Affinity DataKi: 32nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 41nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 41nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 49nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 57nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 61nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 68nMAssay Description:Binding affinity of compound towards Factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 101nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 116nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 124nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 125nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 128nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 140nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 141nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 155nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 162nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 185nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 197nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 240nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 246nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 290nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 310nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 368nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 373nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 497nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: >2.00E+4nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: >2.00E+4nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-beta(Homo sapiens (Human))
Sanofi-Aventis Research And Development
Curated by ChEMBL
Sanofi-Aventis Research And Development
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of HSP90beta in human SKBR3 cells assessed as down regulation of HER2 expression levels after 24 hrs by FACS analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 68nMAssay Description:In vitro inhibitory activity against Factor XaMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-beta(Homo sapiens (Human))
Sanofi-Aventis Research And Development
Curated by ChEMBL
Sanofi-Aventis Research And Development
Curated by ChEMBL
Affinity DataIC50: 900nMAssay Description:Inhibition of HSP90beta in human SKBR3 cells assessed as down regulation of HER2 expression levels after 24 hrs by FACS analysisMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-beta(Homo sapiens (Human))
Sanofi-Aventis Research And Development
Curated by ChEMBL
Sanofi-Aventis Research And Development
Curated by ChEMBL
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of HSP90beta in human SKBR3 cells assessed as down regulation of HER2 expression levels after 24 hrs by FACS analysisMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-beta(Homo sapiens (Human))
Sanofi-Aventis Research And Development
Curated by ChEMBL
Sanofi-Aventis Research And Development
Curated by ChEMBL
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of HSP90beta in human SKBR3 cells assessed as down regulation of HER2 expression levels after 24 hrs by FACS analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 3.69E+3nMAssay Description:Inhibitory concentration of the compound against alpha tryptase was determinedMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-beta(Homo sapiens (Human))
Sanofi-Aventis Research And Development
Curated by ChEMBL
Sanofi-Aventis Research And Development
Curated by ChEMBL
Affinity DataIC50: 7.60E+3nMAssay Description:Inhibition of human Hsp90beta after overnight incubation by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-beta(Homo sapiens (Human))
Sanofi-Aventis Research And Development
Curated by ChEMBL
Sanofi-Aventis Research And Development
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of HSP90beta in human SKBR3 cells assessed as down regulation of HER2 expression levels after 24 hrs by FACS analysisMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-beta(Homo sapiens (Human))
Sanofi-Aventis Research And Development
Curated by ChEMBL
Sanofi-Aventis Research And Development
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of HSP90beta in human SKBR3 cells assessed as down regulation of HER2 expression levels after 24 hrs by FACS analysisMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-beta(Homo sapiens (Human))
Sanofi-Aventis Research And Development
Curated by ChEMBL
Sanofi-Aventis Research And Development
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of HSP90beta in human SKBR3 cells assessed as down regulation of HER2 expression levels after 24 hrs by FACS analysisMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-beta(Homo sapiens (Human))
Sanofi-Aventis Research And Development
Curated by ChEMBL
Sanofi-Aventis Research And Development
Curated by ChEMBL
Affinity DataKd: 0.350nMAssay Description:Binding affinity to human Hsp90beta after overnight incubation by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-beta(Homo sapiens (Human))
Sanofi-Aventis Research And Development
Curated by ChEMBL
Sanofi-Aventis Research And Development
Curated by ChEMBL
Affinity DataKd: 7.30nMAssay Description:Binding affinity to human Hsp90beta after overnight incubation by fluorescence polarization assayMore data for this Ligand-Target Pair