cccc1C |r,wU:5.4,3.3,(-7.78,.49,;-6.29,.89,;-5.2,-.2,;-3.72,.19,;-4.56,1.6,;-5.89,2.37,;-4.41,2.77,;-3.32,1.68,;-1.83,2.08,;-1.43,3.57,;.06,3.97,;1.15,2.88,;.75,1.39,;-.74,.99,;2.63,3.28,;3.26,4.68,;4.79,4.52,;5.11,3.02,;6.45,2.25,;6.45,.71,;7.78,-.06,;5.11,-.06,;3.78,.71,;3.78,2.25,;5.11,-1.6,;6.45,-2.37,;7.78,-1.6,;6.45,-3.91,;5.11,-4.68,;3.78,-3.91,;3.78,-2.37,;2.44,-1.6,)|
CN1C[C@H]2C[C@@H]1CN2c1ccc(cc1)-c1n[nH]c2cc(=O)n(nc12)-c1c(C)cccc1F |r,wD:5.4,3.3,(-7.78,.49,;-6.29,.89,;-5.2,-.2,;-3.72,.19,;-4.56,1.6,;-5.89,2.37,;-4.41,2.77,;-3.32,1.68,;-1.83,2.08,;-1.43,3.57,;.06,3.97,;1.15,2.88,;.75,1.39,;-.74,.99,;2.63,3.28,;3.26,4.68,;4.79,4.52,;5.11,3.02,;6.45,2.25,;6.45,.71,;7.78,-.06,;5.11,-.06,;3.78,.71,;3.78,2.25,;5.11,-1.6,;3.78,-2.37,;2.44,-1.6,;3.78,-3.91,;5.11,-4.68,;6.45,-3.91,;6.45,-2.37,;7.78,-1.6,)|
CN1CCN(CC1(C)C)c1ccc(cc1)-c1n[nH]c2cc(=O)n(nc12)-c1c(C)cccc1F |(-7.78,.49,;-6.29,.89,;-5.2,-.2,;-3.72,.19,;-3.32,1.68,;-4.41,2.77,;-5.89,2.37,;-5.49,3.86,;-7.38,2.77,;-1.83,2.08,;-1.43,3.57,;.06,3.97,;1.15,2.88,;.75,1.39,;-.74,.99,;2.63,3.28,;3.26,4.68,;4.79,4.52,;5.11,3.02,;6.45,2.25,;6.45,.71,;7.78,-.06,;5.11,-.06,;3.78,.71,;3.78,2.25,;5.11,-1.6,;3.78,-2.37,;2.44,-1.6,;3.78,-3.91,;5.11,-4.68,;6.45,-3.91,;6.45,-2.37,;7.78,-1.6,)|
C[C@H]1CN(C[C@@H](C)N1C)c1ccc(cc1)-c1n[nH]c2cc(=O)n(nc12)-c1c(C)cccc1F |r,wU:1.0,5.5,(-6.98,3.46,;-5.89,2.37,;-4.41,2.77,;-3.32,1.68,;-3.72,.19,;-5.2,-.2,;-5.6,-1.69,;-6.29,.89,;-7.78,.49,;-1.83,2.08,;-1.43,3.57,;.06,3.97,;1.15,2.88,;.75,1.39,;-.74,.99,;2.63,3.28,;3.26,4.68,;4.79,4.52,;5.11,3.02,;6.45,2.25,;6.45,.71,;7.78,-.06,;5.11,-.06,;3.78,.71,;3.78,2.25,;5.11,-1.6,;3.78,-2.37,;2.44,-1.6,;3.78,-3.91,;5.11,-4.68,;6.45,-3.91,;6.45,-2.37,;7.78,-1.6,)|
CN1C2CC1CN(C2)c1ccc(cc1)-c1n[nH]c2cc(=O)n(nc12)-c1c(C)cccc1F |(-7.78,.49,;-6.29,.89,;-5.89,2.37,;-4.56,1.6,;-5.2,-.2,;-3.72,.19,;-3.32,1.68,;-4.41,2.77,;-1.83,2.08,;-1.43,3.57,;.06,3.97,;1.15,2.88,;.75,1.39,;-.74,.99,;2.63,3.28,;3.26,4.68,;4.79,4.52,;5.11,3.02,;6.45,2.25,;6.45,.71,;7.78,-.06,;5.11,-.06,;3.78,.71,;3.78,2.25,;5.11,-1.6,;3.78,-2.37,;2.44,-1.6,;3.78,-3.91,;5.11,-4.68,;6.45,-3.91,;6.45,-2.37,;7.78,-1.6,)|
COc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc(cc1)N1CCOCC1 |(1.52,-3.27,;2.29,-1.93,;3.83,-1.93,;4.6,-3.27,;6.14,-3.27,;6.91,-1.93,;6.14,-.6,;6.91,.73,;4.6,-.6,;3.83,.73,;2.29,.73,;1.52,2.07,;.02,2.39,;-.14,3.92,;1.26,4.55,;2.29,3.4,;3.83,3.4,;4.6,2.07,;6.14,2.07,;-1.07,1.3,;-2.56,1.7,;-3.65,.61,;-3.25,-.88,;-1.76,-1.28,;-.67,-.19,;-4.34,-1.97,;-5.83,-1.57,;-6.91,-2.66,;-6.52,-4.15,;-5.03,-4.55,;-3.94,-3.46,)|
Cc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc(OCC2CNCCN2)cc1 |(2.64,-1.6,;3.98,-2.37,;3.98,-3.91,;5.31,-4.68,;6.64,-3.91,;6.64,-2.37,;7.98,-1.6,;5.31,-1.6,;5.31,-.06,;3.98,.71,;3.98,2.25,;2.83,3.28,;3.46,4.68,;4.99,4.52,;5.31,3.02,;6.64,2.25,;6.64,.71,;7.98,-.06,;1.35,2.88,;.26,3.97,;-1.23,3.57,;-1.63,2.08,;-3.12,1.68,;-3.52,.19,;-5,-.2,;-6.09,.89,;-7.58,.49,;-7.98,-1,;-6.89,-2.09,;-5.4,-1.69,;-.54,.99,;.95,1.39,)|
CN1CCN(CC1)c1ccc(cc1F)-c1n[nH]c2cc(=O)n(nc12)-c1c(C)cccc1F |(-7.26,-4.89,;-6.17,-3.8,;-6.57,-2.31,;-5.48,-1.22,;-3.99,-1.62,;-3.59,-3.11,;-4.68,-4.2,;-2.9,-.53,;-3.3,.95,;-2.21,2.04,;-.73,1.64,;-.33,.16,;-1.42,-.93,;-1.02,-2.42,;.36,2.73,;.2,4.26,;1.61,4.89,;2.64,3.75,;4.18,3.75,;4.95,2.41,;6.49,2.41,;4.18,1.08,;2.64,1.08,;1.87,2.41,;4.95,-.26,;4.18,-1.59,;2.64,-1.59,;4.95,-2.92,;6.49,-2.92,;7.26,-1.59,;6.49,-.26,;7.26,1.08,)|
CN(C)Cc1cc(ccc1N1CCN(C)CC1)-c1n[nH]c2cc(=O)n(nc12)-c1c(C)cccc1F |(1.56,-1.73,;.47,-2.82,;.87,-4.31,;-1.02,-2.42,;-1.42,-.93,;-.33,.16,;-.73,1.64,;-2.21,2.04,;-3.3,.95,;-2.9,-.53,;-3.99,-1.62,;-5.48,-1.22,;-6.57,-2.31,;-6.17,-3.8,;-7.26,-4.89,;-4.68,-4.2,;-3.59,-3.11,;.36,2.73,;.2,4.26,;1.61,4.89,;2.64,3.75,;4.18,3.75,;4.95,2.41,;6.49,2.41,;4.18,1.08,;2.64,1.08,;1.87,2.41,;4.95,-.26,;4.18,-1.59,;2.64,-1.59,;4.95,-2.92,;6.49,-2.92,;7.26,-1.59,;6.49,-.26,;7.26,1.08,)|
CNCc1cc(ccc1N1CCN(C)CC1)-c1n[nH]c2cc(=O)n(nc12)-c1c(C)cccc1F |(.87,-4.31,;.47,-2.82,;-1.02,-2.42,;-1.42,-.93,;-.33,.16,;-.73,1.64,;-2.21,2.04,;-3.3,.95,;-2.9,-.53,;-3.99,-1.62,;-5.48,-1.22,;-6.57,-2.31,;-6.17,-3.8,;-7.26,-4.89,;-4.68,-4.2,;-3.59,-3.11,;.36,2.73,;.2,4.26,;1.61,4.89,;2.64,3.75,;4.18,3.75,;4.95,2.41,;6.49,2.41,;4.18,1.08,;2.64,1.08,;1.87,2.41,;4.95,-.26,;4.18,-1.59,;2.64,-1.59,;4.95,-2.92,;6.49,-2.92,;7.26,-1.59,;6.49,-.26,;7.26,1.08,)|
COc1cccc(C)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc(nc1)N1CCN(C)CC1 |(1.87,-2.92,;2.64,-1.59,;4.18,-1.59,;4.95,-2.92,;6.49,-2.92,;7.26,-1.59,;6.49,-.26,;7.26,1.08,;4.95,-.26,;4.18,1.08,;2.64,1.08,;1.87,2.41,;.36,2.73,;.2,4.26,;1.61,4.89,;2.64,3.75,;4.18,3.75,;4.95,2.41,;6.49,2.41,;-.73,1.64,;-.33,.16,;-1.42,-.93,;-2.9,-.53,;-3.3,.95,;-2.21,2.04,;-3.99,-1.62,;-5.48,-1.22,;-6.57,-2.31,;-6.17,-3.8,;-7.26,-4.89,;-4.68,-4.2,;-3.59,-3.11,)|
CCc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc(nc1)N1CCN(C)CC1 |(1.87,-2.92,;2.64,-1.59,;4.18,-1.59,;4.95,-2.92,;6.49,-2.92,;7.26,-1.59,;6.49,-.26,;7.26,1.08,;4.95,-.26,;4.18,1.08,;2.64,1.08,;1.87,2.41,;.36,2.73,;.2,4.26,;1.61,4.89,;2.64,3.75,;4.18,3.75,;4.95,2.41,;6.49,2.41,;-.73,1.64,;-2.21,2.04,;-3.3,.95,;-2.9,-.53,;-1.42,-.93,;-.33,.16,;-3.99,-1.62,;-5.48,-1.22,;-6.57,-2.31,;-6.17,-3.8,;-7.26,-4.89,;-4.68,-4.2,;-3.59,-3.11,)|
CN1CCN(CC1)c1ccc(cn1)-c1n[nH]c2cc(=O)n(nc12)-c1c(C)cc(cc1F)C#N |(-7.64,-4.54,;-6.56,-3.45,;-6.95,-1.96,;-5.87,-.88,;-4.38,-1.27,;-3.98,-2.76,;-5.07,-3.85,;-3.29,-.18,;-1.8,-.58,;-.71,.51,;-1.11,1.99,;-2.6,2.39,;-3.69,1.3,;-.02,3.08,;-.18,4.61,;1.22,5.24,;2.25,4.1,;3.79,4.1,;4.56,2.76,;6.1,2.76,;3.79,1.43,;2.25,1.43,;1.48,2.76,;4.56,.09,;3.79,-1.24,;2.25,-1.24,;4.56,-2.57,;6.13,-2.62,;6.87,-1.24,;6.1,.09,;6.87,1.43,;6.9,-3.95,;7.67,-5.29,)|
CN1CCN(CC1)c1ccc(cn1)-c1n[nH]c2cc(=O)n(nc12)-c1c(O)cccc1F |(-7.26,-4.89,;-6.17,-3.8,;-6.57,-2.31,;-5.48,-1.22,;-3.99,-1.62,;-3.59,-3.11,;-4.68,-4.2,;-2.9,-.53,;-3.3,.95,;-2.21,2.04,;-.73,1.64,;-.33,.16,;-1.42,-.93,;.36,2.73,;.2,4.26,;1.61,4.89,;2.64,3.75,;4.18,3.75,;4.95,2.41,;6.49,2.41,;4.18,1.08,;2.64,1.08,;1.87,2.41,;4.95,-.26,;4.18,-1.59,;2.64,-1.59,;4.95,-2.92,;6.49,-2.92,;7.26,-1.59,;6.49,-.26,;7.26,1.08,)|
CCN1CCN(CC1)c1ccc(cn1)-c1n[nH]c2cc(=O)n(nc12)-c1c(C)cccc1F |(-8,-4.49,;-6.52,-4.89,;-5.43,-3.8,;-5.83,-2.31,;-4.74,-1.22,;-3.25,-1.62,;-2.85,-3.11,;-3.94,-4.2,;-2.16,-.53,;-2.56,.95,;-1.47,2.04,;.02,1.64,;.42,.16,;-.67,-.93,;1.11,2.73,;.95,4.26,;2.35,4.89,;3.38,3.75,;4.92,3.75,;5.69,2.41,;7.23,2.41,;4.92,1.08,;3.38,1.08,;2.61,2.41,;5.69,-.26,;4.92,-1.59,;3.38,-1.59,;5.69,-2.92,;7.23,-2.92,;8,-1.59,;7.23,-.26,;8,1.08,)|
CC(=O)N1CCN(CC1)c1ccc(cn1)-c1n[nH]c2cc(=O)n(nc12)-c1c(C)cccc1F |(-6.12,-5.63,;-6.52,-4.15,;-8,-3.75,;-5.43,-3.06,;-5.83,-1.57,;-4.74,-.48,;-3.25,-.88,;-2.85,-2.37,;-3.94,-3.46,;-2.16,.21,;-2.56,1.7,;-1.47,2.79,;.02,2.39,;.42,.9,;-.67,-.19,;1.11,3.48,;.95,5.01,;2.35,5.63,;3.38,4.49,;4.92,4.49,;5.69,3.16,;7.23,3.16,;4.92,1.82,;3.38,1.82,;2.61,3.16,;5.69,.49,;4.92,-.85,;3.38,-.85,;5.69,-2.18,;7.23,-2.18,;8,-.85,;7.23,.49,;8,1.82,)|
Cc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc(nc1)N1CCN(CC1)C1COC1 |(3.41,-.82,;4.95,-.82,;5.72,-2.15,;7.26,-2.15,;8.03,-.82,;7.26,.51,;8.03,1.85,;5.72,.51,;4.95,1.85,;3.41,1.85,;2.64,3.18,;1.13,3.5,;.97,5.03,;2.38,5.66,;3.41,4.52,;4.95,4.52,;5.72,3.18,;7.26,3.18,;.04,2.41,;-1.44,2.81,;-2.53,1.72,;-2.13,.24,;-.65,-.16,;.44,.93,;-3.22,-.85,;-4.71,-.45,;-5.8,-1.54,;-5.4,-3.03,;-3.91,-3.43,;-2.82,-2.34,;-6.49,-4.12,;-8.03,-4.12,;-8.03,-5.66,;-6.49,-5.66,)|
Cc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc(nc1)N1CCS(=O)(=O)CC1 |(2.29,-1.93,;3.83,-1.93,;4.6,-3.27,;6.14,-3.27,;6.91,-1.93,;6.14,-.6,;6.91,.73,;4.6,-.6,;3.83,.73,;2.29,.73,;1.52,2.07,;.02,2.39,;-.14,3.92,;1.26,4.55,;2.29,3.4,;3.83,3.4,;4.6,2.07,;6.14,2.07,;-1.07,1.3,;-2.56,1.7,;-3.65,.61,;-3.25,-.88,;-1.76,-1.28,;-.67,-.19,;-4.34,-1.97,;-5.83,-1.57,;-6.91,-2.66,;-6.52,-4.15,;-6.91,-5.63,;-5.43,-5.24,;-5.03,-4.55,;-3.94,-3.46,)|
CCS(=O)(=O)N1CCN(CC1)c1ccc(cn1)-c1n[nH]c2cc(=O)n(nc12)-c1c(C)cccc1F |(-5.24,8.93,;-3.73,8.61,;-3.25,7.14,;-1.79,7.62,;-4.72,6.66,;-2.78,5.68,;-3.81,4.53,;-3.33,3.07,;-1.83,2.75,;-.8,3.89,;-1.27,5.36,;-1.35,1.28,;-2.38,.14,;-1.9,-1.33,;-.4,-1.65,;.63,-.5,;.16,.96,;.08,-3.11,;-.83,-4.36,;.08,-5.6,;1.54,-5.13,;2.88,-5.9,;4.21,-5.13,;5.54,-5.9,;4.21,-3.59,;2.88,-2.82,;1.54,-3.59,;5.54,-2.82,;5.54,-1.28,;4.21,-.51,;6.88,-.51,;8.21,-1.28,;8.21,-2.82,;6.88,-3.59,;6.88,-5.13,)|
Cc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc(nc1)N1CCN(CC1)C1CCOC1 |(3.68,-1.6,;5.01,-2.37,;5.01,-3.91,;6.35,-4.68,;7.68,-3.91,;7.68,-2.37,;9.02,-1.6,;6.35,-1.6,;6.35,-.06,;5.01,.71,;5.01,2.25,;3.87,3.28,;4.5,4.68,;6.03,4.52,;6.35,3.02,;7.68,2.25,;7.68,.71,;9.02,-.06,;2.38,2.88,;1.29,3.97,;-.19,3.57,;-.59,2.08,;.5,.99,;1.98,1.39,;-2.08,1.68,;-3.17,2.77,;-4.66,2.37,;-5.05,.89,;-3.97,-.2,;-2.48,.19,;-6.54,.49,;-7.67,1.54,;-9.02,.79,;-8.72,-.72,;-7.19,-.91,)|
CN1CCN(CC1)c1ccc(cn1)-c1n[nH]c2cc(=O)n(nc12)-c1c(F)cccc1Cl |(-7.26,-4.89,;-6.17,-3.8,;-6.57,-2.31,;-5.48,-1.22,;-3.99,-1.62,;-3.59,-3.11,;-4.68,-4.2,;-2.9,-.53,;-3.3,.95,;-2.21,2.04,;-.73,1.64,;-.33,.16,;-1.42,-.93,;.36,2.73,;.2,4.26,;1.61,4.89,;2.64,3.75,;4.18,3.75,;4.95,2.41,;6.49,2.41,;4.18,1.08,;2.64,1.08,;1.87,2.41,;4.95,-.26,;6.49,-.26,;7.26,1.08,;7.26,-1.59,;6.49,-2.92,;4.95,-2.92,;4.18,-1.59,;2.64,-1.59,)|
CN1CCN(CC1)c1ccc(cn1)-c1n[nH]c2cc(=O)n(nc12)-c1c(C)cc(Cl)cc1F |(-7.26,-4.89,;-6.17,-3.8,;-6.57,-2.31,;-5.48,-1.22,;-3.99,-1.62,;-3.59,-3.11,;-4.68,-4.2,;-2.9,-.53,;-1.42,-.93,;-.33,.16,;-.73,1.64,;-2.21,2.04,;-3.3,.95,;.36,2.73,;.2,4.26,;1.61,4.89,;2.64,3.75,;4.18,3.75,;4.95,2.41,;6.49,2.41,;4.18,1.08,;2.64,1.08,;1.87,2.41,;4.95,-.26,;4.18,-1.59,;2.64,-1.59,;4.95,-2.92,;6.49,-2.92,;7.26,-4.26,;7.26,-1.59,;6.49,-.26,;7.26,1.08,)|
CN1C2CCC1CN(C2)c1ccc(cn1)-c1n[nH]c2cc(=O)n(nc12)-c1c(C)cccc1F |(-7.26,-4.89,;-6.17,-3.8,;-6.57,-2.31,;-5.34,-1.98,;-4.36,-3,;-4.68,-4.2,;-3.59,-3.11,;-3.99,-1.62,;-5.48,-1.22,;-2.9,-.53,;-3.3,.95,;-2.21,2.04,;-.73,1.64,;-.33,.16,;-1.42,-.93,;.36,2.73,;.2,4.26,;1.61,4.89,;2.64,3.75,;4.18,3.75,;4.95,2.41,;6.49,2.41,;4.18,1.08,;2.64,1.08,;1.87,2.41,;4.95,-.26,;4.18,-1.59,;2.64,-1.59,;4.95,-2.92,;6.49,-2.92,;7.26,-1.59,;6.49,-.26,;7.26,1.08,)|
CCc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1cnc(nc1)N1CCN(C)CC1 |(1.87,-2.92,;2.64,-1.59,;4.18,-1.59,;4.95,-2.92,;6.49,-2.92,;7.26,-1.59,;6.49,-.26,;7.26,1.08,;4.95,-.26,;4.18,1.08,;2.64,1.08,;1.87,2.41,;.36,2.73,;.2,4.26,;1.61,4.89,;2.64,3.75,;4.18,3.75,;4.95,2.41,;6.49,2.41,;-.73,1.64,;-2.21,2.04,;-3.3,.95,;-2.9,-.53,;-1.42,-.93,;-.33,.16,;-3.99,-1.62,;-5.48,-1.22,;-6.57,-2.31,;-6.17,-3.8,;-7.26,-4.89,;-4.68,-4.2,;-3.59,-3.11,)|
COc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1cnc(nc1)N1CCOCC1 |(1.52,-3.27,;2.29,-1.93,;3.83,-1.93,;4.6,-3.27,;6.14,-3.27,;6.91,-1.93,;6.14,-.6,;6.91,.73,;4.6,-.6,;3.83,.73,;2.29,.73,;1.52,2.07,;.02,2.39,;-.14,3.92,;1.26,4.55,;2.29,3.4,;3.83,3.4,;4.6,2.07,;6.14,2.07,;-1.07,1.3,;-2.56,1.7,;-3.65,.61,;-3.25,-.88,;-1.76,-1.28,;-.67,-.19,;-4.34,-1.97,;-5.83,-1.57,;-6.91,-2.66,;-6.52,-4.15,;-5.03,-4.55,;-3.94,-3.46,)|
CCc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc(cc1)N1CCN(CCO)CC1 |(2.81,-2.92,;3.58,-1.59,;5.12,-1.59,;5.89,-2.92,;7.43,-2.92,;8.2,-1.59,;7.43,-.26,;8.2,1.08,;5.89,-.26,;5.12,1.08,;3.58,1.08,;2.81,2.41,;1.31,2.73,;1.15,4.26,;2.55,4.89,;3.58,3.75,;5.12,3.75,;5.89,2.41,;7.43,2.41,;.22,1.64,;-1.27,2.04,;-2.36,.95,;-1.96,-.53,;-.47,-.93,;.62,.16,;-3.05,-1.62,;-4.54,-1.22,;-5.63,-2.31,;-5.23,-3.8,;-6.32,-4.89,;-7.8,-4.49,;-8.2,-3,;-3.74,-4.2,;-2.65,-3.11,)|
COc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc(cc1)N1CCN(CCO)CC1 |(2.81,-2.92,;3.58,-1.59,;5.12,-1.59,;5.89,-2.92,;7.43,-2.92,;8.2,-1.59,;7.43,-.26,;8.2,1.08,;5.89,-.26,;5.12,1.08,;3.58,1.08,;2.81,2.41,;1.31,2.73,;1.15,4.26,;2.55,4.89,;3.58,3.75,;5.12,3.75,;5.89,2.41,;7.43,2.41,;.22,1.64,;-1.27,2.04,;-2.36,.95,;-1.96,-.53,;-.47,-.93,;.62,.16,;-3.05,-1.62,;-4.54,-1.22,;-5.63,-2.31,;-5.23,-3.8,;-6.32,-4.89,;-7.8,-4.49,;-8.2,-3,;-3.74,-4.2,;-2.65,-3.11,)|
COc1cc(cc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc(cc1)N1CCN(CCO)CC1)C#N |(2.43,-2.57,;3.2,-1.24,;4.74,-1.24,;5.51,-2.57,;7.08,-2.62,;7.82,-1.24,;7.05,.09,;7.82,1.43,;5.51,.09,;4.74,1.43,;3.2,1.43,;2.43,2.76,;.92,3.08,;.76,4.61,;2.17,5.24,;3.2,4.1,;4.74,4.1,;5.51,2.76,;7.05,2.76,;-.17,1.99,;-1.66,2.39,;-2.74,1.3,;-2.35,-.18,;-.86,-.58,;.23,.51,;-3.43,-1.27,;-4.92,-.88,;-6.01,-1.96,;-5.61,-3.45,;-6.7,-4.54,;-8.19,-4.14,;-8.59,-2.65,;-4.12,-3.85,;-3.04,-2.76,;7.85,-3.95,;8.62,-5.29,)|
COc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc(cc1)N1CCN(CC(C)(C)O)CC1 |(3.36,-2.58,;4.13,-1.24,;5.67,-1.24,;6.44,-2.58,;7.98,-2.58,;8.75,-1.24,;7.98,.09,;8.75,1.42,;6.44,.09,;5.67,1.42,;4.13,1.42,;3.36,2.76,;1.85,3.08,;1.69,4.61,;3.1,5.24,;4.13,4.09,;5.67,4.09,;6.44,2.76,;7.98,2.76,;.76,1.99,;-.73,2.39,;-1.81,1.3,;-1.42,-.19,;.07,-.59,;1.16,.5,;-2.51,-1.28,;-3.99,-.88,;-5.08,-1.97,;-4.68,-3.46,;-5.77,-4.54,;-7.26,-4.15,;-8.35,-5.24,;-7.66,-2.66,;-8.75,-3.75,;-3.2,-3.85,;-2.11,-2.77,)|
CCc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc(cc1)N1CCN(CC(C)(C)O)CC1 |(3.36,-2.58,;4.13,-1.24,;5.67,-1.24,;6.44,-2.58,;7.98,-2.58,;8.75,-1.24,;7.98,.09,;8.75,1.42,;6.44,.09,;5.67,1.42,;4.13,1.42,;3.36,2.76,;1.85,3.08,;1.69,4.61,;3.1,5.24,;4.13,4.09,;5.67,4.09,;6.44,2.76,;7.98,2.76,;.76,1.99,;-.73,2.39,;-1.81,1.3,;-1.42,-.19,;.07,-.59,;1.16,.5,;-2.51,-1.28,;-3.99,-.88,;-5.08,-1.97,;-4.68,-3.46,;-5.77,-4.54,;-7.26,-4.15,;-8.35,-5.24,;-7.66,-2.66,;-8.75,-3.75,;-3.2,-3.85,;-2.11,-2.77,)|
Cc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc(cc1)N1CC2CCC(C1)N2CCO |(3.58,-1.59,;5.12,-1.59,;5.89,-2.92,;7.43,-2.92,;8.2,-1.59,;7.43,-.26,;8.2,1.08,;5.89,-.26,;5.12,1.08,;3.58,1.08,;2.81,2.41,;1.31,2.73,;1.15,4.26,;2.55,4.89,;3.58,3.75,;5.12,3.75,;5.89,2.41,;7.43,2.41,;.22,1.64,;-1.27,2.04,;-2.36,.95,;-1.96,-.53,;-.47,-.93,;.62,.16,;-3.05,-1.62,;-4.54,-1.22,;-5.63,-2.31,;-4.39,-1.98,;-3.42,-3,;-3.74,-4.2,;-2.65,-3.11,;-5.23,-3.8,;-6.32,-4.89,;-7.8,-4.49,;-8.2,-3,)|
Cc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc(nc1)N1CCN(CCO)CC1 |(3.93,-1.24,;5.47,-1.24,;6.24,-2.58,;7.78,-2.58,;8.55,-1.24,;7.78,.09,;8.55,1.42,;6.24,.09,;5.47,1.42,;3.93,1.42,;3.16,2.76,;1.65,3.08,;1.49,4.61,;2.9,5.24,;3.93,4.09,;5.47,4.09,;6.24,2.76,;7.78,2.76,;.56,1.99,;.96,.5,;-.13,-.59,;-1.62,-.19,;-2.01,1.3,;-.92,2.39,;-2.7,-1.28,;-4.19,-.88,;-5.28,-1.97,;-4.88,-3.46,;-5.97,-4.54,;-7.46,-4.15,;-8.55,-5.24,;-3.39,-3.85,;-2.31,-2.77,)|
COCCN1CCN(CC1)c1ccc(cn1)-c1n[nH]c2cc(=O)n(nc12)-c1c(C)cccc1F |(-9.29,-4.84,;-7.8,-5.24,;-6.71,-4.15,;-5.23,-4.54,;-4.14,-3.46,;-4.54,-1.97,;-3.45,-.88,;-1.96,-1.28,;-1.56,-2.77,;-2.65,-3.85,;-.87,-.19,;.62,-.59,;1.7,.5,;1.31,1.99,;-.18,2.39,;-1.27,1.3,;2.4,3.08,;2.23,4.61,;3.64,5.24,;4.67,4.09,;6.21,4.09,;6.98,2.76,;8.52,2.76,;6.21,1.42,;4.67,1.42,;3.9,2.76,;6.98,.09,;6.21,-1.24,;4.67,-1.24,;6.98,-2.58,;8.52,-2.58,;9.29,-1.24,;8.52,.09,;9.29,1.42,)|
CN1CCN(CC1CO)c1ccc(cc1)-c1n[nH]c2cc(=O)n(nc12)-c1c(C)cccc1F |(-7.43,.49,;-5.95,.89,;-4.86,-.2,;-3.37,.19,;-2.97,1.68,;-4.06,2.77,;-5.55,2.37,;-6.64,3.46,;-8.12,3.06,;-1.48,2.08,;-1.09,3.57,;.4,3.97,;1.49,2.88,;1.09,1.39,;-.39,.99,;2.98,3.28,;3.61,4.68,;5.14,4.52,;5.46,3.02,;6.79,2.25,;6.79,.71,;8.12,-.06,;5.46,-.06,;4.12,.71,;4.12,2.25,;5.46,-1.6,;4.12,-2.37,;2.79,-1.6,;4.12,-3.91,;5.46,-4.68,;6.79,-3.91,;6.79,-2.37,;8.12,-1.6,)|
COc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc(cc1)N1CCN(C)C(CO)C1 |(1.46,-2.37,;2.79,-1.6,;4.12,-2.37,;4.12,-3.91,;5.46,-4.68,;6.79,-3.91,;6.79,-2.37,;8.12,-1.6,;5.46,-1.6,;5.46,-.06,;4.12,.71,;4.12,2.25,;2.98,3.28,;3.61,4.68,;5.14,4.52,;5.46,3.02,;6.79,2.25,;6.79,.71,;8.12,-.06,;1.49,2.88,;.4,3.97,;-1.09,3.57,;-1.48,2.08,;-.39,.99,;1.09,1.39,;-2.97,1.68,;-3.37,.19,;-4.86,-.2,;-5.95,.89,;-7.43,.49,;-5.55,2.37,;-6.64,3.46,;-8.12,3.06,;-4.06,2.77,)|
Cc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc(cc1)N1CCN2C(COC2=O)C1 |(2.89,-1.6,;4.22,-2.37,;4.22,-3.91,;5.56,-4.68,;6.89,-3.91,;6.89,-2.37,;8.22,-1.6,;5.56,-1.6,;5.56,-.06,;4.22,.71,;4.22,2.25,;3.08,3.28,;3.7,4.68,;5.24,4.52,;5.56,3.02,;6.89,2.25,;6.89,.71,;8.22,-.06,;1.59,2.88,;.5,3.97,;-.99,3.57,;-1.38,2.08,;-.3,.99,;1.19,1.39,;-2.87,1.68,;-3.27,.19,;-4.76,-.2,;-5.85,.89,;-5.45,2.37,;-6.74,3.21,;-7.94,2.24,;-7.38,.8,;-8.22,-.49,;-3.96,2.77,)|
COc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc(cc1)N1CCN2C(COC2=O)C1 |(2.57,-2.28,;3.34,-.95,;4.88,-.95,;5.65,-2.28,;7.19,-2.28,;7.96,-.95,;7.19,.39,;7.96,1.72,;5.65,.39,;4.88,1.72,;3.34,1.72,;2.57,3.06,;1.06,3.38,;.9,4.91,;2.31,5.53,;3.34,4.39,;4.88,4.39,;5.65,3.06,;7.19,3.06,;-.03,2.29,;-1.51,2.69,;-2.6,1.6,;-2.2,.11,;-.72,-.29,;.37,.8,;-3.29,-.98,;-2.89,-2.47,;-3.98,-3.56,;-5.47,-3.16,;-5.87,-1.67,;-7.41,-1.59,;-7.96,-3.03,;-6.76,-4,;-6.84,-5.53,;-4.78,-.58,)|
COc1cc(cc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc(cc1)N1CCN2C(COC2=O)C1)C#N |(2.18,-2.28,;2.95,-.95,;4.49,-.95,;5.26,-2.28,;6.83,-2.33,;7.57,-.95,;6.8,.39,;7.57,1.72,;5.26,.39,;4.49,1.72,;2.95,1.72,;2.18,3.06,;.68,3.38,;.52,4.91,;1.92,5.53,;2.95,4.39,;4.49,4.39,;5.26,3.06,;6.8,3.06,;-.41,2.29,;-1.9,2.69,;-2.99,1.6,;-2.59,.11,;-1.1,-.29,;-.01,.8,;-3.68,-.98,;-3.28,-2.47,;-4.37,-3.56,;-5.86,-3.16,;-6.25,-1.67,;-7.79,-1.59,;-8.34,-3.03,;-7.15,-4,;-7.23,-5.53,;-5.17,-.58,;7.6,-3.66,;8.37,-4.99,)|
CN1CCN(CC1C(C)(C)O)c1ccc(cc1)-c1n[nH]c2cc(=O)n(nc12)-c1c(C)cccc1F |(-7.78,.49,;-6.29,.89,;-5.89,2.37,;-4.41,2.77,;-3.32,1.68,;-3.72,.19,;-5.2,-.2,;-5.6,-1.69,;-4.51,-2.78,;-7.09,-2.09,;-6,-3.18,;-1.83,2.08,;-1.43,3.57,;.06,3.97,;1.15,2.88,;.75,1.39,;-.74,.99,;2.63,3.28,;3.26,4.68,;4.79,4.52,;5.11,3.02,;6.45,2.25,;6.45,.71,;7.78,-.06,;5.11,-.06,;3.78,.71,;3.78,2.25,;5.11,-1.6,;3.78,-2.37,;2.44,-1.6,;3.78,-3.91,;5.11,-4.68,;6.45,-3.91,;6.45,-2.37,;7.78,-1.6,)|
COc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc(cc1)N1CCN(C)C(C1)C(C)(C)O |(1.11,-2.37,;2.44,-1.6,;3.78,-2.37,;3.78,-3.91,;5.11,-4.68,;6.45,-3.91,;6.45,-2.37,;7.78,-1.6,;5.11,-1.6,;5.11,-.06,;3.78,.71,;3.78,2.25,;2.63,3.28,;3.26,4.68,;4.79,4.52,;5.11,3.02,;6.45,2.25,;6.45,.71,;7.78,-.06,;1.15,2.88,;.06,3.97,;-1.43,3.57,;-1.83,2.08,;-.74,.99,;.75,1.39,;-3.32,1.68,;-4.41,2.77,;-5.89,2.37,;-6.29,.89,;-7.78,.49,;-5.2,-.2,;-3.72,.19,;-5.6,-1.69,;-4.51,-2.78,;-7.09,-2.09,;-6,-3.18,)|
COc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc(cc1)N1CCN(C)C(C1)C(C)(C)OC |(1.11,-2.37,;2.44,-1.6,;3.78,-2.37,;3.78,-3.91,;5.11,-4.68,;6.45,-3.91,;6.45,-2.37,;7.78,-1.6,;5.11,-1.6,;5.11,-.06,;3.78,.71,;3.78,2.25,;2.63,3.28,;3.26,4.68,;4.79,4.52,;5.11,3.02,;6.45,2.25,;6.45,.71,;7.78,-.06,;1.15,2.88,;.06,3.97,;-1.43,3.57,;-1.83,2.08,;-.74,.99,;.75,1.39,;-3.32,1.68,;-4.41,2.77,;-5.89,2.37,;-6.29,.89,;-7.78,.49,;-5.2,-.2,;-3.72,.19,;-5.6,-1.69,;-4.51,-2.78,;-7.09,-2.09,;-6,-3.18,;-4.91,-4.27,)|
CN1CCN(CC1CO)c1ccc(cn1)-c1n[nH]c2cc(=O)n(nc12)-c1c(C)cccc1F |(-7.43,.49,;-5.95,.89,;-4.86,-.2,;-3.37,.19,;-2.97,1.68,;-4.06,2.77,;-5.55,2.37,;-6.64,3.46,;-8.12,3.06,;-1.48,2.08,;-.39,.99,;1.09,1.39,;1.49,2.88,;.4,3.97,;-1.09,3.57,;2.98,3.28,;3.61,4.68,;5.14,4.52,;5.46,3.02,;6.79,2.25,;6.79,.71,;8.12,-.06,;5.46,-.06,;4.12,.71,;4.12,2.25,;5.46,-1.6,;4.12,-2.37,;2.79,-1.6,;4.12,-3.91,;5.46,-4.68,;6.79,-3.91,;6.79,-2.37,;8.12,-1.6,)|
Cc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc(nc1)N1CCN2C(COC2=O)C1 |(2.89,-1.6,;4.22,-2.37,;4.22,-3.91,;5.56,-4.68,;6.89,-3.91,;6.89,-2.37,;8.22,-1.6,;5.56,-1.6,;5.56,-.06,;4.22,.71,;4.22,2.25,;3.08,3.28,;3.7,4.68,;5.24,4.52,;5.56,3.02,;6.89,2.25,;6.89,.71,;8.22,-.06,;1.59,2.88,;1.19,1.39,;-.3,.99,;-1.38,2.08,;-.99,3.57,;.5,3.97,;-2.87,1.68,;-3.27,.19,;-4.76,-.2,;-5.85,.89,;-5.45,2.37,;-6.74,3.21,;-7.94,2.24,;-7.38,.8,;-8.22,-.49,;-3.96,2.77,)|
CN1CCN(C(CO)C1)c1ccc(cc1)-c1n[nH]c2cc(=O)n(nc12)-c1c(C)cccc1F |(-7.78,.49,;-6.29,.89,;-5.89,2.37,;-4.41,2.77,;-3.32,1.68,;-3.72,.19,;-2.63,-.89,;-3.02,-2.38,;-5.2,-.2,;-1.83,2.08,;-1.43,3.57,;.06,3.97,;1.15,2.88,;.75,1.39,;-.74,.99,;2.63,3.28,;3.26,4.68,;4.79,4.52,;5.11,3.02,;6.45,2.25,;6.45,.71,;7.78,-.06,;5.11,-.06,;3.78,.71,;3.78,2.25,;5.11,-1.6,;3.78,-2.37,;2.44,-1.6,;3.78,-3.91,;5.11,-4.68,;6.45,-3.91,;6.45,-2.37,;7.78,-1.6,)|
CN1CCN(CC1C(O)=O)c1ccc(cc1)-c1n[nH]c2cc(=O)n(nc12)-c1c(C)cccc1F |(-7.78,.49,;-6.29,.89,;-5.89,2.37,;-4.41,2.77,;-3.32,1.68,;-3.72,.19,;-5.2,-.2,;-5.6,-1.69,;-7.09,-2.09,;-4.51,-2.78,;-1.83,2.08,;-1.43,3.57,;.06,3.97,;1.15,2.88,;.75,1.39,;-.74,.99,;2.63,3.28,;3.26,4.68,;4.79,4.52,;5.11,3.02,;6.45,2.25,;6.45,.71,;7.78,-.06,;5.11,-.06,;3.78,.71,;3.78,2.25,;5.11,-1.6,;3.78,-2.37,;2.44,-1.6,;3.78,-3.91,;5.11,-4.68,;6.45,-3.91,;6.45,-2.37,;7.78,-1.6,)|
COc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc(cc1)N1CCN2C(CN(C)CC2=O)C1 |(2,-2.37,;3.33,-1.6,;4.67,-2.37,;4.67,-3.91,;6,-4.68,;7.34,-3.91,;7.34,-2.37,;8.67,-1.6,;6,-1.6,;6,-.06,;4.67,.71,;4.67,2.25,;3.52,3.28,;4.15,4.68,;5.68,4.52,;6,3.02,;7.34,2.25,;7.34,.71,;8.67,-.06,;2.04,2.88,;.95,3.97,;-.54,3.57,;-.94,2.08,;.15,.99,;1.64,1.39,;-2.43,1.68,;-2.83,.19,;-4.31,-.2,;-5.4,.89,;-5,2.37,;-6.09,3.46,;-7.58,3.06,;-8.67,4.15,;-7.98,1.58,;-6.89,.49,;-7.29,-1,;-3.52,2.77,)|
Cc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc(cc1)N1CCN2CCOC[C@@H]2C1 |r,wU:32.36,(2.64,-1.6,;3.98,-2.37,;3.98,-3.91,;5.31,-4.68,;6.64,-3.91,;6.64,-2.37,;7.98,-1.6,;5.31,-1.6,;5.31,-.06,;3.98,.71,;3.98,2.25,;2.83,3.28,;3.46,4.68,;4.99,4.52,;5.31,3.02,;6.64,2.25,;6.64,.71,;7.98,-.06,;1.35,2.88,;.26,3.97,;-1.23,3.57,;-1.63,2.08,;-.54,.99,;.95,1.39,;-3.12,1.68,;-4.21,2.77,;-5.69,2.37,;-6.09,.89,;-7.58,.49,;-7.98,-1,;-6.89,-2.09,;-5.4,-1.69,;-5,-.2,;-3.52,.19,)|
Cc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc(cc1)N1CCN2CCOC[C@H]2C1 |r,wD:32.36,(2.64,-1.6,;3.98,-2.37,;3.98,-3.91,;5.31,-4.68,;6.64,-3.91,;6.64,-2.37,;7.98,-1.6,;5.31,-1.6,;5.31,-.06,;3.98,.71,;3.98,2.25,;2.83,3.28,;3.46,4.68,;4.99,4.52,;5.31,3.02,;6.64,2.25,;6.64,.71,;7.98,-.06,;1.35,2.88,;.26,3.97,;-1.23,3.57,;-1.63,2.08,;-.54,.99,;.95,1.39,;-3.12,1.68,;-4.21,2.77,;-5.69,2.37,;-6.09,.89,;-7.58,.49,;-7.98,-1,;-6.89,-2.09,;-5.4,-1.69,;-5,-.2,;-3.52,.19,)|
COc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc(cc1)N1CCN2CCOC[C@@H]2C1 |r,wU:33.37,(1.31,-2.37,;2.64,-1.6,;3.98,-2.37,;3.98,-3.91,;5.31,-4.68,;6.64,-3.91,;6.64,-2.37,;7.98,-1.6,;5.31,-1.6,;5.31,-.06,;3.98,.71,;3.98,2.25,;2.83,3.28,;3.46,4.68,;4.99,4.52,;5.31,3.02,;6.64,2.25,;6.64,.71,;7.98,-.06,;1.35,2.88,;.26,3.97,;-1.23,3.57,;-1.63,2.08,;-.54,.99,;.95,1.39,;-3.12,1.68,;-4.21,2.77,;-5.69,2.37,;-6.09,.89,;-7.58,.49,;-7.98,-1,;-6.89,-2.09,;-5.4,-1.69,;-5,-.2,;-3.52,.19,)|
COc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc(cc1)N1CCN2CCOC[C@H]2C1 |r,wD:33.37,(1.31,-2.37,;2.64,-1.6,;3.98,-2.37,;3.98,-3.91,;5.31,-4.68,;6.64,-3.91,;6.64,-2.37,;7.98,-1.6,;5.31,-1.6,;5.31,-.06,;3.98,.71,;3.98,2.25,;2.83,3.28,;3.46,4.68,;4.99,4.52,;5.31,3.02,;6.64,2.25,;6.64,.71,;7.98,-.06,;1.35,2.88,;.26,3.97,;-1.23,3.57,;-1.63,2.08,;-.54,.99,;.95,1.39,;-3.12,1.68,;-4.21,2.77,;-5.69,2.37,;-6.09,.89,;-7.58,.49,;-7.98,-1,;-6.89,-2.09,;-5.4,-1.69,;-5,-.2,;-3.52,.19,)|
Cc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc(cc1)N1CCn2ccnc2C1 |(2.39,-1.6,;3.72,-2.37,;3.72,-3.91,;5.05,-4.68,;6.39,-3.91,;6.39,-2.37,;7.72,-1.6,;5.05,-1.6,;5.05,-.06,;3.72,.71,;3.72,2.25,;2.58,3.28,;3.2,4.68,;4.73,4.52,;5.05,3.02,;6.39,2.25,;6.39,.71,;7.72,-.06,;1.09,2.88,;-0,3.97,;-1.49,3.57,;-1.89,2.08,;-.8,.99,;.69,1.39,;-3.37,1.68,;-4.46,2.77,;-5.95,2.37,;-6.35,.89,;-7.72,.19,;-7.48,-1.33,;-5.96,-1.58,;-5.26,-.2,;-3.77,.19,)|
Cc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc(cc1)N1CCC(O)CC1 |(2.64,-1.59,;4.18,-1.59,;4.95,-2.92,;6.49,-2.92,;7.26,-1.59,;6.49,-.26,;7.26,1.08,;4.95,-.26,;4.18,1.08,;2.64,1.08,;1.87,2.41,;.36,2.73,;.2,4.26,;1.61,4.89,;2.64,3.75,;4.18,3.75,;4.95,2.41,;6.49,2.41,;-.73,1.64,;-2.21,2.04,;-3.3,.95,;-2.9,-.53,;-1.42,-.93,;-.33,.16,;-3.99,-1.62,;-5.48,-1.22,;-6.57,-2.31,;-6.17,-3.8,;-7.26,-4.89,;-4.68,-4.2,;-3.59,-3.11,)|
COc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc(cc1)N1CCC(O)CC1 |(1.87,-2.92,;2.64,-1.59,;4.18,-1.59,;4.95,-2.92,;6.49,-2.92,;7.26,-1.59,;6.49,-.26,;7.26,1.08,;4.95,-.26,;4.18,1.08,;2.64,1.08,;1.87,2.41,;.36,2.73,;.2,4.26,;1.61,4.89,;2.64,3.75,;4.18,3.75,;4.95,2.41,;6.49,2.41,;-.73,1.64,;-2.21,2.04,;-3.3,.95,;-2.9,-.53,;-1.42,-.93,;-.33,.16,;-3.99,-1.62,;-5.48,-1.22,;-6.57,-2.31,;-6.17,-3.8,;-7.26,-4.89,;-4.68,-4.2,;-3.59,-3.11,)|
COc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc(cc1)N1CCC(C)(O)CC1 |(2.07,-2.92,;2.84,-1.59,;4.38,-1.59,;5.15,-2.92,;6.69,-2.92,;7.46,-1.59,;6.69,-.26,;7.46,1.08,;5.15,-.26,;4.38,1.08,;2.84,1.08,;2.07,2.41,;.56,2.73,;.4,4.26,;1.81,4.89,;2.84,3.75,;4.38,3.75,;5.15,2.41,;6.69,2.41,;-.53,1.64,;-2.01,2.04,;-3.1,.95,;-2.7,-.53,;-1.22,-.93,;-.13,.16,;-3.79,-1.62,;-5.28,-1.22,;-6.37,-2.31,;-5.97,-3.8,;-7.46,-3.4,;-7.06,-4.89,;-4.48,-4.2,;-3.39,-3.11,)|
COc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc(cc1)N1CCC(C)(CC1)OC |(2.61,-2.92,;3.38,-1.59,;4.92,-1.59,;5.69,-2.92,;7.23,-2.92,;8,-1.59,;7.23,-.26,;8,1.08,;5.69,-.26,;4.92,1.08,;3.38,1.08,;2.61,2.41,;1.11,2.73,;.95,4.26,;2.35,4.89,;3.38,3.75,;4.92,3.75,;5.69,2.41,;7.23,2.41,;.02,1.64,;-1.47,2.04,;-2.56,.95,;-2.16,-.53,;-.67,-.93,;.42,.16,;-3.25,-1.62,;-4.74,-1.22,;-5.83,-2.31,;-5.43,-3.8,;-6.91,-3.4,;-3.94,-4.2,;-2.85,-3.11,;-6.52,-4.89,;-8,-4.49,)|
Cc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc(cc1)N1CCC(CC1)N1CCOCC1 |(3.93,-.3,;5.47,-.3,;6.24,-1.63,;7.78,-1.63,;8.55,-.3,;7.78,1.03,;8.55,2.37,;6.24,1.03,;5.47,2.37,;3.93,2.37,;3.16,3.7,;1.65,4.02,;1.49,5.55,;2.9,6.18,;3.93,5.03,;5.47,5.03,;6.24,3.7,;7.78,3.7,;.56,2.93,;-.93,3.33,;-2.01,2.24,;-1.62,.75,;-.13,.36,;.96,1.44,;-2.7,-.34,;-4.19,.06,;-5.28,-1.03,;-4.88,-2.51,;-3.39,-2.91,;-2.31,-1.82,;-5.97,-3.6,;-7.46,-3.2,;-8.55,-4.29,;-8.15,-5.78,;-6.66,-6.18,;-5.57,-5.09,)|
CN1CCN(CC1)C1CCN(CC1)c1ccc(cc1)-c1n[nH]c2cc(=O)n(nc12)-c1c(C)cccc1F |(-8.89,-6.52,;-7.8,-5.43,;-8.2,-3.95,;-7.11,-2.86,;-5.63,-3.26,;-5.23,-4.74,;-6.32,-5.83,;-4.54,-2.17,;-4.94,-.68,;-3.85,.41,;-2.36,.01,;-1.96,-1.48,;-3.05,-2.57,;-1.27,1.1,;-1.67,2.59,;-.58,3.68,;.91,3.28,;1.31,1.79,;.22,.7,;2,4.37,;1.84,5.9,;3.24,6.52,;4.27,5.38,;5.81,5.38,;6.58,4.05,;8.12,4.05,;5.81,2.71,;4.27,2.71,;3.5,4.05,;6.58,1.38,;5.81,.04,;4.27,.04,;6.58,-1.29,;8.12,-1.29,;8.89,.04,;8.12,1.38,;8.89,2.71,)|
COc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc(cc1)N1CCC(CC1)N1CCOCC1 |(3.16,-1.63,;3.93,-.3,;5.47,-.3,;6.24,-1.63,;7.78,-1.63,;8.55,-.3,;7.78,1.03,;8.55,2.37,;6.24,1.03,;5.47,2.37,;3.93,2.37,;3.16,3.7,;1.65,4.02,;1.49,5.55,;2.9,6.18,;3.93,5.03,;5.47,5.03,;6.24,3.7,;7.78,3.7,;.56,2.93,;-.93,3.33,;-2.01,2.24,;-1.62,.75,;-.13,.36,;.96,1.44,;-2.7,-.34,;-4.19,.06,;-5.28,-1.03,;-4.88,-2.51,;-3.39,-2.91,;-2.31,-1.82,;-5.97,-3.6,;-7.46,-3.2,;-8.55,-4.29,;-8.15,-5.78,;-6.66,-6.18,;-5.57,-5.09,)|
COc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc(cc1)N1CCC(CC1)N1CCN(C)CC1 |(3.5,-1.29,;4.27,.04,;5.81,.04,;6.58,-1.29,;8.12,-1.29,;8.89,.04,;8.12,1.38,;8.89,2.71,;6.58,1.38,;5.81,2.71,;4.27,2.71,;3.5,4.05,;2,4.37,;1.84,5.9,;3.24,6.52,;4.27,5.38,;5.81,5.38,;6.58,4.05,;8.12,4.05,;.91,3.28,;-.58,3.68,;-1.67,2.59,;-1.27,1.1,;.22,.7,;1.31,1.79,;-2.36,.01,;-3.85,.41,;-4.94,-.68,;-4.54,-2.17,;-3.05,-2.57,;-1.96,-1.48,;-5.63,-3.26,;-7.11,-2.86,;-8.2,-3.95,;-7.8,-5.43,;-8.89,-6.52,;-6.32,-5.83,;-5.23,-4.74,)|
COc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc(cc1)N1CCC(C)(N)CC1 |(1.87,-2.7,;2.64,-1.36,;4.18,-1.36,;4.95,-2.7,;6.49,-2.7,;7.26,-1.36,;6.49,-.03,;7.26,1.3,;4.95,-.03,;4.18,1.3,;2.64,1.3,;1.87,2.64,;.36,2.96,;.2,4.49,;1.61,5.12,;2.64,3.97,;4.18,3.97,;4.95,2.64,;6.49,2.64,;-.73,1.87,;-2.21,2.27,;-3.3,1.18,;-2.9,-.31,;-1.42,-.71,;-.33,.38,;-3.99,-1.4,;-5.48,-1,;-6.57,-2.09,;-6.17,-3.58,;-6.17,-5.12,;-7.26,-4.66,;-4.68,-3.97,;-3.59,-2.89,)|
COc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc(cc1)N1CCC(C)(CC1)N(C)C |(2.61,-2.18,;3.38,-.85,;4.92,-.85,;5.69,-2.18,;7.23,-2.18,;8,-.85,;7.23,.49,;8,1.82,;5.69,.49,;4.92,1.82,;3.38,1.82,;2.61,3.16,;1.11,3.48,;.95,5.01,;2.35,5.63,;3.38,4.49,;4.92,4.49,;5.69,3.16,;7.23,3.16,;.02,2.39,;-1.47,2.79,;-2.56,1.7,;-2.16,.21,;-.67,-.19,;.42,.9,;-3.25,-.88,;-4.74,-.48,;-5.83,-1.57,;-5.43,-3.06,;-5.43,-4.6,;-3.94,-3.46,;-2.85,-2.37,;-6.52,-4.15,;-6.12,-5.63,;-8,-3.75,)|
COc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1cnc(s1)N1CCOCC1 |(.13,-2.8,;.9,-1.46,;2.44,-1.46,;3.21,-2.8,;4.75,-2.8,;5.52,-1.46,;4.75,-.13,;5.52,1.2,;3.21,-.13,;2.44,1.2,;.9,1.2,;.13,2.54,;-1.38,2.86,;-1.54,4.39,;-.13,5.02,;.9,3.87,;2.44,3.87,;3.21,2.54,;4.75,2.54,;-2.47,1.77,;-3.99,2.01,;-4.69,.64,;-3.6,-.45,;-2.23,.25,;-3.84,-1.97,;-5.28,-2.52,;-5.52,-4.05,;-4.32,-5.02,;-2.88,-4.46,;-2.64,-2.94,)|
