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Found 245 with Last Name = 'jackson' and Initial = 'dy'
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50060228((5S,8R,13R,15aS)-8-{[(2R,3S)-1-Acetyl-3-(4-hydroxy...)
Affinity DataIC50:  0.5nMAssay Description:Inhibition of purified alpha-4 beta-1 binding to VCAM-1 was determined in an ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50060185((6S,9R,14R,16aS)-9-[(S)-2-Acetylamino-3-(4-hydroxy...)
Affinity DataIC50:  1nMAssay Description:Inhibition of purified alpha-4 beta-1 binding to VCAM-1 was determined in an ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50119092(4-Methyl-piperazine-1-carboxylic acid 4-[(S)-2-car...)
Affinity DataIC50:  1.10nMAssay Description:Inhibitory activity against alpha4-beta1 integrin (vascular cell adhesion molecule) in ELISA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50108219((5S,8R,13R)-8-[(S)-2-Acetylamino-3-(4-hydroxy-phen...)
Affinity DataIC50:  2nMAssay Description:Inhibitory activity against alpha4-beta1 integrin (vascular cell adhesion molecule) in ELISA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50060226((5S,8R,13R,15aS)-8-[(S)-2-Acetylamino-3-(4-hydroxy...)
Affinity DataIC50:  2nMAssay Description:Inhibition of purified alpha-4 beta-1 binding to VCAM-1 was determined in an ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50060183((5S,8R,13R,15aS)-8-[(S)-2-Acetylamino-3-(4-hydroxy...)
Affinity DataIC50:  3nMAssay Description:Inhibition of purified alpha-4 beta-1 binding to VCAM-1 was determined in an ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50108219((5S,8R,13R)-8-[(S)-2-Acetylamino-3-(4-hydroxy-phen...)
Affinity DataIC50:  3nMAssay Description:Inhibition of purified alpha-4 beta-1 binding to VCAM-1 was determined in an ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50060230((5S,8R,13R,15aS)-8-{[(2R,3R)-1-Acetyl-3-(4-hydroxy...)
Affinity DataIC50:  4nMAssay Description:Inhibition of purified alpha-4 beta-1 binding to VCAM-1 was determined in an ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50060233((5S,8R,13R,15aS)-8-[(S)-2-Acetylamino-3-(4-hydroxy...)
Affinity DataIC50:  4nMAssay Description:Inhibition of purified alpha-4 beta-1 binding to VCAM-1 was determined in an ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50060168((5S,8R,13R,15aS)-8-[(S)-2-Amino-3-(4-hydroxy-pheny...)
Affinity DataIC50:  4nMAssay Description:Inhibition of purified alpha-4 beta-1 binding to VCAM-1 was determined in an ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50060179((5S,8R,13R,15aS)-8-[(S)-2-Amino-3-(4-hydroxy-3-iod...)
Affinity DataIC50:  4nMAssay Description:Inhibition of purified alpha-4 beta-1 binding to VCAM-1 was determined in an ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50422231(CHEMBL1790844)
Affinity DataIC50:  5nMAssay Description:Inhibition of purified alpha-4 beta-1 binding to VCAM-1 was determined in an ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50060203((5S,8R,13R,15aS)-8-[(S)-2-Amino-3-(4-hydroxy-pheny...)
Affinity DataIC50:  5nMAssay Description:Inhibition of purified alpha-4 beta-1 binding to VCAM-1 was determined in an ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50060173((5S,8R,13R,15aS)-8-[(S)-2-Amino-3-(4-hydroxy-pheny...)
Affinity DataIC50:  5nMAssay Description:Inhibition of purified alpha-4 beta-1 binding to VCAM-1 was determined in an ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50060196((5S,8R,13R,15aS)-8-[(S)-2-Amino-3-(3-chloro-4-hydr...)
Affinity DataIC50:  7nMAssay Description:Inhibition of purified alpha-4 beta-1 binding to VCAM-1 was determined in an ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50060228((5S,8R,13R,15aS)-8-{[(2R,3S)-1-Acetyl-3-(4-hydroxy...)
Affinity DataIC50:  8nMAssay Description:Inhibition of fluorescently labeled alpha4-beta1 positive Ramos cells binding to immobilized VCAM-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50060202((4R,9R)-4-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propio...)
Affinity DataIC50:  8nMAssay Description:Inhibition of alpha4-beta1 binding to VCAM-1 in ELISA.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50060193((5S,8R,13R,15aS)-8-[(S)-2-Amino-3-(3-fluoro-4-hydr...)
Affinity DataIC50:  8nMAssay Description:Inhibition of purified alpha-4 beta-1 binding to VCAM-1 was determined in an ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50116502(CHEMBL407428 | [22-Amino-4-carbamoyl-19-(4-hydroxy...)