COc1cc(C)c(cn1)-n1nc2c(n[nH]c2cc1=O)-c1ccc(cc1)N1CCNCC1
CN1CCC(=CC1)c1ccc(cc1)-c1n[nH]c2cc(=O)n(nc12)-c1cnccc1C |c:4|
COc1ccncc1-n1nc2c(n[nH]c2cc1=O)-c1ccc(cc1)C1=CCN(C)CC1 |t:28|
COc1ccncc1-n1nc2c(n[nH]c2cc1=O)-c1ccc(cc1)-c1cnn(C)c1
COc1cnccc1-n1nc2c(n[nH]c2cc1=O)-c1ccc(cc1)N1CCN(C)CC1
COc1cccc(F)c1-n1nc2c(n[nH]c2c(C)c1=O)-c1ccc(cc1)N1CCN(C)CC1 |(1.87,-3.02,;2.64,-1.68,;4.18,-1.68,;4.95,-3.02,;6.49,-3.02,;7.26,-1.68,;6.49,-.35,;7.26,.98,;4.95,-.35,;4.18,.98,;2.64,.98,;1.87,2.32,;.36,2.64,;.2,4.17,;1.61,4.8,;2.64,3.65,;4.18,3.65,;4.95,4.98,;4.95,2.32,;6.49,2.32,;-.73,1.55,;-2.21,1.95,;-3.3,.86,;-2.9,-.63,;-1.42,-1.03,;-.33,.06,;-3.99,-1.72,;-5.48,-1.32,;-6.57,-2.41,;-6.17,-3.9,;-7.26,-4.98,;-4.68,-4.29,;-3.59,-3.21,)|
COc1cccc(F)c1-n1nc2c(n[nH]c2c(C)c1=O)-c1ccc(cc1)N1CCOCC1 |(1.52,-3.36,;2.29,-2.03,;3.83,-2.03,;4.6,-3.36,;6.14,-3.36,;6.91,-2.03,;6.14,-.69,;6.91,.64,;4.6,-.69,;3.83,.64,;2.29,.64,;1.52,1.97,;.02,2.29,;-.14,3.82,;1.26,4.45,;2.29,3.31,;3.83,3.31,;4.6,4.64,;4.6,1.97,;6.14,1.97,;-1.07,1.2,;-2.56,1.6,;-3.65,.51,;-3.25,-.97,;-1.76,-1.37,;-.67,-.28,;-4.34,-2.06,;-5.83,-1.66,;-6.91,-2.75,;-6.52,-4.24,;-5.03,-4.64,;-3.94,-3.55,)|
CN1CCc2ccc(cc2C1)-c1n[nH]c2cc(=O)n(nc12)-c1c(C)cccc1F |(-3.34,-4.94,;-3.74,-3.46,;-5.23,-3.06,;-5.63,-1.57,;-4.54,-.48,;-4.94,1.01,;-3.85,2.1,;-2.36,1.7,;-1.96,.21,;-3.05,-.88,;-2.65,-2.37,;-1.27,2.79,;-1.43,4.32,;-.02,4.94,;1.01,3.8,;2.55,3.8,;3.32,2.47,;4.86,2.47,;2.55,1.13,;1.01,1.13,;.24,2.47,;3.32,-.2,;2.55,-1.54,;1.01,-1.54,;3.32,-2.87,;4.86,-2.87,;5.63,-1.54,;4.86,-.2,;5.63,1.13,)|
CN1CCc2ccc(cc2C1)-c1n[nH]c2cc(=O)n(nc12)-c1c(C)cccc1F |(-3.34,-4.2,;-3.74,-2.71,;-5.23,-2.31,;-5.63,-.83,;-4.54,.26,;-4.94,1.75,;-3.85,2.84,;-2.36,2.44,;-1.96,.95,;-3.05,-.14,;-2.65,-1.62,;-1.27,3.53,;-1.43,5.06,;-.02,5.69,;1.01,4.54,;2.55,4.54,;3.32,3.21,;4.86,3.21,;2.55,1.88,;1.01,1.88,;.24,3.21,;3.32,.54,;2.55,-.79,;1.01,-.79,;3.32,-2.13,;4.86,-2.13,;5.63,-.79,;4.86,.54,;5.63,1.88,)|
COc1cc(F)cc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc2CCN(C)Cc2c1 |(.24,-2.87,;1.01,-1.54,;2.55,-1.54,;3.32,-2.87,;4.86,-2.87,;5.63,-4.2,;5.63,-1.54,;4.86,-.2,;5.63,1.13,;3.32,-.2,;2.55,1.13,;1.01,1.13,;.24,2.47,;-1.27,2.79,;-1.43,4.32,;-.02,4.94,;1.01,3.8,;2.55,3.8,;3.32,2.47,;4.86,2.47,;-2.36,1.7,;-3.85,2.1,;-4.94,1.01,;-4.54,-.48,;-5.63,-1.57,;-5.23,-3.06,;-3.74,-3.46,;-3.34,-4.94,;-2.65,-2.37,;-3.05,-.88,;-1.96,.21,)|
COc1cc(cc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc2CCN(C)Cc2c1)C#N |(-.15,-2.57,;.62,-1.24,;2.16,-1.24,;2.93,-2.57,;4.5,-2.62,;5.24,-1.24,;4.47,.09,;5.24,1.43,;2.93,.09,;2.16,1.43,;.62,1.43,;-.15,2.76,;-1.66,3.08,;-1.82,4.61,;-.41,5.24,;.62,4.1,;2.16,4.1,;2.93,2.76,;4.47,2.76,;-2.74,1.99,;-4.23,2.39,;-5.32,1.3,;-4.92,-.18,;-6.01,-1.27,;-5.61,-2.76,;-4.12,-3.16,;-3.73,-4.65,;-3.04,-2.07,;-3.43,-.58,;-2.35,.51,;5.27,-3.95,;6.04,-5.29,)|
CCc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc2CCN(C)Cc2c1 |(.24,-2.87,;1.01,-1.54,;2.55,-1.54,;3.32,-2.87,;4.86,-2.87,;5.63,-1.54,;4.86,-.2,;5.63,1.13,;3.32,-.2,;2.55,1.13,;1.01,1.13,;.24,2.47,;-1.27,2.79,;-1.43,4.32,;-.02,4.94,;1.01,3.8,;2.55,3.8,;3.32,2.47,;4.86,2.47,;-2.36,1.7,;-3.85,2.1,;-4.94,1.01,;-4.54,-.48,;-5.63,-1.57,;-5.23,-3.06,;-3.74,-3.46,;-3.34,-4.94,;-2.65,-2.37,;-3.05,-.88,;-1.96,.21,)|
Cc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc2CCNCc2c1 |(1.01,-2.27,;2.55,-2.27,;3.32,-3.6,;4.86,-3.6,;5.63,-2.27,;4.86,-.94,;5.63,.4,;3.32,-.94,;2.55,.4,;1.01,.4,;.24,1.73,;-1.27,2.05,;-1.43,3.58,;-.02,4.21,;1.01,3.06,;2.55,3.06,;3.32,1.73,;4.86,1.73,;-2.36,.96,;-3.85,1.36,;-4.94,.27,;-4.54,-1.22,;-5.63,-2.31,;-5.23,-3.79,;-3.74,-4.19,;-2.65,-3.1,;-3.05,-1.61,;-1.96,-.53,)|
Cc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc2CCN(CCO)Cc2c1 |(1.01,-.59,;2.55,-.59,;3.32,-1.93,;4.86,-1.93,;5.63,-.59,;4.86,.74,;5.63,2.07,;3.32,.74,;2.55,2.07,;1.01,2.07,;.24,3.41,;-1.27,3.73,;-1.43,5.26,;-.02,5.89,;1.01,4.74,;2.55,4.74,;3.32,3.41,;4.86,3.41,;-2.36,2.64,;-3.85,3.04,;-4.94,1.95,;-4.54,.46,;-5.63,-.63,;-5.23,-2.11,;-3.74,-2.51,;-3.34,-4,;-1.85,-4.4,;-1.46,-5.89,;-2.65,-1.42,;-3.05,.06,;-1.96,1.15,)|
Cc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc2CCN(Cc2c1)C1CC(N)C1 |(.73,-.96,;2.07,-1.73,;2.07,-3.27,;3.4,-4.04,;4.73,-3.27,;4.73,-1.73,;6.07,-.96,;3.4,-.96,;3.4,.58,;2.07,1.35,;2.07,2.89,;.92,3.92,;1.55,5.33,;3.08,5.17,;3.4,3.66,;4.73,2.89,;4.73,1.35,;6.07,.58,;-.56,3.52,;-1.65,4.61,;-3.14,4.21,;-3.54,2.73,;-5.03,2.33,;-5.43,.84,;-4.34,-.25,;-2.85,.15,;-2.45,1.64,;-.96,2.04,;-4.73,-1.74,;-6.07,-2.51,;-5.3,-3.84,;-5.7,-5.33,;-3.96,-3.07,)|
Cc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc2CCN(Cc2c1)C1CNC1 |(.73,-1.5,;2.07,-2.27,;2.07,-3.81,;3.4,-4.58,;4.73,-3.81,;4.73,-2.27,;6.07,-1.5,;3.4,-1.5,;3.4,.04,;2.07,.81,;2.07,2.35,;.92,3.38,;1.55,4.79,;3.08,4.63,;3.4,3.12,;4.73,2.35,;4.73,.81,;6.07,.04,;-.56,2.98,;-1.65,4.07,;-3.14,3.67,;-3.54,2.18,;-5.03,1.79,;-5.43,.3,;-4.34,-.79,;-2.85,-.39,;-2.45,1.1,;-.96,1.49,;-4.73,-2.28,;-6.07,-3.05,;-5.3,-4.38,;-3.96,-3.61,)|
CC(CO)N1CCc2ccc(cc2C1)-c1n[nH]c2cc(=O)n(nc12)-c1c(C)cccc1F |(-6.15,-2.78,;-4.66,-2.38,;-3.57,-3.47,;-2.08,-3.07,;-4.26,-.89,;-5.35,.19,;-4.95,1.68,;-3.46,2.08,;-3.06,3.57,;-1.58,3.97,;-.49,2.88,;-.89,1.39,;-2.37,.99,;-2.77,-.5,;1,3.28,;1.63,4.68,;3.16,4.52,;3.48,3.02,;4.81,2.25,;4.81,.71,;6.15,-.06,;3.48,-.06,;2.14,.71,;2.14,2.25,;3.48,-1.6,;2.14,-2.37,;.81,-1.6,;2.14,-3.91,;3.48,-4.68,;4.81,-3.91,;4.81,-2.37,;6.15,-1.6,)|
COc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc2CCN(CC(F)F)Cc2c1 |(.24,-1.93,;1.01,-.59,;2.55,-.59,;3.32,-1.93,;4.86,-1.93,;5.63,-.59,;4.86,.74,;5.63,2.07,;3.32,.74,;2.55,2.07,;1.01,2.07,;.24,3.41,;-1.27,3.73,;-1.43,5.26,;-.02,5.89,;1.01,4.74,;2.55,4.74,;3.32,3.41,;4.86,3.41,;-2.36,2.64,;-3.85,3.04,;-4.94,1.95,;-4.54,.46,;-5.63,-.63,;-5.23,-2.11,;-3.74,-2.51,;-3.34,-4,;-1.85,-4.4,;-1.46,-5.89,;-.76,-3.31,;-2.65,-1.42,;-3.05,.06,;-1.96,1.15,)|
Cc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc2CCN(Cc2c1)C1CCOCC1 |(1.01,-1.27,;2.34,-2.04,;2.34,-3.58,;3.68,-4.35,;5.01,-3.58,;5.01,-2.04,;6.34,-1.27,;3.68,-1.27,;3.68,.27,;2.34,1.04,;2.34,2.58,;1.2,3.61,;1.83,5.02,;3.36,4.86,;3.68,3.35,;5.01,2.58,;5.01,1.04,;6.34,.27,;-.29,3.21,;-1.38,4.3,;-2.86,3.91,;-3.26,2.42,;-4.75,2.02,;-5.15,.53,;-4.06,-.56,;-2.57,-.16,;-2.17,1.33,;-.69,1.73,;-4.46,-2.05,;-5.95,-2.44,;-6.34,-3.93,;-5.26,-5.02,;-3.77,-4.62,;-3.37,-3.13,)|
CN1CCC(CC1)N1CCc2ccc(cc2C1)-c1n[nH]c2cc(=O)n(nc12)-c1c(C)cccc1F |(-5.65,-5.76,;-5.26,-4.28,;-6.34,-3.19,;-5.95,-1.7,;-4.46,-1.3,;-3.37,-2.39,;-3.77,-3.88,;-4.06,.19,;-5.15,1.28,;-4.75,2.76,;-3.26,3.16,;-2.86,4.65,;-1.38,5.05,;-.29,3.96,;-.69,2.47,;-2.17,2.07,;-2.57,.58,;1.2,4.36,;1.83,5.76,;3.36,5.6,;3.68,4.1,;5.01,3.33,;5.01,1.79,;6.34,1.02,;3.68,1.02,;2.34,1.79,;2.34,3.33,;3.68,-.52,;2.34,-1.29,;1.01,-.52,;2.34,-2.83,;3.68,-3.6,;5.01,-2.83,;5.01,-1.29,;6.34,-.52,)|
Cc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc2CCN(Cc2c1)C(=O)CN1CCOCC1 |(.81,.02,;2.14,-.75,;2.14,-2.29,;3.48,-3.06,;4.81,-2.29,;4.81,-.75,;6.15,.02,;3.48,.02,;3.48,1.56,;2.14,2.33,;2.14,3.87,;1,4.9,;1.63,6.31,;3.16,6.15,;3.48,4.64,;4.81,3.87,;4.81,2.33,;6.15,1.56,;-.49,4.5,;-1.58,5.59,;-3.06,5.19,;-3.46,3.71,;-4.95,3.31,;-5.35,1.82,;-4.26,.73,;-2.77,1.13,;-2.37,2.62,;-.89,3.02,;-4.66,-.76,;-6.15,-1.16,;-3.57,-1.85,;-3.97,-3.33,;-5.46,-3.73,;-5.85,-5.22,;-4.76,-6.31,;-3.28,-5.91,;-2.88,-4.42,)|
CN1CCc2ccc(cc2C1)-c1n[nH]c2cc(=O)n(nc12)-c1c(C)cc(cc1F)C#N |(-3.73,-4.65,;-4.12,-3.16,;-5.61,-2.76,;-6.01,-1.27,;-4.92,-.18,;-5.32,1.3,;-4.23,2.39,;-2.74,1.99,;-2.35,.51,;-3.43,-.58,;-3.04,-2.07,;-1.66,3.08,;-1.82,4.61,;-.41,5.24,;.62,4.1,;2.16,4.1,;2.93,2.76,;4.47,2.76,;2.16,1.43,;.62,1.43,;-.15,2.76,;2.93,.09,;2.16,-1.24,;.62,-1.24,;2.93,-2.57,;4.5,-2.62,;5.24,-1.24,;4.47,.09,;5.24,1.43,;5.27,-3.95,;6.04,-5.29,)|
Cc1cc(cc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc2CCNCc2c1)C#N |(.62,-1.24,;2.16,-1.24,;2.93,-2.57,;4.5,-2.62,;5.24,-1.24,;4.47,.09,;5.24,1.43,;2.93,.09,;2.16,1.43,;.62,1.43,;-.15,2.76,;-1.66,3.08,;-1.82,4.61,;-.41,5.24,;.62,4.1,;2.16,4.1,;2.93,2.76,;4.47,2.76,;-2.74,1.99,;-4.23,2.39,;-5.32,1.3,;-4.92,-.18,;-6.01,-1.27,;-5.61,-2.76,;-4.12,-3.16,;-3.04,-2.07,;-3.43,-.58,;-2.35,.51,;5.27,-3.95,;6.04,-5.29,)|
Cc1cc(cc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc2CCN(Cc2c1)C(=O)CO)C#N |(.62,-.59,;2.16,-.59,;2.93,-1.93,;4.5,-1.97,;5.24,-.59,;4.47,.74,;5.24,2.07,;2.93,.74,;2.16,2.07,;.62,2.07,;-.15,3.41,;-1.66,3.73,;-1.82,5.26,;-.41,5.89,;.62,4.74,;2.16,4.74,;2.93,3.41,;4.47,3.41,;-2.74,2.64,;-4.23,3.04,;-5.32,1.95,;-4.92,.46,;-6.01,-.63,;-5.61,-2.11,;-4.12,-2.51,;-3.04,-1.42,;-3.43,.06,;-2.35,1.15,;-3.73,-4,;-4.82,-5.09,;-2.24,-4.4,;-1.84,-5.89,;5.27,-3.31,;6.04,-4.64,)|
CC(O)C(=O)N1CCc2ccc(cc2C1)-c1n[nH]c2cc(=O)n(nc12)-c1c(C)cc(cc1F)C#N |(-1.15,-3.31,;-2.24,-4.4,;-1.84,-5.89,;-3.73,-4,;-4.82,-5.09,;-4.12,-2.51,;-5.61,-2.11,;-6.01,-.63,;-4.92,.46,;-5.32,1.95,;-4.23,3.04,;-2.74,2.64,;-2.35,1.15,;-3.43,.06,;-3.04,-1.42,;-1.66,3.73,;-1.82,5.26,;-.41,5.89,;.62,4.74,;2.16,4.74,;2.93,3.41,;4.47,3.41,;2.16,2.07,;.62,2.07,;-.15,3.41,;2.93,.74,;2.16,-.59,;.62,-.59,;2.93,-1.93,;4.5,-1.97,;5.24,-.59,;4.47,.74,;5.24,2.07,;5.27,-3.31,;6.04,-4.64,)|
Cc1cc(cc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc2CCN(Cc2c1)C(=O)CN)C#N |(.62,.15,;2.16,.15,;2.93,-1.18,;4.5,-1.23,;5.24,.15,;4.47,1.48,;5.24,2.82,;2.93,1.48,;2.16,2.82,;.62,2.82,;-.15,4.15,;-1.66,4.47,;-1.82,6,;-.41,6.63,;.62,5.49,;2.16,5.49,;2.93,4.15,;4.47,4.15,;-2.74,3.38,;-4.23,3.78,;-5.32,2.69,;-4.92,1.21,;-6.01,.12,;-5.61,-1.37,;-4.12,-1.77,;-3.04,-.68,;-3.43,.81,;-2.35,1.9,;-3.73,-3.26,;-4.82,-4.35,;-2.24,-3.66,;-1.15,-2.57,;5.27,-2.56,;6.04,-3.9,)|
C[C@H](N)C(=O)N1CCc2ccc(cc2C1)-c1n[nH]c2cc(=O)n(nc12)-c1c(C)cc(cc1F)C#N |r,wD:1.1,(10.02,3.24,;8.69,2.47,;8.69,.93,;7.36,3.24,;7.36,4.78,;6.02,2.47,;6.02,.93,;4.69,.16,;3.36,.93,;2.02,.16,;.69,.93,;.69,2.47,;2.02,3.24,;3.36,2.47,;4.69,3.24,;-.65,3.24,;-.81,4.77,;-2.31,5.09,;-3.08,3.76,;-4.59,3.44,;-5.06,1.97,;-6.57,1.65,;-4.03,.83,;-2.53,1.15,;-2.05,2.61,;-4.51,-.64,;-3.48,-1.78,;-1.97,-1.46,;-3.96,-3.24,;-5.46,-3.56,;-6.49,-2.42,;-6.02,-.96,;-7.05,.19,;-5.94,-5.03,;-6.41,-6.49,)|
CN1Cc2cc(ccc2C[C@H]1CO)-c1n[nH]c2cc(=O)n(nc12)-c1c(C)cccc1F |r,wD:10.12,(-3.77,-2.38,;-3.37,-.89,;-1.88,-.5,;-1.48,.99,;0,1.39,;.4,2.88,;-.69,3.97,;-2.17,3.57,;-2.57,2.08,;-4.06,1.68,;-4.46,.19,;-5.95,-.2,;-7.04,.89,;1.89,3.28,;2.52,4.68,;4.05,4.52,;4.37,3.02,;5.7,2.25,;5.7,.71,;7.04,-.06,;4.37,-.06,;3.03,.71,;3.03,2.25,;4.37,-1.6,;3.03,-2.37,;1.7,-1.6,;3.03,-3.91,;4.37,-4.68,;5.7,-3.91,;5.7,-2.37,;7.04,-1.6,)|
Cc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc2C[C@H]3COC(=O)N3Cc2c1 |r,wD:23.31,(1.1,-1.6,;2.43,-2.37,;2.43,-3.91,;3.77,-4.68,;5.1,-3.91,;5.1,-2.37,;6.43,-1.6,;3.77,-1.6,;3.77,-.06,;2.43,.71,;2.43,2.25,;1.29,3.28,;1.91,4.68,;3.45,4.52,;3.77,3.02,;5.1,2.25,;5.1,.71,;6.43,-.06,;-.2,2.88,;-1.29,3.97,;-2.78,3.57,;-3.17,2.08,;-4.66,1.68,;-5.06,.19,;-6.43,-.5,;-6.19,-2.03,;-4.67,-2.27,;-3.97,-3.64,;-3.97,-.89,;-2.48,-.5,;-2.09,.99,;-.6,1.39,)|
CN1Cc2cc(ccc2CC1(C)C)-c1n[nH]c2cc(=O)n(nc12)-c1c(C)cccc1F |(-4.39,-2.38,;-3.99,-.89,;-2.5,-.5,;-2.11,.99,;-.62,1.39,;-.22,2.88,;-1.31,3.97,;-2.8,3.57,;-3.19,2.08,;-4.68,1.68,;-5.08,.19,;-6.41,-.58,;-6.41,.96,;1.27,3.28,;1.89,4.68,;3.43,4.52,;3.75,3.02,;5.08,2.25,;5.08,.71,;6.41,-.06,;3.75,-.06,;2.41,.71,;2.41,2.25,;3.75,-1.6,;2.41,-2.37,;1.08,-1.6,;2.41,-3.91,;3.75,-4.68,;5.08,-3.91,;5.08,-2.37,;6.41,-1.6,)|
CN1Cc2cc(ccc2C[C@@H]1CO)-c1n[nH]c2cc(=O)n(nc12)-c1c(C)cccc1F |r,wU:10.12,(-3.77,-2.38,;-3.37,-.89,;-1.88,-.5,;-1.48,.99,;0,1.39,;.4,2.88,;-.69,3.97,;-2.17,3.57,;-2.57,2.08,;-4.06,1.68,;-4.46,.19,;-5.95,-.2,;-7.04,.89,;1.89,3.28,;2.52,4.68,;4.05,4.52,;4.37,3.02,;5.7,2.25,;5.7,.71,;7.04,-.06,;4.37,-.06,;3.03,.71,;3.03,2.25,;4.37,-1.6,;3.03,-2.37,;1.7,-1.6,;3.03,-3.91,;4.37,-4.68,;5.7,-3.91,;5.7,-2.37,;7.04,-1.6,)|
COC[C@@H]1Cc2ccc(cc2CN1C)-c1n[nH]c2cc(=O)n(nc12)-c1c(C)cccc1F |r,wD:3.2,(-7.78,.49,;-6.29,.89,;-5.2,-.2,;-3.72,.19,;-3.32,1.68,;-1.83,2.08,;-1.43,3.57,;.06,3.97,;1.15,2.88,;.75,1.39,;-.74,.99,;-1.14,-.5,;-2.63,-.89,;-3.02,-2.38,;2.63,3.28,;3.26,4.68,;4.79,4.52,;5.11,3.02,;6.45,2.25,;6.45,.71,;7.78,-.06,;5.11,-.06,;3.78,.71,;3.78,2.25,;5.11,-1.6,;3.78,-2.37,;2.44,-1.6,;3.78,-3.91,;5.11,-4.68,;6.45,-3.91,;6.45,-2.37,;7.78,-1.6,)|
Cc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc2C[C@H]3COCCN3Cc2c1 |r,wD:23.31,(1.36,-1.6,;2.69,-2.37,;2.69,-3.91,;4.02,-4.68,;5.36,-3.91,;5.36,-2.37,;6.69,-1.6,;4.02,-1.6,;4.02,-.06,;2.69,.71,;2.69,2.25,;1.54,3.28,;2.17,4.68,;3.7,4.52,;4.02,3.02,;5.36,2.25,;5.36,.71,;6.69,-.06,;.06,2.88,;-1.03,3.97,;-2.52,3.57,;-2.92,2.08,;-4.41,1.68,;-4.8,.19,;-6.29,-.2,;-6.69,-1.69,;-5.6,-2.78,;-4.11,-2.38,;-3.72,-.89,;-2.23,-.5,;-1.83,.99,;-.34,1.39,)|
CN1Cc2cc(ccc2CC1=O)-c1n[nH]c2cc(=O)n(nc12)-c1c(C)cccc1F |(-4.31,-2.38,;-3.91,-.89,;-2.43,-.5,;-2.03,.99,;-.54,1.39,;-.14,2.88,;-1.23,3.97,;-2.72,3.57,;-3.12,2.08,;-4.6,1.68,;-5,.19,;-6.49,-.2,;1.35,3.28,;1.97,4.68,;3.5,4.52,;3.82,3.02,;5.16,2.25,;5.16,.71,;6.49,-.06,;3.82,-.06,;2.49,.71,;2.49,2.25,;3.82,-1.6,;2.49,-2.37,;1.16,-1.6,;2.49,-3.91,;3.82,-4.68,;5.16,-3.91,;5.16,-2.37,;6.49,-1.6,)|
CN1CCc2ccc(cc2C1)-c1n[nH]c2cc(=O)n(nc12)-c1c(C)cccc1F |(-5.06,-2.38,;-4.66,-.89,;-5.75,.19,;-5.35,1.68,;-3.86,2.08,;-3.46,3.57,;-1.97,3.97,;-.89,2.88,;-1.28,1.39,;-2.77,.99,;-3.17,-.5,;.6,3.28,;1.23,4.68,;2.76,4.52,;3.08,3.02,;4.41,2.25,;4.41,.71,;5.75,-.06,;3.08,-.06,;1.75,.71,;1.75,2.25,;3.08,-1.6,;1.75,-2.37,;.41,-1.6,;1.75,-3.91,;3.08,-4.68,;4.41,-3.91,;4.41,-2.37,;5.75,-1.6,)|
CN1CCc2ccc(cc2C1CO)-c1n[nH]c2cc(=O)n(nc12)-c1c(C)cccc1F |(-5.06,-2.38,;-4.66,-.89,;-5.75,.19,;-5.35,1.68,;-3.86,2.08,;-3.46,3.57,;-1.97,3.97,;-.89,2.88,;-1.28,1.39,;-2.77,.99,;-3.17,-.5,;-2.08,-1.58,;-2.48,-3.07,;.6,3.28,;1.23,4.68,;2.76,4.52,;3.08,3.02,;4.41,2.25,;4.41,.71,;5.75,-.06,;3.08,-.06,;1.75,.71,;1.75,2.25,;3.08,-1.6,;1.75,-2.37,;.41,-1.6,;1.75,-3.91,;3.08,-4.68,;4.41,-3.91,;4.41,-2.37,;5.75,-1.6,)|
Cc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc2CCN3C(COC3=O)c2c1 |(.55,-1.6,;1.89,-2.37,;1.89,-3.91,;3.22,-4.68,;4.56,-3.91,;4.56,-2.37,;5.89,-1.6,;3.22,-1.6,;3.22,-.06,;1.89,.71,;1.89,2.25,;.74,3.28,;1.37,4.68,;2.9,4.52,;3.22,3.02,;4.56,2.25,;4.56,.71,;5.89,-.06,;-.74,2.88,;-1.83,3.97,;-3.32,3.57,;-3.72,2.08,;-5.21,1.68,;-5.61,.19,;-4.52,-.89,;-3.03,-.5,;-2.19,-1.79,;-3.16,-2.98,;-4.6,-2.43,;-5.89,-3.27,;-2.63,.99,;-1.14,1.39,)|
CN1CCc2ccc(cc2C1CN)-c1n[nH]c2cc(=O)n(nc12)-c1c(C)cccc1F |(-5.06,-2.38,;-4.66,-.89,;-5.75,.19,;-5.35,1.68,;-3.86,2.08,;-3.46,3.57,;-1.97,3.97,;-.89,2.88,;-1.28,1.39,;-2.77,.99,;-3.17,-.5,;-2.08,-1.58,;-2.48,-3.07,;.6,3.28,;1.23,4.68,;2.76,4.52,;3.08,3.02,;4.41,2.25,;4.41,.71,;5.75,-.06,;3.08,-.06,;1.75,.71,;1.75,2.25,;3.08,-1.6,;1.75,-2.37,;.41,-1.6,;1.75,-3.91,;3.08,-4.68,;4.41,-3.91,;4.41,-2.37,;5.75,-1.6,)|
CN1CCc2ncc(cc2C1)-c1n[nH]c2cc(=O)n(nc12)-c1c(C)cccc1F |(-3.34,-4.94,;-3.74,-3.46,;-5.23,-3.06,;-5.63,-1.57,;-4.54,-.48,;-4.94,1.01,;-3.85,2.1,;-2.36,1.7,;-1.96,.21,;-3.05,-.88,;-2.65,-2.37,;-1.27,2.79,;-1.43,4.32,;-.02,4.94,;1.01,3.8,;2.55,3.8,;3.32,2.47,;4.86,2.47,;2.55,1.13,;1.01,1.13,;.24,2.47,;3.32,-.2,;2.55,-1.54,;1.01,-1.54,;3.32,-2.87,;4.86,-2.87,;5.63,-1.54,;4.86,-.2,;5.63,1.13,)|
CN1CCc2ccc(-c3n[nH]c4cc(=O)n(nc34)-c3c(C)cccc3F)c(F)c2C1 |(-3.34,-4.94,;-3.74,-3.46,;-5.23,-3.06,;-5.63,-1.57,;-4.54,-.48,;-4.94,1.01,;-3.85,2.1,;-2.36,1.7,;-1.27,2.79,;-1.43,4.32,;-.02,4.94,;1.01,3.8,;2.55,3.8,;3.32,2.47,;4.86,2.47,;2.55,1.13,;1.01,1.13,;.24,2.47,;3.32,-.2,;2.55,-1.54,;1.01,-1.54,;3.32,-2.87,;4.86,-2.87,;5.63,-1.54,;4.86,-.2,;5.63,1.13,;-1.96,.21,;-.47,-.19,;-3.05,-.88,;-2.65,-2.37,)|
CN1CCc2cc(F)c(cc2C1)-c1n[nH]c2cc(=O)n(nc12)-c1c(C)cccc1F |(-3.34,-4.94,;-3.74,-3.46,;-5.23,-3.06,;-5.63,-1.57,;-4.54,-.48,;-4.94,1.01,;-3.85,2.1,;-4.25,3.58,;-2.36,1.7,;-1.96,.21,;-3.05,-.88,;-2.65,-2.37,;-1.27,2.79,;-1.43,4.32,;-.02,4.94,;1.01,3.8,;2.55,3.8,;3.32,2.47,;4.86,2.47,;2.55,1.13,;1.01,1.13,;.24,2.47,;3.32,-.2,;2.55,-1.54,;1.01,-1.54,;3.32,-2.87,;4.86,-2.87,;5.63,-1.54,;4.86,-.2,;5.63,1.13,)|
COc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc2CCN(C)Cc2c1F |(.24,-2.87,;1.01,-1.54,;2.55,-1.54,;3.32,-2.87,;4.86,-2.87,;5.63,-1.54,;4.86,-.2,;5.63,1.13,;3.32,-.2,;2.55,1.13,;1.01,1.13,;.24,2.47,;-1.27,2.79,;-1.43,4.32,;-.02,4.94,;1.01,3.8,;2.55,3.8,;3.32,2.47,;4.86,2.47,;-2.36,1.7,;-3.85,2.1,;-4.94,1.01,;-4.54,-.48,;-5.63,-1.57,;-5.23,-3.06,;-3.74,-3.46,;-3.34,-4.94,;-2.65,-2.37,;-3.05,-.88,;-1.96,.21,;-.47,-.19,)|
COc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1cc2CN(C)CCc2cc1F |(.24,-2.87,;1.01,-1.54,;2.55,-1.54,;3.32,-2.87,;4.86,-2.87,;5.63,-1.54,;4.86,-.2,;5.63,1.13,;3.32,-.2,;2.55,1.13,;1.01,1.13,;.24,2.47,;-1.27,2.79,;-1.43,4.32,;-.02,4.94,;1.01,3.8,;2.55,3.8,;3.32,2.47,;4.86,2.47,;-2.36,1.7,;-1.96,.21,;-3.05,-.88,;-2.65,-2.37,;-3.74,-3.46,;-3.34,-4.94,;-5.23,-3.06,;-5.63,-1.57,;-4.54,-.48,;-4.94,1.01,;-3.85,2.1,;-4.25,3.58,)|
Cc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc2CN(CCc2c1)C1CNC1 |(2.12,-.79,;3.66,-.79,;4.43,-2.13,;5.97,-2.13,;6.74,-.79,;5.97,.54,;6.74,1.87,;4.43,.54,;3.66,1.87,;2.12,1.87,;1.35,3.21,;-.16,3.53,;-.32,5.06,;1.09,5.69,;2.12,4.54,;3.66,4.54,;4.43,3.21,;5.97,3.21,;-1.24,2.44,;-2.73,2.84,;-3.82,1.75,;-3.42,.26,;-4.51,-.83,;-4.11,-2.32,;-2.62,-2.71,;-1.54,-1.63,;-1.93,-.14,;-.85,.95,;-5.2,-3.4,;-6.74,-3.4,;-6.74,-4.94,;-5.2,-4.94,)|
CN1CC(C1)N1CCc2cc(ccc2C1)-c1n[nH]c2cc(=O)n(nc12)-c1c(C)cccc1F |(-8.29,-1.17,;-6.8,-.77,;-6.03,.57,;-4.7,-.2,;-5.47,-1.54,;-3.21,.19,;-2.12,-.89,;-.63,-.5,;-.23,.99,;1.25,1.39,;1.65,2.88,;.56,3.97,;-.92,3.57,;-1.32,2.08,;-2.81,1.68,;3.14,3.28,;3.77,4.68,;5.3,4.52,;5.62,3.02,;6.95,2.25,;6.95,.71,;8.29,-.06,;5.62,-.06,;4.29,.71,;4.29,2.25,;5.62,-1.6,;4.29,-2.37,;2.95,-1.6,;4.29,-3.91,;5.62,-4.68,;6.95,-3.91,;6.95,-2.37,;8.29,-1.6,)|
Cc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1ccc2CN(CCc2c1)C1CCOCC1 |(2.64,-1.6,;3.98,-2.37,;3.98,-3.91,;5.31,-4.68,;6.64,-3.91,;6.64,-2.37,;7.98,-1.6,;5.31,-1.6,;5.31,-.06,;3.98,.71,;3.98,2.25,;2.83,3.28,;3.46,4.68,;4.99,4.52,;5.31,3.02,;6.64,2.25,;6.64,.71,;7.98,-.06,;1.35,2.88,;.26,3.97,;-1.23,3.57,;-1.63,2.08,;-3.12,1.68,;-3.52,.19,;-2.43,-.89,;-.94,-.5,;-.54,.99,;.95,1.39,;-5,-.2,;-6.09,.89,;-7.58,.49,;-7.98,-1,;-6.89,-2.09,;-5.4,-1.69,)|
CN1CCC(CC1)N1CCc2cc(ccc2C1)-c1n[nH]c2cc(=O)n(nc12)-c1c(C)cccc1F |(-8.72,-1.4,;-7.23,-1,;-6.84,.49,;-5.35,.89,;-4.26,-.2,;-4.66,-1.69,;-6.15,-2.09,;-2.77,.19,;-1.68,-.89,;-.2,-.5,;.2,.99,;1.69,1.39,;2.09,2.88,;1,3.97,;-.49,3.57,;-.89,2.08,;-2.37,1.68,;3.58,3.28,;4.2,4.68,;5.73,4.52,;6.05,3.02,;7.39,2.25,;7.39,.71,;8.72,-.06,;6.05,-.06,;4.72,.71,;4.72,2.25,;6.05,-1.6,;4.72,-2.37,;3.39,-1.6,;4.72,-3.91,;6.05,-4.68,;7.39,-3.91,;7.39,-2.37,;8.72,-1.6,)|
CN1Cc2ccc(cc2C1)-c1n[nH]c2cc(=O)n(nc12)-c1c(C)cccc1F |(-4.93,-4.7,;-4.53,-3.21,;-5.5,-2.02,;-4.66,-.72,;-5.06,.76,;-3.97,1.85,;-2.48,1.45,;-2.09,-.03,;-3.17,-1.12,;-3.09,-2.66,;-1.4,2.54,;-1.56,4.07,;-.15,4.7,;.88,3.56,;2.42,3.56,;3.19,2.22,;4.73,2.22,;2.42,.89,;.88,.89,;.11,2.22,;3.19,-.45,;2.42,-1.78,;.88,-1.78,;3.19,-3.11,;4.73,-3.11,;5.5,-1.78,;4.73,-.45,;5.5,.89,)|
CN1CCN(CC1)c1cccc(c1)-c1n[nH]c2cc(=O)n(nc12)-c1c(C)cccc1F |(-4.71,-4.82,;-4.31,-3.33,;-5.4,-2.24,;-5,-.76,;-3.52,-.36,;-2.43,-1.45,;-2.83,-2.93,;-3.12,1.13,;-4.21,2.22,;-3.81,3.71,;-2.32,4.1,;-1.23,3.02,;-1.63,1.53,;.26,3.41,;.88,4.82,;2.41,4.66,;2.73,3.15,;4.07,2.38,;4.07,.84,;5.4,.07,;2.73,.07,;1.4,.84,;1.4,2.38,;2.73,-1.47,;1.4,-2.24,;.07,-1.47,;1.4,-3.78,;2.73,-4.55,;4.07,-3.78,;4.07,-2.24,;5.4,-1.47,)|
COc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1cccc(c1)N1CCN(C)CC1 |(-1.27,-2.24,;.07,-1.47,;1.4,-2.24,;1.4,-3.78,;2.73,-4.55,;4.07,-3.78,;4.07,-2.24,;5.4,-1.47,;2.73,-1.47,;2.73,.07,;1.4,.84,;1.4,2.38,;.26,3.41,;.88,4.82,;2.41,4.66,;2.73,3.15,;4.07,2.38,;4.07,.84,;5.4,.07,;-1.23,3.02,;-2.32,4.1,;-3.81,3.71,;-4.21,2.22,;-3.12,1.13,;-1.63,1.53,;-3.52,-.36,;-5,-.76,;-5.4,-2.24,;-4.31,-3.33,;-4.71,-4.82,;-2.83,-2.93,;-2.43,-1.45,)|
CCc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1cccc(c1)N1CCN(C)CC1 |(-1.27,-2.24,;.07,-1.47,;1.4,-2.24,;1.4,-3.78,;2.73,-4.55,;4.07,-3.78,;4.07,-2.24,;5.4,-1.47,;2.73,-1.47,;2.73,.07,;1.4,.84,;1.4,2.38,;.26,3.41,;.88,4.82,;2.41,4.66,;2.73,3.15,;4.07,2.38,;4.07,.84,;5.4,.07,;-1.23,3.02,;-2.32,4.1,;-3.81,3.71,;-4.21,2.22,;-3.12,1.13,;-1.63,1.53,;-3.52,-.36,;-5,-.76,;-5.4,-2.24,;-4.31,-3.33,;-4.71,-4.82,;-2.83,-2.93,;-2.43,-1.45,)|
CN1C2CCC1CN(C2)c1cccc(c1)-c1n[nH]c2cc(=O)n(nc12)-c1c(C)cccc1F |(-4.71,-4.82,;-4.31,-3.33,;-5.4,-2.24,;-4.38,-1.65,;-3.41,-1.92,;-2.83,-2.93,;-2.43,-1.45,;-3.52,-.36,;-5,-.76,;-3.12,1.13,;-4.21,2.22,;-3.81,3.71,;-2.32,4.1,;-1.23,3.02,;-1.63,1.53,;.26,3.41,;.88,4.82,;2.41,4.66,;2.73,3.15,;4.07,2.38,;4.07,.84,;5.4,.07,;2.73,.07,;1.4,.84,;1.4,2.38,;2.73,-1.47,;1.4,-2.24,;.07,-1.47,;1.4,-3.78,;2.73,-4.55,;4.07,-3.78,;4.07,-2.24,;5.4,-1.47,)|
COc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1cccc(c1)N1CC2CCC(C1)N2C |(-1.27,-2.24,;.07,-1.47,;1.4,-2.24,;1.4,-3.78,;2.73,-4.55,;4.07,-3.78,;4.07,-2.24,;5.4,-1.47,;2.73,-1.47,;2.73,.07,;1.4,.84,;1.4,2.38,;.26,3.41,;.88,4.82,;2.41,4.66,;2.73,3.15,;4.07,2.38,;4.07,.84,;5.4,.07,;-1.23,3.02,;-2.32,4.1,;-3.81,3.71,;-4.21,2.22,;-3.12,1.13,;-1.63,1.53,;-3.52,-.36,;-5,-.76,;-5.4,-2.24,;-4.38,-1.65,;-3.41,-1.92,;-2.83,-2.93,;-2.43,-1.45,;-4.31,-3.33,;-4.71,-4.82,)|
COc1cc(cc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1cccc(c1)N1CC2CCC(C1)N2C)C#N |(-1.27,-.83,;.07,-.06,;1.4,-.83,;1.4,-2.37,;2.73,-3.2,;4.07,-2.37,;4.07,-.83,;5.4,-.06,;2.73,-.06,;2.73,1.48,;1.4,2.25,;1.4,3.79,;.26,4.82,;.88,6.22,;2.41,6.06,;2.73,4.56,;4.07,3.79,;4.07,2.25,;5.4,1.48,;-1.23,4.42,;-2.32,5.51,;-3.81,5.11,;-4.21,3.62,;-3.12,2.53,;-1.63,2.93,;-3.52,1.04,;-5,.65,;-5.4,-.84,;-4.38,-.25,;-3.41,-.52,;-2.83,-1.53,;-2.43,-.04,;-4.31,-1.93,;-4.71,-3.42,;2.73,-4.74,;2.73,-6.28,)|
COc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1cccc(c1)N1CCCC(N)C1 |(-1.27,-2.09,;.07,-1.32,;1.4,-2.09,;1.4,-3.63,;2.73,-4.4,;4.07,-3.63,;4.07,-2.09,;5.4,-1.32,;2.73,-1.32,;2.73,.22,;1.4,.99,;1.4,2.53,;.26,3.56,;.88,4.97,;2.41,4.81,;2.73,3.3,;4.07,2.53,;4.07,.99,;5.4,.22,;-1.23,3.16,;-2.32,4.25,;-3.81,3.85,;-4.21,2.36,;-3.12,1.28,;-1.63,1.67,;-3.52,-.21,;-5,-.61,;-5.4,-2.1,;-4.31,-3.19,;-2.79,-2.83,;-1.7,-3.92,;-2.43,-1.3,)|
COc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1cccc(c1)N1CCC(N)CC1 |(-1.27,-2.24,;.07,-1.47,;1.4,-2.24,;1.4,-3.78,;2.73,-4.55,;4.07,-3.78,;4.07,-2.24,;5.4,-1.47,;2.73,-1.47,;2.73,.07,;1.4,.84,;1.4,2.38,;.26,3.41,;.88,4.82,;2.41,4.66,;2.73,3.15,;4.07,2.38,;4.07,.84,;5.4,.07,;-1.23,3.02,;-2.32,4.1,;-3.81,3.71,;-4.21,2.22,;-3.12,1.13,;-1.63,1.53,;-3.52,-.36,;-5,-.76,;-5.4,-2.24,;-4.31,-3.33,;-4.71,-4.82,;-2.83,-2.93,;-2.43,-1.45,)|
COc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1cccc(c1)N1CCC(O)CC1 |(-1.27,-2.24,;.07,-1.47,;1.4,-2.24,;1.4,-3.78,;2.73,-4.55,;4.07,-3.78,;4.07,-2.24,;5.4,-1.47,;2.73,-1.47,;2.73,.07,;1.4,.84,;1.4,2.38,;.26,3.41,;.88,4.82,;2.41,4.66,;2.73,3.15,;4.07,2.38,;4.07,.84,;5.4,.07,;-1.23,3.02,;-2.32,4.1,;-3.81,3.71,;-4.21,2.22,;-3.12,1.13,;-1.63,1.53,;-3.52,-.36,;-5,-.76,;-5.4,-2.24,;-4.31,-3.33,;-4.71,-4.82,;-2.83,-2.93,;-2.43,-1.45,)|
CN1CCN(CC1)c1cccc(-c2n[nH]c3cc(=O)n(nc23)-c2c(C)cccc2F)c1F |(-4.71,-4.82,;-4.31,-3.33,;-5.4,-2.24,;-5,-.76,;-3.52,-.36,;-2.43,-1.45,;-2.83,-2.93,;-3.12,1.13,;-4.21,2.22,;-3.81,3.71,;-2.32,4.1,;-1.23,3.02,;.26,3.41,;.88,4.82,;2.41,4.66,;2.73,3.15,;4.07,2.38,;4.07,.84,;5.4,.07,;2.73,.07,;1.4,.84,;1.4,2.38,;2.73,-1.47,;1.4,-2.24,;.07,-1.47,;1.4,-3.78,;2.73,-4.55,;4.07,-3.78,;4.07,-2.24,;5.4,-1.47,;-1.63,1.53,;-.54,.44,)|
CN1CCN(CC1)c1ccc(F)c(c1)-c1n[nH]c2cc(=O)n(nc12)-c1c(C)cccc1F |(-4.71,-5.21,;-4.31,-3.72,;-5.4,-2.63,;-5,-1.14,;-3.52,-.74,;-2.43,-1.83,;-2.83,-3.32,;-3.12,.74,;-4.21,1.83,;-3.81,3.32,;-2.32,3.72,;-1.92,5.21,;-1.23,2.63,;-1.63,1.14,;.26,3.03,;.88,4.44,;2.41,4.27,;2.73,2.77,;4.07,2,;4.07,.46,;5.4,-.31,;2.73,-.31,;1.4,.46,;1.4,2,;2.73,-1.85,;1.4,-2.62,;.07,-1.85,;1.4,-4.16,;2.73,-4.93,;4.07,-4.16,;4.07,-2.62,;5.4,-1.85,)|
COc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1cccc(N2CCN(C)CC2)c1F |(-1.27,-2.24,;.07,-1.47,;1.4,-2.24,;1.4,-3.78,;2.73,-4.55,;4.07,-3.78,;4.07,-2.24,;5.4,-1.47,;2.73,-1.47,;2.73,.07,;1.4,.84,;1.4,2.38,;.26,3.41,;.88,4.82,;2.41,4.66,;2.73,3.15,;4.07,2.38,;4.07,.84,;5.4,.07,;-1.23,3.02,;-2.32,4.1,;-3.81,3.71,;-4.21,2.22,;-3.12,1.13,;-3.52,-.36,;-5,-.76,;-5.4,-2.24,;-4.31,-3.33,;-4.71,-4.82,;-2.83,-2.93,;-2.43,-1.45,;-1.63,1.53,;-.54,.44,)|
COc1cccc(F)c1-n1nc2c(n[nH]c2cc1=O)-c1cc(ccc1F)N1CCN(C)CC1 |(-1.27,-2.62,;.07,-1.85,;1.4,-2.62,;1.4,-4.16,;2.73,-4.93,;4.07,-4.16,;4.07,-2.62,;5.4,-1.85,;2.73,-1.85,;2.73,-.31,;1.4,.46,;1.4,2,;.26,3.03,;.88,4.44,;2.41,4.27,;2.73,2.77,;4.07,2,;4.07,.46,;5.4,-.31,;-1.23,2.63,;-1.63,1.14,;-3.12,.74,;-4.21,1.83,;-3.81,3.32,;-2.32,3.72,;-1.92,5.21,;-3.52,-.74,;-5,-1.14,;-5.4,-2.63,;-4.31,-3.72,;-4.71,-5.21,;-2.83,-3.32,;-2.43,-1.83,)|
COc1cc2CCN(C)Cc2cc1Nc1ncc(Cl)c(n1)N1CC(C)(CC(O)=O)c2ccccc12
COc1cc2CCN(C)Cc2cc1Nc1ncc(Cl)c(n1)N1C[C@](C)(CC(O)=O)c2ccccc12
COc1cc2CCN(C)Cc2cc1Nc1ncc(Cl)c(n1)N1C[C@@](C)(CC(O)=O)c2ccccc12
CN1CCc2cc(F)c(Nc3ncc(Cl)c(n3)N3CC(C)(CC(O)=O)c4ccccc34)cc2C1
CN1CCc2cc(F)c(Nc3ncc(Cl)c(n3)N3C[C@@](C)(CC(O)=O)c4ccccc34)cc2C1
COc1cc2CCN(C)Cc2cc1Nc1ncc(Cl)c(n1)N1CC(C(O)=O)c2ccccc12
COc1cc2CCN(C)Cc2cc1Nc1ncc(Cl)c(n1)N1CC(CC(O)=O)c2ccccc12
COc1cc2CCN(C)Cc2cc1Nc1ncc(Cl)c(n1)N1CC(C)(CC(O)=O)c2cc(F)ccc12
COc1cc2CCN(C)Cc2cc1Nc1ncc(Cl)c(n1)N1CC(C)(CC(O)=O)c2ccc(F)cc12
Cc1ccc2[nH]ncc2c1-c1ccn2nc(NC(=O)[C@@H]3C[C@@H]3F)cc2n1 |r|
CCc1c(F)c(F)c2[nH]ncc2c1-c1ccn2nc(NC(=O)[C@@H]3C[C@@H]3F)cc2n1 |r|
Cc1ccc2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)cn2n1 |r|
CCc1c(F)cc2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)cn2n1 |r|
Cc1c(F)cc2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)cn2n1 |r|
CCc1c(F)c(F)c2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)cn2n1 |r|
CCc1c(F)c(N(C)C)c2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)cn2n1 |r|
Cc1c(F)c(F)c2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)cn2n1 |r|
CSc1c(F)cc2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)cn2n1 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2nc(ccc2n1)-c1c(Cl)c(F)cc2[nH]ncc12 |r|
Nc1c(F)cc2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)cn2n1 |r|
CCN(C)c1c(F)c(CC)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3n2)c2cn[nH]c12 |r|
CCOc1c(F)c(CC)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3n2)c2cn[nH]c12 |r|
CCOc1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3n2)c2cn[nH]c12 |r|
CCN(C)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3n2)c2cn[nH]c12 |r|
CN(C)c1c(F)c(C)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3n2)c2cn[nH]c12 |r|
CCOc1c(F)c(C)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3n2)c2cn[nH]c12 |r|
CN(C)c1c(F)c(c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3n2)c2cn[nH]c12)C(F)(F)F |r|
CSc1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3n2)c2cn[nH]c12 |r|
CSc1c(F)c(F)c2[nH]ncc2c1-c1ccc2nc(NC(=O)[C@@H]3C[C@@H]3F)cn2n1 |r|
CN(C)c1c(F)c(Cl)c(-c2ccc3nc(NC(=O)[C@@H]4C[C@@H]4F)cn3n2)c2cn[nH]c12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2nc(ccc2n1)-c1c(Cl)c(F)c(F)c2[nH]ncc12 |r|
Cc1ccc2[nH]ncc2c1-c1cn2cc(NC(=O)[C@@H]3C[C@@H]3F)nc2cn1 |r|
CCc1c(F)cc2[nH]ncc2c1-c1cn2cc(NC(=O)[C@@H]3C[C@@H]3F)nc2cn1 |r|
CCc1c(F)c(N(C)C)c2[nH]ncc2c1-c1cn2cc(NC(=O)[C@@H]3C[C@@H]3F)nc2cn1 |r|
CSc1c(F)c(SC)c2[nH]ncc2c1-c1cn2cc(NC(=O)[C@@H]3C[C@@H]3F)nc2cn1 |r|
CSc1c(F)cc2[nH]ncc2c1-c1cn2cc(NC(=O)[C@@H]3C[C@@H]3F)nc2cn1 |r|
CCc1c(F)c(F)c2[nH]ncc2c1-c1cn2cc(NC(=O)[C@@H]3C[C@@H]3F)nc2cn1 |r|
CSc1c(F)c(C)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
Cc1c(F)cc2[nH]ncc2c1-c1cn2cc(NC(=O)[C@@H]3C[C@@H]3F)nc2cn1 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ncc2n1)-c1c(Cl)c(F)cc2[nH]ncc12 |r|
CN(C)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CCOc1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
Cc1c(F)c(F)c2[nH]ncc2c1-c1cn2cc(NC(=O)[C@@H]3C[C@@H]3F)nc2cn1 |r|
CSc1c(F)c(F)c2[nH]ncc2c1-c1cn2cc(NC(=O)[C@@H]3C[C@@H]3F)nc2cn1 |r|
CCc1c(F)c(SC)c2[nH]ncc2c1-c1cn2cc(NC(=O)[C@@H]3C[C@@H]3F)nc2cn1 |r|
CSc1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CSc1c(F)c(N(C)C)c2[nH]ncc2c1-c1cn2cc(NC(=O)[C@@H]3C[C@@H]3F)nc2cn1 |r|
CN(C)c1c(F)c(c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12)C(F)(F)F |r|
CCN(C)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CCN(C)c1c(F)c(c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12)C(F)(F)F |r|
CCN(C)c1c(F)c(CC)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CCOc1c(F)c(CC)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CCN(C)c1c(F)c(C)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CN(C)c1c(F)c(C)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CCOc1c(F)c(C)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
Cc1c(F)c(c2[nH]ncc2c1-c1cn2cc(NC(=O)[C@@H]3C[C@@H]3F)nc2cn1)C(F)(F)F |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ncc2n1)-c1c(Br)c(F)c(F)c2[nH]ncc12 |r|
CCN(C)c1c(F)c(SC)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ncc2n1)-c1c(Cl)c(F)c(F)c2[nH]ncc12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ncc2n1)-c1c(Br)c(F)cc2[nH]ncc12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ncc2n1)-c1c(c(F)cc2[nH]ncc12)C(F)(F)F |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ncc2n1)-c1c(Cl)c(F)c(N2CCCC2)c2[nH]ncc12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ncc2n1)-c1c(Cl)c(F)c(N2CCCCC2)c2[nH]ncc12 |r|
OCCCNc1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ncc2n1)-c1c(Cl)c(F)c(N2CCC2)c2[nH]ncc12 |r|
CN(C1CC1)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CNc1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ncc2n1)-c1c(Cl)c(F)c(N2CCSCC2)c2[nH]ncc12 |r|
CC(C)Nc1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CC(C)N(C)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CC(=C)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CC(C)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CC(Nc1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12)C#N |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ncc2n1)-c1c(Cl)c(F)c(-n2cccc2)c2[nH]ncc12 |r|
Nc1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ncc2n1)-c1c(Cl)c(F)c(NCC#N)c2[nH]ncc12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ncc2n1)-c1c(Cl)c(F)c(Cn2ncnn2)c2[nH]ncc12 |r|
CC(C)(O)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ncc2n1)-c1c(Cl)c(F)c(C=C)c2[nH]ncc12 |r|
CC(=O)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ncc2n1)-c1c(Cl)c(F)c(C2CC2)c2[nH]ncc12 |r|
CCOC(C)(C)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
COC(C)(C)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CC(C)(C)Nc1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ncc2n1)-c1c(Cl)c(F)c(NC2CC2)c2[nH]ncc12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ncc2n1)-c1c(Cl)c(F)c(N2CCC(F)C2)c2[nH]ncc12 |r,w:25.28|
Cn1cccc1-c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r,wD:22.24,20.20,(8.84,-.67,;8.44,-2.16,;9.35,-3.41,;8.44,-4.65,;6.98,-4.18,;6.98,-2.64,;5.64,-1.87,;4.31,-2.64,;4.31,-4.18,;2.98,-1.87,;1.64,-2.64,;2.98,-.33,;1.64,.44,;.31,-.33,;-1.02,.44,;-2.49,-.03,;-3.39,1.21,;-4.93,1.21,;-5.7,2.55,;-4.93,3.88,;-7.24,2.55,;-8.58,1.78,;-8.58,3.32,;-9.35,4.65,;-2.49,2.46,;-1.02,1.98,;.31,2.75,;1.64,1.98,;4.31,.44,;4.63,1.95,;6.16,2.11,;6.79,.7,;5.64,-.33,)|
CC(c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12)n1ncnn1 |r|
CC#Cc1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CC(C)c1c(F)c(C)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CC(=C)c1c(F)c(C)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CC(C)Nc1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CC(C)Nc1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@H]4F)nc3cn2)c2cn[nH]c12 |r|
CC(C)Nc1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@H]4C[C@H]4F)nc3cn2)c2cn[nH]c12 |r|
CCCc1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
Cc1cccn1-c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r,wD:22.24,20.20,(8.84,-.67,;8.44,-2.16,;9.35,-3.41,;8.44,-4.65,;6.98,-4.18,;6.98,-2.64,;5.64,-1.87,;4.31,-2.64,;4.31,-4.18,;2.98,-1.87,;1.64,-2.64,;2.98,-.33,;1.64,.44,;.31,-.33,;-1.02,.44,;-2.49,-.03,;-3.39,1.21,;-4.93,1.21,;-5.7,2.55,;-4.93,3.88,;-7.24,2.55,;-8.58,1.78,;-8.58,3.32,;-9.35,4.65,;-2.49,2.46,;-1.02,1.98,;.31,2.75,;1.64,1.98,;4.31,.44,;4.63,1.95,;6.16,2.11,;6.79,.7,;5.64,-.33,)|
CN(C)C(=O)c1ccn(c1)-c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CC(CO)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
COCC(C)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CC(CF)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CC(C)CNc1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CCCNc1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
C\C=C\c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CCNc1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
C[C@H]1COC[C@@H]1OC(=O)Nc1cn2cc(ncc2n1)-c1c(Cl)c(F)c(N(C)C)c2[nH]ncc12 |r|
CN(C)C(=O)Cc1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CN(C)C(=O)CSc1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CC(F)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ncc2n1)-c1c(Cl)c(F)c(C(=C)C(F)(F)F)c2[nH]ncc12 |r|
CC(C)Nc1c(F)c(C)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CNCc1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CN(C)Cc1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CCc1c(F)c(C(C)=C)c2[nH]ncc2c1-c1cn2cc(NC(=O)[C@@H]3C[C@@H]3F)nc2cn1 |r|
CCc1c(F)c(C(C)C)c2[nH]ncc2c1-c1cn2cc(NC(=O)[C@@H]3C[C@@H]3F)nc2cn1 |r|
CCc1c(F)c(NC(C)C)c2[nH]ncc2c1-c1cn2cc(NC(=O)[C@@H]3C[C@@H]3F)nc2cn1 |r|
Cn1ccc(c1)-c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ncc2n1)-c1c(Cl)c(F)c(-c2cc[nH]c2)c2[nH]ncc12 |r|
Cn1nccc1-c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r,wD:22.24,20.20,(8.86,-.57,;8.46,-2.06,;9.43,-3.39,;8.46,-4.72,;6.9,-4.21,;6.9,-2.57,;5.57,-1.8,;4.23,-2.57,;4.23,-4.11,;2.9,-1.8,;1.56,-2.57,;2.9,-.26,;1.56,.51,;.23,-.26,;-1.1,.51,;-2.57,.04,;-3.47,1.28,;-5.01,1.28,;-5.78,2.62,;-5.01,3.95,;-7.32,2.62,;-8.66,1.85,;-8.66,3.39,;-9.43,4.72,;-2.57,2.53,;-1.1,2.05,;.23,2.82,;1.56,2.05,;4.23,.51,;4.55,2.02,;6.08,2.18,;6.71,.77,;5.57,-.26,)|
CC(C)(CO)Nc1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CC(C)(C)C(=O)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ncc2n1)-c1c(Cl)c(F)c(OC2CC2)c2[nH]ncc12 |r|
CSc1c(F)c(Cl)c(-c2cn3cc(NC(=O)OC4COCC4C)nc3cn2)c2cn[nH]c12
OCCNc1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ncc2n1)-c1c(Cl)c(F)c(NC2CCC2)c2[nH]ncc12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ncc2n1)-c1c(Cl)c(F)c(NC2CCCC2)c2[nH]ncc12 |r|
COCCNc1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CC(c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12)C(F)(F)F |r|
CC(CO)Nc1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
COCC(C)Nc1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
C[C@H]1[C@@H]([C@H]1c1cnn(C)c1)C(=O)Nc1cn2cc(ncc2n1)-c1c(Cl)c(F)c(N(C)C)c2[nH]ncc12 |r|
C[C@@H]1[C@@H]([C@H]1c1cnn(C)c1)C(=O)Nc1cn2cc(ncc2n1)-c1c(Cl)c(F)c(N(C)C)c2[nH]ncc12 |r|
CC(C)(F)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ncc2n1)-c1c(Cl)c(F)c(C2=CCCC2)c2[nH]ncc12 |r,t:25|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ncc2n1)-c1c(Cl)c(F)c(Cn2ccnc2)c2[nH]ncc12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ncc2n1)-c1c(Cl)c(F)c(NN2CCOCC2)c2[nH]ncc12 |r|
CC(C)Oc1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
NC(=O)Cc1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CC(C)=Cc1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r,wD:20.21,18.17,(9.45,-2.82,;8.12,-2.05,;8.12,-.51,;6.78,-2.82,;5.53,-2.1,;4.21,-2.87,;4.21,-4.41,;2.87,-2.1,;1.54,-2.87,;2.87,-.56,;1.54,.21,;.21,-.56,;-1.13,.21,;-2.59,-.27,;-3.5,.98,;-5.04,.98,;-5.81,2.31,;-5.04,3.64,;-7.35,2.31,;-8.68,1.54,;-8.68,3.08,;-9.45,4.41,;-2.59,2.22,;-1.13,1.75,;.21,2.52,;1.54,1.75,;4.21,.21,;4.53,1.71,;6.06,1.87,;6.68,.47,;5.54,-.56,)|
FC(F)CNc1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ncc2n1)-c1c(Cl)c(F)c(C2CC2(F)Br)c2[nH]ncc12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ncc2n1)-c1c(Cl)c(F)c(NCC=C)c2[nH]ncc12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ncc2n1)-c1c(Cl)c(F)c(C2CCCC2)c2[nH]ncc12 |r|
CN1CCN(CC1)Nc1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
FCCNc1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CC(CO)(CO)Nc1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CC(C)c1c(F)cc(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
Cn1nccc1Nc1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CC(CCO)Nc1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CSc1c(F)c(C(C)C)c2[nH]ncc2c1-c1cn2cc(NC(=O)[C@@H]3C[C@@H]3F)nc2cn1 |r|
CC(C)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@H]4[C@H](C)[C@@H]4c4cnn(C)c4)nc3cn2)c2cn[nH]c12 |r|
CC(C)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@H]4[C@@H](C)[C@@H]4c4cnn(C)c4)nc3cn2)c2cn[nH]c12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ncc2n1)-c1c(Cl)c(F)c(Cn2cccc2)c2[nH]ncc12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ncc2n1)-c1c(Cl)c(F)c(Cn2cccn2)c2[nH]ncc12 |r|
OC(c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12)C(F)(F)F |r|
OC1CCN(C1)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r,w:1.0|
O[C@@H]1CCN(C1)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ncc2n1)-c1c(Cl)c(F)c(C2=CC(=O)CC2)c2[nH]ncc12 |r,t:25|
COC(C)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CC(N(C)C(C)=O)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
OC(C1CC1)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ncc2n1)-c1c(Cl)c(F)c(Nc2ccn[nH]2)c2[nH]ncc12 |r|
CC(C)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@H]4C[C@H]4F)nc3cn2)c2cn[nH]c12 |r|
CC(C)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@H]4F)nc3cn2)c2cn[nH]c12 |r|
CC(C)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CN(c1ccn[nH]1)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CN(c1ccnn1COCC[Si](C)(C)C)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CN(c1ccnn1C)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CC(C)C(=O)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CC(C)C(O)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
O[C@@H]1CCC(C1)Nc1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
Cc1nccn1Cc1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
OC1(CCCC1)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CC(C)c1c(F)c(c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12)C(F)(F)F |r|
CC(C(F)F)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CC(C)Cc1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
COC(C(C)C)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CC(C)C(F)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
COCCC(C)Nc1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ncc2n1)-c1c(Cl)c(F)c(NC2CC(F)C2)c2[nH]ncc12 |r,wD:3.4,1.0,(-10.44,2.69,;-9.67,1.36,;-9.67,-.18,;-8.34,.59,;-6.8,.59,;-6.03,-.74,;-6.03,1.92,;-4.49,1.92,;-3.58,.68,;-2.12,1.15,;-.78,.39,;.55,1.15,;.55,2.69,;-.78,3.46,;-2.12,2.69,;-3.58,3.17,;1.88,.39,;1.88,-1.15,;.55,-1.92,;3.22,-1.92,;3.22,-3.46,;4.55,-1.15,;5.89,-1.92,;7.22,-1.15,;8.71,-1.55,;9.11,-.07,;10.44,.7,;7.62,.33,;4.55,.39,;5.7,1.42,;5.07,2.82,;3.54,2.66,;3.22,1.15,)|
COC(C1CC1)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
C\C=C(/C)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CC(C=C)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CCC(C)Nc1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
Cc1cccn1Cc1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
Cc1cn(Cc2c(F)c(Cl)c(-c3cn4cc(NC(=O)[C@@H]5C[C@@H]5F)nc4cn3)c3cn[nH]c23)cn1 |r|
Cc1cnn(Cc2c(F)c(Cl)c(-c3cn4cc(NC(=O)[C@@H]5C[C@@H]5F)nc4cn3)c3cn[nH]c23)c1 |r|
O[C@H]1CCN(C1)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
OC1CCCC1c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ncc2n1)-c1c(Cl)c(F)c(NC2CCOC2)c2[nH]ncc12 |r|
COC1CCCC1c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
O[C@H]1CCC(C1)Nc1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CC(C(=O)N(C)C)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
C[C@H](c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12)n1ncnn1 |r|
C[C@@H](c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12)n1ncnn1 |r|
CC(C#N)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
C[C@H](c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12)n1cnnn1 |r|
C[C@@H](c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12)n1cnnn1 |r|
CC(C(N)=O)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CC(CF)Nc1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ncc2n1)-c1c(Cl)c(F)c(-c2ccco2)c2[nH]ncc12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ncc2n1)-c1c(Cl)c(F)c(-c2cnoc2)c2[nH]ncc12 |r|
O[C@H]1CC[C@H](C1)Nc1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
OC1CCC(=C1)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r,c:4|
Cc1ccn(Cc2c(F)c(Cl)c(-c3cn4cc(NC(=O)[C@@H]5C[C@@H]5F)nc4cn3)c3cn[nH]c23)n1 |r|
COC(c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12)C(F)(F)F |r|
CN(C1CCOC1)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CC(c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12)n1nccn1 |r|
CC(c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12)n1cncn1 |r|
O[C@H]1CN(C[C@@H]1O)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
COC1CCN(C1)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r,w:2.1|
CO[C@@H]1CCN(C1)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CO[C@H]1CCN(C1)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CC(Nc1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12)C1CC1 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ncc2n1)-c1c(Cl)c(F)c(NC2CC(F)(F)C2)c2[nH]ncc12 |r|
CN(C1CC1)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
OC(C#C)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CC(NC(C)=O)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CC(C)(C#N)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
Cc1ccc(o1)-c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2c[nH]nc12 |r|
CSc1c(F)c(C(C)=C)c2[nH]ncc2c1-c1cn2cc(NC(=O)[C@@H]3C[C@@H]3F)nc2cn1 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ncc2n1)-c1c(Cl)c(F)c(\C=C\C=C)c2[nH]ncc12 |r|
C[C@@H](c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12)C(F)(F)F |r|
C[C@H](c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12)C(F)(F)F |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ncc2n1)-c1c(Cl)c(F)c(NCC2CC2)c2[nH]ncc12 |r|
COC[C@H](C)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
COC[C@@H](C)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CCOC(c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12)C(F)(F)F |r|
FC(c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12)C(F)(F)F |r|
CO[C@H]1CN(C[C@@H]1OC)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ncc2n1)-c1c(Cl)c(F)c(-c2ccoc2)c2[nH]ncc12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ncc2n1)-c1c(Cl)c(F)c(C=C=C)c2[nH]ncc12 |r|
CN(C1CC1)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@H]4F)nc3cn2)c2cn[nH]c12 |r|
CN(C1CC1)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@H]4C[C@H]4F)nc3cn2)c2cn[nH]c12 |r|
OC(C1CCCOC1)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CSc1c(F)c(NC(C)C)c2[nH]ncc2c1-c1cn2cc(NC(=O)[C@@H]3C[C@@H]3F)nc2cn1 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ncc2n1)-c1c(Cl)c(F)c(C2=COCCO2)c2[nH]ncc12 |r,t:25|
CC(c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12)n1cccn1 |r|
CN([C@@H]1CC[C@H](O)C1)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CC(=C)c1c(F)c(c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12)C(F)(F)F |r|
Cc1cc(co1)-c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
OCC#Cc1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ncc2n1)-c1c(Cl)c(F)c(NCC#C)c2[nH]ncc12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ncc2n1)-c1c(Cl)c(F)c(C2CCCO2)c2[nH]ncc12 |r|
CC(Nc1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12)C(F)F |r|
OC1COC(C1)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CC1(C)CN(C1)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CC(C)(CCl)CNc1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CC(c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12)n1cc(C)cn1 |r|
CC(c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12)n1nccc1C |r|
CC(c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12)n1ccc(C)n1 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ncc2n1)-c1c(Cl)c(F)c(N2CC(F)(F)C2)c2[nH]ncc12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ncc2n1)-c1c(Cl)c(F)c(CC#N)c2[nH]ncc12 |r|
COCC#Cc1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ncc2n1)-c1c(Cl)c(F)c(C2OCC=C2)c2[nH]ncc12 |r,c:28|
CCC(=O)NC(C)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
OCCC(=O)Nc1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CC(NC=O)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
OCC\C=C\c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CC(C)=C(C)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r,wD:21.22,19.18,(8.83,-3.85,;7.5,-3.08,;6.16,-3.85,;7.5,-1.54,;8.83,-.77,;6.16,-.77,;4.83,-1.54,;4.83,-3.08,;3.49,-.77,;2.16,-1.54,;3.49,.77,;2.16,1.54,;.83,.77,;-.51,1.54,;-1.97,1.06,;-2.88,2.31,;-4.42,2.31,;-5.19,.98,;-4.42,-.36,;-6.73,.98,;-8.06,.21,;-8.06,1.75,;-8.83,3.08,;-1.97,3.56,;-.51,3.08,;.83,3.85,;2.16,3.08,;4.83,1.54,;5.15,3.05,;6.68,3.21,;7.31,1.8,;6.16,.77,)|
C[Si](C)(C)C#CCc1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
C[Si](C)(C)C#CC(O)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CC(O)C(C)Nc1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CC1(C)CC(CO1)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CC(c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12)n1ccnc1 |r|
CC(c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12)n1ccnc1C |r|
CC[Si](CC)(CC)C\C=C\c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CC(C(F)F)N(C)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CCC(C)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ncc2n1)-c1c(Cl)c(F)c(C2COCCO2)c2[nH]ncc12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ncc2n1)-c1c(Cl)c(F)c(C2CCCOC2)c2[nH]ncc12 |r|
CC(c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12)n1cnc(C)c1 |r|
FC(C#N)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CC(=O)NC(C#N)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ncc2n1)-c1c(Cl)c(F)c(N2CC3(C2)CC(F)(F)C3)c2[nH]ncc12 |r|
CC(NS(C)(=O)=O)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CC(=C(F)F)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r,wD:21.22,19.18,(8.83,-1.72,;7.5,-2.49,;7.5,-4.03,;8.83,-4.8,;6.16,-4.8,;6.16,-1.72,;4.83,-2.49,;4.83,-4.03,;3.49,-1.72,;2.16,-2.49,;3.49,-.18,;2.16,.59,;.83,-.18,;-.51,.59,;-1.97,.12,;-2.88,1.36,;-4.42,1.36,;-5.19,2.69,;-4.42,4.03,;-6.73,2.69,;-8.06,1.93,;-8.06,3.47,;-8.83,4.8,;-1.97,2.61,;-.51,2.13,;.83,2.9,;2.16,2.13,;4.83,.59,;5.15,2.1,;6.68,2.26,;7.31,.85,;6.16,-.18,)|
C[C@@H](O)[C@@H](O)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ncc2n1)-c1c(Cl)c(F)c(CC#C)c2[nH]ncc12 |r|
CC(C)C(C)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CC(C)=C(C)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r,wD:21.22,19.18,(8.83,-4.8,;7.5,-4.03,;6.16,-4.8,;7.5,-2.49,;8.83,-1.72,;6.16,-1.72,;4.83,-2.49,;4.83,-4.03,;3.49,-1.72,;2.16,-2.49,;3.49,-.18,;2.16,.59,;.83,-.18,;-.51,.59,;-1.97,.12,;-2.88,1.36,;-4.42,1.36,;-5.19,2.69,;-4.42,4.03,;-6.73,2.69,;-8.06,1.93,;-8.06,3.47,;-8.83,4.8,;-1.97,2.61,;-.51,2.13,;.83,2.9,;2.16,2.13,;4.83,.59,;5.15,2.1,;6.68,2.26,;7.31,.85,;6.16,-.18,)|
CC(=O)NCc1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ncc2n1)-c1c(Cl)c(F)c(C=O)c2[nH]ncc12 |r|
CCOC(=O)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CO[C@H](C)[C@@H](C)N(C)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CO[C@@H](C)[C@@H](C)N(C)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CC(NC1(CC1)C#N)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CC(=O)OCCc1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ncc2n1)-c1c(Cl)c(F)c(NC(=O)OCC2c3ccccc3-c3ccccc23)c2[nH]ncc12 |r|
FC(F)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
OC(C#N)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CC(NC(=O)C1CCC1)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ncc2n1)-c1c(Cl)c(F)c(C2CC2F)c2[nH]ncc12 |r|
CC(C)Nc1c(F)c(c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12)C(F)(F)F |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ncc2n1)-c1c(Cl)c(F)c(C2CCOC2)c2[nH]ncc12 |r|
CC(NC(=O)C(F)(F)F)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CSCc1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CSC(C)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CS(=O)Cc1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CS(=O)(=O)Cc1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CNC(=O)N(C)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CO[C@H](C)[C@@H](OC)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CC(NC(=O)C(F)F)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
Cc1ncc([nH]1)-c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CC(c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12)S(C)(=O)=O |r|
CC(c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12)S(C)=O |r|
CCNC(=O)C(C)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ncc2n1)-c1c(Cl)c(F)c(C(NC(=O)C(F)(F)F)C#N)c2[nH]ncc12 |r|
COC(=O)C(C(=O)NC1CCC1)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
F[C@H]1C[C@H]1C(=O)NC(C#N)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
F[C@H]1C[C@H]1C(=O)Nc1cn2cc(ncc2n1)-c1c(Cl)c(F)c(C(NC(=O)C2CC2)C#N)c2[nH]ncc12 |r|
FC(F)C(=O)NC(C#N)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CCOc1c(F)c(SC)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12 |r|
CCOc1c(F)c(SC)c2[nH]ncc2c1-c1cn2cc(NC(=O)[C@@H]3C[C@@H]3F)nc2cn1 |r|
COc1nc2CCN(C)Cc2cc1Nc1ncc2cccc(-c3ccccc3)c2n1
COc1nc2CCN(C)Cc2cc1Nc1ncc2cccc(-c3cnn4ccccc34)c2n1
COc1nc2CCN(C)Cc2cc1Nc1ncc2cccc(-c3ccc4n(C)ncc4c3)c2n1
COc1nc2CCN(C)Cc2cc1Nc1ncc2cccc(-c3ccccc3F)c2n1
COc1ccccc1-c1cccc2cnc(Nc3cc4CN(C)CCc4nc3OC)nc12
COc1cccc(c1)-c1cccc2cnc(Nc3cc4CN(C)CCc4nc3OC)nc12
COc1nc2CCN(C)Cc2cc1Nc1ncc2cccc(C3=CCOCC3)c2n1 |t:24|
COc1nc2CCN(C)Cc2cc1Nc1ncc2cccc(-c3cnn(C)c3)c2n1
COc1nc2CCN(C)Cc2cc1Nc1ncc2cccc(-c3cccnc3)c2n1
COc1nc2CCN(C)Cc2cc1Nc1ncc2cccc(-c3ccc(=O)n(C)c3)c2n1
COc1nc2CCN(C)Cc2cc1Nc1ncc2cccc(C3CCOCC3)c2n1
CNC(=O)c1ccccc1-c1cccc2cnc(Nc3cc4CN(C)CCc4nc3OC)nc12
COC(=O)c1cccc(c1)-c1cccc2cnc(Nc3cc4CN(C)CCc4nc3OC)nc12
CNC(=O)c1cccc(c1)-c1cccc2cnc(Nc3cc4CN(C)CCc4nc3OC)nc12 |$;HN;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;$|
COc1nc2CCN(C)Cc2cc1Nc1ncc2cccc(C3=CCN(CC3)C(=O)OC(C)(C)C)c2n1 |t:24|
COc1nc2CCN(C)Cc2cc1Nc1ncc2cccc(C(C)=C)c2n1
COc1nc2CCN(C)Cc2cc1Nc1ncc2cccc(C3=CCN(CC3)C(C)=O)c2n1 |t:24|
COc1nc2CCN(C)Cc2cc1Nc1ncc2cccc(-c3ccccc3OC(F)(F)F)c2n1
COc1nc2CCN(C)Cc2cc1Nc1ncc2cccc(-c3ccccc3SC)c2n1
COc1cccc(F)c1-c1cccc2cnc(Nc3cc4CN(C)CCc4nc3OC)nc12 |(6.67,-.38,;5.33,.38,;4,-.38,;4,-1.93,;2.67,-2.69,;1.33,-1.93,;1.33,-.38,;,.39,;2.67,.38,;2.67,1.93,;4,2.69,;4,4.23,;2.67,5,;1.33,4.23,;,5,;-1.33,4.23,;-1.33,2.69,;-2.67,1.93,;-2.67,.38,;-1.33,-.38,;-1.33,-1.93,;,-2.69,;,-4.23,;1.33,-5,;-1.33,-5,;-2.67,-4.23,;-2.67,-2.69,;-4,-1.93,;-4,-.38,;-5.33,.38,;-6.67,-.38,;,1.93,;1.33,2.69,)|
COc1nc2CCN(C)Cc2cc1Nc1ncc2cccc(-c3ccccc3OCc3ccccc3)c2n1
COc1nc2CCN(C)Cc2cc1Nc1ncc2cccc(-c3cccnc3OC)c2n1
COc1nc2CCN(C)Cc2cc1Nc1ncc2cccc(N3CCCC3=O)c2n1
COc1ccccc1-c1nccc2cnc(Nc3cc4CN(C)CCc4nc3OC)nc12
COc1nc2CCN(C)Cc2cc1Nc1ncc2ccnc(C3=CCOCC3)c2n1 |t:24|
COc1nc2CCN(C)Cc2cc1Nc1ncc2ccnc(C3=CN(C)C(=O)CC3)c2n1 |t:24|
COc1nc2CCN(C)Cc2cc1Nc1ncc2cccc(-c3ccn(C)n3)c2n1
COc1nc2CCN(C)Cc2cc1Nc1ncc2cccc(NCC3CCOCC3)c2n1
COc1nc2CCN(C)Cc2cc1Nc1ncc2cccc(N3Cc4ccccc4C3=O)c2n1
COc1nc2CCN(C)Cc2cc1Nc1ncc2ccnc(N3CCCCC3)c2n1
COc1nc2CCN(C)Cc2cc1Nc1ncc2ccnc(-c3cccnc3OC)c2n1
COc1nc2CCN(C)Cc2cc1Nc1ncc2ccnc(N3CCOCC3)c2n1
COc1nc2CCN(C)Cc2cc1Nc1ncc2cccc(-c3ccccn3)c2n1
COc1nc2CCN(C)Cc2cc1Nc1ncc2cccc(NCc3ccccc3)c2n1
COc1nc2CCN(C)Cc2cc1Nc1ncc2cccc(NCC(C)C)c2n1
COc1nc2CCN(C)Cc2cc1Nc1ncc2cccc(-c3cccc(Cl)n3)c2n1
COc1nc2CCN(C)Cc2cc1Nc1ncc2ccnc(NCC(C)(C)C)c2n1
COc1nc2CCN(C)Cc2cc1Nc1ncc2ccnc(N[C@@H](C)C(C)(C)C)c2n1 |r|
COc1nc2CCN(C)Cc2cc1Nc1ncc2ccnc(-c3cc(C)nn3C)c2n1
CCOc1nc2CCN(C)Cc2cc1Nc1ncc2cccc(-c3ccccc3OC)c2n1
COc1ccccc1-c1cccc2cnc(Nc3cnc4CCN(C)Cc4c3)nc12
COc1ccccc1-c1cccc2cnc(Nc3cc4CN(C)CCc4nc3C)nc12
CCOc1nc2CCN(C)Cc2cc1Nc1ncc2cccc(-c3cccnc3OC)c2n1
COc1ncccc1-c1cccc2cnc(Nc3cc4CN(C)CCc4nc3C)nc12
CN1CCc2[nH]c(=O)c(Nc3ncc4ccnc(N5CCOCC5)c4n3)cc2C1
CCOc1nc2CCN(C)Cc2cc1Nc1ncc2ccnc(NCC(C)(C)C)c2n1
COc1nc2CCN(C)Cc2cc1Nc1ncc2cccc(-c3cnn(C)c3C)c2n1
CCOc1nc2CCN(C)Cc2cc1Nc1ncc2cccc(-c3ccc(=O)n(C)c3)c2n1
CCOc1nc2CCN(C)Cc2cc1Nc1ncc2cccc(-c3cnn(C)c3C)c2n1
CCOc1nc2CCN(C)Cc2cc1Nc1ncc2ccnc(N[C@@H](CO)C(C)(C)C)c2n1 |r|
CCOc1nc2CCN(C)Cc2cc1Nc1ncc2ccnc(N[C@H](C)C(C)(C)C)c2n1 |r|
COc1nc2CCN(C)Cc2cc1Nc1ncc2cccc(Cc3ccccc3)c2n1
CN1CCc2[nH]c(=O)c(Nc3ncc4cccc(-c5cnn(C)c5C)c4n3)cc2C1
COc1ccccc1-c1nccc2cnc(Nc3cc4CN(C)CCc4[nH]c3=O)nc12
CN1CCc2[nH]c(=O)c(Nc3ncc4ccnc(N5CCCCC5)c4n3)cc2C1
CN1CCc2[nH]c(=O)c(Nc3ncc4ccnc(NCC(C)(C)C)c4n3)cc2C1
CCOc1nc2CCN(C)Cc2cc1Nc1ncc2ccnc(N3CC(C)(C)C3)c2n1
CCOc1nc2CCN(C)Cc2cc1Nc1ncc2cccc(-c3c(C)nn(C)c3C)c2n1 |(-6.7,.38,;-5.37,-.38,;-4.03,.38,;-2.7,-.38,;-2.7,-1.93,;-1.37,-2.69,;-1.37,-4.23,;-.03,-5,;1.3,-4.23,;2.63,-5,;1.3,-2.69,;-.03,-1.93,;-.03,-.38,;-1.37,.38,;-1.37,1.93,;-.03,2.69,;-.03,4.23,;1.3,5,;2.63,4.23,;3.97,5,;5.3,4.23,;5.3,2.69,;3.97,1.93,;3.97,.38,;2.72,-.52,;1.23,-.12,;3.2,-1.98,;4.74,-1.98,;5.51,-3.32,;5.21,-.52,;6.7,-.12,;2.63,2.69,;1.3,1.93,)|
CN1CCc2c(C1)cc(Nc1ncc3ccnc(N4CCCCC4)c3n1)c(=O)n2C
CN1CCc2c(C1)cc(Nc1ncc3ccnc(N4CCOCC4)c3n1)c(=O)n2C
CN1CCc2[nH]c(=O)c(Nc3ncc4ccnc(NCC(C)(C)CO)c4n3)cc2C1
CN1CCc2[nH]c(=O)c(Nc3ncc4ccnc(N5CCSCC5)c4n3)cc2C1
CN1CCc2[nH]c(=O)c(Nc3ncc4ccnc(N5CCCCCC5)c4n3)cc2C1
CN1CCc2[nH]c(=O)c(Nc3ncc4ccnc(N5CCC(F)(F)CC5)c4n3)cc2C1
CN1CCc2[nH]c(=O)c(Nc3ncc4ccnc(C5=CCCCC5)c4n3)cc2C1 |t:18|
C[C@@H]1CCCCN1c1nccc2cnc(Nc3cc4CN(C)CCc4[nH]c3=O)nc12 |r|
CN1CCc2[nH]c(=O)c(Nc3ncc4ccnc(NCC5(C)CC5)c4n3)cc2C1
CN1CCc2c(C1)cc(Nc1ncc3ccnc(N4CCC(F)(F)CC4)c3n1)c(=O)n2C
CN1CCc2c(C1)cc(Nc1ncc3ccnc(N4CCCCCC4)c3n1)c(=O)n2C
CN1CCc2c(C1)cc(Nc1ncc3ccnc(C4=CCCCC4)c3n1)c(=O)n2C |t:19|
Cn1c2CCN(CCO)Cc2cc(Nc2ncc3ccnc(N4CCC(F)(F)CC4)c3n2)c1=O
Cn1c2CCN(CCO)Cc2cc(Nc2ncc3ccnc(N4CCCCC4)c3n2)c1=O
Cn1c2CCN(CCO)Cc2cc(Nc2ncc3ccnc(N4CCSCC4)c3n2)c1=O
CN1CCc2c(C1)cc(Nc1ncc3ccnc(N4CCC(F)(F)C4)c3n1)c(=O)n2C
CN1CCc2c(C1)cc(Nc1ncc3ccnc(N4CC5CC5C4)c3n1)c(=O)n2C
COCCn1c2CCN(C)Cc2cc(Nc2ncc3ccnc(N4CCC(F)(F)CC4)c3n2)c1=O
CCOc1nc2CCN(C)Cc2cc1Nc1ncc2ccnc(N[C@H](CO)C(C)C)c2n1 |r|
CCOc1nc2CCN(C)Cc2cc1Nc1ncc2ccnc(N[C@@H](CO)C(C)C)c2n1 |r|
COc1nc2CCN(C)Cc2cc1Nc1ncc2ccnc(N[C@H](CO)C(C)C)c2n1 |r|
COc1nc2CCN(C)Cc2cc1Nc1ncc2ccnc(N[C@@H](CO)C(C)C)c2n1 |r|
COc1nc2CCN(C)Cc2cc1Nc1ncc2ccnc(N[C@H](CO)C(C)(C)C)c2n1 |r|
COc1nc2CCN(C)Cc2cc1Nc1ncc2ccnc(N[C@@H](CO)C(C)(C)C)c2n1 |r|
CCOc1nc2CCN(C)Cc2cc1Nc1ncc2ccnc(N[C@@H]3CCC[C@H]3O)c2n1 |r|
CCOc1nc2CCN(C)Cc2cc1Nc1ncc2ccnc(N[C@@H]3CC[C@@H](O)C3)c2n1 |r|
CCOc1nc2CCN(C)Cc2cc1Nc1ncc2ccnc(NCC(C)(C)CO)c2n1
CCOc1nc2CCN(C)Cc2cc1Nc1ncc2ccnc(N[C@H]3CC[C@@H](O)C3)c2n1 |r|
COc1nc2CCN(C)Cc2cc1Nc1ncc2ccnc(N[C@@H]3CCC[C@H]3O)c2n1 |r|
COc1nc2CCN(C)Cc2cc1Nc1ncc2ccnc(N[C@@H]3CC[C@@H](O)C3)c2n1 |r|
COc1nc2CCN(C)Cc2cc1Nc1ncc2ccnc(N3CCC[C@H]3CO)c2n1 |r|
COc1nc2CCN(C)Cc2cc1Nc1ncc2ccnc(N[C@@H]3CCC[C@@H]3O)c2n1 |r|
COc1nc2CCN(C)Cc2cc1Nc1ncc2ccnc(N[C@H]3CCC[C@H]3O)c2n1 |r|
COc1nc2CCN(C)Cc2cc1Nc1ncc2ccnc(N[C@H]3CCC[C@@H]3O)c2n1 |r|
CCOc1nc2CCN(C)Cc2cc1Nc1ncc2ccnc(N3CCC[C@H]3CO)c2n1 |r|
COC[C@@H]1CCCN1c1nccc2cnc(Nc3cc4CN(C)CCc4nc3OC)nc12 |r|
COc1nc2CCN(C)Cc2cc1Nc1ncc2ccnc(N3CC(F)(F)C[C@H]3CO)c2n1 |r|
COc1nc2CCN(C)Cc2cc1Nc1ncc2ccnc(NC(C)(C)CO)c2n1
CC[C@H](CO)Nc1nccc2cnc(Nc3cc4CN(C)CCc4nc3OC)nc12 |r|
COc1nc2CCN(C)Cc2cc1Nc1ncc2ccnc(NCC(C)(C)O)c2n1
COc1cc2CCN(C)Cc2cc1Nc1ncc2ccnc(N[C@@H](CO)C(C)C)c2n1 |r|
[2H]C5([2H])N(C)C([2H])([2H])C([2H])([2H])N(c4ccc3[nH]c(c2c(N)c1ccsc1[nH]c2=O)nc3c4)C5([2H])[2H]
[2H]C5([2H])CN(c4ccc3[nH]c(c2c(N)c1ccsc1[nH]c2=O)nc3c4)CC([2H])([2H])N5C
[2H]C1([2H])CN(C)CC([2H])([2H])N1c5ccc4[nH]c(c3c(N)c2ccsc2[nH]c3=O)nc4c5
[2H]c5cc4c(N)c(c3nc2c([2H])c(N1CCN(C)CC1)c([2H])cc2[nH]3)c(=O)[nH]c4s5
CN(C)CCNc1ccc(Nc2ncc3CCN(Cc3n2)c2cnc3OCCNc3c2C)cc1F
Cc1cc(Nc2cc3CN(CCc3cn2)c2cnc3OCCNc3c2Cl)ccc1NC(=O)CN1CCC1
Cc1cc(Nc2ncc3CCN(Cc3n2)c2cnc3OCCNc3c2C)ccc1NC(=O)CN1CCC1
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3ccc(NCCN4CCOCC4)c(F)c3)cc2C1
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3cnc(CS(C)(=O)=O)c(Cl)c3)nc2C1
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3ccc(NCCN4CCOCC4)c(F)c3)nc2C1
CC(C)N1CCc2cc(Nc3cc4CN(CCc4cn3)c3cnc4OCCNc4c3C)nn2CC1=O
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3ccc(NC(=O)C4(C)COC4)nc3)nc2C1
Cc1cc(Nc2cc3CN(CCc3cn2)c2cnc3OCCNc3c2C)ccc1NC(=O)CN1CCC1
Cc1cc(Nc2ncc3CCN(Cc3n2)c2cnc3OCCNc3c2C)ccc1NC(=O)CN1CCCC1
CN(C)[C@@H]1CCN(C1)C(=O)c1ccc(Nc2cc3CN(CCc3cn2)c2cnc3OCCNc3c2C)cc1 |r|
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3ccc(NC(=O)CN4CCOCC4)cc3)nc2C1
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3ccc4c(CNC4(C)C)c3)nc2C1
CN(C)CCNc1ccc(Nc2cc3CN(CCc3cn2)c2cnc3OCCNc3c2C)cc1C
Cc1cc(Nc2cc3CN(CCc3cn2)c2cnc3OCCNc3c2C)ccc1NCCN1CCOCC1
CN(C)CC(=O)Nc1ccc(Nc2ncc3CCN(Cc3n2)c2cnc3OCCNc3c2C)cc1C
CN(CCN1CCOCC1)c1ccc(Nc2ncc3CCN(Cc3n2)c2cnc3OCCNc3c2C)cc1C
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3ccc(nc3)C3(CC3)S(C)(=O)=O)nc2C1
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3cnc(CS(C)(=O)=O)c(F)c3)nc2C1
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3ccc(nc3)C(C)(C)S(C)(=O)=O)nc2C1
Cc1cc(Nc2ncc3CCN(Cc3n2)c2cnc3OCCNc3c2C)cnc1CS(C)(=O)=O
CN1CCc2cc(Nc3ncc4CCN(Cc4n3)c3cnc4OCCNc4c3C)nn2CC1=O
Cc1cc(Nc2ncc3CCN(Cc3n2)c2cnc3OCCNc3c2C)ccc1NCCN1CCOCC1
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3ccc(cc3)S(C)(=O)=O)nc2C1
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3ccc(OCS(C)(=O)=O)cc3)nc2C1
CN(C)CCNc1ccc(Nc2cc3CN(CCc3cn2)c2cnc3OCCNc3c2C)cn1
Cc1cc(Nc2cc3CN(CCc3cn2)c2cnc3OCCNc3c2C)ccc1C(=O)NCCN1CCOCC1
CN(C)CCNc1ncc(Nc2ncc3CCN(Cc3n2)c2cnc3OCCNc3c2C)cc1C
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3ccc(NC(=O)CN4CCOCC4)c(c3)C(F)(F)F)nc2C1
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3ccc4CN(CC(C)(C)O)Cc4c3)nc2C1
CN(C)CC(=O)Nc1ccc(Nc2cc3CN(CCc3cn2)c2cnc3OCCNc3c2C)cn1
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3ccc(NC(=O)CN4CCOCC4)nc3)cc2C1
CN(C)CC(=O)Nc1ccc(Nc2cc3CN(CCc3cn2)c2cnc3OCCNc3c2C)cc1C
Cc1cc(Nc2cc3CN(CCc3cn2)c2cnc3OCCNc3c2C)ccc1NC(=O)CN1CCOCC1
CN1CC(C1)NC(=O)c1ccc(Nc2ncc3CCN(Cc3n2)c2cnc3OCCNc3c2C)cc1C
Cc1cc(Nc2ncc3CCN(Cc3n2)c2cnc3OCCNc3c2C)cnc1NCCN1CCOCC1
CN1CCc2cc(Nc3cc4CN(CCc4cn3)c3cnc4OCCNc4c3Cl)nn2CC1=O
CN(C)C1CN(C1)C(=O)c1ccc(Nc2ncc3CCN(Cc3n2)c2cnc3OCCNc3c2C)cc1C
Cc1cc(Nc2ncc3CCN(Cc3n2)c2cnc3OCCNc3c2C)ccc1C(=O)NCCN1CCOCC1
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3ccc(CS(=O)(=O)C4CC4)nc3)nc2C1
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3ccc(CS(=O)(=O)CC4(C)COC4)cc3)nc2C1
CN(C)[C@@H]1CCN(C1)C(=O)c1ccc(Nc2ncc3CCN(Cc3n2)c2cnc3OCCNc3c2C)cc1 |r|
CN(CCN1CCOCC1)c1ncc(Nc2ncc3CCN(Cc3n2)c2cnc3OCCNc3c2C)cc1C
COCCNC(=O)c1ccc(Nc2ncc3CCN(Cc3n2)c2cnc3OCCNc3c2C)cc1
CNCc1cccc(Nc2ncc3CCN(Cc3n2)c2cnc3OCCNc3c2C)c1
CN1Cc2ccc(Nc3cc4CN(CCc4cn3)c3cnc4OCCNc4c3C)cc2C1
Cc1cc(Nc2ncc3CCN(Cc3n2)c2cnc3OCCNc3c2C)ccc1NC(=O)CN1CCOCC1
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3ccnc(CS(C)(=O)=O)c3)nc2C1
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3cccc(CS(C)(=O)=O)c3)nc2C1
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3ccc(CS(C)(=O)=O)nc3)cc2C1
CN1CCC(O)(CC1)c1ccc(Nc2cc3CN(CCc3cn2)c2cnc3OCCNc3c2C)cc1
CNCc1ccc(Nc2ncc3CCN(Cc3n2)c2cnc3OCCNc3c2C)cc1
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3ccnc(c3)N3CCOCC3)cc2C1
CN1CCN(CC1)c1ccc(Nc2ncc3CCN(Cc3n2)c2cnc3OCCNc3c2C)cc1
CN(C)CC(=O)Nc1ccc(Nc2ncc3CCN(Cc3n2)c2cnc3OCCNc3c2C)cn1
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3ccc(CS(C)(=O)=O)cc3)cc2C1
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3ccc(CS(C)(=O)=O)nc3)nc2C1
CN(C)Cc1ccc(Nc2ncc3CCN(Cc3n2)c2cnc3OCCNc3c2C)cc1
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3cccc(CN4CCOCC4)c3)nc2C1
CN1CCN(CC1)c1cccc(Nc2ncc3CCN(Cc3n2)c2cnc3OCCNc3c2C)c1
CN1CCc2ccc(Nc3ncc4CCN(Cc4n3)c3cnc4OCCNc4c3C)cc2CC1
CS(=O)(=O)Cc1ccc(Nc2ncc3CCN(Cc3n2)c2cnc3OCCNc3c2Cl)cc1
CN1CCN(Cc2ccc(Nc3ncc4CCN(Cc4n3)c3cnc4OCCNc4c3C)cc2)CC1
CN(C)Cc1cccc(Nc2ncc3CCN(Cc3n2)c2cnc3OCCNc3c2C)c1
CN1CCN(Cc2cccc(Nc3ncc4CCN(Cc4n3)c3cnc4OCCNc4c3C)c2)CC1
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3ccnc(c3)C(C)(C)O)nc2C1
CN1CCc2cc(Nc3cc4CN(CCc4cn3)c3cnc4OCCNc4c3C)nn2CC1=O
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3ccc(CS(C)(=O)=O)cc3)nc2C1
Cc1c2NCCOc2ncc1N1CCc2cnc(NC3CCN(Cc4cnn(C)c4)CC3)nc2C1
COC(=O)Nc1ccc(Nc2ncc3CCN(Cc3n2)c2cnc3OCCNc3c2C)cc1
CN1CCN(CC1)c1cc(Nc2ncc3CCN(Cc3n2)c2cnc3OCCNc3c2C)ccn1
CC(=O)Nc1ccc(Nc2ncc3CCN(Cc3n2)c2cnc3OCCNc3c2C)cn1
CNC(=O)c1ccc(Nc2ncc3CCN(Cc3n2)c2cnc3OCCNc3c2C)cc1F
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3ccnc(c3)S(C)(=O)=O)nc2C1
Cc1c(cnc2OCCNc12)N1CCc2cnc(Nc3ccnc(c3)C3CCOCC3)nc2C1
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3ccnc(c3)N3CCOCC3)nc2C1
COCc1cncc(c1)N1CCc2cnc(Nc3ccc(C4CCOCC4)c(CO)c3)nc2C1
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3cccc(c3)S(C)(=O)=O)nc2C1
CCc1cc(Nc2ncc3CCN(Cc3n2)c2cnc3OCCNc3c2C)ccc1N1CCC(O)CC1
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3ccc4CS(=O)(=O)Cc4c3)nc2C1
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3cccc(c3)C(C)(C)O)nc2C1
COCCOc1ccc(Nc2ncc3CCN(Cc3n2)c2cnc3OCCNc3c2C)cc1CO
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3ccc4COCCc4c3)nc2C1
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3ccc4C(=O)NCc4c3)nc2C1
CC(C)N1CCc2cc(Nc3ncc4CCN(Cc4n3)c3sncc3C)nn2CC1=O
CN1CCc2ncc(Nc3ncc4CCN(Cc4n3)c3cnc4OCCNc4c3)cc2C1
CN1CCc2ncc(Nc3ncc4CCN(Cc4n3)c3cnc4OCC(=O)Nc4c3C)cc2C1
CC(C)N1CCc2cc(Nc3ncc4CCN(Cc4n3)c3cnc4OCCNc4c3C)nn2CC1=O
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3ccc(OC[C@@H]4COCCO4)cc3)nc2C1 |r|
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3ccc(N4CCC(O)CC4)c(CC#N)c3)nc2C1
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3ccc4COCc4c3)nc2C1
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3ccc4COC(C)(C)c4c3)nc2C1
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3ccc(OC4CCOCC4)cc3)nc2C1
CN1CCc2ncc(Nc3ncc4CCN(Cc4n3)c3cnc4OCCOc4c3C)cc2C1
CN1Cc2cc(Nc3ncc4CCN(Cc4n3)c3cnc4OCCNc4c3C)ccc2C1=O
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3ccc(OCCN4CCOCC4)cc3)nc2C1
COCCOc1ccc(Nc2ncc3CCN(Cc3n2)c2cnc3OCCNc3c2C)cc1
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3ccc(CN4CCOCC4)cc3)nc2C1
CN1CCC(CC1)c1ccc(Nc2ncc3CCN(Cc3n2)c2cnc3OCCNc3c2C)cc1
CN1CCc2ncc(Nc3ncc4CCN(Cc4n3)c3cnc4OCCN(C)c4c3C)cc2C1
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3ccc(nc3)N3CCC(O)CC3)nc2C1
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3ccc(cc3)N3CCC(CC3)OC(F)(F)F)nc2C1
CN1Cc2ccc(Nc3ncc4CCN(Cc4n3)c3cnc4OCCNc4c3C)cc2C1
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3cnc4CCN(CC(F)F)Cc4c3)nc2C1
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3cnc4CCN(CC(F)(F)F)Cc4c3)nc2C1
CN1CCC(CC1)c1ccc(Nc2ncc3CCN(Cc3n2)c2cnc3OCCNc3c2C)cc1CO
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3cnc4CCNCc4c3)nc2C1
CN1CCc2ncc(Nc3cc4CN(CCc4cn3)c3cnc4OCCNc4c3C)cc2C1
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3cnc4CCC(O)Cc4c3)nc2C1
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3ccc(cc3)N3CCC(O)CC3)nc2C1
CN1CCC(CC1)c1ccc(Nc2ncc3CCN(Cc3n2)c2cnc3OCCNc3c2C)cc1CC#N
COC1CCN(CC1)c1ccc(Nc2ncc3CCN(Cc3n2)c2cnc3OCCNc3c2C)cc1
CN1CCc2ncc(Nc3ncc4CCN(Cc4n3)c3cnn(C)c3)cc2C1
CN1CCc2ncc(Nc3ncc4CCN(Cc4n3)c3cnc4OCCNc4c3C)cc2C1
CN1CCc2ncc(Nc3ncc4CCN(Cc4n3)c3cncc(N)c3C)cc2C1
COc1cccc(F)c1N1CCc2cnc(Nc3ccc(cc3)C3CCN(C)CC3)nc2C1
CN1CCc2ncc(Nc3ncc4CCN(Cc4n3)c3cnccc3C)cc2C1
CN1CCc2ncc(Nc3ncc4CCN(Cc4n3)c3sncc3C)cc2C1
COc1cccc(F)c1N1CCc2cnc(Nc3cnc4CCN(C)Cc4c3)nc2C1
Cc1cc(Nc2ncc3CCN(Cc3n2)c2cnc3OCCNc3c2Cl)ccc1NC(=O)CN1CCC1
Cc1cc(Nc2cc3CN(CCc3cn2)c2cnc3OCCNc3c2Cl)ccc1NC(=O)CN1CCOCC1
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3ccc(CN4CC(C)(O)C4)cc3)nc2C1
CN(C)CCNc1ccc(Nc2cc3CN(CCc3cn2)c2cnc3OCCNc3c2C)cc1F
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3ccc(CN4CCCC4)cc3)nc2C1
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3ccc(Cn4cncn4)cc3)nc2C1
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3ccc(Cn4ccnc4)cc3)nc2C1
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3ccc(CS(N)(=O)=O)cc3)nc2C1
CN1CCc2ncc(Nc3ncc4CCN(Cc4n3)c3ccccn3)cc2C1
CNC(=O)c1ccc(Nc2ncc3CCN(Cc3n2)c2cnc3OCCNc3c2Cl)cc1C
CN(C)C(=O)Cn1nc(Nc2cc3CN(CCc3cn2)c2cnc3OCCNc3c2Cl)cc1C
CS(=O)(=O)Cc1ccc(Nc2ncc3CCN(Cc3n2)c2cnc3OCCNc3c2C2CC2)cc1
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3ccc(CO)cc3)nc2C1
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3ccc(CCO)cc3)nc2C1
COCCS(=O)(=O)Cc1ccc(Nc2ncc3CCN(Cc3n2)c2cnc3OCCNc3c2C)cc1
CS(=O)(=O)Cc1ccc(Nc2ncc3CCN(Cc3n2)c2cnc3cnccn23)cc1
COCCOCCS(=O)(=O)Cc1ccc(Nc2ncc3CCN(Cc3n2)c2cnc3OCCNc3c2C)cc1
Cc1c(cnc2c(F)c[nH]c12)N1CCc2cnc(Nc3ccc(CS(C)(=O)=O)cc3)nc2C1
Cc1c2NCC3(CC3)Oc2ncc1N1CCc2cnc(Nc3ccc(CS(C)(=O)=O)cc3)nc2C1
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3cc4CCN(CC(F)F)C(=O)Cn4n3)cc2C1
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3cc4CCN(C5CC5)C(=O)Cn4n3)cc2C1
Cc1c(cnc2C(=O)CCNc12)N1CCc2cnc(Nc3ccc(CS(C)(=O)=O)cc3)nc2C1
Cc1c2NCCC(O)c2ncc1N1CCc2cnc(Nc3ccc(CS(C)(=O)=O)cc3)nc2C1
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3ccc(Cn4cncn4)cc3)cc2C1
CCc1c2NCCOc2ncc1N1CCc2cnc(Nc3ccc(CS(C)(=O)=O)cc3)nc2C1
Cn1ccc2c(ccnc12)N1CCc2cnc(Nc3ccc(CS(C)(=O)=O)cc3)nc2C1
COCCOCCS(=O)(=O)c1ccc(Nc2ncc3CCN(Cc3n2)c2cnc3OCCNc3c2C)cc1
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3ccc(CC#N)cc3)nc2C1
Cc1cc(Nc2ncc3CCN(Cc3n2)c2cnc3OCCNc3c2C)ccc1CC#N
CN(C)S(=O)(=O)Cc1ccc(Nc2cc3CN(CCc3cn2)c2cnc3OCCNc3c2C)cc1
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3ccc(CC(=O)N4CC(F)(F)C4)cc3)nc2C1
Cc1c2NCCOc2ncc1N1Cc2nc(Nc3ccc(CS(C)(=O)=O)cc3)ncc2C(F)(F)C1
COCCN1CCc2cc(Nc3cc4CN(CCc4cn3)c3cnc4OCCNc4c3C)nn2CC1=O
CN(C)CCS(=O)(=O)Cc1ccc(Nc2ncc3CCN(Cc3n2)c2cnc3OCCNc3c2C)cc1
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3ccc(CC(=O)N4CC(F)C4)cc3)nc2C1
CN1Cc2cc(Nc3ncc4CCN(Cc4n3)c3cnc4OCCNc4c3C)ccc2CS1(=O)=O
C[C@@H](c1ccc(Nc2ncc3CCN(Cc3n2)c2cnc3OCCNc3c2C)cc1)S(C)(=O)=O |r|
C[C@H](c1ccc(Nc2ncc3CCN(Cc3n2)c2cnc3OCCNc3c2C)cc1)S(C)(=O)=O |r|
Clc1c2NCCOc2ncc1N1CCc2cnc(Nc3ccc(cc3)-c3nnc(o3)C3CC3)nc2C1
Cc1c(cnc2oc(=O)[nH]c12)N1CCc2cnc(Nc3ccc(CS(C)(=O)=O)cc3)nc2C1
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3ccc(CCS(C)(=O)=O)cc3)nc2C1
COCCOCC(=O)Nc1ccc(Nc2ncc3CCN(Cc3n2)c2cnc3OCCNc3c2C)cc1C
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3ccc(CC(=O)N4CCC4)cc3)nc2C1
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3ccc(CC(=O)N4CC5(COC5)C4)cc3)nc2C1
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3ccc(CC(=O)N4CC(C4)N4CCOCC4)cc3)nc2C1
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3cccc(CS(C)(=N)=O)c3)nc2C1
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3ccc(cc3)[C@H]3CCCS3(=O)=O)cc2C1 |r|
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3ccc(cc3)[C@@H]3CCCS3(=O)=O)cc2C1 |r|
Cc1c(cnc2nc[nH]c12)N1CCc2cnc(Nc3ccc(CS(C)(=O)=O)cc3)cc2C1
COCCS(=O)(=O)Cc1ccc(Nc2cc3CN(CCc3cn2)c2cnc3OCCNc3c2C)cc1
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3ccc(CC(=O)N4CC(C)(O)C4)cc3)nc2C1
CC(C)OC1CN(C1)C(=O)Cc1ccc(Nc2ncc3CCN(Cc3n2)c2cnc3OCCNc3c2C)cc1
COCC1CN(C1)C(=O)Cc1ccc(Nc2ncc3CCN(Cc3n2)c2cnc3OCCNc3c2C)cc1
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3ccc(CS(=O)(=O)C4CC4)cn3)cc2C1
Cc1cc(Nc2ncc3CCN(Cc3n2)c2cnc3OCCNc3c2Cl)ccc1CS(C)(=O)=O
Cc1cc(Nc2ncc3CCN(Cc3n2)c2cnc3OCCNc3c2C)ccc1CS(C)(=O)=O
Cc1cc(Nc2cc3CN(CCc3cn2)c2cnc3OCCNc3c2C)ccc1CS(C)(=O)=O
CC1N(CCc2cnc(Nc3ccc(CS(C)(=O)=O)cc3)nc12)c1cnc2OCCNc2c1C
COC1CN(C1)C(=O)Cc1ccc(Nc2ncc3CCN(Cc3n2)c2cnc3OCCNc3c2C)cc1
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3ccc(cc3)C(C)(C)C#N)nc2C1
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3ccc(Cn4ccnn4)cc3)nc2C1
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3ccc(Cn4nccn4)cc3)nc2C1
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3ccc(cc3)C(C)(C)S(C)(=O)=O)nc2C1
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3ccc(Cn4cccn4)cc3)nc2C1
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3ccc(CN4CCOC4=O)cc3)nc2C1
CN(C)C(=O)Cc1ccc(Nc2ncc3CCN(Cc3n2)c2cnc3OCCNc3c2C)cc1
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3ccc(CS(C)(=O)=O)c(F)c3)nc2C1
Cc1c2NCCOc2ncc1N1CCc2cnc(Nc3cccc(Cn4ccnc4)c3)nc2C1
CN1CCC(CC1)c1ncc(s1)-c1cnc(N)c(OCc2ccncc2)n1
CN1CCC(CC1)c1ncc(s1)-c1cnc(N)c(OCc2ccncc2)c1
CN1CCC(CC1)c1ncc(s1)-c1cnc(N)c(OCc2cccc(c2)C#CC(C)(C)O)c1
CC(Oc1cc(cnc1N)-c1cnc(s1)C1CCN(C)CC1)c1ccncc1
CN1CCC(CC1)c1ncc(s1)-c1cnc(N)c(OCc2ccc(F)cc2)c1
CN1CCC(CC1)c1ncc(s1)-c1cnc(N)c(OC(C)(C)c2ccncc2)c1
Nc1ncc(cc1OCc1ccncc1)-c1cnc(s1)C1CCNCC1
CN1CCC(CC1)c1ncc(s1)-c1cnc(N)c(OCc2ccnc(Cl)c2)c1
COc1ccc(COc2cc(cnc2N)-c2cnc(s2)C2CCN(C)CC2)cc1
CN1CCC(CC1)c1ncc(s1)-c1cnc(N)c(OCc2ccnc(c2)C#CC(C)(C)O)c1
CN1CCC(CC1)c1ncc(s1)-c1cnc(N)c(OCc2cncc(c2)C#CC(C)(C)O)c1
CN1CCN(CC1)c1ncc(s1)-c1cnc(N)c(OCc2ccncc2)c1
Nc1ncc(cc1OCc1ccncc1)-c1cnc(s1)C1CCOCC1
CN1CCC(CC1)n1cc(c(N)n1)-c1cnc(N)c(OCc2ccncc2)n1
CN1CCC(CC1)c1nc(C)c(s1)-c1cnc(N)c(OCc2ccncc2)n1
CCC(C)(O)C#Cc1cccc(COc2cc(cnc2N)-c2cnc(s2)C2CCN(C)CC2)c1
CSc1ncc(s1)-c1cnc(N)c(OCc2cccc(c2)C#CC(C)(C)O)c1
CC(C)(O)C#Cc1cccc(COc2cc(cnc2N)-c2cnc(Oc3ccccc3)s2)c1
CN1CCC(CC1)c1ncc(s1)-c1cnc(N)c(OCc2cc(ccc2F)C#CC(C)(C)O)c1
CCC(C)c1ncc(s1)-c1cnc(N)c(OCc2cccc(c2)C#CC(C)(C)O)c1
CC(C)c1ncc(s1)-c1cnc(N)c(OCc2cc(ccc2F)C#CC(C)(C)O)c1
CC1CN(CCN1C)c1ncc(s1)-c1cnc(N)c(OCc2cccc(c2)C#CC(C)(C)O)c1
CC(C)(O)C#Cc1cccc(COc2cc(cnc2N)-c2cnc(s2)C2CCOCC2)c1
CN1CCCN(CC1)c1ncc(s1)-c1cnc(N)c(OCc2cccc(c2)C#CC(C)(C)O)c1
CN1CCN(CC1)c1ncc(s1)-c1cnc(N)c(OCc2cccc(c2)C#CC(C)(C)O)c1
CC1CN(CC(C)N1C)c1ncc(s1)-c1cnc(N)c(OCc2cccc(c2)C#CC(C)(C)O)c1
CC(C)(O)C#Cc1cccc(COc2cc(cnc2N)-c2cnc(s2)C2CCN(CC(F)(F)F)CC2)c1
CN1CCC(CC1)c1ncc(s1)-c1cnc(N)c(OCc2cccc(c2)C#CC2(O)CC2)c1
CC(C)(O)C#Cc1cccc(COc2cc(cnc2N)-c2cnc(s2)N2CCCCC2)c1
CC(C)(O)C#Cc1cccc(COc2cc(cnc2N)-c2cnc(s2)C2CCCCC2)c1
CC(C)(O)C#Cc1ccc(F)c(COc2cc(cnc2N)-c2cnc(s2)C2CCNCC2)c1
CN1CCC(CC1)n1cc(cn1)-c1cnc(N)c(OCc2cccc(c2)C#CC(C)(C)O)c1
CN1CCC(CC1)c1ncc(s1)-c1cnc(N)c(OCc2cccc(c2)C#CC(C)(O)C(F)(F)F)c1
CN1CCC(CC1)c1ncc(s1)-c1cnc(N)c(OCc2cccc(c2)C#CC2(O)CCCC2)c1
Cc1ncc(s1)-c1cnc(N)c(OCc2ccncc2)c1
CC(C)c1ncc(s1)-c1cnc(N)c(OCc2ccncc2)c1
Nc1ncc(cc1OCc1ccncc1)-c1cnc(s1)C1CCCCC1
CN1CCC(CC1)c1ncc(s1)-c1cnc(N)c(OCc2cccc(c2)C#CC2(O)CCCCC2)c1
CN1CCC(CC1)c1ncc(s1)-c1cnc(N)c(OCc2ccnc(c2)C#C)c1
CN1CCC(CC1)c1ncc(s1)-c1cnc(N)c(OCc2cccc(c2)C#CC2(O)CCC2)c1
CC(C)c1ncc(s1)-c1cnc(N)c(OCc2cccc(c2)C#CC(C)(C)O)c1
CC(C)(O)C#Cc1cccc(COc2cc(cnc2N)-c2cnc(s2)C2CCNCC2)c1
CN1CCC(CC1)c1ccc(nc1)-c1cnc(N)c(OCc2ccncc2)c1
CC(C)c1ncc(s1)-c1cnc(N)c(OCc2cncc(c2)C#CC(C)(C)O)c1
Nc1ncc(cc1OCc1cc(ccc1F)C#CC1(O)CC1)-c1cnc(s1)C1CCOCC1
Nc1ncc(cc1OCc1cccc(c1)C#CC1(O)CC1)-c1cnn(c1)C1CCOCC1
CN1CCC(CC1)c1ncc(s1)-c1cnc(N)c(OCc2cc(ccc2F)C#CC2(O)CC2)c1
CC(C)(O)C#Cc1cccc(COc2cc(cnc2N)-c2cnc(s2)C2CCCCN2)c1
Nc1ncc(cc1OCc1cccc(c1)C#CC1(O)CC1)-c1cnc(s1)C1CCOCC1
Nc1ncc(cc1OCc1cc(ccc1F)C#CC1(O)CC1)-c1cnn(c1)C1CCOCC1
Nc1ncc(cc1OCc1cccc(c1)C#CC1(O)CC1)-c1cnc(s1)C1CCNCC1
Nc1ncc(cc1OCc1cc(ccc1F)C#CC1(O)CC1)-c1cnc(s1)C1CCNCC1
Nc1ncc(cc1OCc1cccc(c1)C#CC1(O)CC1)-c1cnn(c1)C1CCNCC1
CN1CCC(CC1)c1ncc(s1)-c1cnc(N)c(OCc2cc(ccc2Cl)C#CC(C)(C)O)c1
CC(C)(O)C#Cc1cccc(COc2cc(cnc2N)-c2cnc(s2)C2CCCNC2)c1
CN1CCC(CC1)c1ncc(s1)-c1cnc(N)c(OCc2cc(F)cc(c2)C#CC(C)(C)O)c1
CN1CCC(CC1)c1ccnc(c1)-c1cnc(N)c(OCc2cccc(c2)C#CC(C)(C)O)c1
COc1ccc(cc1COc1cc(cnc1N)-c1cnc(s1)C1CCN(C)CC1)C#CC(C)(C)O
CN1CCC(CC1)c1ncc(s1)-c1cnc(N)c(OCc2cc(ccc2C)C#CC(C)(C)O)c1
CN1CCC(CC1)c1ncc(s1)-c1cnc(N)c(OCc2cccc(c2)C#CC2(O)CCCCC2=O)c1
CN1CCC(CC1)c1nc(C)c(s1)-c1cnc(N)c(OCc2cccc(c2)C#CC(C)(C)O)c1
CC1CN(C)CCN1c1ncc(s1)-c1cnc(N)c(OCc2cccc(c2)C#CC(C)(C)O)c1
CN1CCC(CC1)c1ncc(s1)-c1cnc(N)c(OCc2cccc(c2)C#CC(C)(O)C=C)c1
CN1CCC(CC1)c1ncc(s1)-c1cnc(N)c(OCc2cccc(c2)C#CC2(O)CCCC2=O)c1
CN1CCC(CC1)c1cnc(s1)-c1cnc(N)c(OCc2cccc(c2)C#CC(C)(C)O)c1
CC(C)c1ncc(s1)-c1cnc(N)c(OCc2cc(ccc2CN)C#CC(C)(C)O)c1
CN1CCN(CC1)C1CCN(CC1)c1ncc(s1)-c1cnc(N)c(OCc2cccc(c2)C#CC(C)(C)O)c1
CC(C)c1ncc(s1)-c1cnc(N)c(OCc2cc(CN)cc(c2)C#CC(C)(C)O)c1
CN1CCC(CC1)c1ncc(s1)-c1cnc(N)c(OCc2cc(C)cc(c2)C#CC(C)(C)O)c1
CN1CCC(C1)c1ncc(s1)-c1cnc(N)c(OCc2cccc(c2)C#CC(C)(C)O)c1
CN1CCC(CC1)n1cc(cn1)-c1cnc(N)c(OCc2cc(ccc2F)C#CC(C)(C)O)c1
CN1CCC(CC1)n1cc(cn1)-c1cnc(N)c(OCc2cccc(c2)C#CC(C)(O)CF)c1
CN1CCC(CC1)c1ncc(s1)-c1cnc(N)c(OCc2ccc(F)c(c2)C#CC(C)(C)O)c1
CN1CCC(CC1)c1ncc(s1)-c1cnc(N)c(OCc2cc(ccc2C(F)(F)F)C#CC(C)(C)O)c1
CN1CCC(CC1)c1ncc(s1)-c1cnc(N)c(OCc2cc(ccc2OC(F)F)C#CC(C)(C)O)c1
CC(C)(O)C#Cc1cccc(COc2cc(cnc2N)-c2cnn(c2)C2CCNCC2)c1
CC(C)(O)C#Cc1cccc(COc2cc(cnc2N)-c2cnn(c2)C2CCOCC2)c1
CC(C)(O)C#Cc1cc(CN)cc(COc2cc(cnc2N)-c2cnc(s2)C2CCOCC2)c1
CN(C)Cc1cc(COc2cc(cnc2N)-c2cnc(s2)C2CCOCC2)cc(c1)C#CC(C)(C)O
CN1CCC(CC1)c1ncc(s1)-c1cnc(N)c(OCc2cc(CN)cc(c2)C#CC(C)(C)O)c1
CC(C)(O)C#Cc1ccc(CN)c(COc2cc(cnc2N)-c2cnc(s2)C2CCOCC2)c1
Nc1ncc(cc1OCc1ccncc1)-c1cccc(c1)N1CCOCC1=O
CN(C)CCNC(=O)c1c(C)cc(cc1C)-c1cnc(N)c(Oc2cnn(c2)C2CCN(C)CC2)n1
CNS(=O)(=O)c1cc(C)cc(c1)-c1cnc(N)c(Oc2cnn(c2)C2CCN(C)CC2)n1
CNC(=O)c1c(C)cc(cc1C)-c1cnc(N)c(Oc2cnn(c2)C2CCN(C)CC2)n1
CN1CCC(CC1)n1cc(Oc2nc(cnc2N)-c2cc(C)c(C(=O)NCCN3CCCC3)c(C)c2)cn1
CN1CCC(CC1)n1cc(Oc2nc(cnc2N)-c2cc(C)c(C(=O)NCCN3CCCCC3)c(C)c2)cn1
CN1CCC(CC1)n1cc(Oc2nc(cnc2N)-c2cc(C)cc(c2)S(N)(=O)=O)cn1
CNS(=O)(=O)c1cc(OC)cc(c1)-c1cnc(N)c(Oc2cnn(c2)C2CCN(C)CC2)n1
CNS(=O)(=O)c1cc(cc(C)c1C)-c1cnc(N)c(Oc2cnn(c2)C2CCN(C)CC2)n1
CN1CCC(CC1)n1cc(Oc2nc(cnc2N)-c2cc(C)cc(c2)S(=O)(=O)NCCN2CCCCC2)cn1
CN1CCC(CC1)n1cc(Oc2nc(cnc2N)-c2cc(C)cc(c2)S(=O)(=O)NCCC#N)cn1
CN1CCC(CC1)n1cc(Oc2nc(cnc2N)-c2cc(C)cc(c2)C2(CC2)NS(C)(=O)=O)cn1
CN1CCC(CC1)n1cc(Oc2nc(cnc2N)-c2cc(C)cc(CCNS(C)(=O)=O)c2)cn1
CNS(=O)(=O)c1cc(C)cc(c1)-c1cnc(N)c(Oc2cnn(c2)C2CCNCC2)n1
CNS(=O)(=O)c1cc(C)cc(c1)-c1cnc(N)c(Oc2cnn(c2)[C@H]2C[C@@H]3CC[C@H](C2)N3C)n1 |r,TLB:32:31:28.27:24.30.25|
CCNS(=O)(=O)c1cc(C)cc(c1)-c1cnc(N)c(Oc2cnn(c2)C2CCN(C)CC2)n1
CNS(=O)(=O)c1cc(OC(C)C)cc(c1)-c1cnc(N)c(Oc2cnn(c2)C2CCN(C)CC2)n1
CN(C)CCNC(=O)c1cc(cc(C)c1C)-c1cnc(N)c(Oc2cnn(c2)C2CCN(C)CC2)n1
CNS(=O)(=O)c1cc(cc(F)c1C)-c1cnc(N)c(Oc2cnn(c2)C2CCN(C)CC2)n1
CN1CCC(CC1)n1cc(Oc2nc(cnc2N)-c2cc(C)c(CNS(C)(=O)=O)c(C)c2)cn1
CN1CCC(CC1)n1cc(Oc2nc(cnc2N)-c2cc(C)cc(c2)C2(CC2)NS(=O)(=O)c2ccccc2)cn1
CONC(=O)c1c(C)cc(cc1C)-c1cnc(N)c(Oc2cnn(c2)C2CCN(C)CC2)n1
CNc1cc(cc(c1)S(=O)(=O)NC)-c1cnc(N)c(Oc2cnn(c2)C2CCN(C)CC2)n1
CNS(=O)(=O)c1cc(cc(c1)-c1cnc(N)c(Oc2cnn(c2)C2CCN(C)CC2)n1)N1CCCC1
CNS(=O)(=O)c1cc(C)cc(c1)-c1cnc(N)c(Oc2cnn(c2)C2CCN(CC2)C2CC2)n1
CN1CCC(CC1)n1cc(Oc2nc(cnc2N)-c2cc(C)cc(c2)C2(CC2)NS(=O)(=O)CC(F)(F)F)cn1
CNC(=O)NCc1c(C)cc(cc1C)-c1cnc(N)c(Oc2cnn(c2)C2CCN(C)CC2)n1
CCN1CCC(CC1)n1cc(Oc2nc(cnc2N)-c2cc(C)cc(c2)S(=O)(=O)NC)cn1
CNS(=O)(=O)c1cc(C)cc(c1)-c1cnc(N)c(Oc2cnn(c2)C2CCN(CC3COC3)CC2)n1
CN1CCC(CC1)n1cc(Oc2nc(cnc2N)-c2cc(C)c(C3COC(=O)N3)c(C)c2)cn1
CNS(=O)(=O)c1cc(cc(c1)C(C)(C)C)-c1cnc(N)c(Oc2cnn(c2)C2CCN(C)CC2)n1
CN1CCC(CC1)n1cc(Oc2nc(cnc2N)-c2cc(C)c(CNS(=O)(=O)C3CCOCC3)c(C)c2)cn1
CN1CCC(CC1)n1cc(Oc2nc(cnc2N)-c2cc(C)c(CNS(=O)(=O)C3CC3)c(C)c2)cn1
CN(C)CCNC(=O)c1c(C)cc(cc1C(F)F)-c1cnc(N)c(Oc2cnn(c2)C2CCN(C)CC2)n1
CN1CCC(CC1)n1cc(Oc2nc(cnc2N)-c2cc(C)c(C(=O)NCCN3CC[C@@H](F)C3)c(C)c2)cn1 |r|
CN1CCC(CC1)n1cc(Oc2nc(cnc2N)-c2cc(C)c(C3COCC(=O)N3)c(C)c2)cn1
CCNC(=O)NCc1c(C)cc(cc1C)-c1cnc(N)c(Oc2cnn(c2)C2CCN(C)CC2)n1
CN1CCC(CC1)n1cc(Oc2nc(cnc2N)-c2cc(C)c(CNC(=O)NC3CCCC3)c(C)c2)cn1
CN1CCC(CC1)n1cc(Oc2nc(cnc2N)-c2cc(C)c(CNS(=O)(=O)c3ccccc3)c(C)c2)cn1
COc1ccc(cc1)S(=O)(=O)NCc1c(C)cc(cc1C)-c1cnc(N)c(Oc2cnn(c2)C2CCN(C)CC2)n1
CN1CCC(CC1)n1cc(Oc2nc(cnc2N)-c2cc(C)c(CNS(=O)(=O)C3CCCC3)c(C)c2)cn1
CNS(=O)(=O)c1cc(cc(c1)-c1cnc(N)c(Oc2cnn(c2)C2CCN(C)CC2)n1)N1CCCCC1
CNS(=O)(=O)c1cc(cc(c1)-c1cnc(N)c(Oc2cnn(c2)C2CCN(C)CC2)n1)N1CCOCC1
CNS(=O)(=O)c1cc(cc(c1)-c1cnc(N)c(Oc2cnn(c2)C2CCN(C)CC2)n1)N1CCC[C@H]1C |r|
CN1CCC(CC1)n1cc(Oc2nc(cnc2N)-c2cc(C)c(CNC(=O)c3ccccc3)c(C)c2)cn1
CN1CCC(CC1)n1cc(Oc2nc(cnc2N)-c2cc(C)c(CNC(C)=O)c(C)c2)cn1
CN1CCC(CC1)n1cc(Oc2nc(cnc2N)-c2ccc(CNS(C)(=O)=O)c(C)c2)cn1
CNC(=O)NCc1ccc(cc1C)-c1cnc(N)c(Oc2cnn(c2)C2CCN(C)CC2)n1
CN1CCC(CC1)n1cc(Oc2nc(cnc2N)-c2cc(C)c(CNCC(F)(F)F)c(C)c2)cn1
CNS(=O)(=O)c1cc(cc(c1)-c1cnc(N)c(Oc2cnn(c2)C2CCN(C)CC2)n1)N1CCOC[C@H]1C |r|
CN1CCC(CC1)n1cc(Oc2nc(cnc2N)-c2cc(C)cc(c2)[Si](C)(C)O)cn1
CN1CCC(CC1)n1cc(Oc2nc(cnc2N)-c2cc(C)c(CNC(=O)NCC(F)(F)F)c(C)c2)cn1
CN1CCC(CC1)n1cc(Oc2nc(cnc2N)-c2cc(C)cc(c2)C(C)(C)O)cn1
CN1CCC(CC1)n1cc(Oc2nc(cnc2N)-c2cc(C)c(CNC(=O)NC(C)(C)C)c(C)c2)cn1
CN1CCC(CC1)n1cc(Oc2nc(cnc2N)-c2cc(C)cc(c2)C2(O)COC2)cn1
CN1CCC(CC1)n1cc(Oc2nc(cnc2N)-c2cc(C)c(CNC3COC3)c(C)c2)cn1
CN1CCC(CC1)n1cc(Oc2nc(cnc2N)-c2cc(C)c(CNc3ccn(C)n3)c(C)c2)cn1
CN1CCC(CC1)n1cc(Oc2nc(cnc2N)-c2cc(C)c(CNc3cnn(C)c3)c(C)c2)cn1
CN1CCC(CC1)n1cc(Oc2nc(cnc2N)-c2cc(C)cc(c2)C2(O)CCOCC2)cn1
C[C@@H]1COCCN1c1cc(cc(c1)C1(O)COC1)-c1cnc(N)c(Oc2cnn(c2)C2CCN(C)CC2)n1 |r|
CN1CCC(CC1)n1cc(Oc2nc(cnc2N)-c2cc(C)c(CNC3(C)COC3)c(C)c2)cn1
CN1CCC(CC1)n1cc(Oc2nc(cnc2N)-c2cc(C)cc(c2)[C@@H]2CCC(=O)N2)cn1 |r|
CN1CCC(CC1)n1cc(Oc2nc(cnc2N)-c2cc(C)cc(c2)[C@H]2CCC(=O)N2)cn1 |r|
CN(C)S(=O)(=O)NCc1c(C)cc(cc1C)-c1cnc(N)c(Oc2cnn(c2)C2CCN(C)CC2)n1
CN1CCC(CC1)n1cc(Oc2nc(cnc2N)-c2cc(C)c(c(C)c2)C2(O)COC2)cn1
CN1CCC(CC1)n1cc(Oc2nc(cnc2N)-c2cc(C)c(CNC(=O)NC3(CC3)C(F)(F)F)c(C)c2)cn1
CN1CCC(CC1)n1cc(Oc2nc(cnc2N)-c2cc(C)cc(c2)C2(O)CCCC2)cn1
CN1CCC(CC1)n1cc(Oc2nc(cnc2N)-c2cc(C)c(N3CCOCC3)c(C)c2)cn1
CN1CCC(CC1)n1cc(Oc2nc(cnc2N)-c2cc(C)c(CNc3ncco3)c(C)c2)cn1
CN1CCC(CC1)n1cc(Oc2nc(cnc2N)-c2cc(C)c(CNc3ncn(C)n3)c(C)c2)cn1
CN1CCC(CC1)n1cc(Oc2nc(cnc2N)-c2cc(C)cc(c2)C2(O)CCOC2)cn1
CN1CCC(CC1)n1cc(Oc2nc(cnc2N)-c2cc(C)cc(c2)C(C)(O)CO)cn1
CN1CCC(CC1)n1cc(Oc2nc(cnc2N)-c2cc(C)c(CNS(=O)(=O)N3CCOCC3)c(C)c2)cn1
CN1CCC(CC1)n1cc(Oc2nc(cnc2N)-c2cc(cc(c2)C2(O)COC2)N2CCOCC2)cn1
CN1CCC(CC1)n1cc(Oc2nc(cnc2N)-c2cc(C)c(C)c(c2)C2(O)COC2)cn1
CN1CCC(CC1)n1cc(Oc2nc(cnc2N)-c2cc(C)cc(c2)[C@]2(O)CCOC2)cn1
CN1CCC(CC1)n1cc(Oc2nc(cnc2N)-c2cc(C)cc(c2)[C@@]2(O)CCOC2)cn1
CN1CCC(CC1)n1cc(Oc2nc(cnc2N)-c2cc(C)c(C3=CCOCC3)c(C)c2)cn1 |t:25|
COC[C@@H]1COCCN1c1cc(cc(c1)C1(O)COC1)-c1cnc(N)c(Oc2cnn(c2)C2CCN(C)CC2)n1 |r|
CN1CCC(CC1)n1cc(Oc2nc(cnc2N)-c2cc(C)c(N3CC4(COC4)C3)c(C)c2)cn1
CN1CCC(CC1)n1cc(Oc2nc(cnc2N)-c2cc(cc(c2)C2(O)COC2)N2CC3(COC3)C2)cn1
CN1CCC(CC1)n1cc(Oc2nc(cnc2N)-c2cc(cc(c2)C2(O)COC2)C2CCOCC2)cn1
C[C@@H]1COCCN1c1cc(cc(c1)[C@]1(O)CCOC1)-c1cnc(N)c(Oc2cnn(c2)C2CCN(C)CC2)n1
C[C@H]1COCCN1c1cc(cc(c1)[C@]1(O)CCOC1)-c1cnc(N)c(Oc2cnn(c2)C2CCN(C)CC2)n1
CC#Cc1c(C)cc(cc1C1(O)COC1)-c1cnc(N)c(Oc2cnn(c2)C2CCN(C)CC2)n1
COCc1cc(cc(c1)C1(O)COC1)-c1cnc(N)c(Oc2cnn(c2)C2CCN(C)CC2)n1
CN1CCC(CC1)n1cc(Oc2nc(cnc2N)-c2cc(C)c(N3CC4(COC4)C3)c(c2)C2(O)CCOC2)cn1
CN1CCC(CC1)n1cc(Oc2nc(cnc2N)-c2cc(C)c(Cl)c(c2)C2(O)COC2)cn1
CN1CCC(CC1)n1cc(Oc2nc(cnc2N)-c2cc(cc(c2)C2(O)COC2)N2CCC[C@H]2CO)cn1 |r|
CN1CCC(CC1)n1cc(Oc2nc(cnc2N)-c2cc(C)c(C3=CCOCC3)c(c2)C2(O)COC2)cn1 |t:25|
CN1CCC(CC1)n1cc(Oc2nc(cnc2N)-c2cc(C)c(C3OCCO3)c(c2)C2(O)COC2)cn1
CN1CCC(CC1)n1cc(Oc2nc(cnc2N)-c2cc(C)cc(c2)C2(O)CCCOC2)cn1
C[C@@H]1COCCN1c1cc(cc(c1)C1(O)CCCOC1)-c1cnc(N)c(Oc2cnn(c2)C2CCN(C)CC2)n1 |r|
C[C@H]1COCCN1c1cc(cc(c1)[C@@]1(O)CCCOC1)-c1cnc(N)c(Oc2cnn(c2)C2CCN(C)CC2)n1
C[C@@H]1COCCN1c1cc(cc(c1)[C@@]1(O)CCCOC1)-c1cnc(N)c(Oc2cnn(c2)C2CCN(C)CC2)n1
CN1CCC(CC1)n1cc(Oc2nc(cnc2N)-c2cc(cc(c2)C2(O)COC2)N2CCCC2=O)cn1
CN1CCC(CC1)n1cc(Oc2nc(cnc2N)-c2cc(C)c(N3CC4(C3)CCOCC4)c(c2)C2(O)CCOC2)cn1
CN1CCC(CC1)n1cc(Oc2nc(cnc2N)-c2cc(C)c(F)c(c2)C2(O)CCOC2)cn1
CC1OCCC1(O)c1cc(cc(c1)-c1cnc(N)c(Oc2cnn(c2)C2CCN(C)CC2)n1)N1CCOC[C@H]1C |r|
C[C@H]1OCC[C@]1(O)c1cc(cc(c1)-c1cnc(N)c(Oc2cnn(c2)C2CCN(C)CC2)n1)N1CCOC[C@H]1C
C[C@@H]1OCC[C@@]1(O)c1cc(cc(c1)-c1cnc(N)c(Oc2cnn(c2)C2CCN(C)CC2)n1)N1CCOC[C@H]1C
CN1CCC(CC1)n1cc(Oc2nc(cnc2N)-c2cc(C)c(N3CCOCC3)c(c2)C2(O)CCOC2)cn1
CN1CCC(CC1)n1cc(Oc2nc(cnc2N)-c2cc(C)c(N3CCOCC3)c(c2)[C@@]2(O)CCOC2)cn1
CN1CCC(CC1)n1cc(Oc2nc(cnc2N)-c2cc(C)c(N3CCOCC3)c(c2)[C@]2(O)CCOC2)cn1
CN1CCC(CC1)n1cc(Oc2nc(cnc2N)-c2cc(cc(c2)C2(O)CCOC2)N2CCCOCC2)cn1
CCN(CC)c1cc(cc(CNC)n1)-c1cnc(N)c(Oc2cnn(c2)C2CCN(C)CC2)n1
CNCc1cc(cc(n1)N1CCC[C@H]1C)-c1cnc(N)c(Oc2cnn(c2)C2CCN(C)CC2)n1 |r|
C[C@@H]1COCCN1c1cc(cc(n1)C(C)(C)O)-c1cnc(N)c(Oc2cnn(c2)C2CCN(C)CC2)n1 |r|
C[C@@H]1COCCN1c1cc(cc(n1)C1(O)COC1)-c1cnc(N)c(Oc2cnn(c2)C2CCN(C)CC2)n1 |r|
CCn1cc(-c2cc(N)c3nnc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)cn1
COc1ccncc1-c1cc(N)c2nnc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1
CCc1ccncc1-c1cc(N)c2nnc(NC3CCOC3)cc2c1
N#Cc1ccncc1-c1cc(N)c2nnc(NC(=O)C3CC3F)cc2c1
Cc1cc(N)ncc1-c1cc(N)c2nnc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1
CCc1cc(N)c2nnc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1
Nc1cc(C2CC2)cc2cc(NC(=O)C3CC3F)nnc12
CC(C)NC(=O)Nc1cc2cc(-c3cnn(C)c3)cc(N)c2nn1
CC(C)OC(=O)Nc1cc2cc(-c3cnn(C)c3)cc(N)c2nn1
Cn1cc(-c2cc(N)c3nnc(NC(=O)N4CCCC4)cc3c2)cn1
CCc1ccncc1-c1cc(N)c2nnc(NC(=O)NC(C)C)cc2c1
CCc1ccncc1-c1cc(N)c2nnc(NC(=O)NC3CCOC3)cc2c1
CCc1ccncc1-c1cc(N)c2nnc(NC(=O)N3CCCC3)cc2c1
CCc1ccncc1-c1cc(N)c2nnc(NC(=O)NCC(F)(F)F)cc2c1
Cc1cnsc1-c1cc(N)c2nnc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1
CCc1ccncc1-c1cc(N)c2nnc(NC(C)C)cc2c1
Cc1cnccc1-c1cc(N)c2nnc(NC(=O)[C@@H]3C[C@@H]3F)cc2c1
Cn1cc(-c2cc(N)c3nnc(NC(=O)[C@@H]4C[C@@H]4F)cc3c2)cn1
Cn1cc(-c2cc(N)c3nnc(NC(=O)C4CC4C#N)cc3c2)cn1
CCc1ccncc1-c1cc(N)c2nnc(NC(=O)C3CC3C#N)cc2c1
CCc1ccncc1-c1cc(N)c2nnc(NC(=O)C3CC3F)cc2c1
Nc1cc(-c2cnccc2C2CC2)cc2cc(NC(=O)C3CC3F)nnc12
Cc1c(N)cncc1-c1cc(N)c2nnc(NC(=O)[C@@H]3C[C@H]3C#N)cc2c1
Cc1c(N)cncc1-c1cc(N)c2nnc(NC(=O)[C@H]3C[C@@H]3C#N)cc2c1
Cc1ccncc1-c1cc(C)c2nnc(NC(=O)C3CC3)cc2c1
Cc1ccncc1-c1cc(N)c2nnc(NC(=O)C3CC3)cc2c1
Cc1ccncc1-c1cc(Cl)c2nnc(NC(=O)C3CC3)cc2c1
Cc1ccncc1-c1ccc2nnc(NC(=O)C3CC3)cc2c1
Cc1c(N)cncc1-c1ccc2nnc(Nc3cc4n(n3)CC(=O)N(C(C)C)CC4)cc2c1
Cc1c(N)cncc1-c1cc(N)c2nnc(Nc3cc4n(n3)CC(=O)N(C(C)C)CC4)cc2c1
Cn1cnc2c(-c3cnc(Nc4ccc(N5CCOCC5)cc4)c(C(N)=O)n3)cccc21
Cc1nc(Nc2ccc(N3CCOCC3)cc2)c(C(N)=O)nc1-c1cccc2c1ncn2C
COc1nc(Nc2ccc(N3CCOCC3)cc2)c(C(N)=O)nc1-c1cccc2c1ncn2C
CN(C)CCOc1nc(Nc2ccc(N3CCOCC3)cc2)c(C(N)=O)nc1-c1cccc2c1ncn2C
Cn1cnc2c(-c3nc(C(N)=O)c(Nc4ccc(N5CCOCC5)cc4)nc3C3CC3)cccc21
Cc1nc(Nc2ccc(N3CCOCC3)cc2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(N3CCOCC3)cc2)c(C(N)=O)nc1-c1cccc2c1ncn2C
CNc1nc(Nc2ccc(N3CCOCC3)cc2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CSc1nc(Nc2ccc(N3CCOCC3)cc2)c(C(N)=O)nc1-c1cccc2c1ncn2C
CCNc1nc(Nc2ccc(N3CCOCC3)cc2)c(C(N)=O)nc1-c1cccc2c1ncn2C
Cn1cnc2c(-c3nc(C(N)=O)c(Nc4ccc(N5CCOCC5)cc4)nc3NC3CC3)cccc21
Cn1cnc2c(-c3nc(C(N)=O)c(Nc4ccc(N5CCOCC5)cc4)nc3N)cccc21
C[C@@H](O)CNc1nc(Nc2ccc(N3CCOCC3)cc2)c(C(N)=O)nc1-c1cccc2c1ncn2C
C[C@H](O)CNc1nc(Nc2ccc(N3CCOCC3)cc2)c(C(N)=O)nc1-c1cccc2c1ncn2C
Cn1cnc2c(-c3nc(C(N)=O)c(Nc4ccc(N5CCOCC5)cc4)nc3NCC(F)(F)F)cccc21
Cn1cnc2c(-c3nc(C(N)=O)c(Nc4ccc(N5CCOCC5)cc4)nc3NCC(F)F)cccc21
CN(C)CCNc1nc(Nc2ccc(N3CCOCC3)cc2)c(C(N)=O)nc1-c1cccc2c1ncn2C
Cn1cnc2c(-c3nc(C(N)=O)c(Nc4ccc(N5CCOCC5)cc4)nc3NCCO)cccc21
C#CCNc1nc(Nc2ccc(N3CCOCC3)cc2)c(C(N)=O)nc1-c1cccc2c1ncn2C
C[C@@H]1C[C@H]1Nc4nc(Nc3ccc(N2CCOCC2)cc3)c(C(N)=O)nc4c5cccc6c5ncn6C
C[C@H]1C[C@@H]1Nc4nc(Nc3ccc(N2CCOCC2)cc3)c(C(N)=O)nc4c5cccc6c5ncn6C
Cn1cnc2c(-c3nc(C(N)=O)c(Nc4ccc(N5CCOCC5)cc4)nc3NCC#N)cccc21
C[C@@H](F)CNc1nc(Nc2ccc(N3CCOCC3)cc2)c(C(N)=O)nc1-c1cccc2c1ncn2C
C[C@H](F)CNc1nc(Nc2ccc(N3CCOCC3)cc2)c(C(N)=O)nc1-c1cccc2c1ncn2C
Cn1cnc2c(-c3nc(C(N)=O)c(Nc4ccc(N5CCOCC5)cc4)nc3NCC3COC3)cccc21
C#Cc1nc(Nc2ccc(N3CCOCC3)cc2)c(C(N)=O)nc1-c1cccc2c1ncn2C
Cn1cnc2c(-c3nc(C(N)=O)c(Nc4ccc(N5CCOCC5)cc4)nc3C(F)F)cccc21
Cn1cnc2c(-c3nc(C(N)=O)c(Nc4ccc(N5CCOCC5)cc4)nc3Cl)cccc21
Cn1cc(Nc2nc(Nc3ccc(N4CCOCC4)cc3)c(C(N)=O)nc2-c2cccc3c2ncn3C)cn1
Cn1cnc2c(-c3nc(C(N)=O)c(Nc4ccc(N5CCOCC5)cc4)nc3Nc3ccccn3)cccc21
Cn1cnc2c(-c3nc(C(N)=O)c(Nc4ccc(N5CCOCC5)cc4)nc3C3COC3)cncc21
CCOc1nc(Nc2ccc(N3CCOCC3)cc2)c(C(N)=O)nc1-c1cncc2c1ncn2C
Cn1cnc2c(-c3nc(C(N)=O)c(Nc4ccc(N5CCOCC5)cc4)nc3C(F)(F)F)cncc21
CSc1nc(Nc2ccc(N3CCOCC3)cc2)c(C(N)=O)nc1-c1cncc2c1ncn2C
Cn1cnc2c(-c3nc(C(N)=O)c(Nc4ccc(N5CCOCC5)cc4)nc3NC3(C)CC3)cncc21
Cn1cnc2c(-c3nc(C(N)=O)c(Nc4ccc(N5CCOCC5)cc4)nc3C#N)cncc21
Cn1cnc2c(-c3nc(C(N)=O)c(Nc4ccc(N5CCOCC5)cc4)nc3NC3CC3)cncc21
Cn1cnc2c(-c3nc(C(N)=O)c(Nc4ccc(N5CCOCC5)cc4)nc3N)cncc21
Cn1cnc2c(-c3cnc(Nc4ccc(N5CCOCC5)cc4)c(C(N)=O)n3)cncc21
COc1nc(Nc2ccc(N3CCOCC3)cc2)c(C(N)=O)nc1-c1cncc2c1ncn2C
Cn1cnc2c(-c3nc(C(N)=O)c(Nc4ccc(N5CCOCC5)cc4)nc3C3CC3)cncc21
Cn1cnc2c(-c3nc(C(N)=O)c(Nc4ccc(N5CCOCC5)cc4)nc3C(F)F)cncc21
Cc1nc(Nc2ccc(N3CCOCC3)cc2)c(C(N)=O)nc1-c1nncc2c1ncn2C
Cc1nc(Nc2ccc(N3CCOCC3)cc2)c(C(N)=O)nc1-c1cnnc2c1ncn2C
CNc1nc(Nc2ccc(N3CCOCC3)cc2)c(C(N)=O)nc1-c1cnnc2c1ncn2C
CCn1cnc2c(-c3nc(C(N)=O)c(Nc4ccc(N5CCOCC5)cc4)nc3NC)cncc21
CNc1nc(Nc2ccc(N3CCOCC3)cc2)c(C(N)=O)nc1-c1cncc2c1ncn2C1CC1
CNc1nc(Nc2ccc(N3CCOCC3)cc2)c(C(N)=O)nc1-c1cncc2c1ncn2C(F)F
CNc1nc(Nc2ccc(N3CCOCC3)cc2)c(C(N)=O)nc1-c1ccc(Cl)c2c1ncn2C
CNc1nc(Nc2ccc(N3CCOCC3)cc2)c(C(N)=O)nc1-c1ccc(C#N)c2c1ncn2C
CNc1nc(Nc2ccc(N3CCOCC3)cc2)c(C(N)=O)nc1-c1cnc(C)c2c1ncn2C
CNc1nc(Nc2ccc(N3CCOCC3)cc2F)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(N3CCOCC3)c(F)c2F)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(N3CCOCC3)c(C)c2F)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(N3CCOCC3)c(Cl)c2F)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2cc(F)c(N3CCOCC3)c(F)c2F)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2cc(C)c(N3CCOCC3)cc2F)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2cc(F)c(N3CCOCC3)c(F)c2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(N3CCOCC3)c(Cl)c2)c(C(N)=O)nc1-c1cccc2c1ncn2C
CNc1nc(Nc2ccc(N3CCOCC3)c(Cl)c2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(N3CCOCC3)c(C)c2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2cc(C)c(N3CCOCC3)c(C)c2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(N3CCOCC3)c(C#N)c2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(N3CCOCC3)c(OC)c2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(N3CCOCC3)c(C(F)F)c2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(N3CCOCC3)cc2C)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(N3CCOCC3)cc2OC)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(N3CCOCC3)cc2Cl)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2cnc(N3CCOCC3)c(C)c2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2cnc(N3CCOC[C@@H]3C)c(C)c2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2cnc(N3CCO[C@@H](C)C3)c(C)c2)c(C(N)=O)nc1-c1cncc2c1ncn2C
C[C@@H]1COCCN1c1ccc(Nc2nc(C3CC3)c(-c3cncc4c3ncn4C)nc2C(N)=O)cn1
CNc1nc(Nc2cnc(N3CCOCC3)c(C#N)c2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(N3CCCOCC3)cc2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2cnc(N3CCOC[C@H]3C)c(C)c2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(N3C[C@H]4C[C@@H]3CO4)cc2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(N3C[C@@H]4C[C@H]3CO4)cc2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(N3C[C@@H]4C[C@H]3CO4)cc2F)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(N3C[C@@H]4C[C@H]3CO4)c(F)c2F)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2cc(F)c(N3C[C@@H]4C[C@H]3CO4)c(F)c2F)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(N3CC4CC(C3)O4)cc2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(N3CC4CCC(C3)O4)cc2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(N3CC4(COC4)C3)cc2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccccc2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(OC(F)F)cc2)c(C(N)=O)nc1-c1cncc2c1ncn2C
Cn1cnc2c(-c3nc(C(N)=O)c(Nc4ccc(C(C)(C)O)cc4)nc3C3CC3)cncc21
CNc1nc(Nc2ccc(OC(C)C)cc2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(OS(C)(=O)=O)cc2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(OCCOC)cc2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(OCCN(C)C)cc2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(OCCO)cc2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(OCCN3CCOCC3)cc2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(N)cc2)c(C(N)=O)nc1-c1cccc2c1ncn2C
CNc1nc(Nc2ccc(N(C)CCOC)cc2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(N(CCOC)CCOC)cc2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccnc(C)c2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccnc(OC)c2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2cc(C)nc(OC)c2)c(C(N)=O)nc1-c1cnnc2c1ncn2C
CNc1nc(Nc2cc(C)nc(C)c2)c(C(N)=O)nc1-c1cncc2c1ncn2C
Cc1cc(Nc2nc(C3CC3)c(-c3cncc4c3ncn4C)nc2C(N)=O)cc(C)n1
CNc1nc(Nc2cc(C)nc(OC)c2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2cc(C)nc(OCCOC)c2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2cc(C)nc(C#N)c2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2cc(C)c(=O)n(C)c2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(=O)n(C(F)F)c2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(N3C[C@H]4C[C@@H]3CN4C)cc2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(N3CC4CCC(C3)N4C)cc2)c(C(N)=O)nc1-c1cncc2c1ncn2C
C[C@@H]1CN(c2ccc(Nc3nc(C(F)(F)F)c(-c4cncc5c4ncn5C)nc3C(N)=O)cc2)C[C@H](C)N1
CNc1nc(Nc2cc(F)c(N3C[C@@H](C)N[C@@H](C)C3)c(F)c2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(N3C4CCC3CN(C)C4)cc2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(N3C[C@@H]4C[C@H]3CN4C)cc2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2cc(C)c(N3C[C@@H](C)N[C@@H](C)C3)c(C)c2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(N(C)CCN(C)C)cc2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(N3CC(N(C)C)C3)cc2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(N3C[C@@H](C)N[C@@H](C)C3)c(C#N)c2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(N3CCC(N4CCN(C)CC4)CC3)c(F)c2F)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2cnc(N3CCN(C(C)C)CC3)c(C)c2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2cnc(N3CCN(C)CC3)c(OC)c2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2cnc(N3C[C@H]4C[C@@H]3CN4C)c(C)c2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2cnc(N3C[C@H]4C[C@@H]3CN4C)c(Cl)c2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2cnc3c(c2)CN(C)C3)c(C(N)=O)nc1-c1cncc2c1ncn2C
CCN1Cc2cc(Nc3nc(NC)c(-c4cncc5c4ncn5C)nc3C(N)=O)cnc2C1
CNc1nc(Nc2cnc3c(c2)CN(C(C)C)C3)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(CN(C)C)cc2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(CN3CCCC3)cc2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(CN3CCOCC3)cc2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(CN3CCN(C)CC3)cc2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(CN3CC4(COC4)C3)cc2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc3nc(Nc2ccc([C@@H](C)N1CCN(C)CC1)cc2)c(C(N)=O)nc3c4cncc5c4ncn5C
CNc3nc(Nc2ccc([C@H](C)N1CCN(C)CC1)cc2)c(C(N)=O)nc3c4cncc5c4ncn5C
CNc3nc(Nc2ccc([C@@H](C)N1CCOCC1)cc2)c(C(N)=O)nc3c4cncc5c4ncn5C
CNc3nc(Nc2ccc([C@H](C)N1CCOCC1)cc2)c(C(N)=O)nc3c4cncc5c4ncn5C
CNc1nc(Nc2ccc(C(C)(C)N3CCN(C)CC3)cc2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(C(C)(C)N3CCOCC3)cc2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(CN3CC[C@@H](F)C3)cc2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(CN3CC[C@H](F)C3)cc2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(CN3CCC(F)(F)C3)cc2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(CN3CCN(C)[C@@H](C)C3)cc2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(CN3CCN(C)[C@H](C)C3)cc2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(CN3CCOCC3)nc2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(CN3CCN(C)CC3)cc2F)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(CN3CCN(C)CC3)c(Cl)c2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(CN3CCOCC3)cc2F)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(CN3CCOCC3)c(F)c2F)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(CN3C[C@@H]4C[C@H]3CO4)cc2F)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(CN3C[C@H]4C[C@@H]3CO4)cc2F)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(CN3C[C@H]4C[C@@H]3CO4)c(F)c2F)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(CN3CC4(COC4)C3)cc2Cl)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(CCN3CCOCC3)cc2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(CCN3CCN(C)CC3)cc2)c(C(N)=O)nc1-c1cncc2c1ncn2C
Cn1cnc2c(-c3nc(C(N)=O)c(Nc4ccc(CN5CCCC5)cc4)nc3C3CC3)cncc21
CN1CCN(Cc2ccc(Nc3nc(C4CC4)c(-c4cncc5c4ncn5C)nc3C(N)=O)cc2)CC1
COc1nc(Nc2ccc(CN3CCN(C)CC3)cc2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CN1CCN(Cc2ccc(Nc3nc(C(F)F)c(-c4cncc5c4ncn5C)nc3C(N)=O)cc2)CC1
Cn1cnc2c(-c3nc(C(N)=O)c(Nc4ccc(CN5CCOCC5)cc4)nc3C(F)F)cncc21
COc1nc(Nc2ccc(CN3CCOCC3)cc2F)c(C(N)=O)nc1-c1cncc2c1ncn2C
COc1nc(Nc2ccc(CN3CCOCC3)c(F)c2F)c(C(N)=O)nc1-c1cncc2c1ncn2C
Cc1nc(Nc2ccc([C@@H]3COCCN3C)cc2)c(C(N)=O)nc1-c1cccc2c1ncn2C
Cc3nc(Nc2ccc([C@H]1COCCN1C)cc2)c(C(N)=O)nc3c4cccc5c4ncn5C
Cc1nc(Nc2ccc([C@@H]3CN(C)CCO3)cc2)c(C(N)=O)nc1-c1cccc2c1ncn2C
Cc3nc(Nc2ccc([C@H]1CN(C)CCO1)cc2)c(C(N)=O)nc3c4cccc5c4ncn5C
CNc1nc(Nc2ccc(OC3CCNCC3)cc2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(OC3CCN(C(C)=O)CC3)cc2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(OC3CCN(C)CC3)cc2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(OC3CCN(C(=O)CO)CC3)cc2)c(C(N)=O)nc1-c1cncc2c1ncn2C
COc1nc(Nc2ccc(OC3CCN(C)CC3)cc2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CN1CCC(Oc2ccc(Nc3nc(C4CC4)c(-c4cncc5c4ncn5C)nc3C(N)=O)cc2)CC1
CNc1nc(Nc2cc(F)c(OC3CCN(C)CC3)c(F)c2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(OC3CCN(C(C)C)CC3)cc2)c(C(N)=O)nc1-c1cncc2c1ncn2C
Cc1nc(Nc2ccc(OC[C@@H]3C[C@@H](O)CN3C)cc2)c(C(N)=O)nc1-c1cccc2c1ncn2C
Cc1nc(Nc2ccc(OC[C@H]3C[C@H](O)CN3C)cc2)c(C(N)=O)nc1-c1cccc2c1ncn2C
CO[C@H]1C[C@H](COc2ccc(Nc3nc(C)c(-c4cccc5c4ncn5C)nc3C(N)=O)cc2)N(C)C1
CO[C@@H]1C[C@@H](COc2ccc(Nc3nc(C)c(-c4cccc5c4ncn5C)nc3C(N)=O)cc2)N(C)C1
CNc1nc(Nc2cccc(N3CCN(C)CC3)c2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2cccc(N3CCN(C)CC3)c2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(-n3cnc(C)c3)cc2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc3nncn3c2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(C(C)(C)O)cc2)c(C(N)=O)nc1-c1cncc2c1ncn2C
Cn1cnc2c(-c3nc(C(N)=O)c(Nc4ccc(C(C)(C)O)nc4)nc3C3CC3)cncc21
Cc1nc(Nc2ccc3c(c2)CS(=N)(=O)C3)c(C(N)=O)nc1-c1cccc2c1ncn2C
CCS(=N)(=O)c4c(C)cc(Nc3nc(C)c(c1cccc2c1ncn2C)nc3C(N)=O)cc4C
CCS(=N)(=O)c4c(C)cc(Nc3nc(C)c(c1cccc2c1ncn2C)nc3C(N)=O)cc4C
CNc1nc(Nc2ccc3c(c2)CS(=O)(=O)C3)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc3c(c2)CS(=O)(=O)N3C)c(C(N)=O)nc1-c1cncc2c1ncn2C
CN1c2ccc(Nc3nc(C4CC4)c(-c4cncc5c4ncn5C)nc3C(N)=O)cc2CS1(=O)=O
COc1nc(Nc2ccc3c(c2)CS(=O)(=O)N3C)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(N3CCS(=O)(=O)CC3)cc2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(N=S(C)(C)=O)cc2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(N=S(C)(C)=O)cc2F)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(N=S(C)(C)=O)c(F)c2F)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(N3CCCS3(=O)=O)cc2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(N3CCCCS3(=O)=O)cc2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(S(C)(=O)=O)cc2F)c(C(N)=O)nc1-c1cncc2c1ncn2C
CC[S@@](=N)(=O)c1ccc(Nc2nc(NC)c(-c3cncc4c3ncn4C)nc2C(N)=O)cc1
CC[S@](=N)(=O)c1ccc(Nc2nc(NC)c(-c3cncc4c3ncn4C)nc2C(N)=O)cc1
CNc2nc(Nc1ccc(S(=N)(=O)C(C)C)cc1)c(C(N)=O)nc2c3cncc4c3ncn4C
CNc2nc(Nc1ccc(S(=N)(=O)C(C)C)cc1)c(C(N)=O)nc2c3cncc4c3ncn4C
CNc1nc(Nc2ccc(S(=N)(=O)C(C)(C)C)cc2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2ccc(C3(S(C)(=O)=O)CC3)cc2)c(C(N)=O)nc1-c1cncc2c1ncn2C
COc1nc(Nc2ccc(C3(S(C)(=O)=O)CC3)cc2)c(C(N)=O)nc1-c1cncc2c1ncn2C
COc1nc(Nc2cnn(C)c2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2cnn(C3CCOCC3)c2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2cnn(C(C)C)c2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2cnn(C3CCS(=O)(=O)CC3)c2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2cnn(C3CCN(C)CC3)c2)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2cn(C3CCN(C)CC3)nc2C)c(C(N)=O)nc1-c1cccc2c1ncn2C
CNc1nc(Nc2cn(C)nc2C)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2cn(CC(F)(F)F)nc2C)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2cn(CC(F)F)nc2C)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2cnn(CC(F)F)c2C)c(C(N)=O)nc1-c1cncc2c1ncn2C
CNc1nc(Nc2cn(C(C)(C)C#N)nc2C)c(C(N)=O)nc1-c1cncc2c1ncn2C
Cc1nn(C)cc1Nc1nc(C2CC2)c(-c2cncc3c2ncn3C)nc1C(N)=O
Cc5c(Nc4nc(C1CC1)c(c2cncc3c2ncn3C)nc4C(N)=O)cnn5CC(F)(F)F
Cc1c(cn(n1)CC(F)(F)F)Nc2c(nc(c(n2)C3CC3)c4cncc5c4ncn5C)C(=O)N
Cc1nn(CC(F)F)cc1Nc1nc(C2CC2)c(-c2cncc3c2ncn3C)nc1C(N)=O
Cc1nn(C(C)(C)C#N)cc1Nc1nc(C2CC2)c(-c2cncc3c2ncn3C)nc1C(N)=O
Cc1nn(C2(C#N)CC2)cc1Nc1nc(C2CC2)c(-c2cncc3c2ncn3C)nc1C(N)=O
Cc1c(Nc2nc(C3CC3)c(-c3cncc4c3ncn4C)nc2C(N)=O)cnn1C
Cc1n[nH]cc1Nc1nc(C2CC2)c(-c2cncc3c2ncn3C)nc1C(N)=O
Cc1nn(C[C@@H](F)CF)cc1Nc1nc(C2CC2)c(-c2cncc3c2ncn3C)nc1C(N)=O
Cc1nn(C[C@H](F)CF)cc1Nc1nc(C2CC2)c(-c2cncc3c2ncn3C)nc1C(N)=O
Cc1c(Nc2nc(C3CC3)c(-c3cncc4c3ncn4C)nc2C(N)=O)cnn1C[C@@H](F)CF
Cc1c(Nc2nc(C3CC3)c(-c3cncc4c3ncn4C)nc2C(N)=O)cnn1C[C@H](F)CF
Cc5c(Nc4nc(C1CC1)c(c2cncc3c2ncn3C)nc4C(N)=O)cnn5C6COC6
Cc2nn(C1COC1)cc2Nc6nc(C3CC3)c(c4cncc5c4ncn5C)nc6C(N)=O
Cc1c(Nc2nc(C3CC3)c(-c3cncc4c3ncn4C)nc2C(N)=O)cnn1CC(F)F
Cc5c(Nc4nc(C1CC1)c(c2cncc3c2ncn3C)nc4C(N)=O)cnn5CCC(F)F
Cc1nn(CCC(F)F)cc1Nc5nc(C2CC2)c(c3cncc4c3ncn4C)nc5C(N)=O
Cc1nn(C2CCOCC2)cc1Nc1nc(C2CC2)c(-c2cncc3c2ncn3C)nc1C(N)=O
Cc1c(Nc2nc(C3CC3)c(-c3cncc4c3ncn4C)nc2C(N)=O)cnn1C1CCOCC1
Cc5c(Nc4nc(C1CC1)c(c2cccc3c2ncn3C)nc4C(N)=O)cnn5C6CCN(C)CC6
Cc2nn(C1CCN(C)CC1)cc2Nc6nc(C3CC3)c(c4cccc5c4ncn5C)nc6C(N)=O
COC1=CC2C(C=C1)N=CC1C(C3C=C(N4CCC(N(C)C)CC4)C=CC3)=NN(C3=CC(C)C(C)C=C3)C12
COC1=CC2C(C=C1)N=CC1C(C3C=C(N4CCN(C)CC4)C=CC3)=NN(C3=CC(C)C(C)C=C3)C12
COC1=CC2c3c(c(-c4cccc(OC)c4)nn3C3C=C(N4CCC(N(C)C)CC4)C=CC3)C=NC2C=C1
COC1=CC2c3c(c(-c4cccc(OC)c4)nn3C3C=C(N4CCN(C)CC4)C=CC3)C=NC2C=C1
COC1=CC2c3c(c(-c4cccc(OC)c4)nn3C3C=C(N4CCC(N(C)C)CC4)C=CC3C)C=NC2C=C1
COC1=CC2c3c(c(-c4cccc(OC)c4)nn3C3C=C(N4CCN(C)CC4)C=CC3C)C=NC2C=C1
CC1C=CC(N2N=C(c3ccc(N4CCN(C)CC4)cc3)C3C=NC4C=CC=CC4C32)=CC1C
CC1C=CC(N2N=C(c3ccc(N4CCNCC4)cc3)C3C=NC4C=CC=CC4C32)=CC1C
COC1=CC2C(C=C1)N=CC1C(c3ccc(OCCN(C)C)c(OC)c3)=NN(C3=CC(C)C(C)C=C3)C12
COC1=CC2C(C=C1)N=CC1C(c3ccc(OCCN4CCOCC4)c(OC)c3)=NN(C3=CC(C)C(C)C=C3)C12
COC1=CC2C(C=C1)N=CC1C(c3ccc(OCCCN4CCOCC4)c(OC)c3)=NN(C3=CC(C)C(C)C=C3)C12
COC1=CC2c3c(c(C4=CC(OC)C(OC)C=C4)nn3C3C=C4CCNCC4=CC3)C=NC2C=C1
COC1=CC2c3c(c(C4=CC(OC)C(OC)C=C4)nn3C3C=C4CNCC4=CC3)C=NC2C=C1
CN(C)C(=O)c1cc(ccc1N)-c1cnc2NCC3(CCCC3)c2c1
CN(C)C(=O)c1cc(ccc1N)-c1cnc2NCC3(CC3)c2c1
O=C1COCCN1c1cccc(-c2cnc3c(c2)C2(CC2)CN3)c1
CN(C)C(=O)c1cc(ccc1N)-c1cnc2NCC3(CCC3)c2c1
O=C1COCCN1c1cccc(-c2cnc3c(c2)C2(CCC2)CN3)c1
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2)C2(CC2)CN3)c1F
CN(CCO)C(=O)c1c(N)ccc(-c2cnc3c(c2)C2(CC2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)C2(CC2)CN3)c1F
O=C1COCCN1c1cccc(-c2cnc3c(c2)C2(CC2)CN3)c1F
Nc1cc(-c2cnc3c(c2)C2(CC2)CN3)cc(-c2ncccc2CO)c1
NS(=O)(=O)Cc1ccc(-c2cnc3c(c2)C2(CC2)CN3)cc1
CN(CCO)C(=O)c1cccc(-c2cnc3c(c2)C2(CC2)CN3)c1F
CC1(C)C(=O)Nc2ccc(-c3cnc4c(c3)C3(CC3)CN4)cc21
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2)C2(CC2)CN3)c1Cl
CC1Nc2ncc(-c3ccc(N)c(C(=O)N(C)C)c3F)cc2C12CC2
CN(C)C(=O)c1cc(CO)cc(-c2cnc3c(c2)C2(CC2)CN3)c1
Nc1ccc(-c2cnc3c(c2)C2(CC2)CN3)c(F)c1C(=O)N1CCCC1CO
CN(C)C(=O)c1cc(-c2cnc3c(c2)C2(CC2)CN3)ccc1CO
CN(C(=O)c1c(N)ccc(-c2cnc3c(c2)C2(CC2)CN3)c1F)C(C)(C)CO
CC1(O)C(=O)Nc2ccc(-c3cnc4c(c3)C3(CC3)CN4)cc21
CN(C)S(=O)(=O)c1cccc(-c2cnc3c(c2)C2(CC2)CN3)c1F
CNS(=O)(=O)c1cccc(-c2cnc3c(c2)C2(CC2)CN3)c1F
O=C1Nc2ccc(-c3cnc4c(c3)C3(CC3)CN4)cc2C1(O)C1CC1
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2)C2(CN3)CC2(C)C)c1F
CC1CNC(=O)N1c1c(N)ccc(-c2cnc3c(c2Cl)C2(CC2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2)C2(CN3)C3COCC32)c1F
CN(C)C(=O)c1c(N)ccc(c1F)-c1cnc2NCC3(CCCC3)c2c1Cl
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)C2(CC=CC2)CN3)c1F
CN(CC(C)(C)O)C(=O)c1c(N)ccc(-c2cnc3c(c2)C2(CC2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(c1F)-c1cnc2NCC3(CC3)c2c1C
COc1c(-c2ccc(N)c(C(=O)N(C)C)c2F)cnc2c1C1(CC1)CN2
CC(=O)c1cc(-c2cnc3c(c2Cl)C2(CC2)CN3)ccc1N
CC(=O)Nc1cc(C(=O)N(C)C)cc(-c2cnc3c(c2Cl)C2(CC2)CN3)c1
Nc1cc(-c2cnc3c(c2Cl)C2(CC2)CN3)cc(-c2ncccc2CO)c1
CN(CC(C)(C)O)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)C2(CC2)CN3)c1F
CN(CCO)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)C2(CC2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(c1F)-c1cnc2NCC3(CCC3)c2c1Cl
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)[C@@]2(CC[C@H](O)C2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(c1F)-c1cnc2NC[C@@]3(CC[C@H](O)C3)c2c1Cl |r|
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)C2(CN3)CC2CO)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)[C@@]2(CN3)C[C@H]2CO)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)[C@]2(CN3)C[C@@H]2CO)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)[C@]2(CN3)C[C@H]2CO)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)[C@@]2(CN3)C[C@@H]2CO)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)C2(CN3)Cc3ccncc3C2)c1F
O=C1COCCN1c1cccc(-c2cnc3c(c2)C2(CC2)CN3)c1
O=C1CNCCN1c1cccc(-c2cnc3c(c2)C2(CC2)CN3)c1
OCc1cccnc1-c1cccc(-c2cnc3c(c2)C2(CC2)CN3)c1
CN(CCO)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)C2(CCC2)CN3)c1F
CN(CCO)C(=O)c1cccc(-c2cnc3c(c2Cl)C2(CC2)CN3)c1F
CCN(CCO)C(=O)c1cccc(-c2cnc3c(c2Cl)C2(CC2)CN3)c1F
O=C(c1cccc(-c2cnc3c(c2Cl)C2(CC2)CN3)c1F)N(CCO)CCO
O=C(c1cccc(-c2cnc3c(c2Cl)C2(CC2)CN3)c1F)N1CCNCC1
O=C(c1cccc(-c2cnc3c(c2Cl)C2(CC2)CN3)c1F)N1CC(O)C1
CC(=O)NC1CN(C(=O)c2cccc(-c3cnc4c(c3Cl)C3(CC3)CN4)c2F)C1
O=C(c1cccc(-c2cnc3c(c2Cl)C2(CC2)CN3)c1F)N1CC(O)C1
COc1c(-c2ccc(N)c(C(=O)N(C)CCO)c2F)cnc2c1C1(CCC1)CN2
Cc1c(-c2ccc(N)c(C(=O)N(C)C)c2F)cnc2c1C1(CCC1)CN2
CC(=O)Nc1cc(C#N)cc2c(-c3cnc4c(c3)C3(CC3)CN4)cn(C)c12
O=C1NCCN1c1cccc(-c2cnc3c(c2Cl)C2(CC2)CN3)c1
N#Cc1cc2c(-c3cnc4c(c3)C3(CC3)CN4)c[nH]c2cn1
Cn1cccc(-c2cccc(-c3cnc4c(c3Cl)C3(CC3)CN4)c2)c1=O
O=C1NCCCC1c1cccc(-c2cnc3c(c2Cl)C2(CC2)CN3)c1
O=C1NCCCN1c1cccc(-c2cnc3c(c2Cl)C2(CC2)CN3)c1
O=C1CCCCN1c1cccc(-c2cnc3c(c2Cl)C2(CC2)CN3)c1
Nc1cc(-c2cnc3c(c2Cl)C2(CCC(O)C2)CN3)cc(-c2ncccc2CO)c1
Nc1cc(-c2cnc3c(c2Cl)[C@@]2(CC[C@@H](O)C2)CN3)cc(-c2ncccc2CO)c1
Nc1cc(-c2cnc3c(c2Cl)[C@@]2(CC[C@H](O)C2)CN3)cc(-c2ncccc2CO)c1
NS(=O)(=O)c1cccc(-c2cnc3c(c2)C2(CC2)CN3)c1
CS(=O)(=O)c1cccc(-c2cnc3c(c2)C2(CC2)CN3)c1
CC(=O)Nc1ccc(-c2cnc3c(c2)C2(CC2)CN3)cc1C(F)(F)F
NS(=O)(=O)c1ccc(-c2cnc3c(c2)C2(CC2)CN3)cc1
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2)C2(CCC2)CN3)c1F
O=C1NCCCN1c1cccc(-c2cnc3c(c2)C2(CC2)CN3)c1
Cn1cccc(-c2cccc(-c3cnc4c(c3Cl)[C@]3(CC[C@@H](O)C3)CN4)c2)c1=O
Cn1cccc(-c2cccc(-c3cnc4c(c3Cl)[C@@]3(CC[C@H](O)C3)CN4)c2)c1=O
Cn1cccc(-c2cccc(-c3cnc4c(c3Cl)[C@]3(CC[C@H](O)C3)CN4)c2)c1=O
C[C@@H]1CNC(=O)N1c1cccc(-c2cnc3c(c2Cl)C2(CC2)CN3)c1
C[C@H]1CNC(=O)N1c1cccc(-c2cnc3c(c2Cl)C2(CC2)CN3)c1
O=C1NCCCN1c1cccc(-c2cnc3c(c2)C2(CC2)CN3)n1
O=C1NCCN1c1cccc(-c2cnc3c(c2)C2(CC2)CN3)n1
c1cc(-c2cnc3c(c2)C2(CC2)CN3)cc(-c2nnn3c2CNCC3)c1
O=C1NCCC1c1cccc(-c2cnc3c(c2Cl)C2(CC2)CN3)c1
N#Cc1cc2c(-c3cnc4c(c3)C3(CC3)CN4)c[nH]c2cc1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)C2(CCC(N(C)CC(N)=O)C2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)C2(CCC(NCC(N)=O)C2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2)[C@]2(CN3)C[C@@H](O)C2)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2)[C@]2(CN3)C[C@@H](O)C2)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2)[C@]2(CN3)C[C@](C)(O)C2)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2)[C@]2(CN3)C[C@](C)(O)C2)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2)C2(CNC(=O)C2)CN3)c1F
CO[C@H]1C[C@@]2(CNc3ncc(-c4ccc(N)c(C(=O)N(C)C)c4F)c(Cl)c32)C1
CO[C@H]1C[C@@]2(CNc3ncc(-c4ccc(N)c(C(=O)N(C)C)c4F)c(Cl)c32)C1
CO[C@@H]1CC[C@]2(CNc3ncc(-c4ccc(N)c(C(=O)N(C)C)c4F)c(Cl)c32)C1
CO[C@@H]1CC[C@@]2(CNc3ncc(-c4ccc(N)c(C(=O)N(C)C)c4F)c(Cl)c32)C1
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)C2(CCC(C)(O)C2)CN3)c1F
CC(=O)NC1CCC2(CNc3ncc(-c4ccc(N)c(C(=O)N(C)C)c4F)c(Cl)c32)C1
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)[C@@]2(CC[C@@H](C(N)=O)C2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)[C@]2(CC[C@@H](C(N)=O)C2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)[C@@]2(CC[C@H](n4cncn4)C2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)[C@]2(CC[C@@H](n4cncn4)C2)CN3)c1F
C[C@H]1C[C@]12CNc1ncc(-c3ccc(N)c(C(=O)N(C)C)c3F)cc12
C[C@@H]1C[C@@]12CNc1ncc(-c3ccc(N)c(C(=O)N(C)C)c3F)cc12
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2)C2(CN3)CC(O)(C(F)(F)F)C2)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2)C2(CN3)CC(n3cncn3)C2)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)[C@]2(CC[C@@H](n4nccn4)C2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)[C@@]2(CC[C@H](n4nccn4)C2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)[C@]2(CC[C@@H](n4ccnn4)C2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)[C@@]2(CC[C@H](n4ccnn4)C2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)C2(CCC(C#N)C2)CN3)c1F
O=C1NCCC1c1cccc(-c2cnc3c(c2)C2(CC2)CN3)c1F
CC(=O)N1CC2(CNc3ncc(-c4ccc(N)c(C(=O)N(C)C)c4F)cc32)C1
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2)C2(CN3)CC(=CC#N)C2)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2)C2(CN3)CC(CC#N)C2)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2)C2(CN3)CC(C#N)C2)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2)C2(CN3)CC(C(N)=O)C2)c1F
CNC(=O)C1CCC2(CNc3ncc(-c4ccc(N)c(C(=O)N(C)C)c4F)c(Cl)c32)C1
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)C2(CCC(c4ncn[nH]4)C2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)[C@]2(CC[C@@H](C(N)=O)C2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)[C@@]2(CC[C@H](C(N)=O)C2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2)C2(CN3)CC(=CC(N)=O)C2)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2)[C@]2(CN3)C[C@H](CC(N)=O)C2)c1F
CC1CCC2(CNc3ncc(-c4ccc(N)c(C(=O)N(C)C)c4F)c(Cl)c32)C1
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)C2(CCC(=CC#N)C2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)C2(CCC(C(=O)O)C2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)C2(CCC(C(=O)NCCO)C2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)C2(CCC(C(=O)N(C)C)C2)CN3)c1F
Cc1noc(C2CCC3(CNc4ncc(-c5ccc(N)c(C(=O)N(C)C)c5F)c(Cl)c43)C2)n1
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)[C@]2(CC[C@](O)(CC#N)C2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)[C@@]2(CC[C@@](O)(CC#N)C2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)C2(CCC(=CC(N)=O)C2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2)[C@]2(CC[C@H](O)CC2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2)[C@]2(CC[C@H](O)CC2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)C2(C=C(c4cccnc4)CC2)CN3)c1F
COc1c(-c2ccc(N)c(C(=O)N(C)C)c2F)cnc2c1[C@]1(CC[C@H](O)CC1)CN2
COc1c(-c2ccc(N)c(C(=O)N(C)C)c2F)cnc2c1[C@]1(CC[C@H](O)CC1)CN2
Cc1cnn(C2CCC3(CNc4ncc(-c5ccc(N)c(C(=O)N(C)C)c5F)c(Cl)c43)C2)n1
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)C2(CCC(N4CCNC4=O)C2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)[C@]2(CC[C@](O)(Cn4cncn4)C2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)[C@]2(CC[C@@](O)(Cn4cncn4)C2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)C2(CCC(O)(Cn4ccnc4)C2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)C2(CCC(n4ncnc4N)C2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)C2(CCC(n4cnc(N)n4)C2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)C2(CCC(N4CCOCC4)C2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)C2(CCC(N4CCCC4)C2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)[C@]2(CCNC(=O)C2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)[C@@]2(CCNC(=O)C2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)[C@]2(CCC(=O)NC2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)[C@@]2(CCC(=O)NC2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)C2(CCC(N4CCOC4=O)C2)CN3)c1F
Cc1cnn(C2CCC3(CNc4ncc(-c5ccc(N)c(C(=O)N(C)C)c5F)c(Cl)c43)C2)c1
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)C2(CCC(n4cccn4)C2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)C2(CCC(CN)C2)CN3)c1F
C[C@@H]1Nc2ncc(-c3ccc(N)c(C(=O)N(C)C)c3F)cc2C12CC2
C[C@H]1Nc2ncc(-c3ccc(N)c(C(=O)N(C)C)c3F)cc2C12CC2
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)C2(CCC(Cn4cncn4)C2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)C2(CCC(CC#N)C2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)C2(CCC(C)(C#N)C2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)C2(CCC(C)(C(N)=O)C2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)C2(CCC(n4ccc(N)n4)C2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)C2(CCC(n4nccc4N)C2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)[C@]2(CC[C@@H](CC(N)=O)C2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)[C@@]2(CC[C@H](CC(N)=O)C2)CN3)c1F
CN(Cc1cnn(C)c1)C(=O)c1cccc(-c2cnc3c(c2)C2(CC2)CN3)c1F
CCN(C(=O)c1cccc(-c2cnc3c(c2)C2(CC2)CN3)c1F)C1CCC1
N#CCCN(C)C(=O)c1cccc(-c2cnc3c(c2)C2(CC2)CN3)c1F
CC(C)C1CN(C(=O)c2cccc(-c3cnc4c(c3)C3(CC3)CN4)c2F)C1
COC1C[C@@]2(CNc3ncc(-c4ccc(N)c(C(=O)N(C)C)c4F)c(Cl)c32)C[C@@H]1O
COC1C[C@]2(CNc3ncc(-c4ccc(N)c(C(=O)N(C)C)c4F)c(Cl)c32)C[C@H]1O
CN(C(=O)c1cccc(-c2cnc3c(c2)C2(CC2)CN3)c1F)c1cnn(C)c1
CC1CN(C(=O)c2cccc(-c3cnc4c(c3)C3(CC3)CN4)c2F)C1
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)C2(CCC(N4CCCC4=O)C2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)[C@]2(CC[C@@H](O)CC2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)[C@]2(CC[C@@H](O)CC2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)C2(CCC(c4cccnc4)C2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)[C@]2(CC[C@@H](c4cccnc4)C2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)[C@]2(CC[C@H](c4cccnc4)C2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)[C@@]2(CC[C@@H](c4cccnc4)C2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)[C@@]2(CN3)CC(n3ccnn3)[C@@H](O)C2)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)[C@]2(CN3)CC(n3ccnn3)[C@H](O)C2)c1F
O=C(c1cccc(-c2cnc3c(c2)C2(CC2)CN3)c1F)N1CCC12COC2
Cc1cnn(C2CCC3(CC2)CNc2ncc(-c4ccc(N)c(C(=O)N(C)C)c4F)c(Cl)c23)c1
CN(C)C(=O)c1cccc(-c2cnc3c(c2)C2(CC2)CN3)c1F
CC[C@@H]1C[C@@]12CNc1ncc(-c3ccc(N)c(C(=O)N(C)C)c3F)c(Cl)c12
CC[C@H]1C[C@]12CNc1ncc(-c3ccc(N)c(C(=O)N(C)C)c3F)c(Cl)c12
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)C2(CCC(C)(C#N)C2)CN3)c1F
CCC1(C#N)CCC2(CNc3ncc(-c4ccc(N)c(C(=O)N(C)C)c4F)c(Cl)c32)C1
CCC1(C(N)=O)CCC2(CNc3ncc(-c4ccc(N)c(C(=O)N(C)C)c4F)c(Cl)c32)C1
N#CC1CCCN1C(=O)c1cccc(-c2cnc3c(c2)C2(CC2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)[C@]2(CC[C@@](C)(C(N)=O)C2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)[C@@]2(CC[C@](C)(C(N)=O)C2)CN3)c1F
Cc1noc(C2(C)CCC3(CNc4ncc(-c5ccc(N)c(C(=O)N(C)C)c5F)c(Cl)c43)C2)n1
Cc1nc(N)nn1C1CCC2(CNc3ncc(-c4ccc(N)c(C(=O)N(C)C)c4F)c(Cl)c32)C1
Cc1nc(N)n(C2CCC3(CNc4ncc(-c5ccc(N)c(C(=O)N(C)C)c5F)c(Cl)c43)C2)n1
Cc1ccn(C2CCC3(CNc4ncc(-c5ccc(N)c(C(=O)N(C)C)c5F)c(Cl)c43)C2)n1
Cc1ccnn1C1CCC2(CNc3ncc(-c4ccc(N)c(C(=O)N(C)C)c4F)c(Cl)c32)C1
Cc1cc(C#N)n(C2CCC3(CNc4ncc(-c5ccc(N)c(C(=O)N(C)C)c5F)c(Cl)c43)C2)n1
Cc1cc(C#N)nn1C1CCC2(CNc3ncc(-c4ccc(N)c(C(=O)N(C)C)c4F)c(Cl)c32)C1
Cc1cc(C)n(C2CCC3(CNc4ncc(-c5ccc(N)c(C(=O)N(C)C)c5F)c(Cl)c43)C2)n1
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)C2(CCC(n4cc(C(F)(F)F)cn4)C2)CN3)c1F
COc1c(-c2ccc(N)c(C(=O)N(C)C)c2F)cnc2c1C1(CN2)CC1C
CN(Cc1cnn(C)c1)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)C2(CC2)CN3)c1F
Cc1nccn1C1CCC2(CNc3ncc(-c4ccc(N)c(C(=O)N(C)C)c4F)c(Cl)c32)C1
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)C2(CCC(n4ccc(C(F)(F)F)n4)C2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)C2(CCC(n4nccc4C(F)(F)F)C2)CN3)c1F
CCc1cnn(C2CCC3(CNc4ncc(-c5ccc(N)c(C(=O)N(C)C)c5F)c(Cl)c43)C2)c1
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)C2(CCC(n4cc(Cl)cn4)C2)CN3)c1F
O=C(c1cccc(-c2cnc3c(c2)C2(CC2)CN3)c1F)N1CCc2ccccc21
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)C2(CCC(Oc4ccccn4)C2)CN3)c1F
Cn1cc([C@H]2CCCN2C(=O)c2cccc(-c3cnc4c(c3)C3(CC3)CN4)c2F)cn1
Cn1cc([C@@H]2CCCN2C(=O)c2cccc(-c3cnc4c(c3)C3(CC3)CN4)c2F)cn1
Cn1cc([C@H]2CCCCN2C(=O)c2cccc(-c3cnc4c(c3)C3(CC3)CN4)c2F)cn1
Cn1cc([C@@H]2CCCCN2C(=O)c2cccc(-c3cnc4c(c3)C3(CC3)CN4)c2F)cn1
O=C(c1cccc(-c2cnc3c(c2)C2(CC2)CN3)c1F)N1CCc2ccncc21
Cc1cn(C2CCC3(CNc4ncc(-c5ccc(N)c(C(=O)N(C)C)c5F)c(Cl)c43)C2)nc1N
Cc1cnn(C2CCC3(CNc4ncc(-c5ccc(N)c(C(=O)N(C)C)c5F)c(Cl)c43)C2)c1N
Cn1cccc(-c2cccc(-c3cnc4c(c3Cl)[C@]3(CC[C@@](C)(C(N)=O)C3)CN4)c2)c1=O
Cn1cccc(-c2cccc(-c3cnc4c(c3Cl)[C@@]3(CC[C@](C)(C(N)=O)C3)CN4)c2)c1=O
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)C2(CCC(n4cc(C(N)=O)cn4)C2)CN3)c1F
OCc1ccc(-c2cnc3c(c2Cl)C2(CC=CC2)CN3)cc1
CC(C)(O)c1ccc(-c2cnc3c(c2Cl)C2(CC=CC2)CN3)cc1
CS(=O)(=O)c1cccc(-c2cnc3c(c2Cl)C2(CC=CC2)CN3)c1
CCS(=O)(=O)c1cccc(-c2cnc3c(c2Cl)C2(CC=CC2)CN3)c1
CNS(=O)(=O)c1cccc(-c2cnc3c(c2Cl)C2(CC=CC2)CN3)c1
CS(=O)(=O)c1ccc(-c2cnc3c(c2Cl)C2(CC=CC2)CN3)cc1
CCS(=O)(=O)c1ccc(-c2cnc3c(c2Cl)C2(CC=CC2)CN3)cc1
CNS(=O)(=O)c1ccc(-c2cnc3c(c2Cl)C2(CC=CC2)CN3)cc1
CCNS(=O)(=O)c1ccc(-c2cnc3c(c2Cl)C2(CC=CC2)CN3)cc1
N#Cc1cccc(-c2cnc3c(c2Cl)C2(CC=CC2)CN3)c1
N#CC1(C)CCCN1C(=O)c1cccc(-c2cnc3c(c2)C2(CC2)CN3)c1F
CN(C)C(=O)c1ccc(-c2cnc3c(c2Cl)C2(CC=CC2)CN3)cc1Cl
CC(C)[C@@H]1C[C@]12CNc1ncc(-c3ccc(N)c(C(=O)N(C)C)c3F)c(Cl)c12
CC(C)[C@H]1C[C@]12CNc1ncc(-c3ccc(N)c(C(=O)N(C)C)c3F)c(Cl)c12
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)[C@]2(CC[C@@](C)(O)CC2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)[C@]2(CC[C@@](C)(O)CC2)CN3)c1F
CN(C)C(=O)c1cccc(-c2cnc3c(c2Cl)C2(CCC(C)(C(N)=O)C2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)C2(CCC(n4ccccc4=O)C2)CN3)c1F
CCC[C@@H]1C[C@@]12CNc1ncc(-c3ccc(N)c(C(=O)N(C)C)c3F)c(Cl)c12
CCC[C@H]1C[C@]12CNc1ncc(-c3ccc(N)c(C(=O)N(C)C)c3F)c(Cl)c12
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)C2(CN3)CC2c2ccncc2)c1F
CN(C)C(=O)c1cccc(-c2cnc3c(c2Cl)[C@]2(CC[C@@](C)(C(N)=O)C2)CN3)c1F
CN(C)C(=O)c1cccc(-c2cnc3c(c2Cl)[C@@]2(CC[C@](C)(C(N)=O)C2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)C2(CCCCC2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)C2(CN3)CC2c2ccccc2)c1F
CC1(C(N)=O)CCC2(CNc3ncc(-c4cccc(N5CCOCC5=O)c4F)c(Cl)c32)C1
O=S(=O)(c1ccc(-c2cnc3c(c2Cl)C2(CC=CC2)CN3)cc1)n1cccn1
OCC1(c2ccc(-c3cnc4c(c3Cl)C3(CC=CC3)CN4)cc2)CC1
CN(C)C(=O)c1ccc(-c2cnc3c(c2Cl)C2(CC=CC2)CN3)cc1F
CN(C)C(=O)c1ccc(-c2cnc3c(c2Cl)C2(CC=CC2)CN3)c(F)c1
O=S(=O)(Nc1ccc(-c2cnc3c(c2Cl)C2(CC=CC2)CN3)cc1)C1CC1
O=S1(=O)CCCN1c1ccc(-c2cnc3c(c2Cl)C2(CC=CC2)CN3)cc1
O=S(=O)(Nc1cccc(-c2cnc3c(c2Cl)C2(CC=CC2)CN3)c1)C1CC1
CS(=O)(=O)Nc1cccc(-c2cnc3c(c2Cl)C2(CC=CC2)CN3)c1
CC(=O)NCc1cccc(-c2cnc3c(c2Cl)C2(CC=CC2)CN3)c1
CC(=O)NCc1ccc(-c2cnc3c(c2Cl)C2(CC=CC2)CN3)cc1
CC(=O)NCCc1ccc(-c2cnc3c(c2Cl)C2(CC=CC2)CN3)cc1
O=C(NCCO)c1ccc(-c2cnc3c(c2Cl)C2(CC=CC2)CN3)cc1
Clc1c(-c2ccc(-n3cccn3)cc2)cnc2c1C1(CC=CC1)CN2
OCc1ccc(-c2cnc3c(c2Cl)C2(CC=CC2)CN3)c(F)c1
CCC[C@H]1C[C@]12CNc1ncc(-c3ccc(N)c(C(=O)N(C)C)c3F)cc12
CCC[C@@H]1C[C@@]12CNc1ncc(-c3ccc(N)c(C(=O)N(C)C)c3F)cc12
CCC[C@@H]1C[C@]12CNc1ncc(-c3ccc(N)c(C(=O)N(C)C)c3F)cc12
CCC[C@H]1C[C@@]12CNc1ncc(-c3ccc(N)c(C(=O)N(C)C)c3F)cc12
CN(C)S(=O)(=O)Nc1cccc(-c2cnc3c(c2Cl)C2(CC=CC2)CN3)c1
OCc1cccc(-c2cnc3c(c2Cl)C2(CC=CC2)CN3)c1F
Clc1c(-c2ccc(COC3CCOCC3)cc2)cnc2c1C1(CC=CC1)CN2
N#CCCNC(=O)c1ccc(-c2cnc3c(c2Cl)C2(CC=CC2)CN3)cc1
CC(=O)Nc1cccc(-c2cnc3c(c2Cl)C2(CC=CC2)CN3)c1
COCCc1ccc(-c2cnc3c(c2Cl)C2(CC=CC2)CN3)cc1
Nc1ccc(-c2cnc3c(c2Cl)C2(CC=CC2)CN3)cc1
Nc1ccc(-c2cnc3c(c2Cl)C2(CC=CC2)CN3)c(F)c1
CN(C)C(=O)c1cccc(-c2cnc3c(c2Cl)C2(CC=CC2)CN3)c1
CN(C)C(=O)c1cccc(-c2cnc3c(c2Cl)C2(CC=CC2)CN3)c1F
C[C@@H]1C[C@@]12CNc1ncc(-c3ccc(N)c(C(=O)N(C)C)c3F)c(Cl)c12
C[C@H]1C[C@]12CNc1ncc(-c3ccc(N)c(C(=O)N(C)C)c3F)c(Cl)c12
C[C@@H](c1cnn(C)c1)N(C)C(=O)c1cccc(-c2cnc3c(c2)C2(CC2)CN3)c1F
C[C@H](c1cnn(C)c1)N(C)C(=O)c1cccc(-c2cnc3c(c2)C2(CC2)CN3)c1F
O=C(c1ccc(-c2cnc3c(c2Cl)C2(CC=CC2)CN3)cc1Cl)N1CCC(O)CC1
O=C(c1ccc(-c2cnc3c(c2Cl)C2(CC=CC2)CN3)cc1)N1CCOCC1
O=C(c1cccc(-c2cnc3c(c2)C2(CC2)CN3)c1F)N1CCCCC1
Cc1c(-c2ccc(N)c(C(=O)N(C)C)c2F)cnc2c1C1(CCCCC1)CN2
CC(C)[C@@H]1C[C@]12CNc1ncc(-c3ccc(N)c(C(=O)N(C)C)c3F)cc12
CC(C)[C@@H]1C[C@]12CNc1ncc(-c3ccc(N)c(C(=O)N(C)C)c3F)cc12
CC(C)[C@H]1C[C@]12CNc1ncc(-c3ccc(N)c(C(=O)N(C)C)c3F)cc12
CC(C)[C@@H]1C[C@@]12CNc1ncc(-c3ccc(N)c(C(=O)N(C)C)c3F)cc12
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)[C@]2(CC[C@@H](C(N)=O)CC2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)[C@]2(CC[C@@H](C(N)=O)CC2)CN3)c1F
NC(=O)C1(c2cccc(-c3cnc4c(c3Cl)C3(CC=CC3)CN4)c2)CC1
Clc1c(-c2ccc(Oc3ncccn3)cc2)cnc2c1C1(CC=CC1)CN2
Cc1cc(C)n(-c2cccc(-c3cnc4c(c3Cl)C3(CC=CC3)CN4)c2)n1
Cn1cc([C@H]2CCCCN2C(=O)c2c(N)ccc(-c3cnc4c(c3Cl)C3(CC=CC3)CN4)c2F)cn1
Cn1cc([C@@H]2CCCCN2C(=O)c2c(N)ccc(-c3cnc4c(c3Cl)C3(CC=CC3)CN4)c2F)cn1
Cn1cc([C@H]2CCCCN2C(=O)c2cccc(-c3cnc4c(c3Cl)C3(CC=CC3)CN4)c2F)cn1
Cn1cc([C@@H]2CCCCN2C(=O)c2cccc(-c3cnc4c(c3Cl)C3(CC=CC3)CN4)c2F)cn1
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)[C@]2(CC[C@@H](C#N)CC2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)[C@]2(CC[C@@H](C#N)CC2)CN3)c1F
Cc1c(CC#N)ccnc1-c1cccc(-c2cnc3c(c2)C2(CC2)CN3)c1
CC[C@@H]1C[C@@]12CNc1ncc(-c3ccc(N)c(C(=O)N(C)C)c3F)cc12
CC[C@H]1C[C@]12CNc1ncc(-c3ccc(N)c(C(=O)N(C)C)c3F)cc12
CC[C@H]1C[C@@]12CNc1ncc(-c3ccc(N)c(C(=O)N(C)C)c3F)cc12
CC[C@@H]1C[C@]12CNc1ncc(-c3ccc(N)c(C(=O)N(C)C)c3F)cc12
N#CC1CCCCN1C(=O)c1cccc(-c2cnc3c(c2)C2(CC2)CN3)c1F
Cn1cc(C2CCCCN2C(=O)c2cccc(-c3cnc4c(c3)C3(CCC(O)CC3)CN4)c2F)cn1
Cn1cc(C2CCCCN2C(=O)c2cccc(-c3cnc4c(c3Cl)[C@]3(CC[C@@H](O)CC3)CN4)c2F)cn1
Cn1cc(C2CCCCN2C(=O)c2cccc(-c3cnc4c(c3Cl)[C@]3(CC[C@@H](O)CC3)CN4)c2F)cn1
CC(C)(C)c1nnc(-c2cccc(-c3cnc4c(c3Cl)C3(CC=CC3)CN4)c2)o1
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)[C@]2(CC[C@@H](CO)CC2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)[C@]2(CC[C@@H](CO)CC2)CN3)c1F
Cc1c(CC#N)ccnc1-c1cccc(-c2cnc3c(c2Cl)C2(CC=CC2)CN3)c1
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)[C@]2(CC[C@@](C)(C#N)CC2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)[C@]2(CC[C@@](C)(C#N)CC2)CN3)c1F
Cc1c(CC#N)ccnc1-c1cccc(-c2cnc3c(c2)C2(CC2)CN3)c1F
Cc1c(CC#N)ccnc1-c1cccc(-c2cnc3c(c2Cl)C2(CC=CC2)CN3)c1F
Cn1cc(C2CCCCN2C(=O)c2c(N)ccc(-c3cnc4c(c3)C3(CCC(O)CC3)CN4)c2F)cn1
Cn1cc(C2CCCCN2C(=O)c2c(N)ccc(-c3cnc4c(c3)[C@]3(CC[C@H](O)CC3)CN4)c2F)cn1
Cn1cc(C2CCCCN2C(=O)c2c(N)ccc(-c3cnc4c(c3)[C@]3(CC[C@H](O)CC3)CN4)c2F)cn1
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)[C@]2(CC[C@@H](C(C)(C)O)CC2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)[C@]2(CC[C@@H](C(C)(C)O)CC2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)C2(CCC(C)(CO)CC2)CN3)c1F
Cc1cc(CC#N)nn1-c1cccc(-c2cnc3c(c2Cl)C2(CC=CC2)CN3)c1
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)[C@]2(CC[C@@H](CN)CC2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)[C@]2(CC[C@@H](CN)CC2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)[C@]2(CC[C@@H](CO)C2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)[C@]2(CC[C@H](CO)C2)CN3)c1F
CN(Cc1cnn(C2CCNC2)c1)C(=O)c1cccc(-c2cnc3c(c2Cl)C2(CC=CC2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)[C@]2(CC[C@@](C)(C#N)C2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)[C@@]2(CC[C@](C)(C#N)C2)CN3)c1F
CN(Cc1cnn(CCO)c1)C(=O)c1cccc(-c2cnc3c(c2Cl)C2(CC=CC2)CN3)c1F
CN(C)C(=O)C1(c2cccc(-c3cnc4c(c3Cl)C3(CC=CC3)CN4)c2)CC1
N#CC1CCCCN1C(=O)c1cccc(-c2cnc3c(c2Cl)C2(CC=CC2)CN3)c1F
NC(=O)C1(c2cccc(-c3cnc4c(c3Cl)C3(CC=CC3)CN4)c2F)CC1
Cc1c(CC#N)ccnc1-c1cccc(-c2cnc3c(c2Cl)[C@@]2(CC[C@](C)(C#N)C2)CN3)c1F
Cc1c(CC#N)ccnc1-c1cccc(-c2cnc3c(c2Cl)[C@]2(CC[C@@](C)(C#N)C2)CN3)c1F
Cc1c(CC#N)ccnc1-c1cccc(-c2cnc3c(c2Cl)[C@@]2(CC[C@](C)(C(N)=O)C2)CN3)c1F
Cc1c(CC#N)ccnc1-c1cccc(-c2cnc3c(c2Cl)[C@]2(CC[C@@](C)(C(N)=O)C2)CN3)c1F
O=C(N1CCOCC1)C1(c2cccc(-c3cnc4c(c3Cl)C3(CC=CC3)CN4)c2)CC1
N#CCNC(=O)c1ccnc(-c2cccc(-c3cnc4c(c3Cl)C3(CC=CC3)CN4)c2F)c1
CN(CC#N)C(=O)C1(c2cccc(-c3cnc4c(c3Cl)C3(CC=CC3)CN4)c2)CC1
CN(C)CCN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)C2(CCC(C)(C#N)C2)CN3)c1F
CN(CCN1CCOCC1)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)C2(CCC(C)(C#N)C2)CN3)c1F
CN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)C2(CCC(S(C)(=O)=O)CC2)CN3)c1F
Cc1c(CC#N)ccnc1-c1cc(N)cc(-c2cnc3c(c2Cl)[C@]2(CC[C@@](C)(C#N)C2)CN3)c1
Cc1c(CC#N)ccnc1-c1cc(N)cc(-c2cnc3c(c2Cl)[C@@]2(CC[C@](C)(C#N)C2)CN3)c1
CN(C)CCCN(C)C(=O)c1c(N)ccc(-c2cnc3c(c2Cl)C2(CCC(C)(C#N)C2)CN3)c1F
Clc1c(-c2ccc3[nH]nnc3c2)cnc2c1C1(CC=CC1)CN2
O=C1OCc2ccc(-c3cnc4c(c3)C3(CC3)CN4)cc21
CCC1(O)C(=O)Nc2ccc(-c3cnc4c(c3)C3(CC3)CN4)cc21
N#CC1(C)C(=O)Nc2ccc(-c3cnc4c(c3)C3(CC3)CN4)cc21
N#CC1(C2CC2)C(=O)Nc2ccc(-c3cnc4c(c3Cl)C3(CC3)CN4)cc21
CC1(C(N)=O)C(=O)Nc2ccc(-c3cnc4c(c3Cl)C3(CC3)CN4)cc21
N#CC1(C)C(=O)Nc2ccc(-c3cnc4c(c3Cl)C3(CC3)CN4)cc21
O=C1NCCC1c1nc2ccc(-c3cnc4c(c3Cl)C3(CC3)CN4)cc2[nH]1
Clc1c(-c2cccc3[nH]ccc23)cnc2c1C1(CC=CC1)CN2
Clc1c(-c2ccc3[nH]ncc3c2)cnc2c1C1(CC=CC1)CN2
Clc1c(-c2cccc3[nH]ncc23)cnc2c1C1(CC=CC1)CN2
Clc1c(-c2ccc3[nH]ccc3c2)cnc2c1C1(CC=CC1)CN2
CN(C)C(=O)c1nc(-c2cnc3c(c2Cl)C2(CCC(C)(C#N)C2)CN3)ccc1N
Nc1cc(-c2cnc3c(c2Cl)C2(CC2)CN3)nc(N2CCCOC2=O)n1
Nc1ccc(-c2cnc3c(c2)C2(CC2)CN3)nc1C(=O)N1CC[C@@H](O)C1
Nc1ccc(-c2cnc3c(c2)C2(CC2)CN3)nc1C(=O)N1CC[C@H](O)C1
CN(C)C(=O)CNc1ccc(-c2cnc3c(c2)C2(CC2)CN3)cn1
Nc1cc(-c2cnc3c(c2)C2(CC2)CN3)nc(N2CCOC2=O)c1
Nc1cc(-c2cnc3c(c2)C2(CC2)CN3)nc(N2CCCOC2=O)c1
CN(C)C(=O)c1cc(N)cc(-c2cnc3c(c2)C2(CC2)CN3)n1
Nc1cc(-c2cnc3c(c2)C2(CC2)CN3)nc(-c2ncccn2)c1
Cn1cccc(-c2cc(-c3cnc4c(c3Cl)C3(CC3)CN4)cc(N)n2)c1=O
CN(C)C(=O)c1cccc2c(-c3cnc4c(c3)C3(CC3)CN4)c[nH]c12
CN(C)C(=O)c1cccc2c(-c3cnc4c(c3Cl)C3(CC3)CN4)c[nH]c12
O=C1CCCCN1c1cccc2c(-c3cnc4c(c3)C3(CC3)CN4)c[nH]c12
O=C1CCCCN1c1cccc2c(-c3cnc4c(c3Cl)C3(CCC(O)C3)CN4)c[nH]c12
O=C1CCCCN1c1cccc2c(-c3cnc4c(c3Cl)[C@]3(CC[C@@H](O)C3)CN4)c[nH]c12
O=C1CCCCN1c1cccc2c(-c3cnc4c(c3Cl)[C@@]3(CC[C@H](O)C3)CN4)c[nH]c12
CN(C)C(=O)Cc1cccc2c(-c3cnc4c(c3Cl)C3(CC3)CN4)c[nH]c12
O=C1COCCN1c1cccc2c(-c3cnc4c(c3Cl)C3(CC3)CN4)c[nH]c12
O=C1CNCCN1c1cccc2c(-c3cnc4c(c3)C3(CC3)CN4)c[nH]c12
CN1CCN(c2cccc3c(-c4cnc5c(c4Cl)C4(CCC(C(N)=O)C4)CN5)c[nH]c23)C(=O)C1
NC(=O)C1CCC2(CNc3ncc(-c4c[nH]c5c(N6CCNCC6=O)cccc45)c(Cl)c32)C1
CC1CC12CNc1ncc(-c3c[nH]c4c(N5CCNCC5=O)cccc34)cc12
N#Cc1ccc2[nH]cc(-c3cnc4c(c3)C3(CC3)CN4)c2c1
Cc1n[nH]cc1-c1cnc2c(c1Cl)C1(CC=CC1)CN2
COc1c(-c2ccc(N)c(C(=O)N(C)C)n2)cnc2c1C1(CC1)CN2
CN1CCN(c2cc(Cl)cc3c(-c4cnc5c(c4)C4(CC4)CN5)c[nH]c23)C(=O)C1
NC(=O)CCn1cc(-c2cnc3c(c2Cl)C2(CC=CC2)CN3)cn1
Clc1ccc2[nH]cc(-c3cnc4c(c3)C3(CC3)CN4)c2c1
Cc1ccc2[nH]cc(-c3cnc4c(c3)C3(CC3)CN4)c2c1
c1ccc2c(-c3cnc4c(c3)C3(CC3)CN4)c[nH]c2c1
COc1c(-c2c[nH]c3ccc(C#N)cc23)cnc2c1C1(CC1)CN2
Fc1cccc2[nH]cc(-c3cnc4c(c3)C3(CC3)CN4)c12
OCCn1cc(-c2cnc3c(c2Cl)C2(CC=CC2)CN3)cn1
NC(=O)Cn1cc(-c2cnc3c(c2Cl)C2(CC=CC2)CN3)cn1
CN(C)C(=O)Cn1cc(-c2cnc3c(c2Cl)C2(CC=CC2)CN3)cn1
CC(C)(O)Cn1cc(-c2cnc3c(c2Cl)C2(CC=CC2)CN3)cn1
Cc1[nH]ncc1-c1cnc2c(c1)C1(CC1)CN2
N#Cc1ccc2[nH]nc(-c3cnc4c(c3)C3(CC3)CN4)c2c1
Clc1c(-c2cnn(Cc3ccccc3)c2)cnc2c1C1(CC=CC1)CN2
CN1CCN(c2cc(C#N)cc3c(-c4cnc5c(c4)C4(CC4)CN5)c[nH]c23)C(=O)C1
N#Cc1ccc2[nH]cc(-c3cnc4c(c3Cl)C3(CCC(O)CC3)CN4)c2c1
Cc1n[nH]cc1-c1ccc2[nH]cc(-c3cnc4c(c3)C3(CC3)CN4)c2c1
COCCn1cc(-c2cnc3c(c2Cl)C2(CC=CC2)CN3)cn1
c1nc2c(cc1-c1c[nH]c3ccc(C4CC4)cc13)C1(CC1)CN2
c1cc2[nH]cc(-c3cnc4c(c3)C3(CC3)CN4)c2cn1
CC1(C#N)CCC2(CNc3ncc(-c4c[nH]c5ccc(C#N)cc45)c(Cl)c32)C1
CS(=N)(=O)c1ccc2[nH]cc(-c3cnc4c(c3)C3(CC3)CN4)c2c1
c1ccc2c(c1)nnn2-c1cnc2c(c1)C1(CC1)CN2
c1cc2c(-c3cnc4c(c3)C3(CC3)CN4)c[nH]c2cn1
c1nnc(-c2ccc3[nH]cc(-c4cnc5c(c4)C4(CC4)CN5)c3c2)o1
Cn1cnnc1-c1ccc2[nH]cc(-c3cnc4c(c3)C3(CC3)CN4)c2c1
Cc1cc2[nH]cc(-c3cnc4c(c3)C3(CC3)CN4)c2cc1-c1cnn(C)c1
CC1(C(N)=O)CCC2(CNc3ncc(-c4c[nH]c5ccc(C#N)cc45)c(Cl)c32)C1
Fc1ccc2[nH]cc(-c3cnc4c(c3)C3(CC3)CN4)c2c1
CN(C)C(=O)c1ccc2[nH]cc(-c3cnc4c(c3)C3(CC3)CN4)c2c1
N#Cc1cc(N(C)S(C)(=O)=O)c2[nH]cc(-c3cnc4c(c3)C3(CC3)CN4)c2c1
N#Cc1cc(N(C)S(C)(=O)=O)c2c(c1)c(-c1cnc3c(c1)C1(CC1)CN3)cn2C
N#CCc1ccc2[nH]cc(-c3cnc4c(c3)C3(CC3)CN4)c2c1
CN(c1ccc2c(c1)ncn2-c1cnc2c(c1)C1(CC1)CN2)c1cnn(C)c1
N#Cc1ccc2ccn(-c3cnc4c(c3)C3(CC3)CN4)c2c1
Cn1cc(Nc2ccc3c(c2)N=CC3c2cnc3c(c2)C2(CC2)CN3)cn1
COc1cccc(F)c1-c1nccc(C(=O)Nc2cc(F)ccc2N2C[C@@H]3C[C@H]2CN3)c1F
COc1cccc(F)c1-c1nccc(C(=O)Nc2cc(F)ccc2N2C[C@H]3C[C@@H]2CN3)c1F
COc1cccc(F)c1-c1cccc(C(=O)Nc2cc(F)ccc2N2C[C@H]3C[C@@H]2CN3)c1F
COc1ccc(Cl)c(F)c1-c1nccc(C(=O)Nc2cc(F)ccc2N2C[C@H]3C[C@@H]2CN3)c1F
COc1ccc(F)c(F)c1-c1nccc(C(=O)Nc2cc(F)ccc2N2C[C@H]3C[C@@H]2CN3)c1F
COc1cccc(Cl)c1-c1nccc(C(=O)Nc2cc(F)ccc2N2C[C@H]3C[C@@H]2CN3)c1F
COc1cccc(F)c1-c1nccc(C(=O)Nc2ccc3c(nc(C)n3C)c2N2C[C@H]3C[C@@H]2CN3)c1F
COc1cccc(F)c1-c1nccc(C(=O)Nc2ccc3c(nc(C)n3C)c2N2CCC(N)CC2)c1F
COc1cccc(F)c1-c1nccc(C(=O)Nc2ccc3c(nc(C)n3C)c2N2CCC[C@H]2CO)c1F
COc1cccc(F)c1-c1nccc(C(=O)Nc2ccc3c(nc(C)n3C)c2N2CC[C@H](N)C2)c1F
COCCn1c(C)nc2c(N3CC[C@H](N)C3)c(NC(=O)c3ccnc(-c4c(F)cccc4OC)c3F)ccc21
COc1cccc(F)c1-c1nccc(C(=O)Nc2ccc(-c3cnccc3C#N)cc2N2CC[C@H](N)C2)c1F
COc1cccc(F)c1-c1nccc(C(=O)Nc2ccc(-c3cnccc3C#N)cc2N2C[C@@H](N)C[C@H]2CO)c1F
COc1cccc(F)c1-c1nccc(C(=O)Nc2ccc3c(nc(-c4ccncc4F)n3C)c2N2CC[C@H](N)C2)c1F
COCc1nc2c(N3CC[C@H](N)C3)c(NC(=O)c3ccnc(-c4c(F)cccc4OC)c3F)ccc2n1C
Cn1c(C(F)(F)F)nc2c(N3CCC[C@H]3CN)c(NC(=O)c3ccnn(-c4c(F)cccc4F)c3=O)ccc21
COc1cccc(F)c1-n1nccc(C(=O)Nc2ccc3c(nc(C(F)(F)F)n3C)c2N2CC[C@H](N)C2)c1=O
Cn1c(-c2ccncc2F)nc2c(N3CC[C@H](N)C3)c(NC(=O)c3ccnn(-c4c(F)cccc4F)c3=O)ccc21
Cn1c(-c2ccncc2F)nc2c(N3CCC[C@H]3CN)c(NC(=O)c3ccnn(-c4c(F)cccc4F)c3=O)ccc21
COCc1nc2c(N3CC[C@H](N)C3)c(NC(=O)c3ccnn(-c4c(F)cccc4F)c3=O)ccc2n1C
COCCn1c(C)nc2c(N3CCC[C@H]3CN)c(NC(=O)c3ccnn(-c4c(F)cccc4F)c3=O)ccc21
CC(C)c1nc2c(N3CC[C@H](N)C3)c(NC(=O)c3ccnn(-c4c(F)cccc4F)c3=O)ccc2n1C
Cc1nc2c(N3CC[C@H](N)C3)c(NC(=O)c3ccnn(-c4c(F)cccc4F)c3=O)ccc2n1C1CCOCC1
Cc5nc4c(N1CC[C@H](N)C1)c(NC(=O)c3ccnn(c2c(F)cccc2F)c3=O)ccc4n5C6CC6
Cc1nc2c(N3CC[C@H](N)C3)c(NC(=O)c3ccnn(-c4c(Cl)cccc4Cl)c3=O)ccc2n1C
COc1ccc(F)cc1-n1nccc(C(=O)Nc2ccc3c(nc(C)n3C)c2N2CC[C@H](N)C2)c1=O
COc1cccc(F)c1-n1cccc(C(=O)Nc2cc(F)ccc2N2C[C@H]3C[C@@H]2CN3)c1=O
COc1cccc(F)c1-n1cccc(C(=O)Nc2cc(F)c3nn(C)cc3c2N2C[C@H]3C[C@@H]2CN3)c1=O
COc1cccc(F)c1-n1cccc(C(=O)Nc2cc(F)c3c(cnn3C)c2N2C[C@H]3C[C@@H]2CN3)c1=O
COc1cccc(F)c1-n1cccc(C(=O)Nc2ccc3c(nc(C)n3C)c2N2CCC[C@H]2CN)c1=O
COc1cccc(F)c1-c1nc(C(=O)Nc2cc(F)ccc2N2C[C@@H]3C[C@H]2CN3)cs1
COc1cccc(F)c1-c1csc(C(=O)Nc2cc(F)ccc2N2C[C@@H]3C[C@H]2CN3)n1
COc1cccc(F)c1-n1nc(C(=O)Nc2ccc3c(nc(C)n3C)c2N2CC[C@H](N)C2)ccc1=O
Cc1nc2c(N3CCC[C@@H](N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1C
Cc1nc2c(N3C[C@@H](N)C[C@H]3CO)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1C
Cc1nc2c(N3CCN(C)CC3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1C
Cc1nc2c(N(C)[C@@H]3CCCNC3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1C
Cc1nc2c(N3CCNCC3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1C
Cc1nc2c(N3CC[C@H](N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1C
Cc1nc2c(N3CC[C@@H](N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1C
Cc1nc2c(N3CCC(N)CC3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1C
Cc1nc2c(N3C[C@@H]4C[C@H]3CN4)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1C
Cc1nc2c(N3CCC(C)(N)CC3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1C
Cc1nc2c(N3CC[C@](C)(N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1C
Cc1nc2c(N3CCC4(CC3)CNC4)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1C
Cc1nc2c(N3CC4CNCC4C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1C
Cc1nc2c(N3C[C@H]4C[C@@H]3CN4)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1C
Cc1nc2c(N3CCNC4(CC4)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1C
Cc1nc2c(N3CC[C@H](O)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1C
Cc1nc2c(N3CCNC(=O)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1C
Cc1nc2c(N3CCCC4(CNC4)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1C
Cc1nc2c(N3CCC4(CNC4)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1C
Cc1nc2c(N(C)CC3CNC3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1C
Cn1ncc2c(N3C[C@@H]4C[C@H]3CN4)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc21
Cc1nc2c(N3CC[C@H](N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1C1CCOCC1
COCCn1c(C)nc2c(N3CC[C@H](N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc21
Cc1nc2c(N3CC[C@@](C)(N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1C
CC1=NC2C(N3C[C@H](N)C4(CC4)C3)=C(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)C=CC2N1C
Cc1nc2c(N3CC[C@@H](NC(=O)CN)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1C
Cc1nc2c(N3CCC[C@H]3CN)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1C
Cc1nc2c(N3C[C@H](N)C(F)(F)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1C
Cc1nc2c(N3CCC(N)C(F)(F)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1C
Cc1nc2c(N3CC(N)CC(F)(F)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1C
Cn1c(C2CC2)nc2c(N3CC[C@H](N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc21
Cn1c(C(C)(C)C)nc2c(N3CC[C@H](N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc21
Cn1c(C(C)(C)C)nc2c(N3CC[C@@H](N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc21
Cn1c(C(C)(C)C)nc2c(N3CC[C@@](C)(N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc21
Cn1c(C(C)(C)C)nc2c(N3CC[C@@](C)(N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc21
Cn1c(C(C)(C)C)nc2c(N3CC[C@@H](O)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc21
Cn1c(C(C)(C)C)nc2c(N3CCC[C@H]3CN)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc21
C[C@@H]1CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3c2nc(C(C)(C)C)n3C)C[C@@H]1N
Cn1c(C(C)(C)C)nc2c(N3CCC(N)(CO)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc21
Cc1nc2c(N3CC[C@H](N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1C1CCN(C)CC1
Cc1nc2c(N3CC[C@H](N)C3)c(NC(=O)c3ccc(=O)n(-c4c(Cl)cccc4Cl)n3)ccc2n1C
Cc1nc2c(N3CC[C@@H](N)C3)c(NC(=O)c3ccc(=O)n(-c4c(Cl)cccc4Cl)n3)ccc2n1C
CC(C)c1nc2c(N3CC[C@@H](N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1C
CC(C)c1nc2c(N3C[C@@H](C)[C@@H](N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1C
CC(C)c1nc2c(N3C[C@H](C)[C@@H](N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1C
CC(C)c1nc2c(N3CC4C[C@]4(N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1C
CC(C)c1nc2c(N3C[C@H](N)C4(COC4)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1C
CC(C)n1cc2c(N3CC[C@@H](N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1
CC(C)c1nc2c(N3CC[C@H](CN)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1C
CC(C)c1nc2c(N3CC[C@@H](CN)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1C
CC(C)c1nc2c(N3CC[C@@H](O)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1C
CC(C)c1nc2c(N3CC4[C@@H](N)[C@@H]4C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1C
CC(C)c1nc2c(N3CC4C(N)C4C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1C
CC(C)c1nc2c(N3CC[C@@H](N)C3)c(NC(=O)c3nn(-c4c(F)cccc4F)c(=O)cc3Cl)ccc2n1C
CC[C@@]1(N)CCN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3c2nc(C(C)C)n3C)C1
CC[C@]1(N)CCN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3c2nc(C(C)C)n3C)C1
CC(C)c1nc2c(N3CC[C@@](C)(N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1C
CC(C)c1nc2c(N3CC[C@](N)(CO)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1C
CC(C)c1nc2c(N3CC[C@](N)(CO)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1C
CC(C)c1nc2c(N3CC[C@@H](N(C)C)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1C
CN[C@@H]1CCN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3c2nc(C(C)C)n3C)C1
CC(C)c1nc2c(N3CC[C@@H](NC(=O)CCN)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1C
CC(C)c1nc2c(N3CC[C@@H](NCC(C)(C)O)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1C
CC(C)c1nc2c(N3CC[C@@H](NCCO)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1C
CC(C)c1nc2c(N3CC[C@@H](NC(=O)CN)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1C
CC(C)c1nc2c(N3CC[C@H](N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1C
CC(C)c1nc2c(N3CCC(N)CC3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1C
CC(C)c1nc2c(N3CCC[C@H]3CN)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1C
CC(C)c1nc2c(N3CC[C@H]4NCC[C@H]43)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1C
CC(C)c1nc2c(N3CCC4(CCNC4)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1C
CC(C)c1nc2c(N3C[C@H]4CNC[C@H]4C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1C
CC(C)c1nc2c(N3CC[C@](N)(C(F)(F)F)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1C
CC(C)c1nc2c(N3CC[C@](N)(C(F)(F)F)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1C
CC(C)c1nc2c(N3CC[C@@](C)(O)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1C
CC(C)c1nc2c(N3CC(F)(F)C[C@H]3CN)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1C
CC(C)c1nc2c(N3CC(N)C(O)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1C
CC(C)c1nc2c(N3CC[C@@H](N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)cc(F)c2n1C
CC(C)c1nc2c(N3CC(F)(F)C[C@H]3CN)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)cc(F)c2n1C
CC(C)c1nc2c(N3C[C@@H]4[C@H](N)[C@@H]4C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)cc(F)c2n1C
Cn1c(C2(C(F)(F)F)CC2)nc2c(N3CC[C@@H](N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc21
Cn1c(C2(C(F)(F)F)CC2)nc2c(N3C[C@H](N)C(C)(C)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc21
C[C@@H]1CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3c2nc(C2(C(F)(F)F)CC2)n3C)C[C@@H]1N
Cn1c(C2(C(F)(F)F)CC2)nc2c(N3C[C@H](N)C4(CC4)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc21
Cc1nc2c(N3C[C@H](N)C(C)(C)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1[C@H]1CCOC1
Cc1nc2c(N3C[C@H](N)C4(CC4)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1C1CCOCC1
Cc1nc2c(N3C[C@H](N)C4(CC4)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1[C@H]1CCOC1
C[C@@H]1CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3c2ncn3C2CCOCC2)C[C@@H]1N
CC(C)n1cnc2c(N3C[C@@H](C)[C@@H](N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc21
Cn1c(C(C)(C)F)nc2c(N3CC[C@@H](N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc21
Cn1c(CC(F)(F)F)nc2c(N3CC[C@@H](N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc21
Cn1c(C(C)(C)F)nc2c(N3CC[C@@H](N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)cc(F)c21
Cn1c(C(C)(C)C(F)(F)F)nc2c(N3CC[C@@H](N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc21
Cn1c(C(F)F)nc2c(N3CC[C@@H](N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc21
Cn1c(C2CC2)nc2c(N3CC[C@@H](N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc21
Cn1c(C(F)F)nc2c(N3CC[C@H](N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc21
CSCc1nc2c(N3CC[C@@H](N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1C
CC(C)c1nc2c(N3CC[C@@H](N)C3)c(NC(=O)c3ccnn(-c4c(F)cccc4F)c3=O)ccc2n1C
COc1cccc(F)c1-c1nccc(C(=O)Nc2ccc3c(nc(C(F)F)n3C)c2N2CC[C@@H](N)C2)c1F
COc1cccc(F)c1-c1nccc(C(=O)Nc2ccc3c(nc(CS(C)(=O)=O)n3C)c2N2CC[C@@H](N)C2)c1F
C[C@@H]1CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3c2cnn3C)C[C@@H]1N
Cn1ncc2c(N3CC[C@@H](N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc21
Cn1ncc2c(N3CCC(N)CC3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)cc(F)c21
Cn1ncc2c(N3CCC[C@@H](N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)cc(F)c21
C[C@@H]1CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)cc(F)c3c2cnn3C)C[C@@H]1N
[2H]C([2H])([2H])n1ncc2c(N3C[C@@H](C)[C@@H](N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc21
[2H]C([2H])([2H])n1ncc2c(N3C[C@H](N)C4(CC4)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc21
C[C@H]1CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3c2cnn3C)C[C@@H]1N
Cn1ncc2c(N3C[C@H](N)C4(CC4)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc21
Cn1cc2c(N3CC[C@@H](N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1
Cn1cc2c(N3CCC[C@@H](N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1
Cn1cc2c(N3CCC(N)CC3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1
[2H]C([2H])([2H])n1cc2c(N3C[C@@H](C)[C@@H](N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1
CC(C)n1ncc2c(N3CC[C@@H](N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc21
CC(C)n1ncc2c(N3C[C@@H](C)[C@@H](N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc21
CC(C)n1ncc2c(N3CCC[C@@H]3CN)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc21
CC(C)n1ncc2c(N3C[C@H](N)C4(CC4)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc21
CC(C)n1ncc2c(N3CCC[C@@H](N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc21
CC(C)n1ncc2c(N3CCC(N)CC3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc21
Cc1cc(NC(=O)c2ccc(=O)n(-c3c(F)cccc3F)n2)c(N2CC[C@@H](N)C2)c2cnn(C(C)C)c12
CC(C)n1ncc2c(N3C[C@H](N)C(C)(C)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc21
CC(C)n1ncc2c(N3C[C@@H](N)C(C)(C)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc21
CC(C)n1ncc2c(N3CC[C@@H](N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)cc(F)c21
CC(C)n1ncc2c(N3C[C@H](N)C4(CC4)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)cc(F)c21
CC(C)n1nc(Cl)c2c(N3CC[C@@H](N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)cc(F)c21
CC(C)n1nc(Cl)c2c(N3C[C@@H](C)[C@@H](N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc21
Cc1nn(C(C)C)c2ccc(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)c(N3C[C@@H](C)[C@@H](N)C3)c12
CC(C)n1ncc2c(N3C[C@@H](C)[C@@H](N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)cc(F)c21
CC(C)n1ncc2c(N3C[C@@H]4NCCO[C@H]4C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc21
Cc1nn(C(C)C)c2ccc(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)c(N3CC[C@@H](N)C3)c12
CC[C@@H]1CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3c2cnn3C(C)C)C[C@@H]1N
CC[C@@H]1CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3c2cnn3C(C)C)C[C@@H]1N
CC(C)n1nc(F)c2c(N3C[C@@H](C)[C@@H](N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc21
CC(C)n1nc(F)c2c(N3C[C@H](N)C4(CC4)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc21
CO[C@H]1CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3c2cnn3C(C)C)C[C@@H]1N
CO[C@@H]1CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3c2cnn3C(C)C)C[C@H]1N
Cc1nn(C(C)C)c2ccc(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)c(N3C[C@H](N)C4(CC4)C3)c12
CC[C@H]1CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)cc(F)c3c2cnn3C(C)C)C[C@H]1N
CC(C)n1ncc2c(N3CC[C@@H](CN)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)cc(F)c21
CO[C@H]1CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3c2cnn3C(C)C)C[C@H]1N
CC(C)n1ncc2c(N3CC(N)C4(COC4)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc21
CC(C)n1ncc2c(N3CC[C@H](N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc21
CC(C)n1ncc2c(N3CC[C@@](C)(N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc21
CC(C)n1ncc2c(N3C[C@H](C)[C@@H](N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc21
CC(C)n1ncc2c(N3C[C@H](N)C4(CC4)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc21
CC(C)n1ncc2c(N3C[C@@H]4[C@@H](N)[C@@H]4C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc21
CC(C)n1ncc2c(N3C[C@@H](N)C[C@H]3CO)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc21
CC(C)n1ncc2c(N3CC[C@@H](NCCO)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc21
CC(C)n1ncc2c(N3C[C@@H](C)[C@@H](NCCO)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc21
CC(C)n1ncc2c(N3C[C@@H](C)[C@@H](N)C3)c(NC(=O)c3ccc(=O)n(-c4ccccc4F)n3)ccc21
CC[C@@H]1CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)cc(F)c3c2cnn3C(C)C)C[C@@H]1N
CC(C)n1ncc2c(N3CCC(N)CC3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)cc(F)c21
Cc1nn(C(C)C)c2c(F)cc(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)c(N3C[C@@H](C)[C@@H](N)C3)c12
CC(C)n1ncc2c(N3C[C@H]4CNC[C@H]4C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)cc(F)c21
CC(C)n1cc2c(N3CC[C@@](C)(N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1
CC(C)n1cc2c(N3CC[C@@H](CN)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)cc(F)c2n1
CC(C)n1cc2c(N3CC[C@@H](N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)cc(F)c2n1
CC(C)n1nc2c(F)cc(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)c(N3CC[C@@H](N)C3)c2c1Cl
CC(C)n1cc2c(N3C[C@@H](C)[C@@H](N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1
CC(C)n1cc2c(N3CCC[C@@H]3CN)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1
Cc1cc(NC(=O)c2ccc(=O)n(-c3c(F)cccc3F)n2)c(N2CC[C@@H](N)C2)c2cn(C(C)C)nc12
CC(C)n1cc2c(N3C[C@H](N)C(C)(C)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1
CC(C)n1cc2c(N3C[C@@H](N)C(C)(C)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1
CC(C)n1cc2c(N3C[C@H](N)C4(CC4)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1
CC(C)n1cc2c(N3CCC(N)CC3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1
CC(C)n1cc2c(N3C[C@H](C)[C@@H](N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1
CC(C)n1cc2c(N3CCC[C@@H](N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1
CC(C)n1cc2c(N3C[C@@H]4C[C@H]3CN4)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)cc(F)c2n1
C[C@@H]1CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3nn(C(C)(C)C)cc23)C[C@@H]1N
CC(C)(C)n1cc2c(N3C[C@H](N)C4(CC4)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1
CC1(C)CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3nn(C(C)(C)C)cc23)C[C@@H]1N
CC1(C)CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3nn(C(C)(C)C)cc23)C[C@H]1N
C[C@H]1CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3nn(C(C)(C)C)cc23)C[C@@H]1N
CC(C)(C)n1cc2c(N3CCC[C@@H](N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1
CC(C)(C)n1cc2c(N3CCC(N)CC3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1
CC(C)(C)n1cc2c(N3CC[C@@H](N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1
CC(C)(C)n1cc2c(N3C[C@@H](N)C4(CC4)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1
CCC(C)(C)n1cc2c(N3C[C@H](C)[C@@H](N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1
CCC(C)(C)n1cc2c(N3C[C@@H](C)[C@@H](N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1
C[C@@H]1CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3nn(C(C)(C)C(C)(C)C)cc23)C[C@@H]1N
CC(C)(C)C(C)(C)n1cc2c(N3C[C@H](N)C4(CC4)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1
CC(C)C(C)(C)n1cc2c(N3C[C@@H](C)[C@@H](N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1
CC(C)C(C)(C)n1cc2c(N3C[C@H](N)C4(CC4)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1
N[C@H]1CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3c2cnn3[C@H]2CCOC2)CC12CC2
N[C@H]1CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3c2cnn3[C@@H]2CCOC2)CC12CC2
N[C@H]1CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3c2cnn3C2CCOCC2)CC12CC2
C[C@@H]1CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3c2cnn3[C@@H]2CCCOC2)C[C@@H]1N
C[C@@H]1CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3c2cnn3[C@H]2CCCOC2)C[C@@H]1N
C[C@@H]1CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3c2cnn3[C@H]2CCOC2)C[C@@H]1N
CC[C@H](C)n1ncc2c(N3C[C@@H](C)[C@@H](N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc21
CC[C@@H](C)n1ncc2c(N3C[C@@H](C)[C@@H](N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc21
C[C@@H]1CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3c2cnn3C2COC2)C[C@@H]1N
C[C@H]1CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3c2cnn3[C@@H]2CCOC2)C[C@@H]1N
C[C@H]1CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3c2cnn3[C@H]2CCOC2)C[C@@H]1N
C[C@@H]1CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3c2cnn3C2CCOCC2)C[C@@H]1N
C[C@@H]1CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3c2cnn3[C@@H]2CCOC2)C[C@@H]1N
N[C@@H]1CCCN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3c2cnn3[C@H]2CCOC2)C1
N[C@@H]1CCCN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3c2cnn3[C@@H]2CCOC2)C1
NC1CCN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3c2cnn3[C@@H]2CCOC2)CC1
NC1CCN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3c2cnn3[C@H]2CCOC2)CC1
CC1(C)CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3c2cnn3[C@@H]2CCOC2)C[C@@H]1N
CC1(C)CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3c2cnn3[C@@H]2CCOC2)C[C@H]1N
CC1(C)CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3c2cnn3[C@H]2CCOC2)C[C@@H]1N
CC1(C)CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3c2cnn3[C@H]2CCOC2)C[C@H]1N
N[C@H]1CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3c2cnn3[C@H]2CCCOC2)CC12CC2
N[C@H]1CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3c2cnn3[C@@H]2CCCOC2)CC12CC2
C[C@H]1CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3c2cnn3C2CCOCC2)C[C@@H]1N
N[C@@H]1CCN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3c2cnn3C2CCOCC2)C1
[2H]C([2H])([2H])C([2H])(n5ncc4c(N1C[C@@H](C)[C@@H](N)C1)c(NC(=O)c3ccc(=O)n(c2c(F)cccc2F)n3)ccc45)C([2H])([2H])[2H]
[2H]C([2H])([2H])C([2H])(n6ncc5c(N2C[C@H](N)C1(CC1)C2)c(NC(=O)c4ccc(=O)n(c3c(F)cccc3F)n4)ccc56)C([2H])([2H])[2H]
[2H]C([2H])([2H])C(n6ncc5c(N2C[C@H](N)C1(CC1)C2)c(NC(=O)c4ccc(=O)n(c3c(F)cccc3F)n4)ccc56)C([2H])([2H])[2H]
[2H]C([2H])([2H])C(n5ncc4c(N1C[C@@H](C)[C@@H](N)C1)c(NC(=O)c3ccc(=O)n(c2c(F)cccc2F)n3)ccc45)C([2H])([2H])[2H]
[2H]C([2H])([2H])C(n5ncc4c(N1C[C@H](N)C(C)(C)C1)c(NC(=O)c3ccc(=O)n(c2c(F)cccc2F)n3)ccc45)C([2H])([2H])[2H]
[2H]C([2H])([2H])C(n5ncc4c(N1C[C@@H](N)C(C)(C)C1)c(NC(=O)c3ccc(=O)n(c2c(F)cccc2F)n3)ccc45)C([2H])([2H])[2H]
[2H]C([2H])([2H])C([2H])(n5ncc4c(N1C[C@H](N)C(C)(C)C1)c(NC(=O)c3ccc(=O)n(c2c(F)cccc2F)n3)ccc45)C([2H])([2H])[2H]
[2H]C([2H])([2H])C([2H])(n5ncc4c(N1C[C@@H](N)C(C)(C)C1)c(NC(=O)c3ccc(=O)n(c2c(F)cccc2F)n3)ccc45)C([2H])([2H])[2H]
COCCn1ncc2c(N3C[C@@H](C)[C@@H](N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc21
COCCn1ncc2c(N3CCC(N)CC3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)cc(F)c21
COCCn1ncc2c(N3CC[C@@H](N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc21
COCCn1ncc2c(N3CCC[C@@H](N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)cc(F)c21
N[C@@H]1CCN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3c2cnn3C2CCCC2)C1
C[C@@H]1CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3c2cnn3C2CCCC2)C[C@@H]1N
CCn1ncc2c(N3CC[C@@H](N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)cc(F)c21
N[C@@H]1CCN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3c2cnn3CC(F)(F)F)C1
C[C@@H]1CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3c2cnn3CC(F)(F)F)C[C@@H]1N
CCn1ncc2c(N3CC[C@@H](N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc21
COCCn1ncc2c(N3CC[C@@H](N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)cc(F)c21
CC(C)Cn1ncc2c(N3CC[C@@H](N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc21
N[C@@H]1CCN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3c2cnn3CC2CC2)C1
C[C@@H]1CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3c2cnn3C2CCC2)C[C@@H]1N
C[C@@H]1CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3c2cnn3C2CCCCC2)C[C@@H]1N
C[C@@H]1CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3c2cnn3C2CC2)C[C@@H]1N
N#Cc1ccncc1-c1ccc(NC(=O)c2ccc(=O)n(-c3c(F)cccc3F)n2)c(N2CC[C@@H](N)C2)c1
N[C@H]1CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3c2cnn3C2CC2)CC12CC2
N[C@@H]1CCN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3c2cnn3C2CC2)C1
CC(C)(C)n1ncc2c(N3C[C@H](N)C4(CC4)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc21
C[C@@H]1CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3c2cnn3C(C)(C)C)C[C@@H]1N
C[C@@H]1CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3nn(C45CCC(CC4)CC5)cc23)C[C@@H]1N
C[C@@H]1CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3nn(C45CC6CC(CC(C6)C4)C5)cc23)C[C@@H]1N
C[C@@H]1CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3nn(C45CCC(CC4)C5)cc23)C[C@@H]1N
C[C@@H]1CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3nn(C4CC(F)(F)C4)cc23)C[C@@H]1N
C[C@@H]1CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3nn(C4CCN(C)CC4)cc23)C[C@@H]1N
C[C@H]1CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3nn(C4CC(F)(F)C4)cc23)C[C@@H]1N
C[C@H]1CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3nn(C4(C)CC4)cc23)C[C@@H]1N
CC1(n2cc3c(N4C[C@H](N)C5(CC5)C4)c(NC(=O)c4ccc(=O)n(-c5c(F)cccc5F)n4)ccc3n2)CC1
C[C@H]1CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3nn(C45CCC(CC4)C5)cc23)C[C@@H]1N
N[C@H]1CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3nn(C4(C(F)(F)F)CC4)cc23)CC12CC2
CC1(C)CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3nn(C4(C(F)(F)F)CC4)cc23)C[C@@H]1N
C[C@@H]1CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3nn(C4(C(F)(F)F)CC4)cc23)C[C@@H]1N
C[C@@H]1CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3nn(C45CC(C4)C5)cc23)C[C@@H]1N
C[C@@H]1CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3nn(C4(C)CCC4)cc23)C[C@@H]1N
C[C@@H]1CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3nn(C45CC(C)(C4)C5)cc23)C[C@@H]1N
C[C@@H]1CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3nn(C45CC(C(F)(F)F)(C4)C5)cc23)C[C@@H]1N
C[C@H]1CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3nn(C45CC(C4)C5)cc23)C[C@@H]1N
C[C@H]1CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3nn(C4(C)CCC4)cc23)C[C@@H]1N
CC1(C)CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3nn([C@@H]4CCOC4)cc23)C[C@@H]1N
CC1(C)CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3nn([C@@H]4CCOC4)cc23)C[C@H]1N
CC1(C)CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3nn([C@H]4CCOC4)cc23)C[C@@H]1N
CC1(C)CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3nn([C@H]4CCOC4)cc23)C[C@H]1N
C[C@H]1CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3nn([C@@H]4CCOC4)cc23)C[C@@H]1N
C[C@H]1CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3nn([C@H]4CCOC4)cc23)C[C@@H]1N
COCCn1cc2c(N3CC[C@@H](N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1
CCn1cc2c(N3CC[C@@H](N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1
N[C@@H]1CCN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3nn(CC4CC4)cc23)C1
CC(C)Cn1cc2c(N3CC[C@@H](N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1
C[C@@H]1CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3nn(C4CCC(F)(F)CC4)cc23)C[C@@H]1N
C[C@@H]1CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3nn(C4CCCC4)cc23)C[C@@H]1N
CC1(C)CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3nn(C4CC4)cc23)C[C@@H]1N
CC1(C)CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3nn(C4CC4)cc23)C[C@H]1N
N[C@H]1CN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3nn(C4CC4)cc23)CC12CC2
N[C@@H]1CCN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3nn(C4CCOCC4)cc23)C1
N[C@@H]1CCN(c2c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc3nn(CC(F)(F)F)cc23)C1
[2H]C([2H])([2H])C(n1cc2c(N3C[C@H](N)C4(CC4)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc2n1)C([2H])([2H])[2H]
CC(C)n1nnc2c(N3C[C@H](N)C4(CC4)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc21
CC(C)n1nnc2c(N3C[C@@H](C)[C@@H](N)C3)c(NC(=O)c3ccc(=O)n(-c4c(F)cccc4F)n3)ccc21
N#Cc1ccncc1-c1ccc(NC(=O)c2ccc(=O)n(-c3c(F)cccc3F)n2)c(N2CCNCC2)c1
N#Cc1ccncc1-c1ccc(NC(=O)c2ccc(=O)n(-c3c(F)cccc3F)n2)c(N2CC[C@@H](N)C2)c1
N#Cc1ccncc1-c1ccc(NC(=O)c2ccc(=O)n(-c3c(F)cccc3F)n2)c(N2CC[C@H](N)C2)c1
N#Cc1ccncc1-c1ccc(NC(=O)c2ccc(=O)n(-c3c(F)cccc3F)n2)c(N2CCC[C@@H](N)C2)c1
N#Cc1ccncc1-c1ccc(NC(=O)c2ccc(=O)n(-c3c(F)cccc3F)n2)c(N2CCC(N)CC2)c1
N#Cc1ccncc1-c1ccc(NC(=O)c2ccc(=O)n(-c3c(F)cccc3F)n2)c(N2C[C@@H](N)C[C@H]2CO)c1
C[C@]1(N)CCN(c2cc(-c3cnccc3C#N)ccc2NC(=O)c2ccc(=O)n(-c3c(F)cccc3F)n2)C1
N#Cc1ccncc1-c1ccc(NC(=O)c2ccc(=O)n(-c3c(F)cccc3F)n2)c(N2CCC(O)CC2)c1
N#Cc1ccncc1-c1ccc(NC(=O)c2ccc(=O)n(-c3c(F)cccc3F)n2)c(N2CCN[C@H](CO)C2)c1
N#Cc1ccncc1-c1ccc(NC(=O)c2ccc(=O)n(-c3c(F)cccc3F)n2)c(N2C[C@H](N)C[C@H]2CO)c1
N#Cc1ccncc1-c1ccc(NC(=O)c2ccc(=O)n(-c3c(F)cccc3F)n2)c(N2CCC(N)(CO)CC2)c1
C[C@]1(O)CCN(c2cc(-c3cnccc3C#N)ccc2NC(=O)c2ccc(=O)n(-c3c(F)cccc3F)n2)C1
C[C@]1(O)CCN(c2cc(-c3cnccc3C#N)ccc2NC(=O)c2ccc(=O)n(-c3c(F)cccc3F)n2)C1
N#Cc1ccncc1-c1ccc(NC(=O)c2ccc(=O)n(-c3c(F)cccc3F)n2)c(N2CC[C@@](N)(CO)C2)c1
N#Cc1ccncc1-c1ccc(NC(=O)c2ccc(=O)n(-c3c(F)cccc3F)n2)c(N2CC[C@@](N)(CO)C2)c1
N#Cc1ccncc1-c1ccc(NC(=O)c2ccc(=O)n(-c3c(F)cccc3F)n2)c(N2CCC(F)(F)[C@@H](N)C2)c1
N#Cc1ccncc1-c1ccc(NC(=O)c2ccc(=O)n(-c3c(F)cccc3F)n2)c(N2CC[C@](N)(C(F)(F)F)C2)c1
N#Cc1ccncc1-c1ccc(NC(=O)c2ccc(=O)n(-c3c(F)cccc3F)n2)c(N2CC[C@](N)(C(F)(F)F)C2)c1
N#Cc1ccncc1-c1ccc(NC(=O)c2ccc(=O)n(-c3c(F)cccc3F)n2)c(N2CCC(NCCO)CC2)c1
N#Cc1ccncc1-c1ccc(NC(=O)c2ccc(=O)n(-c3c(F)cccc3Cl)n2)c(N2C[C@@H](N)C[C@H]2CO)c1
COc1cccc(F)c1c5nccc(C(=O)Nc3ccc(c2cnccc2C#N)cc3N4C[C@@H](N)C[C@H]4CO)n5
Cn1cccc1-c1cc2cc(NC(=O)C3CC3F)ncc2c(N)c1F
C=Cn1cccc1-c1cc2cc(NC(=O)C3CC3F)ncc2c(N)c1F
CCn1cccc1-c1cc2cc(NC(=O)C3CC3F)ncc2c(N)c1F
Cn1cccc1-c1cc2cc(NC(=O)c3ccc(N4CCNCC4)cc3)ncc2c(N)c1F
CN1CCN(c2ccc(C(=O)Nc3cc4cc(-c5cccn5C)c(F)c(N)c4cn3)cc2)CC1
CCn1cccc1-c1cc2cc(NC(=O)C3CCC(F)CC3)ncc2c(N)c1F
Cn1cccc1-c1cc2cc(NC(=O)c3ccc(N4CCOCC4)cc3)ncc2c(N)c1F
CC(C)n1cccc1-c1cc2cc(NC(=O)C3CC3F)ncc2c(N)c1F
CN1CCN(c2ccc(C(=O)Nc3cc4cc(-c5cccn5C)c(F)c(N)c4cn3)nc2)CC1
Cn1cccc1-c1cc2cc(NC(=O)C3CC3F)ncc2c(F)c1C#N
Cc1c(F)c(C(O)C2CC2)c2[nH]ncc2c1-c1cn2cc(NC(=O)[C@@H]3C[C@@H]3F)nc2cn1
COC(c1c(F)c(C)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12)C1CC1
CCOC(C)c1c(F)c(C)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12
COCC(C)c1c(F)c(C)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12
Cc1c(F)c(C(C)C(F)F)c2[nH]ncc2c1-c1cn2cc(NC(=O)[C@@H]3C[C@@H]3F)nc2cn1
Cc1c(F)c(C2CCOC2)c2[nH]ncc2c1-c1cn2cc(NC(=O)[C@@H]3C[C@@H]3F)nc2cn1
Cc1c(F)c(C2=CC(=O)CC2)c2[nH]ncc2c1-c1cn2cc(NC(=O)[C@@H]3C[C@@H]3F)nc2cn1
Cc1c(F)c(C(C)CO)c2[nH]ncc2c1-c1cn2cc(NC(=O)[C@@H]3C[C@@H]3F)nc2cn1
Cc1c(F)c(C2CCCC2O)c2[nH]ncc2c1-c1cn2cc(NC(=O)[C@@H]3C[C@@H]3F)nc2cn1
CNC(C)c1c(F)c(C)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12
Cc1c(F)c(C2=CCCC2)c2[nH]ncc2c1-c1cn2cc(NC(=O)[C@@H]3C[C@@H]3F)nc2cn1
Cc1c(F)c(C(C)N(C)C)c2[nH]ncc2c1-c1cn2cc(NC(=O)[C@@H]3C[C@@H]3F)nc2cn1
Cc1c(F)c(C(C)CN(C)C)c2[nH]ncc2c1-c1cn2cc(NC(=O)[C@@H]3C[C@@H]3F)nc2cn1
CC(C)N(c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12)C1OC(C(=O)O)C(O)C(O)C1O
Cc1c(F)c(C2=CC(O)CC2)c2[nH]ncc2c1-c1cn2cc(NC(=O)[C@@H]3C[C@@H]3F)nc2cn1
COC1CCCC1c1c(F)c(C)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12
CN(C)c1c(F)c(C(F)F)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12
COC(=O)C6OC(N(c4c(F)c(Cl)c(c3cn2cc(NC(=O)[C@@H]1C[C@@H]1F)nc2cn3)c5cn[nH]c45)C(C)C)C(OC(C)=O)C(OC(C)=O)C6OC(C)=O
O=C(Nc1cn2cc(-c3c(C(F)F)c(F)c(C(O)C4CC4)c4[nH]ncc34)ncc2n1)[C@@H]1C[C@@H]1F
CC(C)Nc1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4C(=O)O)nc3cn2)c2cn[nH]c12
Cc1c(F)c(C(C2CC2)N2C(=O)c3ccccc3C2=O)c2[nH]ncc2c1-c1cn2cc(NC(=O)[C@@H]3C[C@@H]3F)nc2cn1
Cc1c(F)c(C(C)CN2C(=O)c3ccccc3C2=O)c2[nH]ncc2c1-c1cn2cc(NC(=O)[C@@H]3C[C@@H]3F)nc2cn1
Cc1c(F)c(C(N)C2CC2)c2[nH]ncc2c1-c1cn2cc(NC(=O)[C@@H]3C[C@@H]3F)nc2cn1
Cc1c(F)c(C(C)CN)c2[nH]ncc2c1-c1cn2cc(NC(=O)[C@@H]3C[C@@H]3F)nc2cn1
Cc1c(F)c(C(C)N)c2[nH]ncc2c1-c1cn2cc(NC(=O)[C@@H]3C[C@@H]3F)nc2cn1
CCN(CC)C(=O)[C@H]1C[C@H]1C(=O)Nc1cn2cc(-c3c(Cl)c(F)c(NC(C)C)c4[nH]ncc34)ncc2n1
CN(C)c4c(F)c(C(F)(F)F)c(c3cn2cc(NC(=O)[C@H]1C[C@H]1F)nc2cn3)c5cn[nH]c45
CC(C)Nc1c(F)c(C(F)F)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12
CCNC(=O)[C@H]1C[C@H]1C(=O)Nc1cn2cc(-c3c(Cl)c(F)c(NC(C)C)c4[nH]ncc34)ncc2n1
CN(C)c4c(F)c(C(F)(F)F)c(c3cn2cc(NC(=O)[C@@H]1C[C@H]1F)nc2cn3)c5cn[nH]c45
CN(C)c4c(F)c(C(F)(F)F)c(c3cn2cc(NC(=O)[C@H]1C[C@@H]1F)nc2cn3)c5cn[nH]c45
COC(=O)[C@H]1C[C@H]1C(=O)Nc1cn2cc(-c3c(Cl)c(F)c(NC(C)C)c4[nH]ncc34)ncc2n1
Cc1c(F)c(NC(C)C)c2[nH]ncc2c1-c1cn2cc(NC(=O)[C@H]3C[C@H]3F)nc2cn1
Cc1c(F)c(NC(C)C)c2[nH]ncc2c1-c1cn2cc(NC(=O)[C@@H]3C[C@H]3F)nc2cn1
Cc1c(F)c(NC(C)C)c2[nH]ncc2c1-c1cn2cc(NC(=O)[C@H]3C[C@@H]3F)nc2cn1
O=C(Nc5cn4cc(c2c(C(F)(F)F)c(F)c(C(O)C1CC1)c3[nH]ncc23)ncc4n5)[C@@H]6C[C@@H]6F
CC(C)Nc1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4CCl)nc3cn2)c2cn[nH]c12
CC(C)Nc1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4CO)nc3cn2)c2cn[nH]c12
CC(C)Nc1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4C(N)=O)nc3cn2)c2cn[nH]c12
CC(C)Nc1c(F)c(CO)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12
NC(c1c(F)c(C(F)F)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12)C1CC1
CC(=O)NC(c1c(F)c(C)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12)C1CC1
CC(=O)Nc1cn2cc(-c3c(Cl)c(F)c(NC(C)C)c4[nH]ncc34)ncc2n1
NC(c4c(F)c(C(F)(F)F)c(c3cn2cc(NC(=O)[C@@H]1C[C@@H]1F)nc2cn3)c5cn[nH]c45)C6CC6
CC(N)c4c(F)c(C(F)(F)F)c(c3cn2cc(NC(=O)[C@@H]1C[C@@H]1F)nc2cn3)c5cn[nH]c45
CC(C)Nc1c(F)c(Cl)c(-c2cn3cc(NC(=O)C4CC4)nc3cn2)c2cn[nH]c12
COC(=O)NC1(C(=O)Nc2cn3cc(-c4c(Cl)c(F)c(NC(C)C)c5[nH]ncc45)ncc3n2)CC1
O=C(Nc1cn2cc(-c3c(C(F)F)c(F)c(C(C4CC4)N4C(=O)c5ccccc5C4=O)c4[nH]ncc34)ncc2n1)[C@@H]1C[C@@H]1F
CC(O)c1c(F)c(C(F)F)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12
CC(c1c(F)c(C(F)F)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12)N1C(=O)c2ccccc2C1=O
N#C[C@H]1CC1C(=O)Nc1cn2cc(-c3c(Cl)c(F)c(NC(C)C)c4[nH]ncc34)ncc2n1
CC(C)Nc1c(F)c(Cl)c(-c2cn3cc(NC(=O)C4(F)CC4)nc3cn2)c2cn[nH]c12
CC(=O)NC(C)c1c(F)c(C(F)F)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12
CC(=O)NC(c1c(F)c(C(F)F)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12)C1CC1
CC(N)c1c(F)c(C(F)F)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12
CC(=O)NC(c4c(F)c(C(F)(F)F)c(c3cn2cc(NC(=O)[C@@H]1C[C@@H]1F)nc2cn3)c5cn[nH]c45)C6CC6
CC(C)Nc1c(F)c(Cl)c(-c2cn3cc(NC(=O)c4ccccc4)nc3cn2)c2cn[nH]c12
CC(C)Nc1c(F)c(Cl)c(-c2cn3cc(NC(=O)c4ccccn4)nc3cn2)c2cn[nH]c12
COC(=O)c1c(F)c(NC(C)C)c2[nH]ncc2c1-c1cn2cc(NC(=O)[C@@H]3C[C@@H]3F)nc2cn1
CC(C)Nc1c(F)c(Cl)c(-c2cn3cc(NC(=O)C4CCC4)nc3cn2)c2cn[nH]c12
CCC(=O)Nc1cn2cc(-c3c(Cl)c(F)c(NC(C)C)c4[nH]ncc34)ncc2n1
CC(C)Nc3c(F)c(Cl)c(c2cn1cc(NC(=O)C(F)(F)F)nc1cn2)c4cn[nH]c34
Cc1c(F)c(C(NC(=O)C2CC2)C2CC2)c2[nH]ncc2c1-c1cn2cc(NC(=O)[C@@H]3C[C@@H]3F)nc2cn1
Cc1c(F)c(C(C)N2C(=O)c3ccccc3C2=O)c2[nH]ncc2c1-c1cn2cc(NC(=O)[C@@H]3C[C@@H]3F)nc2cn1
Cc1c(F)c(C(C)NC(=O)C2CC2)c2[nH]ncc2c1-c1cn2cc(NC(=O)[C@@H]3C[C@@H]3F)nc2cn1
CC(=O)NC(C)c1c(F)c(C)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12
Cc1c(F)c(C(C)NC(=O)C(F)(F)F)c2[nH]ncc2c1-c1cn2cc(NC(=O)[C@@H]3C[C@@H]3F)nc2cn1
N#Cc1c(F)cc2[nH]ncc2c1-c1cn2cc(NC(=O)[C@@H]3C[C@@H]3F)nc2cn1
CC(C)Nc1c(F)c(C(=O)O)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12
CC(C)Nc1c(F)c(Cl)c(-c2cn3cc(NC(=O)C4CCNC4)nc3cn2)c2cn[nH]c12
CC(NC=O)c1c(F)c(C(F)F)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12
CC(NC(=O)C1CC1)c1c(F)c(C(F)F)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12
O=C(NC(c1c(F)c(C(F)F)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12)C1CC1)C1CC1
CC(C)Nc1c(F)c(Cl)c(-c2cn3cc(NC(=O)C4(N)CC4)nc3cn2)c2cn[nH]c12
CC(C)Nc1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@H](C)N)nc3cn2)c2cn[nH]c12
CC(C)Nc1c(F)c(Cl)c(-c2cn3cc(NC(=O)CN)nc3cn2)c2cn[nH]c12
CC(C)Nc1c(F)c(Cl)c(-c2cn3cc(NC(=O)C(C)C)nc3cn2)c2cn[nH]c12
CC(C)Nc1c(F)c(Cl)c(-c2cn3cc(NC(=O)C(C)(C)C)nc3cn2)c2cn[nH]c12
CC(=O)Nc1cn2cc(-c3c(C(F)(F)F)c(F)c(NC(C)C)c4[nH]ncc34)ncc2n1
CC(C)Nc1c(F)c(Cl)c(-c2cn3cc(NC(=O)N4CCOCC4)nc3cn2)c2cn[nH]c12
CC(CO)c1c(F)c(C(F)(F)F)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12
CC(NS(=O)C(C)(C)C)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12
CC(NS(=O)C(C)(C)C)c1c(F)c(C(F)(F)F)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12
CC(C)Nc1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4C(F)F)nc3cn2)c2cn[nH]c12
CC(C)Nc1c(F)c(Cl)c(-c2cn3cc(NC(=O)Cc4cccnc4)nc3cn2)c2cn[nH]c12
CC(C)Nc1c(F)c(Cl)c(-c2cn3cc(NC(=O)CN4CCOCC4)nc3cn2)c2cn[nH]c12
CC(C)Nc1c(F)c(Cl)c(-c2cn3cc(N4CCOCC4)nc3cn2)c2cn[nH]c12
CC(C)Nc1c(F)c(Cl)c(-c2cn3cc(NC(=O)N4CCN(C)CC4)nc3cn2)c2cn[nH]c12
Cc1c(F)c(NC(C)C)c2[nH]ncc2c1-c1cn2cc(NC(=O)Cc3cccnc3)nc2cn1
CC(C)Nc1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4CF)nc3cn2)c2cn[nH]c12
CC(C)Nc1c(F)c(Cl)c(-c2cn3cc(NC(=O)OC(C)C)nc3cn2)c2cn[nH]c12
CC(NC=O)c1c(F)c(C(F)(F)F)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12
CC(C)(C)S(=O)NC(c1c(F)c(C(F)(F)F)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12)C1CC1
CC(CN)c1c(F)c(C(F)(F)F)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12
CC(=O)NCC(C)c1c(F)c(C(F)(F)F)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12
CSCC(=O)Nc4cn3cc(c1c(Cl)c(F)c(NC(C)C)c2[nH]ncc12)ncc3n4
CC(C)Nc1c(F)c(Cl)c(-c2cn3cc(NC4CCOC4)nc3cn2)c2cn[nH]c12
CC(=O)N(C)c1cn2cc(-c3c(Cl)c(F)c(NC(C)C)c4[nH]ncc34)ncc2n1
CC(C)Nc1c(F)c(Cl)c(-c2cn3cc(NC(=O)CN(C)C)nc3cn2)c2cn[nH]c12
CC(C)Nc1c(F)c(C(F)(F)F)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4CO)nc3cn2)c2cn[nH]c12
CSC(C)C(=O)Nc4cn3cc(c1c(Cl)c(F)c(NC(C)C)c2[nH]ncc12)ncc3n4
CC(C)Nc1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H](C)N(C)C)nc3cn2)c2cn[nH]c12
Cc1c(F)c(C(NC(=O)C(F)(F)F)C2CC2)c2[nH]ncc2c1-c1cn2cc(NC(=O)[C@@H]3C[C@@H]3F)nc2cn1
CC(C)Nc1c(F)c(Cl)c(-c2cn3cc(NC(=O)C4CCN4)nc3cn2)c2cn[nH]c12
COCC(=O)Nc1cn2cc(-c3c(Cl)c(F)c(NC(C)C)c4[nH]ncc34)ncc2n1
CCCC(=O)Nc1cn2cc(-c3c(Cl)c(F)c(NC(C)C)c4[nH]ncc34)ncc2n1
CC(C)Nc1c(F)c(Cl)c(-c2cn3cc(NC(=O)C4CCCO4)nc3cn2)c2cn[nH]c12
CC(C)Nc1c(F)c(Cl)c(-c2cn3cc(NC=O)nc3cn2)c2cn[nH]c12
COC(=O)Nc1cn2cc(-c3c(Cl)c(F)c(NC(C)C)c4[nH]ncc34)ncc2n1
CCOC(=O)Nc1cn2cc(-c3c(Cl)c(F)c(NC(C)C)c4[nH]ncc34)ncc2n1
O=CNC(c1c(F)c(C(F)(F)F)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12)C1CC1
CC(C)Nc1c(F)c(Cl)c(-c2cn3cc(NC(=O)CC4COC4)nc3cn2)c2cn[nH]c12
CCCCC(=O)Nc1cn2cc(-c3c(Cl)c(F)c(NC(C)C)c4[nH]ncc34)ncc2n1
O=C(Nc1cn2cc(-c3c(C(F)(F)F)c(F)c(C(O)C4CC4)c4[nH]ncc34)ncc2n1)[C@@H]1C[C@@H]1CO
CCNC(=O)Nc1cn2cc(-c3c(Cl)c(F)c(NC(C)C)c4[nH]ncc34)ncc2n1
CC(C)Nc1c(F)c(Cl)c(-c2cn3cc(NC(=O)N4CCNCC4)nc3cn2)c2cn[nH]c12
CNC(=O)Nc1cn2cc(-c3c(Cl)c(F)c(NC(C)C)c4[nH]ncc34)ncc2n1
CC(C)Nc1c(F)c(Cl)c(-c2cn3cc(NC(=O)C(F)F)nc3cn2)c2cn[nH]c12
CC(C)Nc1c(F)c(Cl)c(-c2cn3cc(NC(=O)C4CCN(C)CC4)nc3cn2)c2cn[nH]c12
CC(C)Nc1c(F)c(Cl)c(-c2cn3cc(NC(=O)N4CCCC4)nc3cn2)c2cn[nH]c12
CC(C)Nc1c(F)c(Cl)c(-c2cn3cc(NC(=O)C4CCOC4)nc3cn2)c2cn[nH]c12
CC(C)Nc1c(F)c(Cl)c(-c2cn3cc(NC(=O)OC4CCC4)nc3cn2)c2cn[nH]c12
COc1c(F)c(C(O)C2CC2)c2[nH]ncc2c1-c1cn2cc(NC(=O)[C@@H]3C[C@@H]3F)nc2cn1
COc1c(F)c(C(C)O)c2[nH]ncc2c1-c1cn2cc(NC(=O)[C@@H]3C[C@@H]3F)nc2cn1
CC(C)Nc1c(F)c(Cl)c(-c2cn3cc(NC(=O)CO)nc3cn2)c2cn[nH]c12
CC(C)Nc1c(F)c(Cl)c(-c2cn3cc(NC(=O)CCO)nc3cn2)c2cn[nH]c12
CC(C)Nc1c(F)c(Cl)c(-c2cn3cc(NC(=O)C4COC4)nc3cn2)c2cn[nH]c12
C[C@H](N[S@@](=O)C(C)(C)C)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12
C[C@@H](N[S@](=O)C(C)(C)C)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12
CC(=O)Nc1cn2cc(-c3c(Cl)c(F)c([C@H](C)N[S@@](=O)C(C)(C)C)c4[nH]ncc34)ncc2n1
CC(=O)Nc1cn2cc(-c3c(Cl)c(F)c([C@@H](C)N[S@](=O)C(C)(C)C)c4[nH]ncc34)ncc2n1
COc1c(F)c(N(C)C)c2[nH]ncc2c1-c1cn2cc(NC(=O)[C@@H]3C[C@@H]3F)nc2cn1
C[C@@H](NC(=O)C(F)(F)F)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12
CC(=O)Nc1cn2cc(-c3c(Cl)c(F)c([C@H](C)NC(=O)C(F)(F)F)c4[nH]ncc34)ncc2n1
CC(=O)Nc1cn2cc(-c3c(Cl)c(F)c([C@@H](C)NC(=O)C(F)(F)F)c4[nH]ncc34)ncc2n1
CC(=O)Nc1cn2cc(-c3c(Cl)c(F)c([C@H](C)NC=O)c4[nH]ncc34)ncc2n1
COc1c(F)c(NC(C)C)c2[nH]ncc2c1-c1cn2cc(NC(=O)[C@@H]3C[C@@H]3F)nc2cn1
CC(=O)N1CC(Oc2c(F)c(Cl)c(-c3cn4cc(NC(=O)[C@@H]5C[C@@H]5F)nc4cn3)c3cn[nH]c23)C1
O=C(Nc1cn2cc(-c3c(Cl)c(F)c(OC4CNC4)c4[nH]ncc34)ncc2n1)[C@@H]1C[C@@H]1F
CC(C)Nc1c(F)c(Cl)c(-c2cn3cc(NC(=O)Cc4cocn4)nc3cn2)c2cn[nH]c12
CC(=O)Nc1cn2cc(-c3c(Cl)c(F)c(OC4CN(C(C)=O)C4)c4[nH]ncc34)ncc2n1
C[C@H](NC(=O)C(F)(F)F)c1c(F)c(Cl)c(-c2cn3cc(NC(=O)[C@@H]4C[C@@H]4F)nc3cn2)c2cn[nH]c12
CC(=O)Nc1cn2cc(-c3c(Cl)c(F)c(OC4CNC4)c4[nH]ncc34)ncc2n1
CC(=O)Nc1cn2cc(-c3c(Cl)c(F)c(OC4CN(C(=O)CO)C4)c4[nH]ncc34)ncc2n1
CCC(=O)N1CC(Oc2c(F)c(Cl)c(-c3cn4cc(NC(C)=O)nc4cn3)c3cn[nH]c23)C1
CC(=O)Nc1cn2cc(-c3c(Cl)c(F)c(CN4CC(O)C4)c4[nH]ncc34)ncc2n1
CC(=O)Nc1cn2cc(-c3c(Cl)c(F)c(CN4CCC(O)C4)c4[nH]ncc34)ncc2n1
CC(=O)Nc1cn2cc(-c3c(Cl)c(F)c(C(O)C4CC4)c4[nH]ncc34)ncc2n1
CC(=O)Nc1cn2cc(-c3c(C(F)F)c(F)c(NC(C)C)c4[nH]ncc34)ncc2n1
N#C[C@H]1C[C@H]1C(=O)Nc1cn2cc(-c3c(C(F)F)c(F)c(NC(C)C)c4[nH]ncc34)ncc2n1
CCC(=O)Nc1cn2cc(-c3c(C(F)F)c(F)c(NC(C)C)c4[nH]ncc34)ncc2n1
CC(C)Nc1c(F)c(C(F)F)c(-c2cn3cc(NC(=O)C4CC4)nc3cn2)c2cn[nH]c12
CC(=O)Nc1cn2cc(-c3c(Cl)c(F)c(CN4CC(C)(O)C4)c4[nH]ncc34)ncc2n1
COc1c(F)c(NC(C)C)c2[nH]ncc2c1-c1cn2cc(NC(C)=O)nc2cn1
CC(=O)Nc1cn2cc(-c3c(Cl)c(F)c(CN4CCC(C)(O)C4)c4[nH]ncc34)ncc2n1
COc1c(F)c(NC(C)C)c2[nH]ncc2c1-c1cn2cc(NC(=O)C3CC3)nc2cn1
CC(=O)Nc1cn2cc(-c3c(Cl)c(F)c(C(C)N4CC(O)C4)c4[nH]ncc34)ncc2n1
CCC(=O)Nc1cn2cc(-c3c(OC)c(F)c(NC(C)C)c4[nH]ncc34)ncc2n1
CC(=O)Nc1cn2cc(-c3c(Cl)c(F)c(C(C)N4CCC(O)C4)c4[nH]ncc34)ncc2n1
COc1c(F)c(NC(C)C)c2[nH]ncc2c1-c1cn2cc(NC(=O)[C@@H]3C[C@@H]3C#N)nc2cn1
C[C@@]12[C@](C[C@@H](O1)n3c4ccccc4c5c3c6n2c7ccccc7c6c8c5C(=O)NC8)(CO)O
C[C@@]12[C@@H]([C@@H](C[C@@H](O1)n3c4ccccc4c5c3c6n2c7ccccc7c6c8c5C(=O)NC8)N(C)C(=O)c9ccccc9)OC
CN1CCN(CC1)CC(=O)N(C)c2ccc(cc2)N/C(=C\3/c4ccc(cc4NC3=O)C(=O)OC)/c5ccccc5
C[C@@]12[C@@H]([C@@H](C[C@@H](O1)n3c4ccccc4c5c3c6n2c7ccccc7c6c8c5C(=O)NC8)NC)OC
Cn1c2nc(Nc3ccc4[nH]ccc4c3)ncc2cc(c1=O)S(=O)(=O)c1ccc(F)cc1F
CC(C)(C)c1cc(NC(=O)Nc2ccc(cc2)-c2cn3c(n2)sc2cc(OCCN4CCOCC4)ccc32)no1
CO[C@@H]1[C@@H](C[C@H]2O[C@]1(C)n1c3ccccc3c3c4[C@H](O)NC(=O)c4c4c5ccccc5n2c4c13)N(C)C(=O)c1ccccc1 |r|
COc1cc2c(ncnc2cc1OCCCN1CCCCC1)N1CCN(CC1)C(=O)Nc1ccc(OC(C)C)cc1
CNC(=O)c1cc(ccn1)Oc2ccc(cc2)NC(=O)Nc3ccc(c(c3)C(F)(F)F)Cl
Cc1cnc2c(NCCN)nc3ccc(C)cc3n12
CC(C)S(=O)(=O)c1ccccc1Nc2c(cnc(n2)Nc3ccc(cc3OC)N4CCC(CC4)N5CCN(CC5)C)Cl
CN1CCN(CC1)CCCOc2cc3c(cc2OC)c(c(cn3)C#N)Nc4cc(c(cc4Cl)Cl)OC
COc1cc(Oc2ccnc3cc(OC)c(OC)cc23)ccc1NC(=O)NC(C)c1nccs1
COc1ccc(cc1)COc2ccc(cc2OC)Cc3cnc(nc3N)N
Cc1ccc(cc1)-n1nc(cc1NC(=O)Nc1ccc(OCCN2CCOCC2)c2ccccc12)C(C)(C)C
CC(C)n1nc(-c2cc3cc(O)ccc3[nH]2)c2c(N)ncnc12
Cn1c(Nc2ccc(cc2)C(F)(F)F)nc2cc(Oc3ccnc(c3)-c3ncc([nH]3)C(F)(F)F)ccc12
Cc1n[nH]c2ccc(cc12)-c1cncc(OC[C@@H](N)Cc2ccccc2)c1 |r|
COc1ccc(c(c1C(=O)c2cnc(nc2N)NC3CCN(CC3)S(=O)(=O)C)F)F
Cn1cnc2c1cc(c(c2F)Nc3ccc(cc3Cl)Br)C(=O)NOCCO
Cc1cn(cn1)-c1cc(NC(=O)c2ccc(C)c(Nc3nccc(n3)-c3cccnc3)c2)cc(c1)C(F)(F)F
Oc1cccc(c1)-c1nc(N2CCOCC2)c2oc3ncccc3c2n1
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(Cl)cc23)c1F
COc1cc2c(Oc3ccc4[nH]c(C)cc4c3F)ncnc2cc1OCCCN1CCCC1
COc1cc2c(cc1OCCCN3CCOCC3)c(ncn2)Nc4ccc(c(c4)Cl)F
OCCn1cc(c(n1)-c1ccncc1)-c1ccc2C(CCc2c1)N=O
CN(C)C/C=C/C(=O)Nc1cc2c(cc1O[C@H]3CCOC3)ncnc2Nc4ccc(c(c4)Cl)F
C=CC(=O)Nc1cc2c(cc1OCCCN3CCOCC3)ncnc2Nc4ccc(c(c4)Cl)F
CS(=O)(=O)N1CCN(Cc2cc3nc(nc(N4CCOCC4)c3s2)-c2cccc3[nH]ncc23)CC1
Cn1cc(cn1)-c1ccc2nnc(Sc3ccc4ncccc4c3)n2n1
c1c[nH]c2c1c(ncn2)c3cnn(c3)[C@H](CC#N)C4CCCC4
Cc1[nH]c(\C=C2/C(=O)Nc3ccc(cc23)S(=O)(=O)Cc2c(Cl)cccc2Cl)c(C)c1C(=O)N1CCC[C@@H]1CN1CCCC1 |r|
Cn1cc(C2=C(C(=O)NC2=O)c2cn(C3CCN(Cc4ccccn4)CC3)c3ccccc23)c2ccccc12 |t:4|
C[C@@H](Oc1cc(sc1C(N)=O)-n1cnc2ccc(CN3CCN(C)CC3)cc12)c1ccccc1C(F)(F)F |r|
CC1(CNc2c1ccc(c2)NC(=O)c3cccnc3NCc4ccncc4)C
OC(=O)c1ccc(Nc2ncc3CN=C(c4cc(Cl)ccc4-c3n2)c2c(F)cccc2F)cc1 |c:13|
COc1c(Cl)cc2c3ccncc3[nH]c2c1NC(=O)c1cccnc1C
CC(C)(C)c1cnc(o1)CSc2cnc(s2)NC(=O)C3CCNCC3
CCOc1cc2ncc(C#N)c(Nc3ccc(OCc4ccccn4)c(Cl)c3)c2cc1NC(=O)\C=C\CN(C)C
CN1c2c(cnc(n2)Nc3cccc(c3)SC)C=C(C1=O)c4c(cccc4Cl)Cl
Nc1nc(N)c2nc(-c3cccc(O)c3)c(nc2n1)-c1cccc(O)c1
COCCOc1cc2c(cc1OCCOC)ncnc2Nc3cccc(c3)C#C
Cc1cnc(nc1Nc2cccc(c2)S(=O)(=O)NC(C)(C)C)Nc3ccc(cc3)OCCN4CCCC4
CN(C)CC(=O)N1CCC(CC1)c1ccc(NC(=O)c2ncc([nH]2)C#N)c(c1)C1=CCCCC1 |t:31|
C[C@@H](O)COc1cn2ncnc(Oc3ccc4[nH]c(C)cc4c3F)c2c1C
CS(=O)c1ccc(cc1)-c1nc(c([nH]1)-c1ccc(F)cc1)-c1ccncc1
O=C(N1CCNCC1)c1ccc(\C=C\c2n[nH]c3ccccc23)cc1
CCn1c(nc2c(ncc(OC[C@H]3CCCNC3)c12)C#CC(C)(C)O)-c1nonc1N |r|
c1cc(c(c(c1)Cl)C2=C3C=CC(=NN3C=NC2=O)Sc4ccc(cc4F)F)Cl
CC1(C(=O)Nc2c(ccc(n2)Nc3c(cnc(n3)Nc4cc(c(c(c4)OC)OC)OC)F)O1)C
CNC(=O)c1c(F)cccc1Nc1nc(Nc2cc3N(CCc3cc2OC)C(=O)CN(C)C)nc2[nH]ccc12
CN1CCN(Cc2ccc(cc2)C(=O)Nc2ccc(C)c(Nc3nccc(n3)-c3cccnc3)c2)CC1
Clc1ccc(Nc2nnc(Cc3ccncc3)c3ccccc23)cc1
CN1CCC(CC1)COc2cc3c(cc2OC)c(ncn3)Nc4ccc(cc4F)Br
C[C@@H]1CCN(C[C@@H]1N(C)c1ncnc2[nH]ccc12)C(=O)CC#N |r|
CS(=O)(=O)CCNCc1ccc(o1)-c1ccc2ncnc(Nc3ccc(OCc4cccc(F)c4)c(Cl)c3)c2c1
CN1CC[C@@H]([C@H](O)C1)c1c(O)cc(O)c2c1oc(cc2=O)-c1ccccc1Cl |r|
Clc1cccc(Cl)c1C(=O)Nc1cn[nH]c1C(=O)NC1CCNCC1
CC[C@H]1N(C2CCCC2)c2nc(Nc3ccc(cc3OC)C(=O)NC3CCN(C)CC3)ncc2N(C)C1=O |r|
COc1cc2c(Oc3ccc(NC(=O)C4(CC4)C(=O)NC4=CCC(F)C=C4)cc3F)ccnc2cc1OCCCN1CCOCC1 |c:26,t:21|
CNC(=O)c1ccccc1Sc2ccc3c(c2)[nH]nc3/C=C/c4ccccn4
CCN(CCCOc1ccc2c(c1)ncnc2Nc3cc(n[nH]3)CC(=O)Nc4cccc(c4)F)CCO
Cc1ccc(cc1Nc2nc(cs2)c3cccnc3)NC(=O)c4ccc(cc4)CN5CCN(CC5)C
C[C@@H](Oc1cc(cnc1N)-c1cnn(c1)C1CCNCC1)c1c(Cl)ccc(F)c1Cl |r|
Fc1ccc(C(=O)NOCC2CC2)c(Nc2ccc(I)cc2Cl)c1F
COCC(=O)NC\C=C\c1ccc2ncnc(Nc3ccc(Oc4ccc(C)nc4)c(C)c3)c2c1
CC[C@H](CO)Nc1nc(NCc2ccccc2)c2ncn(C(C)C)c2n1 |r|
Oc1ccc(cc1)-c1nc(c([nH]1)-c1ccc(F)cc1)-c1ccncc1
NC(=O)c1ccc(cc1)-c1nc(c([nH]1)-c1ccc2OCOc2c1)-c1ccccn1
CC(C)(C)NS(=O)(=O)c1cncc(c1)-c1ccn2nc(N)nc2c1
COc1cc(OC)c(F)c(c1F)-c1ncc2c(n[nH]c2n1)-c1ccc(cc1)N1CCN(C)CC1
CN1CCN(CC1)c1ccc(cc1)-c1n[nH]c2cc(cnc12)-c1ccccc1
CN1CCN(CC1)c1ccc(Nc2ncc3ccc(cc3n2)-c2ccccc2)cc1
COc1cccc(F)c1-c1cc2c(n[nH]c2cn1)-c1cnn(C)c1
CNCc1cc(F)c(c(OC)c1)-c1cc2c(n[nH]c2cn1)-c1cnn(C)c1
NC1CCCN(C1)c1ccccc1NC(=O)c1cccc(c1)-c1ccccc1F
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccccc1N1CCC[C@@H](N)C1 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)ccc1N1CC[C@@H](N)C1 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2n(C)ncc2c1N1CC[C@@H](N)C1 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc2cnn(C)c2cc1N1CC[C@@H](N)C1 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2n(C)cnc2c1N1CC[C@@H](N)C1 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc2sc(C)nc2c1N1CC[C@@H](N)C1 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c2n(C)ncc2c1N1CCC(N)CC1
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c2n(C)ncc2c1N1CCNCC1
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c2n(C)ncc2c1N1CCNC[C@H]1C |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c2n(C)ncc2c1N1C[C@@H](N)C[C@H]1C |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c2n(C)ncc2c1N1CCC[C@H]1CO |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c2n(C)ncc2c1N1C[C@H](N)C[C@H]1CO |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c2n(C)ncc2c1N1CC[C@@H](O)[C@@H]1CN |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1cc(F)c2n(C)ncc2c1N1CC[C@H](N)[C@@H]1CO |r|
[H][C@@]12CN(c3ccccc3NC(=O)c3ccnc(n3)-c3c(F)cccc3OC)[C@@]([H])(CN1)C2 |r|
[H][C@]12CN(c3cc(c(F)cc3NC(=O)c3ccnc(n3)-c3c(F)cccc3OC)-c3cccnc3)[C@]([H])(CN1)C2 |r|
COc1cccc(F)c1-c1nccc(n1)C(=O)Nc1ccc(cc1N1C[C@@H](N)C[C@H]1CO)-c1c(C)nn(C)c1C#N |r|
CN1CCN(CC1)c1ccc2nc([nH]c2c1)-c1c(N)c2sccc2[nH]c1=O
CN1CCN(CC1)c1ccc2nc([nH]c2c1)-c1c(N)c2ccsc2[nH]c1=O
[H][C@]12C[C@H]([C@@H](OC)[C@](C)(O1)n1c3ccccc3c3c4CNC(=O)c4c4c5ccccc5n2c4c13)N(C)CCOCCOCCOCCNC(=O)CCC1=[N+]2C(C=C1)=Cc1c(C)cc(C)n1[B-]2(F)F |r,c:63,65,t:60|
[H][C@]12C[C@@H](NCCOCCOCCOCCNC(=O)CCC3=[N+]4C(C=C3)=Cc3c(C)cc(C)n3[B-]4(F)F)[C@@H](OC)[C@](C)(O1)n1c3ccccc3c3c4CNC(=O)c4c4c5ccccc5n2c4c13 |r,c:24,26,t:21|
[H]/N=C(/N)\SCCCn1cc(c2c1cccc2)C3=C(C(=O)NC3=O)c4cn(c5c4cccc5)C
CN(C)c1ccc(cc1)C(=O)Nc1cccc(NC(=O)COc2ccc3c(c2)occc3=O)c1
CCN1CCC(CC1)c1ncc(s1)-c1cnc(N)c(OCc2ccncc2)c1
CNC(=O)c1cnc(Nc2ccc3ncsc3c2)cc1N[C@H](CO)c1ccccc1 |r|
CCc1cc(Nc2ncc(C(=O)NC)c(N[C@H](CO)c3ccccc3)n2)ccc1C#N |r|
CNC(=O)c1cnc(Nc2ccc3C(=O)OC(C)(C)c3c2)nc1N[C@H](CO)c1ccccc1 |r|
CCNC(=O)c1cnc(Nc2ccc3C(=O)OC(C)(C)c3c2)nc1N[C@H](CO)c1ccccc1 |r|
CC(C)NC(=O)c1cnc(Nc2ccc3C(=O)OC(C)(C)c3c2)nc1N[C@H](CO)c1ccccc1 |r|
CCCNC(=O)c1cnc(Nc2ccc3C(=O)OC(C)(C)c3c2)nc1N[C@H](CO)c1ccccc1 |r|
CCCN(C)C(=O)c1cnc(Nc2ccc3C(=O)OC(C)(C)c3c2)nc1N[C@H](CO)c1ccccc1 |r|
CC1(C)OC(=O)c2ccc(Nc3ncc(C(N)=O)c(N[C@H](CO)c4ccccc4)n3)cc12 |r|
CC1(C)OC(=O)c2ccc(Nc3ncc(C(O)=O)c(N[C@H](CO)c4ccccc4)n3)cc12 |r|
CCOC(=O)c1cnc(Nc2ccc3C(=O)OC(C)(C)c3c2)nc1N[C@H](CO)c1ccccc1 |r|
Cc1noc(n1)-c1cnc(Nc2ccc3C(=O)OC(C)(C)c3c2)nc1N[C@H](CO)c1ccccc1 |r|
CCc1noc(n1)-c1cnc(Nc2ccc3C(=O)OC(C)(C)c3c2)nc1N[C@H](CO)c1ccccc1 |r|
CC(C)c1noc(n1)-c1cnc(Nc2ccc3C(=O)OC(C)(C)c3c2)nc1N[C@H](CO)c1ccccc1 |r|
CC(C)(C)c1noc(n1)-c1cnc(Nc2ccc3C(=O)OC(C)(C)c3c2)nc1N[C@H](CO)c1ccccc1 |r|
CC1(C)OC(=O)c2ccc(Nc3ncc(-c4nc(no4)C4CC4)c(N[C@H](CO)c4ccccc4)n3)cc12 |r|
CC1(C)OC(=O)c2ccc(Nc3ncc(-c4nc(no4)-c4ccc(F)cc4)c(N[C@H](CO)c4ccccc4)n3)cc12 |r|
CC1(C)OC(=O)c2ccc(Nc3ncc(-c4nc(no4)-c4ccncc4)c(N[C@H](CO)c4ccccc4)n3)cc12 |r|
CN1CCC(CC1)c1noc(n1)-c1cnc(Nc2ccc3C(=O)OC(C)(C)c3c2)nc1N[C@H](CO)c1ccccc1 |r|
CC1(C)OC(=O)c2ccc(Nc3ncc(-c4nc(no4)C45CCN(CC4)CC5)c(N[C@H](CO)c4ccccc4)n3)cc12 |r|
Cc1nnc(o1)-c1cnc(Nc2ccc3C(=O)OC(C)(C)c3c2)nc1N[C@H](CO)c1ccccc1 |r|
CC1(C)OC(=O)c2ccc(Nc3ncc(-c4nnc(o4)C4CC4)c(N[C@H](CO)c4ccccc4)n3)cc12 |r|
CN1CCC(CC1)c1nnc(o1)-c1cnc(Nc2ccc3C(=O)OC(C)(C)c3c2)nc1N[C@H](CO)c1ccccc1 |r|
CC1(C)OC(=O)c2ccc(Nc3ncc(-c4nnc(o4)C45CCN(CC4)CC5)c(N[C@H](CO)c4ccccc4)n3)cc12 |r|
CC1(C)OC(=O)c2ccc(Nc3ncc(-c4nnco4)c(N[C@H](CO)c4ccccc4)n3)cc12 |r|
CN1CCN(CC1)c1ccc(cc1)-n1ncc2cc(C#N)c(cc12)-c1c(C)cccc1F |(16.04,-4.16,;15.57,-5.62,;16.6,-6.77,;16.13,-8.23,;14.62,-8.55,;13.59,-7.42,;14.06,-5.95,;14.15,-10.01,;15.19,-11.15,;14.72,-12.62,;13.22,-12.94,;12.18,-11.81,;12.64,-10.35,;12.75,-14.41,;13.66,-15.65,;12.76,-16.9,;11.29,-16.43,;9.95,-17.21,;8.62,-16.44,;7.28,-17.21,;5.95,-17.98,;8.62,-14.9,;9.95,-14.13,;11.28,-14.89,;7.29,-14.13,;7.29,-12.59,;8.63,-11.82,;5.96,-11.82,;4.63,-12.59,;4.63,-14.14,;5.96,-14.9,;5.97,-16.44,)|
COc1cccc(F)c1-c1cc2n(ncc2cc1C#N)-c1cccc(n1)N1CCN(C)CC1 |(19.09,-7.98,;19.08,-9.52,;17.75,-10.28,;16.42,-9.51,;15.08,-10.28,;15.08,-11.84,;16.42,-12.59,;16.43,-14.13,;17.74,-11.82,;19.07,-12.59,;20.4,-11.82,;21.74,-12.59,;23.2,-12.1,;24.11,-13.34,;23.22,-14.6,;21.75,-14.13,;20.41,-14.91,;19.07,-14.14,;17.74,-14.91,;16.41,-15.67,;23.67,-10.64,;22.63,-9.51,;23.1,-8.05,;24.61,-7.71,;25.64,-8.85,;25.18,-10.32,;27.15,-8.52,;28.18,-9.67,;29.68,-9.35,;30.15,-7.89,;31.66,-7.56,;29.12,-6.74,;27.61,-7.07,)|
COc1cccc(F)c1-c1cc2n(ncc2cn1)-c1cccc(n1)N1CC2CCC(C1)N2C
COc1cccc(F)c1-c1cc2n(ncc2cn1)-c1cccc(n1)N1CC[C@@H](C1)N(C)C |r|
[H][C@]12CN(c3cccc(n3)-n3ncc4cnc(cc34)-c3c(F)cccc3OC)[C@]([H])(CN1C)C2 |r|
COc1cccc(F)c1-c1cc2n(ncc2cn1)-c1cccc(n1)N1CCN(C)CC1
CN1CCN(CC1)c1ccc(cc1)-n1ncc2ccc(cc12)-c1c(C)cccc1F
CNC(=O)N1CCN(CC1)c1cccc(n1)-n1ncc2cnc(cc12)-c1c(F)cccc1OC
COC(=O)N1CCN(CC1)c1cccc(n1)-n1ncc2cnc(cc12)-c1c(F)cccc1OC
CNC1CCN(CC1)c1cccc(n1)-n1ncc2cnc(cc12)-c1c(F)cccc1OC
COc1cccc(F)c1-c1cc2n(ncc2cn1)-c1cccc(n1)N1CCCCC1
COc1cccc(F)c1-c1cc2n(ncc2cn1)-c1cccc(n1)N1CCCC1=O
COc1cccc(F)c1-c1cc2n(ncc2cn1)-c1cccc(n1)N1CC2(C1)CCCNC2
COc1cccc(F)c1-c1cc2n(ncc2cn1)-c1cccc(n1)N1CCCC1
COc1cccc(F)c1-c1cc2n(ncc2cn1)-c1cccc(N)n1
COc1cccc(F)c1-c1cc2n(ncc2cn1)-c1cccc(n1)N1CCOCC1
COc1cccc(F)c1-c1cc2n(ncc2cn1)-c1cccc(n1)N1CC(N)C1
COc1cccc(n1)-n1ncc2cnc(cc12)-c1c(F)cccc1OC
COc1cccc(F)c1-c1cc2n(ncc2cn1)-c1cc(Cl)cc(n1)N1CCN(C)CC1
COc1cccc(F)c1-c1cc2n(ncc2cn1)-c1cccc(n1)N1CCNCC1
COc1cccc(F)c1-c1cc2n(ncc2cn1)-c1ccnc(n1)N1CCN(C)CC1
COc1cccc(F)c1-c1cc2n(ncc2cn1)-c1ccnc(c1)N1CCN(C)CC1
COc1cccc(F)c1-c1cc2n(ncc2cn1)-c1ccc(cn1)N1CCN(C)CC1
COc1cccc(F)c1-c1cc2n(ncc2cn1)-c1cccc(c1)N1CCN(C)CC1
COc1cccc(F)c1-c1cc2n(ncc2cn1)-c1ccc(cc1)N1CCOCC1
COc1cccc(F)c1-c1cc2n(ncc2cn1)-c1cnn(C)c1
COc1cccc(F)c1-c1cc2n(ncc2cn1)-c1ccccc1
CCOc1cccc(F)c1-c1cc2n(ncc2cn1)-c1ccc(cc1)N1CCN(C)CC1
COc1cccc(F)c1-c1cc2n(ncc2cn1)-c1ccc(cc1)N1CCN(C)CC1
CNC1CCc2c1ccc(F)c2-c1cc2n(ncc2cn1)-c1ccc(cc1)N1CCN(C)CC1
CN1CCN(CC1)c1ccc(cc1)-n1ncc2cnc(cc12)-c1c(C)cccc1F
CN1CCN(CC1)c1ccc(cc1)-n1ncc2cnc(cc12)-c1c(C)cccc1C
CN1CCN(CC1)c1ccc(cc1)-n1ncc2cnc(cc12)-c1ccccc1C
CN1CCN(CC1)c1ccc(cc1)-n1ncc2cnc(cc12)-c1ccccc1
COc1ccncc1-c1cc2n(ncc2cn1)-c1ccc(cc1)N1CCN(C)CC1
COc1ccncc1-c1ccc2cnn(-c3ccnc(c3)N3CCOCC3)c2c1
C[C@H]1CN(C[C@@H](C)N1C)c1cc(ccn1)-n1ncc2ccc(cc12)-c1cnn2CCCOc12 |r|
CN1CCN(CC1)c1cc(ccn1)-c1n[nH]c2cnc(cc12)-c1cnn2CCCc12
CN1CCN(CC1)c1cc(ccn1)-c1n[nH]c2ccc(cc12)-c1cnn2CCCc12
Cc1c2NCCOc2ncc1-c1cc2\C(=C\c3ccc([nH]3)C3CC3)C(=O)Nc2c(F)c1
COc1cc2CCN(C)Cc2cc1Nc1ncc(C(N)=O)c(NC2CCCC2)n1
CN1CCc2cc(c(cc2C1)Nc3ncc(c(n3)Nc4ccccc4Br)C(=O)N)OC
COc1cc2CCN(C)Cc2cc1Nc1ncc(C(N)=O)c(Nc2ccccc2F)n1
COc1cc2CCN(C)Cc2cc1Nc1ncc(C(N)=O)c(Nc2ccccc2Cl)n1
COc1cc2CCN(C)Cc2cc1Nc1ncc(C(N)=O)c(Nc2ccccc2C)n1
COc1cc2CCN(C)Cc2cc1Nc1ncc(C(N)=O)c(Nc2ccccc2C(F)(F)F)n1
COc1cc2CCN(C)Cc2cc1Nc1ncc(C(N)=O)c(Nc2ccccc2C(C)(C)C)n1
COc1cc2CCN(C)Cc2cc1Nc1ncc(C(N)=O)c(Nc2ccccc2C(C)(F)F)n1
COc1ccccc1Nc1nc(Nc2cc3CN(C)CCc3cc2OC)ncc1C(N)=O
COCc1ccccc1Nc1nc(Nc2cc3CN(C)CCc3cc2OC)ncc1C(N)=O
COC(C)c1ccccc1Nc1nc(Nc2cc3CN(C)CCc3cc2OC)ncc1C(N)=O
CO[C@@H](C)c1ccccc1Nc1nc(Nc2cc3CN(C)CCc3cc2OC)ncc1C(N)=O |r|
COc1cc2CCN(C)Cc2cc1Nc1ncc(C(N)=O)c(Nc2ccccc2N2CCOC2=O)n1
COc1cc2CCN(C)Cc2cc1Nc1ncc(C(N)=O)c(Nc2ccccc2S(N)(=O)=O)n1
COc1cc2CCN(C)Cc2cc1Nc1ncc(C(N)=O)c(Nc2ccccc2C2CCCOC2)n1
COc1cc2CCN(C)Cc2cc1Nc1ncc(C(N)=O)c(Nc2ccccc2C2CCCO2)n1
COc1cc2CCN(C)Cc2cc1Nc1ncc(C(N)=O)c(Nc2ccccc2CO)n1
COc1cc2CCN(C)Cc2cc1Nc1ncc(C(N)=O)c(Nc2ccccc2C(C)(C)O)n1
COc1cc2CCN(C)Cc2cc1Nc1ncc(C(N)=O)c(Nc2c(C)cccc2Br)n1
COc1cc2CCN(C)Cc2cc1Nc1ncc(C(N)=O)c(Nc2c(F)cccc2CO)n1
COc1cc2CCN(C)Cc2cc1Nc1nccc(Nc2ccccc2)n1
COc1cc2CCN(C)Cc2cc1Nc1ncc(C)c(Nc2ccccc2)n1
COc1cc2CCN(C)Cc2cc1Nc1ncc(c(Nc2ccccc2)n1)C(F)(F)F
CNCc1cc(OC)cc2C(=O)N(Cc12)c1cccc(n1)-c1nncn1[C@@H](C)C1CC1
COc1cc2C(=O)N(Cc2c(CN)c1)c1cccc(n1)-c1nncn1[C@@H](C)CC(F)(F)F
CC[C@H](C)n1cnnc1-c1cccc(n1)N1Cc2c(cc(cc2CNC)N(C)C)C1=O |r|
COc1cc2C(=O)N(Cc2c(c1)S(N)(=O)=O)c1cccc(n1)-c1nncn1C(C)C
CC[C@H](C)n1cnnc1-c1cccc(n1)N1Cc2c(cc(cc2CNC)N2CCCC2)C1=O |r|
CC[C@@H](CC(F)(F)F)n1cnnc1-c1cccc(n1)N1Cc2c(cc(OC)cc2CNC)C1=O |r|
CN(C)C(=O)c1c(N)ccc(c1F)-c1cnc2NC[C@@]3(CC[C@](C)(O)C3)c2c1Cl |r|
CN(C)C(=O)c1c(N)ccc(c1F)-c1cnc2NC[C@]3(CC[C@@](C)(O)CC3)c2c1Cl |r,wU:22.24,19.19,(57.58,-11.9,;58.92,-11.13,;58.92,-9.59,;60.26,-11.9,;60.26,-13.44,;61.6,-11.13,;62.94,-11.9,;62.94,-13.45,;64.28,-11.13,;64.27,-9.58,;62.93,-8.81,;61.6,-9.58,;60.27,-8.82,;62.92,-7.27,;61.59,-6.51,;61.58,-4.97,;62.92,-4.18,;63.24,-2.67,;64.77,-2.51,;65.39,-3.92,;66.47,-2.83,;67.95,-3.24,;68.35,-4.71,;69.44,-5.79,;69.83,-4.31,;67.26,-5.8,;65.79,-5.4,;64.25,-4.96,;64.26,-6.5,;65.6,-7.26,)|
CN(C)C(=O)c1c(N)ccc(c1F)-c1cnc2NC[C@@]3(CC[C@@](C)(C3)C#N)c2c1Cl |r|
CN(C)C(=O)c1c(N)ccc(c1F)-c1cnc2NC[C@]3(CC[C@](C)(CC3)C#N)c2c1Cl |r,wU:22.27,19.19,(3.18,-29.71,;4.52,-28.95,;4.52,-27.4,;5.86,-29.72,;5.86,-31.26,;7.2,-28.95,;8.54,-29.72,;8.54,-31.26,;9.89,-28.95,;9.88,-27.39,;8.54,-26.62,;7.2,-27.4,;5.87,-26.63,;8.53,-25.08,;7.19,-24.32,;7.18,-22.78,;8.52,-21.99,;8.84,-20.48,;10.38,-20.32,;11,-21.73,;12.08,-20.64,;13.56,-21.05,;13.96,-22.52,;15.05,-23.6,;12.87,-23.61,;11.39,-23.21,;15.44,-22.12,;16.92,-21.71,;9.86,-22.77,;9.87,-24.31,;11.2,-25.08,)|
CN(C)C(=O)c1c(N)ccc(c1F)-c1cnc2NC[C@@]3(CC[C@@H](C3)C(N)=O)c2c1Cl |r|
CNC(=O)[C@H]1CC[C@@]2(CNc3ncc(c(Cl)c23)-c2ccc(N)c(C(=O)N(C)C)c2F)C1 |r|
CN(C)C(=O)c1c(N)ccc(c1F)-c1cnc2NC[C@@]3(CC[C@@](C)(C3)C(N)=O)c2c1Cl |r|
CN(C)C(=O)c1c(N)ccc(c1F)-c1cnc2NC[C@]3(CC[C@](C)(C3)C(N)=O)c2c1Cl |r|
CN(C)C(=O)c1c(N)ccc(c1F)-c1cnc2NC[C@@]3(CC[C@@H](C3)c3ncn[nH]3)c2c1Cl |r|
CN(C)C(=O)c1c(N)ccc(c1F)-c1cnc2NC[C@@]3(CC[C@]4(C3)CCCNC4=O)c2c1Cl |r|
CN(C)C(=O)c1c(N)ccc(c1F)-c1cnc2NC[C@@]3(CC[C@]4(C3)CCCCNC4=O)c2c1Cl |r|
COc1ccccc1-c1c[nH]c2ncc(cc12)-c1ccc(N)c(c1)C(=O)N(C)C
CCc1c[nH]c2ncc(cc12)-c1ccc(N)c(c1)C(=O)N(C)C
CN(C)C(=O)c1cc(ccc1N)-c1cnc2[nH]ccc2c1
CCc1c[nH]c2ncc(-c3ccc(N)c(c3)C(=O)N(C)C)c(C)c12
CCc1c[nH]c2ncc(-c3ccc(N)c(c3)C(=O)N(C)C)c(CC)c12
CCc1c[nH]c2ncc(-c3ccc(N)c(c3)C(=O)N(C)C)c(Cl)c12
CCc1c[nH]c2ncc(cc12)-c1cccc(c1)C(=O)N(C)C
CCc1c[nH]c2ncc(cc12)-c1ccc(N)c(n1)C(=O)N(C)C
CCc1c[nH]c2ncc(cc12)-c1ccc(N)c(C(=O)N(C)C)c1F
C[C@H]1CC(=O)c2ccc(Nc3cc4c(cnc(OC5CC5)c4cn3)[C@](C)(N)C3CC3)cc2C11CC1 |r|
COc1cc2CCN(C)Cc2cc1Nc1ncc(Cl)c(n1)N1CC(CO)c2ccccc12
Cc1ccncc1-c1cc2cc(NC(=O)C=C3CC(C3)C#N)ncc2c(N)n1 |(5.62,-3.46,;6.96,-2.69,;8.29,-3.46,;9.62,-2.69,;9.62,-1.15,;8.29,-.38,;6.96,-1.15,;5.62,-.38,;4.29,-1.16,;2.96,-.38,;1.63,-1.15,;.29,-.39,;-1.04,-1.16,;-2.37,-.39,;-2.37,1.15,;-3.71,-1.16,;-5.04,-.39,;-6.55,-.79,;-6.95,.69,;-5.44,1.1,;-8.29,1.46,;-9.62,2.23,;.29,1.16,;1.63,1.93,;2.96,1.16,;4.29,1.92,;4.29,3.46,;5.62,1.15,)|
C[C@H]1COC(=O)N1c1cc(N)c2nnc(NC(=O)[C@@H]3C[C@H]3c3cnn(C)c3)cc2c1 |r|
CN1CCc2c(C)cc(cc2C1)-c1cnc(N)c(OCc2ccnc(c2)C#Cc2cccc(F)c2)n1
Cn1cc(cn1)Nc2c(nc(cn2)C3=CCC[C@H](C3)NC(=O)c4ccccc4)C(=O)N
CC(CO)CNC(=O)c1c[nH]c2ncc(cc12)-c1ccc(C2CCOCC2)c(CN(C)C)c1
CCc1c(Cl)[nH]c2nc(C(=O)N(C)C)c(N)cc12
CCc1c(C)[nH]c2nc(C(=O)N(C)C)c(N)cc12
CN(C)C(=O)c1nc2[nH]c(C)cc2cc1N
Cc1c(CC#N)ccnc1-c1cccc(c1F)-c1cnc2NCC3(CC[C@](C)(C3)C(N)=O)c2c1Cl |r|
Cc1c(CC#N)ccnc1-c1cc(N)cc(c1)-c1cnc2NC[C@@]3(CC[C@@](C)(C3)C#N)c2c1Cl |r|
Fc1cc(NC(=O)NCCCN2CCOCC2)ccc1Oc1ccnc2[nH]cc(c12)C(F)(F)F
COc1ccc(-c2c[nH]c3nccc(Oc4c(F)cc(NC5=NCC(C)(CO)CO5)cc4F)c23)c(F)c1 |t:21|
CN(C)C(=O)c1ccc(cc1)-c1c[nH]c2ncc(cc12)-c1ccc2CCNCc2c1
CN(C)C(=O)c1ccc(cc1)-c1c[nH]c2ncc(cc12)-c1ccc2CCN(Cc2c1)[C@H]1CC[C@](C)(O)CC1 |r,wU:30.34,33.38,(-7.52,5.93,;-7.12,4.45,;-5.63,4.05,;-8.21,3.36,;-9.7,3.75,;-7.81,1.87,;-8.9,.78,;-8.5,-.7,;-7.02,-1.1,;-5.92,-.01,;-6.33,1.48,;-6.62,-2.59,;-7.52,-3.84,;-6.62,-5.08,;-5.15,-4.61,;-3.82,-5.37,;-2.5,-4.6,;-2.5,-3.07,;-3.82,-2.3,;-5.15,-3.07,;-1.17,-2.3,;-1.17,-.76,;.16,.01,;1.5,-.76,;2.82,.01,;4.15,-.75,;4.16,-2.29,;2.83,-3.06,;1.5,-2.29,;.17,-3.07,;5.49,-3.06,;6.82,-2.29,;8.16,-3.06,;8.16,-4.6,;9.7,-4.6,;8.93,-5.93,;6.82,-5.37,;5.49,-4.6,)|
CN(C)C1CN(C1)C(=O)c1ccc(cc1)-c1c[nH]c2ncc(cc12)-c1cc(C)c(N2CCN(CC2)C2CCN(C)CC2)c(C)c1
CN1CCC(C1)C(O)c1ccc(cc1)-c1c[nH]c2ncc(cc12)-c1ccc(N2CCN(C)CC2)c(C)c1
[H][C@]12CCc3cc(cc(C)c3N1CCN(C)C2)-c1cnc2[nH]cc(-c3ccc(cc3)C(=O)N(C)C[C@H](C)O)c2c1 |r|
COCCN(C)C(=O)c1ccc(cc1)-c1c[nH]c2ncc(nc12)-c1ccc(cc1)N1CCN(C)CC1
C[C@H](O)CN(C)C(=O)c1ccc(cc1)-c1c[nH]c2ncc(nc12)-c1cc(C)c2CCN(CCN3CCOCC3)Cc2c1 |r|
CCN(CC)CCNC(=O)c1c[nH]c(\C=C2/C(=O)Nc3ccc(cc23)-c2c(F)cccc2OC)c1
C\C(Nc1ccc(cn1)N1CCOCC1)=C1\C(=O)Nc2cnc(cc12)-c1cnccc1C
Oc1ccc(Br)cc1C(=O)N\N=C1/C(=O)Nc2ccc(Cl)cc12
C[C@H]1CCCN1C(=O)c1ccc(N\N=C2/C(=O)Nc3c2cc(C)cc3C)cc1 |r|
O=C(Nc1ccc2NC(=O)CCc2c1)c1n[nH]c2ccccc12
Cc1cccc(NC(=O)c2n[nH]c3ccccc23)c1
CCCC[C@@H](CC)CNC(=O)c1ccc(N\N=C2/C(=O)Nc3ccccc23)cc1 |r|
Cc1nnc2[nH]c(C)c(CC(=O)Nc3ncc(Cc4ccccc4F)s3)c(=O)n12
CC(=O)Nc1cc(Oc2ccc(NC(=O)Cc3ccccc3C(F)(F)F)cc2)ncn1
OC[C@H]1Nc2nc(Nc3ccc(C#N)c(CCCOc4ccccc14)c3)ncc2-c1cn[nH]c1 |r|
OC[C@H]1Nc2nc(Nc3ccc(C#N)c(CCCCOc4ccccc14)c3)ncc2-c1cn[nH]c1 |r|
OC[C@H]1Nc2nc(Nc3ccc(C#N)c(CCCCCOc4ccccc14)c3)ncc2-c1cn[nH]c1 |r|
OC[C@H]1Nc2nc(Nc3ccc(C#N)c(COCCOc4ccccc14)c3)ncc2-c1cn[nH]c1 |r|
CN1CCOc2ccccc2[C@@H](CO)Nc2nc(Nc3ccc(C#N)c(C1)c3)ncc2-c1cn[nH]c1 |r|
Cn1cc(cn1)-c1cnc2Nc3ccc(C#N)c(CCCCOc4ccccc4[C@@H](CO)Nc1n2)c3 |r|
OCCn1cc(cn1)-c1cnc2Nc3ccc(C#N)c(CCCCOc4ccccc4[C@@H](CO)Nc1n2)c3 |r|
CN(C)CCn1cc(cn1)-c1cnc2Nc3ccc(C#N)c(CCCCOc4ccccc4[C@@H](CO)Nc1n2)c3 |r|
CC(C)(O)Cn1cc(cn1)-c1cnc2Nc3ccc(C#N)c(CCCCOc4ccccc4[C@@H](CO)Nc1n2)c3 |r|
OC[C@H]1Nc2nc(Nc3ccc(C#N)c(CCCCOc4ccccc14)c3)ncc2-c1cnn(c1)C1CCNCC1 |r|
Cc1c2NCCOc2ncc1-c1cc2cc(NC(=O)C3CC3)ncc2c(N)c1F
Cc1c2NCCOc2ncc1-c1cc(N)c2cnc(Nc3ccccn3)nc2c1
Cc1c2NCCOc2ncc1-c1cc(N)c2cnc(Nc3cccnc3)nc2c1
Cc1c2NCCOc2ncc1-c1cc(N)c2cnc(Nc3ccncc3)nc2c1
Cc1c2NCCOc2ncc1-c1cc(N)c2cnc(Nc3ccn(C)n3)nc2c1
Cc1c2NCCOc2ncc1-c1cc(N)c2cnc(Nc3cnn(C)c3)nc2c1
CCn1ccc(Nc2ncc3c(N)cc(cc3n2)-c2cnc3OCCNc3c2C)n1
CCn1cc(Nc2ncc3c(N)cc(cc3n2)-c2cnc3OCCNc3c2C)cn1
Cc1nn(C)cc1Nc1ncc2c(N)cc(cc2n1)-c1cnc2OCCNc2c1C
Cc1cc(Nc2ncc3c(N)cc(cc3n2)-c2cnc3OCCNc3c2C)nn1C
Cc1c(Nc2ncc3c(N)cc(cc3n2)-c2cnc3OCCNc3c2C)cnn1C
Cc1c2NCCOc2ncc1-c1cc(N)c2cnc(Nc3cnn(c3)C3CC3)nc2c1
CC(C)n1cc(Nc2ncc3c(N)cc(cc3n2)-c2cnc3OCCNc3c2C)cn1
Nc1cc(cc2nc(Nc3cnn(c3)C3CC3)ncc12)-c1cccnc1
Cc1ccncc1-c1cc(N)c2cnc(Nc3cnn(c3)C3CC3)nc2c1
Cn1cc(cn1)-c1cc(N)c2cnc(Nc3cnn(c3)C3CC3)nc2c1
Cc1c(cnn1C)-c1cc(N)c2cnc(Nc3cnn(c3)C3CC3)nc2c1
Nc1cncc(c1)-c1cc(N)c2cnc(Nc3cnn(c3)C3CC3)nc2c1
Cc1c(N)cncc1-c1cc(N)c2cnc(Nc3cnn(c3)C3CC3)nc2c1
Cc1c2NCCOc2ncc1-c1cc(N)c2cnc(Nc3ccccc3)nc2c1
CNCc1cccc(Nc2ncc3c(N)cc(cc3n2)-c2cnc3OCCNc3c2C)c1
CNCc1ccc(Nc2ncc3c(N)cc(cc3n2)-c2cnc3OCCNc3c2C)cc1
CNCCc1cccc(Nc2ncc3c(N)cc(cc3n2)-c2cnc3OCCNc3c2C)c1
CNCCc1ccc(Nc2ncc3c(N)cc(cc3n2)-c2cnc3OCCNc3c2C)cc1
Cc1c2NCCOc2ncc1-c1cc(N)c2cnc(Nc3ccc4CCNCc4c3)nc2c1
Cc1c2NCCOc2ncc1-c1cc(N)c2cnc(Nc3ccc4CNCCc4c3)nc2c1
CN1CCc2ccc(Nc3ncc4c(N)cc(cc4n3)-c3cnc4OCCNc4c3C)cc2C1
CN1CCc2cc(Nc3ncc4c(N)cc(cc4n3)-c3cnc4OCCNc4c3C)ccc2C1
CCN1CCc2ccc(Nc3ncc4c(N)cc(cc4n3)-c3cnc4OCCNc4c3C)cc2C1
CC(C)N1CCc2ccc(Nc3ncc4c(N)cc(cc4n3)-c3cnc4OCCNc4c3C)cc2C1
COc1cc2CCN(C)Cc2cc1Nc1nc(Nc2ccccc2)c2cc[nH]c2n1
COc1cc2CCN(C)Cc2cc1Nc1nc(Nc2ccccc2F)c2cc[nH]c2n1
COc1cc2CCN(C)Cc2cc1Nc1nc(Nc2ccccc2Cl)c2cc[nH]c2n1
COc1cc2CCN(C)Cc2cc1Nc1nc(Nc2ccccc2C)c2cc[nH]c2n1
COc1cc2CCN(C)Cc2cc1Nc1nc(Nc2ccccc2C(C)(C)C)c2cc[nH]c2n1
COc1ccccc1Nc1nc(Nc2cc3CN(C)CCc3cc2OC)nc2[nH]ccc12
COc1cc2CCN(C)Cc2cc1Nc1nc(Nc2ccccc2OC(C)C)c2cc[nH]c2n1
COc1cc2CCN(C)Cc2cc1Nc1nc(Nc2ccccc2P(C)(C)=O)c2cc[nH]c2n1
COc1cc2CCN(C)Cc2cc1Nc1nc(Nc2ccccc2S(=O)(=O)C(C)C)c2cc[nH]c2n1
COc1cc2CCN(C)Cc2cc1Nc1nc(Nc2ccccc2S(=O)(=O)N(C)C)c2cc[nH]c2n1
CCN(CC)S(=O)(=O)c1ccccc1Nc1nc(Nc2cc3CN(C)CCc3cc2OC)nc2[nH]ccc12
CCCN(CCC)S(=O)(=O)c1ccccc1Nc1nc(Nc2cc3CN(C)CCc3cc2OC)nc2[nH]ccc12
COc1cc2CCN(C)Cc2cc1Nc1nc(Nc2ccccc2S(=O)(=O)N2CCC2)c2cc[nH]c2n1
COc1cc2CCN(C)Cc2cc1Nc1nc(Nc2ccccc2S(=O)(=O)N2CCCC2)c2cc[nH]c2n1
COc1cc2CCN(C)Cc2cc1Nc1nc(Nc2ccccc2S(=O)(=O)N2CC(C)(C)C2)c2cc[nH]c2n1
COc1cc2CCN(C)Cc2cc1Nc1nc(Nc2ccccc2S(=O)(=O)N2CCCCC2)c2cc[nH]c2n1
COc1cc2CCN(C)Cc2cc1Nc1nc(Nc2ccccc2S(=O)(=O)N2CCC(C)(C)CC2)c2cc[nH]c2n1
COc1cc2CCN(C)Cc2cc1Nc1nc(Nc2ccccc2S(=O)(=O)N2CCOCC2)c2cc[nH]c2n1
COc1cc2CCN(C)Cc2cc1Nc1nc(Nc2ccccc2S(=O)(=O)N(C)C)c2c(c[nH]c2n1)-c1ccoc1
COc1cc2CCN(C)Cc2cc1Nc1nc(Nc2ccccc2S(=O)(=O)N(C)C)c2c(c[nH]c2n1)-c1cn[nH]c1
COc1cc2CCN(C)Cc2cc1Nc1nc(Nc2ccccc2S(=O)(=O)N(C)C)c2c(c[nH]c2n1)-c1cnn(C)c1
COc1cc2CCN(C)Cc2cc1Nc1nc(Nc2ccccc2S(=O)(=O)N(C)C)c2c(c[nH]c2n1)-c1c[nH]nc1C
COc1cc2CCN(C)Cc2cc1Nc1nc(Nc2ccccc2S(=O)(=O)N(C)C)c2c(c[nH]c2n1)-c1c(C)noc1C |(-7.33,-1.57,;-6,-.8,;-4.67,-1.57,;-4.67,-3.11,;-3.33,-3.88,;-3.33,-5.42,;-2,-6.19,;-.67,-5.42,;.67,-6.19,;-.67,-3.88,;-2,-3.11,;-2,-1.57,;-3.33,-.8,;-3.33,.74,;-2,1.51,;-.66,.74,;.67,1.52,;2,.75,;2,-.79,;.66,-1.57,;.66,-3.11,;2,-3.87,;3.33,-3.1,;3.33,-1.56,;4.67,-.79,;5.44,.54,;3.9,.54,;6,-1.56,;7.33,-.79,;6,-3.1,;.67,3.05,;1.81,4.08,;1.18,5.49,;-.35,5.33,;-.67,3.82,;-2,3.05,;3.3,3.68,;3.85,2.32,;2.51,1.55,;5.38,2.32,;5.78,3.81,;4.49,4.65,;4.49,6.19,)|
COc1cc2CCN(C)Cc2cc1Nc1nc(Nc2ccccc2S(=O)(=O)N(C)C)c2c(c[nH]c2n1)-c1ccncc1
COc1cc2CCN(C)Cc2cc1Nc1nc(Nc2ccccc2S(=O)(=O)N(C)C)c2c(c[nH]c2n1)-c1cccnc1
COc1cc2CCN(C)Cc2cc1Nc1nc(Nc2ccccc2S(=O)(=O)N(C)C)c2c(c[nH]c2n1)-c1ccc(N)nc1
COc1cc2CCN(C)Cc2cc1Nc1nc(Nc2ccccc2S(=O)(=O)N(C)C)c2c(c[nH]c2n1)-c1ccn(C)c(=O)c1
COc1cc2CCN(C)Cc2cc1Nc1nc(Nc2ccccc2S(=O)(=O)N(C)C)c2c(c[nH]c2n1)-c1ccccc1
COc1cc2CCN(C)Cc2cc1Nc1nc(Nc2ccccc2S(=O)(=O)N(C)C)c2c(c[nH]c2n1)-c1cccnc1C
COc1cc2CCN(C)Cc2cc1Nc1nc(Nc2ccccc2S(=O)(=O)N(C)C)c2c(c[nH]c2n1)-c1cnccc1C
COc1cc2CCN(C)Cc2cc1Nc1nc(Nc2ccccc2S(=O)(=O)N2CCC2)c2c(c[nH]c2n1)-c1cccnc1
COc1cc2CCN(C)Cc2cc1Nc1nc(Nc2ccccc2S(=O)(=O)N2CCCC2)c2c(c[nH]c2n1)-c1cccnc1
CN(C)S(=O)(=O)c1ccccc1Nc1nc(Nc2cc3CN(C)CCc3cc2Cl)nc2[nH]cc(-c3cccnc3)c12
CN(C)S(=O)(=O)c1ccccc1Nc1nc(Nc2ccc3CCN(C)Cc3c2)nc2[nH]cc(-c3cccnc3)c12
CN(C)S(=O)(=O)c1ccccc1Nc1nc(Nc2ccc3CN(C)CCc3c2)nc2[nH]cc(-c3cccnc3)c12
COc1cc2CCN(Cc2cc1Nc1nc(Nc2ccccc2S(=O)(=O)N(C)C)c2c(c[nH]c2n1)-c1cccnc1)C(C)C
COc1ccc(CN(C)C)cc1Nc1nc(Nc2ccccc2S(=O)(=O)N(C)C)c2c(c[nH]c2n1)-c1cccnc1
COc1cc(ccc1Nc1nc(Nc2ccccc2S(=O)(=O)N(C)C)c2c(c[nH]c2n1)-c1cccnc1)N1CCOCC1
CN(C)S(=O)(=O)c1ccccc1Nc1nc(Nc2ccc(cc2)N2CCOCC2)nc2[nH]cc(-c3cccnc3)c12
COc1cc(Nc2nc(Nc3ccccc3S(=O)(=O)N(C)C)c3c(c[nH]c3n2)-c2cccnc2)ccc1N1CCOCC1
CCOc1cc(Nc2nc(Nc3ccccc3S(=O)(=O)N(C)C)c3c(c[nH]c3n2)-c2cccnc2)ccc1N1CCOCC1
CN1CCC(CC1)c1ccc(Nc2ncc3ccc(cc3n2)-c2cccc(c2)C#N)cc1
CN1CCC(CC1)c1ccc(Nc2ncc3ccc(cc3n2)-c2ccccc2C(N)=O)cc1
CN1CCC(CC1)c1ccc(Nc2ncc3ccc(cc3n2)-c2cccc(OC(F)(F)F)c2)cc1
CN1CCC(CC1)c1ccc(Nc2ncc3ccc(cc3n2)-c2cccc(CN)c2)cc1
CN1CCC(CC1)c1ccc(Nc2ncc3ccc(cc3n2)-c2cccc(CO)c2)cc1
CN1CCC(CC1)c1ccc(Nc2ncc3ccc(cc3n2)-c2ccccc2CO)cc1
CN1CCC(CC1)c1ccc(Nc2ncc3ccc(cc3n2)-c2cnc3CCNCc3c2)cc1
COc1cccc(F)c1-c1ccc2cnc(Nc3ccc(cc3)C3CCN(C)CC3)nc2c1
CN1CCC(CC1)c1ccc(Nc2ncc3ccc(cc3n2)-c2cnccc2C)cc1
CN1CCC(CC1)c1ccc(Nc2ncc3ccc(cc3n2)-c2ccncc2C)cc1
COc1ccnc(F)c1-c1ccc2cnc(Nc3ccc(cc3)C3CCN(C)CC3)nc2c1
CN1CCC(CC1)c1ccc(Nc2ncc3ccc(cc3n2)-c2nnn(C)c2C)cc1
CN1CCC(CC1)c1ccc(Nc2ncc3ccc(cc3n2)-c2cnc3COCCn23)cc1
CN1CCC(CC1)c1ccc(Nc2ncc3ccc(cc3n2)-c2cnc[nH]2)cc1
CN1CCC(CC1)c1ccc(Nc2ncc3ccc(cc3n2)-c2cnc(s2)C(C)(C)O)cc1
CN1CCC(CC1)c1ccc(Nc2ncc3ccc(cc3n2)-c2cnn(C)c2)cc1
CN1CCC(CC1)c1ccc(Nc2ncc3ccc(cc3n2)-c2cn[nH]c2)cc1
CCn1cc(cn1)-c1ccc2cnc(Nc3ccc(cc3)C3CCN(C)CC3)nc2c1
CC(C)n1cc(cn1)-c1ccc2cnc(Nc3ccc(cc3)C3CCN(C)CC3)nc2c1
CN1CCC(CC1)c1ccc(Nc2ncc3ccc(cc3n2)-c2cnn(CCO)c2)cc1
CN1CCC(CC1)c1ccc(Nc2ncc3ccc(cc3n2)-c2cnn(C)c2C)cc1
CN1CCC(CC1)c1ccc(Nc2ncc3ccc(cc3n2)-c2c(C)nn(C)c2C)cc1
CN1CCC(CC1)c1ccc(Nc2ncc3ccc(cc3n2)-c2cnn(C)c2C2CC2)cc1
CN1CCC(CC1)c1ccc(Nc2ncc3ccc(cc3n2)-c2cnn3CCCCc23)cc1
CN1CCC(CC1)c1ccc(Nc2ncc3ccc(cc3n2)-c2cnn(C)c2-c2ccccc2)cc1
Cc1c2NCCOc2ncc1-c1ccc2cnc(Nc3ccc4COC(C)(C)c4c3)nc2c1
CN1CCC(CC1)c1ccc(Nc2ncc3ccc(cc3n2)-c2cnc3OCCNc3c2C)cc1
Cc1c2NCCOc2ncc1-c1ccc2cnc(Nc3ccc4COCc4c3)nc2c1
Cc1c2NCCOc2ncc1-c1ccc2cnc(Nc3ccc4CCOCc4c3)nc2c1
Cc1c2NCCOc2ncc1-c1ccc2cnc(Nc3ccc4COCCc4c3)nc2c1
Cc1c2NCCOc2ncc1-c1ccc2cnc(Nc3cnc4COC(C)(C)c4c3)nc2c1
Cc1c2NCCOc2ncc1-c1ccc2cnc(Nc3ccc4C(=O)OC(C)(C)c4c3)nc2c1
CC(=O)Nc1cccc(Nc2ncc3ccc(cc3n2)-c2cnc3OCCNc3c2C)c1
CC(=O)Nc1ccc(Nc2ncc3ccc(cc3n2)-c2cnc3OCCNc3c2C)cc1
CC(=O)Nc1ccc(Nc2ncc3ccc(cc3n2)-c2cnc3OCCNc3c2C)cc1C
CC(=O)Nc1ccc(Nc2ncc3ccc(cc3n2)-c2cnc3OCCNc3c2C)cc1C(F)(F)F
CN(C)CC(=O)Nc1ccc(Nc2ncc3ccc(cc3n2)-c2cnc3OCCNc3c2C)cc1C
Cc1cc(Nc2ncc3ccc(cc3n2)-c2cnc3OCCNc3c2C)ccc1NC(=O)CN1CCC1
Cc1c2NCCOc2ncc1-c1ccc2cnc(Nc3ccc(cc3)N3CCOC3=O)nc2c1
Cc1c2NCCOc2ncc1-c1ccc2cnc(Nc3ccc(cc3)N3CCNC3=O)nc2c1
Cc1cc(Nc2ncc3ccc(cc3n2)-c2cnc3OCCNc3c2C)ccc1C(N)=O
Cc1c2NCCOc2ncc1-c1ccc2cnc(Nc3ccc(CS(C)(=O)=O)nc3)nc2c1
Cc1c2NCCOc2ncc1-c1ccc2cnc(Nc3ccc(cc3)[S@@](C)(=N)=O)nc2c1 |r|
Cc1c2NCCS(=O)(=O)c2ncc1-c1ccc2cnc(Nc3ccc(CS(C)(=O)=O)cc3)nc2c1
Cc1c2NCCC(=O)c2ncc1-c1ccc2cnc(Nc3ccc(CS(C)(=O)=O)cc3)nc2c1
Cc1c2NCCC(O)c2ncc1-c1ccc2cnc(Nc3ccc(CS(C)(=O)=O)cc3)nc2c1
Cc1c2NCCC(F)(F)c2ncc1-c1ccc2cnc(Nc3ccc(CS(C)(=O)=O)cc3)nc2c1
CS(=O)(=O)Cc1ccc(Nc2ncc3ccc(cc3n2)-c2cnc3OCCNc3c2C#N)cc1
CN(C)c1c2NCCOc2ncc1-c1ccc2cnc(Nc3ccc(CS(C)(=O)=O)cc3)nc2c1
COc1c2NCCOc2ncc1-c1ccc2cnc(Nc3ccc(CS(C)(=O)=O)cc3)nc2c1
COc1cc2CCN(C)Cc2cc1Nc1ncc(C(N)=O)c(Nc2cccc3CCOc23)n1
CO[C@H](C)c1ccccc1Nc1nc(Nc2cc3CN(C)CCc3cc2OC)ncc1C(N)=O |r|
CCOc1ccccc1Nc1nc(Nc2cc3CN(C)CCc3cc2OC)ncc1C(N)=O
COCCOc1ccc(-c2cc(C(N)=O)c3ncnc(N[C@H]4CCCNC4)c3n2)c(c1)C#N |r|
CS(=O)(=O)Cc1ccc(cc1)-c1cc(C(N)=O)c2ncnc(N[C@H]3CCCNC3)c2n1 |r|
NC(=O)c1cc(nc2c(N[C@H]3CCCNC3)ncnc12)-c1ccc(cc1)C1(O)CC1 |r|
CN1CCN(CC1)c1ccc(cn1)-c1cc(C(N)=O)c2ncnc(N[C@H]3CCCNC3)c2n1 |r|
COc1ccccc1-c1cc(C(N)=O)c2ncnc(N[C@H]3CCCNC3)c2n1 |r|
NC(=O)c1cc(nc2c(N[C@H]3CCCNC3)ncnc12)-c1ccc(F)cc1 |r|
CC1(C)NC(=O)c2ccc(Nc3ncc(-c4nnco4)c(N[C@H](CO)c4ccccc4)n3)cc12 |r|
OC[C@@H](Nc1nc(Nc2ccc3C(=O)NCc3c2)ncc1-c1nnco1)c1ccccc1 |r|
OC[C@@H](Nc1nc(Nc2ccc3C(=O)NC4(CC4)c3c2)ncc1-c1nnco1)c1ccccc1 |r|
CN1C(=O)c2ccc(Nc3ncc(-c4nnco4)c(N[C@H](CO)c4ccccc4)n3)cc2C1(C)C |r|
CCN1C(=O)c2ccc(Nc3ncc(-c4nnco4)c(N[C@H](CO)c4ccccc4)n3)cc2C1(C)C |r|
CC1(C)N(CC(F)(F)F)C(=O)c2ccc(Nc3ncc(-c4nnco4)c(N[C@H](CO)c4ccccc4)n3)cc12 |r|
Cc1nnc(o1)-c1cnc(Nc2ccc3C(=O)NC(C)(C)c3c2)nc1N[C@H](CO)c1ccccc1 |r|
CC1(C)NC(=O)c2ccc(Nc3ncc(-c4nnc(CCl)o4)c(N[C@H](CO)c4ccccc4)n3)cc12 |r|
CC1(C)NC(=O)c2ccc(Nc3ncc(-c4nnc(o4)C(F)F)c(N[C@H](CO)c4ccccc4)n3)cc12 |r|
CC1(C)NC(=O)c2ccc(Nc3ncc(-c4nnc(o4)C(F)(F)F)c(N[C@H](CO)c4ccccc4)n3)cc12 |r|
CC1(C)NC(=O)c2ccc(Nc3ncc(-c4nnc(o4)C(F)(F)Cl)c(N[C@H](CO)c4ccccc4)n3)cc12 |r|
CC(F)(F)c1nnc(o1)-c1cnc(Nc2ccc3C(=O)NC(C)(C)c3c2)nc1N[C@H](CO)c1ccccc1 |r|
CC1(C)NC(=O)c2ccc(Nc3ncc(-c4nnc(o4)C4CC4)c(N[C@H](CO)c4ccccc4)n3)cc12 |r|
CC1(C)NC(=O)c2ccc(Nc3ncc(-c4nnc(o4)C4(F)CC4)c(N[C@H](CO)c4ccccc4)n3)cc12 |r|
CC1(C)NC(=O)c2ccc(Nc3ncc(-c4nnc(o4)C4CC4(F)F)c(N[C@H](CO)c4ccccc4)n3)cc12 |r|
CC1(C)NC(=O)c2ccc(Nc3ncc(C(=O)NCCO)c(N[C@H](CO)c4ccccc4)n3)cc12 |r|
CC1(C)NC(=O)c2ccc(Nc3ncc(C(=O)NCC(O)C(F)(F)F)c(N[C@H](CO)c4ccccc4)n3)cc12 |r|
CC1(C)NC(=O)c2ccc(Nc3ncc(C(=O)NCC4(O)COC4)c(N[C@H](CO)c4ccccc4)n3)cc12 |r|
CC1(C)NC(=O)c2ccc(Nc3ncc(C(=O)NC[C@H](F)CO)c(N[C@H](CO)c4ccccc4)n3)cc12 |r|
CC(C)(O)[C@H](F)CNC(=O)c1cnc(Nc2ccc3C(=O)NC(C)(C)c3c2)nc1N[C@H](CO)c1ccccc1 |r|
CC1(C)NC(=O)c2ccc(Nc3ncc(C(=O)NCC(F)(F)CO)c(N[C@H](CO)c4ccccc4)n3)cc12 |r|
COCC(C)(C)CNC(=O)c1cnc(Nc2ccc3C(=O)NC(C)(C)c3c2)nc1N[C@H](CO)c1ccccc1 |r|
CC(C)(O)CCCNC(=O)c1cnc(Nc2ccc3C(=O)NC(C)(C)c3c2)nc1N[C@H](CO)c1ccccc1 |r|
CC1(C)NC(=O)c2ccc(Nc3ncc(C(=O)NCCOCCO)c(N[C@H](CO)c4ccccc4)n3)cc12 |r|
CC1(C)NC(=O)c2ccc(Nc3ncc(C(=O)NCCCOCCO)c(N[C@H](CO)c4ccccc4)n3)cc12 |r|
COCCOCCNC(=O)c1cnc(Nc2ccc3C(=O)NC(C)(C)c3c2)nc1N[C@H](CO)c1ccccc1 |r|
CC1(C)NC(=O)c2ccc(Nc3ncc(C(=O)NCCCN4CCOCC4)c(N[C@H](CO)c4ccccc4)n3)cc12 |r|
CN1CCN(CCCNC(=O)c2cnc(Nc3ccc4C(=O)NC(C)(C)c4c3)nc2N[C@H](CO)c2ccccc2)CC1 |r|
CC1(C)NC(=O)c2ccc(Nc3ncc(C(=O)N[C@@H]4C[C@H](CO)[C@@H](O)[C@H]4O)c(N[C@H](CO)c4ccccc4)n3)cc12 |r|
CC1(C)NC(=O)c2ccc(Nc3ncc(C(=O)NC4C(O)OC(CO)C(O)C4O)c(N[C@H](CO)c4ccccc4)n3)cc12 |r|
CC1(C)NC(=O)c2ccc(Nc3ncc(-c4nnco4)c(N[C@H](CO)c4ccccc4F)n3)cc12 |r|
CC1(C)NC(=O)c2ccc(Nc3ncc(-c4nnco4)c(N[C@H](CO)c4cccc(F)c4)n3)cc12 |r|
CC1(C)NC(=O)c2ccc(Nc3ncc(-c4nnco4)c(N[C@H](CO)c4ccc(F)cc4)n3)cc12 |r|
CC1(C)NC(=O)c2ccc(Nc3ncc(-c4nnco4)c(N[C@H](CO)c4ccc(F)c(F)c4)n3)cc12 |r|
CC1(C)NC(=O)c2ccc(Nc3ncc(-c4nnco4)c(N[C@H](CO)c4cc(F)ccc4F)n3)cc12 |r|
CC1(C)NC(=O)c2ccc(Nc3ncc(-c4nnco4)c(N[C@H](CO)c4cc(F)cc(F)c4)n3)cc12 |r|
CC1(C)NC(=O)c2ccc(Nc3ncc(-c4nnco4)c(N[C@H](CO)c4ccc(F)cc4F)n3)cc12 |r|
CC1(C)NC(=O)c2ccc(Nc3ncc(-c4nnco4)c(N[C@H](CO)c4cccc(Cl)c4)n3)cc12 |r|
CC(C)(O)[C@@H](Nc1nc(Nc2ccc3C(=O)NC(C)(C)c3c2)ncc1-c1nnco1)c1ccccc1 |r|
CC1(C)NC(=O)c2ccc(Nc3ncc(-c4nnco4)c(N[C@H](CCO)c4ccccc4)n3)cc12 |r|
N[C@H]1CN(CC[C@H]1F)c1ncnc2[nH]c(Cl)c(-c3cccc(c3)C#N)c12 |r|
C[C@@H]1CCCN1c1cc2C(=O)N(Cc2c(n1)[C@H](N)CN)c1cccc(n1)-c1nnc2CC[C@H](C)n12 |r|
CN1CCC2(CC1)CN(CCO2)c1ncnc2[nH]cc(-c3cccc(c3)C#N)c12
CN1CCC2(CC1)CN(CCO2)c1ncnc2[nH]c(Cl)c(-c3cccc(c3)C#N)c12
Clc1[nH]c2ncnc(N3CCO[C@]4(CCNC4)C3)c2c1-c1cccc(c1)C#N |r|
NC[C@H]1CN(CCO1)c1ncnc2[nH]c(Cl)c(-c3cccc(CO)c3)c12 |r|
Clc1[nH]c2ncnc(N3CCCC4(CNC4)C3)c2c1-c1cccc(c1)C#N
N[C@@H]1CCCCN(C1)c1ncnc2[nH]c(Cl)c(-c3cccc(c3)C#N)c12 |r|
N[C@H]1CCN(C1)c1ncnc2[nH]c(Cl)c(-c3cccc(c3)C#N)c12 |r|
N[C@@H]1CCCN(C1)c1ncnc2[nH]c(Cl)c(-c3cccc(c3)C#N)c12 |r|
N[C@@H]1CCCN(C1)c1ncnc2[nH]cc(-c3cccc(c3)C#N)c12 |r|
O[C@@H]1CCCN(C1)c1ncnc2[nH]cc(-c3cccc(c3)C#N)c12 |r|
C[C@H]1C[C@@H](N)CN(C1)c1ncnc2[nH]c(Cl)c(-c3cccc(c3)C#N)c12 |r|
N[C@@H]1C[C@@H](CN(C1)c1ncnc2[nH]c(Cl)c(-c3cccc(c3)C#N)c12)C(F)(F)F |r|
C[C@H]1C[C@@H](N)CN(C1)c1ncnc2[nH]c(Cl)c(-c3ccccc3)c12 |r|
C[C@H]1C[C@@H](N)CN(C1)c1ncnc2[nH]c(Cl)c(-c3cnn(C)c3)c12 |r|
C[C@H]1C[C@@H](N)CN(C1)c1ncnc2[nH]c(Cl)c(-c3cccc(CO)c3)c12 |r|
C[C@H]1C[C@@H](N)CN(C1)c1ncnc2[nH]c(Cl)c(-c3cccc(C#N)c3C)c12 |r,wD:1.0,3.3,(2.78,-.76,;2.51,.76,;3.69,1.75,;3.42,3.27,;4.6,4.26,;1.98,3.79,;.8,2.8,;1.07,1.29,;-.65,3.33,;-.65,4.87,;-1.98,5.64,;-3.32,4.87,;-3.32,3.33,;-4.46,2.3,;-3.83,.89,;-4.6,-.44,;-2.3,1.05,;-1.49,-.25,;.05,-.25,;.87,-1.51,;.15,-2.92,;-1.39,-2.92,;-2.12,-4.28,;-2.84,-5.64,;-2.21,-1.61,;-3.75,-1.61,;-1.98,2.56,)|
C[C@H]1C[C@@H](N)CN(C1)c1ncnc2[nH]c(Cl)c(-c3cccc(C#N)c3Cl)c12 |r,wD:1.0,3.3,(2.78,-.76,;2.51,.76,;3.69,1.75,;3.42,3.27,;4.6,4.26,;1.98,3.79,;.8,2.8,;1.07,1.29,;-.65,3.33,;-.65,4.87,;-1.98,5.64,;-3.32,4.87,;-3.32,3.33,;-4.46,2.3,;-3.83,.89,;-4.6,-.44,;-2.3,1.05,;-1.49,-.25,;.05,-.25,;.87,-1.51,;.15,-2.92,;-1.39,-2.92,;-2.12,-4.28,;-2.84,-5.64,;-2.21,-1.61,;-3.75,-1.61,;-1.98,2.56,)|
C[C@H]1C[C@@H](N)CN(C1)c1ncnc2[nH]c(Cl)c(-c3cccc(C#N)c3F)c12 |r,wD:1.0,3.3,(2.78,-.76,;2.51,.76,;3.69,1.75,;3.42,3.27,;4.6,4.26,;1.98,3.79,;.8,2.8,;1.07,1.29,;-.65,3.33,;-.65,4.87,;-1.98,5.64,;-3.32,4.87,;-3.32,3.33,;-4.46,2.3,;-3.83,.89,;-4.6,-.44,;-2.3,1.05,;-1.49,-.25,;.05,-.25,;.87,-1.51,;.15,-2.92,;-1.39,-2.92,;-2.12,-4.28,;-2.84,-5.64,;-2.21,-1.61,;-3.75,-1.61,;-1.98,2.56,)|
C[C@H]1CC[C@@H](N)CN1c1ncnc2[nH]c(Cl)c(-c3cccc(c3)C#N)c12 |r|
[H][C@@]12CCCN(c3ncnc4[nH]c(Cl)c(-c5cccc(c5)C#N)c34)[C@]1([H])CCN2 |r|
COc1cc2c(cc1Nc1ncc3c(N)cc(=O)n(-c4ccccc4)c3n1)CN(C)CC2
COc1cc2c(cc1Nc1ncc3c(N)cc(=O)n(-c4ccccc4Cl)c3n1)CN(C)CC2
COc1cc2c(cc1Nc1ncc3c(N)cc(=O)n(-c4ccccc4C(F)(F)F)c3n1)CN(C)CC2
COc1cc2c(cc1Nc1ncc3c(N)cc(=O)n(-c4ccccc4C)c3n1)CN(C)CC2
CCc1ccccc1-n1c(=O)cc(N)c2cnc(Nc3cc4c(cc3OC)CCN(C)C4)nc21
COc1cc2c(cc1Nc1ncc3c(N)cc(=O)n(-c4ccccc4OC)c3n1)CN(C)CC2
COc1cccc(-n2c(=O)cc(N)c3cnc(Nc4cc5c(cc4OC)CCN(C)C5)nc32)c1
COc1ccc(-n2c(=O)cc(N)c3cnc(Nc4cc5c(cc4OC)CCN(C)C5)nc32)cc1
COc1cc2c(cc1Nc1ncc3c(N)cc(=O)n(-c4c(F)cccc4C(F)(F)F)c3n1)CN(C)CC2
COc1cc2c(cc1Nc1ncc3c(N)cc(=O)n(-c4c(OC)cccc4OC)c3n1)CN(C)CC2
COc1cc2c(cc1Nc1ncc3ccc(=O)n(-c4ccccc4C(F)(F)F)c3n1)CN(C)CC2
COc1cc2c(cc1Nc1ncc3c(N)cc(=O)n(Cc4ccccc4)c3n1)CN(C)CC2
COc1cc2c(cc1Nc1ncc3c(N)cc(=O)n([C@H](C)c4ccccc4)c3n1)CN(C)CC2
COc1cc2c(cc1Nc1ncc3c(N)cc(=O)n([C@@H](C)c4ccccc4)c3n1)CN(C)CC2
COc1cc2c(cc1Nc1ncc3c(N)cc(=O)n(Cc4cccc(C(F)(F)F)c4)c3n1)CN(C)CC2
COc1cc2c(cc1Nc1ncc3c(N)cc(=O)n(Cc4ccc(C(F)(F)F)cc4)c3n1)CN(C)CC2
CN1CCc2cc(c(cc2C1)Nc3ncc4c(n3)N(C(=O)C=C4N)Cc5ccccc5C(F)(F)F)OC
COc1cccc(Cn2c(=O)cc(N)c3cnc(Nc4cc5c(cc4OC)CCN(C)C5)nc32)c1
COc1ccc(Cn2c(=O)cc(N)c3cnc(Nc4cc5c(cc4OC)CCN(C)C5)nc32)cc1
COc1ccccc1Cn1c(=O)cc(N)c2cnc(Nc3cc4c(cc3OC)CCN(C)C4)nc21
COc1cc2c(cc1Nc1ncc3c(N)cc(=O)n(Cc4ccccc4F)c3n1)CN(C)CC2
COc1cc2c(cc1Nc1ncc3c(N)cc(=O)n(Cc4ccccc4C)c3n1)CN(C)CC2
COc1cc2c(cc1Nc1ncc3c(N)cc(=O)n(Cc4ccccc4Cl)c3n1)CN(C)CC2
COc1cc2c(cc1Nc1ncc3c(N)cc(=O)n(Cc4ccccc4OC(C)C)c3n1)CN(C)CC2
COc1cc2c(cc1Nc1ncc3c(N)cc(=O)n(Cc4ccc(F)cc4C(F)(F)F)c3n1)CN(C)CC2
COc1cc2c(cc1Nc1ncc3c(N)cc(=O)n(Cc4c(F)cccc4C(F)(F)F)c3n1)CN(C)CC2
CC[C@@H](N)c1cc(N2CCC[C@H]2C)cc2c1CN(c1cccc(-c3nnc4n3[C@@H](C)CC4)n1)C2=O
CC(C)(O)Cn1nccc1-c1ccc2cc1N[C@H](CO)c1ccccc1OCCCCc1cc(ccc1C#N)N2
[2H]C([2H])(O)[C@@H](Nc1nc(Nc2ccc3c(c2)C(C)(C)NC3=O)ncc1-c1nnco1)c1ccc(F)cc1
CN1CCN(c2ccc(-c3cnc4[nH]nc(-c5ccc(C#N)cc5)c4c3)cc2)CC1
CN1CCN(c2ccc(-c3cnc4[nH]nc(-c5ccc(C(F)(F)F)cc5)c4c3)cc2)CC1
CN1CCN(c2ccc(-c3cnc4[nH]nc(-c5ccc(C(F)F)cc5)c4c3)cc2)CC1
CSc1ccccc1-c1n[nH]c2ncc(-c3ccc(N4CCN(C)CC4)cc3)cc12
CC(=O)Nc1cccc(-c2n[nH]c3ncc(-c4ccc(N5CCN(C)CC5)cc4)cc23)c1
CN1CCN(c2ccc(-c3cnc4[nH]nc(-c5ccc(N(C)C)cc5)c4c3)cc2)CC1
CCN(CC)c1ccc(-c2n[nH]c3ncc(-c4ccc(N5CCN(C)CC5)cc4)cc23)cc1
CN(C)Cc1ccc(-c2n[nH]c3ncc(-c4ccc(N5CCN(C)CC5)cc4)cc23)cc1
CSc1ccc(-c2n[nH]c3ncc(-c4ccc(N5CCN(C)CC5)cc4)cc23)cc1
CCOc1ccc(-c2n[nH]c3ncc(-c4ccc(N5CCN(C)CC5)cc4)cc23)cc1
CN1CCN(c2ccc(-c3cnc4[nH]nc(-c5ccc(Oc6ccccc6)cc5)c4c3)cc2)CC1
CN1CCN(c2ccc(-c3cnc4[nH]nc(-c5ccc(OCc6ccccc6)cc5)c4c3)cc2)CC1
CN1CCN(c2ccc(-c3cnc4[nH]nc(-c5ccc(OC(F)F)cc5)c4c3)cc2)CC1
COc1cccc(F)c1-c1n[nH]c2ncc(-c3ccc(N4CCN(C)CC4)cc3)cc12
Cc1ccc(-c2n[nH]c3ncc(-c4ccc(N5CCN(C)CC5)cc4)cc23)cc1
CN1CCN(c2ccc(-c3cnc4[nH]nc(-c5ccc(C6(C#N)CC6)cc5)c4c3)cc2)CC1
CN1CCN(c2ccc(-c3cnc4[nH]nc(-c5ccccc5OC(F)(F)F)c4c3)cc2)CC1
CCOc1ccccc1-c1n[nH]c2ncc(-c3ccc(N4CCN(C)CC4)cc3)cc12
CC(C)Oc1cccc(-c2n[nH]c3ncc(-c4ccc(N5CCN(C)CC5)cc4)cc23)c1
CC(=O)c1cccc(-c2n[nH]c3ncc(-c4ccc(N5CCN(C)CC5)cc4)cc23)c1
COc1ccc(-c2n[nH]c3ncc(-c4ccc(N5CCN(C)CC5)cc4)cc23)cc1
CN1CCN(c2ccc(-c3cnc4[nH]nc(-c5ccc(S(C)(=O)=O)cc5)c4c3)cc2)CC1
COCc1ccc(-c2n[nH]c3ncc(-c4ccc(N5CCN(C)CC5)cc4)cc23)cc1
CN1CCN(c2ccc(-c3cnc4[nH]nc(-c5ccc(OC6CC6)cc5)c4c3)cc2)CC1
CN1CCN(c2ccc(-c3cnc4[nH]nc(-c5ccc(OC(F)(F)F)cc5)c4c3)cc2)CC1
COc1ccc(-c2n[nH]c3ncc(-c4ccc(N5CCN(C)CC5)cc4)cc23)cc1F
COc1ccc(-c2n[nH]c3ncc(-c4ccc(N5CCN(C)CC5)cc4)cc23)c(F)c1F
COc1ccc(-c2n[nH]c3ncc(-c4ccc(N5CCN(C)CC5)cc4)cc23)cc1OC
COc1cc(-c2n[nH]c3ncc(-c4ccc(N5CCN(C)CC5)cc4)cc23)cc(OC)c1OC
CN1CCN(c2ccc(-c3cnc4[nH]nc(-c5ccc6c(c5)OCCO6)c4c3)cc2)CC1
COc1c(F)cc(-c2n[nH]c3ncc(-c4ccc(N5CCN(C)CC5)cc4)cc23)cc1F
COc1ccc(-c2n[nH]c3ncc(-c4ccc(N5CCN(C)CC5)cc4)cc23)c(F)c1
COc1ccc(-c2n[nH]c3ncc(-c4ccc(N5CCN(C)CC5)cc4)cc23)c(C(F)(F)F)c1
COc1ccc(-c2n[nH]c3ncc(-c4ccc(N5CCN(C)CC5)cc4)cc23)cc1Cl
COc1ccc(-c2n[nH]c3ncc(-c4ccc(N5CCN(C)CC5)cc4)cc23)c(Cl)c1
COc1ccc(-c2n[nH]c3ncc(-c4ccc(N5CCN(C)CC5)cc4)cc23)cc1C
COc1ccc(-c2n[nH]c3ncc(-c4ccc(N5CCN(C)CC5)cc4)cc23)cc1C(F)(F)F
COc1ccc(-c2c[nH]c3ncc(-c4ccc(N5CCN(C)CC5)cc4)cc23)cc1OC
COc1ccc(-c2c[nH]c3ncc(-c4ccc(N5CCN(C)CC5)cc4)nc23)cc1OC
COc1ccc(-c2c[nH]c3ncc(-c4ccc(N5CCNCC5)cc4)cc23)cc1OC
COc1ccc(-c2c[nH]c3ncc(-c4ccc(N5CCN(C)CC5)nc4)cc23)cc1OC
COc1ccc(-c2c[nH]c3ncc(-c4ccc(C5CCN(C)CC5)cc4)cc23)cc1OC
COc1ccc(-c2c[nH]c3ncc(-c4ccc(C5CCOCC5)cc4)cc23)cc1OC
COc1ccc(-c2c[nH]c3ncc(-c4ccc(N5CCOCC5)nc4)cc23)cc1OC
COc1ccc(-c2c[nH]c3ncc(-c4ccc(N5CCNCC5)nc4)cc23)cc1OC
COc1ccc(-c2c[nH]c3ncc(-c4ccc(N5CCOCC5)cc4)cc23)cc1OC
COc1ccc(-c2c[nH]c3ncc(-c4cnc(N5CCN(C)CC5)nc4)cc23)cc1OC
COc1ccc(-c2c[nH]c3ncc(-c4ccc(N5CCN(C(=O)N(C)C)CC5)cc4)cc23)cc1OC
COCCN1CCN(c2ccc(-c3cnc4[nH]cc(-c5ccc(OC)c(OC)c5)c4c3)cc2)CC1
COc1ccc(-c2c[nH]c3ncc(-c4ccc(N5CCN(CCO)CC5)cc4)cc23)cc1OC
COc1ccc(-c2c[nH]c3ncc(-c4ccc(S(=O)(=O)N5CCN(C)CC5)cc4)cc23)cc1OC
COc1ccc(-c2c[nH]c3ncc(-c4ccc(CN5CCN(C)CC5)cc4)cc23)cc1OC
COc1ccc(-c2c[nH]c3ncc(-c4ccc(CN5CCOCC5)cc4)cc23)cc1OC
Cc1cc(-c2c[nH]c3ncc(-c4ccc(C5CCN(C6CN(c7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)C6)CC5)cc4)nc23)ccc1C(=O)N(C)C
Cc1cc(-c2c[nH]c3ncc(-c4cc(C)c5c(c4)CN(C)CC5)nc23)ccc1C(=O)N(C)C
Cc1ccc(C(=O)Nc2cccc(C(F)(F)F)c2)cc1Nc1nc(-c2cccnc2)nc2nn(C)cc12
Cc1ccc(C(=O)Nc2cccc(C(F)(F)F)c2)cc1Nc1nc(-c2cccnc2)nc2c1cnn2C
C[C@H]1CC(=O)Nc2cc(C(=O)NCCC3CC3)ccc2N1C(=O)N1CC2CC2C1
Cc1cn(CCN2CCN(CC2)c2ccccc2-c2cc(cc(c2)C(=O)NCCCN2CCCC2)C#N)c2ccccc12
COc1cc(ccc1Nc1nc2ccc(cn2n1)-c1ccc(NC(=O)[C@H](C)c2ccc(F)cc2)cc1)S(C)(=O)=O |r|