Affinity DataIC50:  9nMAssay Description:Inhibitory concentration affording 50% inhibition of alpha4-beta1 integrin binding to VCAM-1, using ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50119089((S)-2-(2-Chloro-benzoylamino)-3-(4-dimethylcarbamo...)
Affinity DataIC50:  9.30nMAssay Description:Inhibitory activity against alpha4-beta1 integrin (vascular cell adhesion molecule) in ELISA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-7(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50108219((5S,8R,13R)-8-[(S)-2-Acetylamino-3-(4-hydroxy-phen...)
Affinity DataIC50:  10nMAssay Description:Inhibitory activity against alpha4-beta7/ MAdCAM integrin (mucosal addressin cell adhesion molecule) in ELISA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-7(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50119096((S)-2-(2-Chloro-benzoylamino)-3-[2'-(4-methyl-pipe...)
Affinity DataIC50:  10nMAssay Description:Inhibitory activity against alpha4-beta7/ MAdCAM integrin (mucosal addressin cell adhesion molecule) in ELISA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-7(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50119093((S)-2-(2-Chloro-benzoylamino)-3-(2'-dimethylaminom...)
Affinity DataIC50:  11nMAssay Description:Inhibitory activity against alpha4-beta7/ MAdCAM integrin (mucosal addressin cell adhesion molecule) in ELISA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-7(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50119092(4-Methyl-piperazine-1-carboxylic acid 4-[(S)-2-car...)
Affinity DataIC50:  12nMAssay Description:Inhibitory activity against alpha4-beta7/ MAdCAM integrin (mucosal addressin cell adhesion molecule) in ELISA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50060219((5S,8R,13R,15aS)-5-Hydroxymethyl-8-[3-(4-hydroxy-p...)
Affinity DataIC50:  13nMAssay Description:Inhibition of purified alpha-4 beta-1 binding to VCAM-1 was determined in an ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50119093((S)-2-(2-Chloro-benzoylamino)-3-(2'-dimethylaminom...)
Affinity DataIC50:  17nMAssay Description:Inhibitory activity against alpha4-beta1 integrin (vascular cell adhesion molecule) in ELISA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50119083((S)-2-(2-Chloro-benzoylamino)-3-(4-phenethylcarbam...)
Affinity DataIC50:  18nMAssay Description:Inhibitory activity against alpha4-beta1 integrin (vascular cell adhesion molecule) in ELISA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50060185((6S,9R,14R,16aS)-9-[(S)-2-Acetylamino-3-(4-hydroxy...)
Affinity DataIC50:  20nMAssay Description:Inhibition of fluorescently labeled alpha4-beta1 positive Ramos cells binding to immobilized VCAM-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50060181((1S,4R,9R,12S)-9-[(S)-2-Amino-3-(4-hydroxy-phenyl)...)
Affinity DataIC50:  20nMAssay Description:Inhibition of purified alpha-4 beta-1 binding to VCAM-1 was determined in an ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50119085((S)-2-(2-Chloro-benzoylamino)-3-(4-propylcarbamoyl...)
Affinity DataIC50:  20nMAssay Description:Inhibitory activity against alpha4-beta7/ MAdCAM integrin (mucosal addressin cell adhesion molecule) in ELISA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-7(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50119089((S)-2-(2-Chloro-benzoylamino)-3-(4-dimethylcarbamo...)
Affinity DataIC50:  22nMAssay Description:Inhibitory activity against alpha4-beta7/ MAdCAM integrin (mucosal addressin cell adhesion molecule) in ELISA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50060175((4R,7S,10S,13R)-13-[(S)-2-Amino-3-(4-hydroxy-pheny...)
Affinity DataIC50:  23nMAssay Description:Inhibition of purified alpha-4 beta-1 binding to VCAM-1 was determined in an ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-7(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50119087((S)-2-(2-Chloro-benzoylamino)-3-(2'-{[2-(4-hydroxy...)
Affinity DataIC50:  25nMAssay Description:Inhibitory activity against alpha4-beta7/ MAdCAM integrin (mucosal addressin cell adhesion molecule) in ELISA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50119087((S)-2-(2-Chloro-benzoylamino)-3-(2'-{[2-(4-hydroxy...)
Affinity DataIC50:  25nMAssay Description:Inhibitory activity against alpha4-beta1 integrin (vascular cell adhesion molecule) in ELISA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50119096((S)-2-(2-Chloro-benzoylamino)-3-[2'-(4-methyl-pipe...)
Affinity DataIC50:  25nMAssay Description:Inhibitory activity against alpha4-beta1 integrin (vascular cell adhesion molecule) in ELISA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-7(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50116474(4-(2-{[22-Amino-13-carboxymethyl-19-(3-guanidino-p...)
Affinity DataIC50:  30nMAssay Description:Ability to block the alpha4-beta7 integrin-MAdCAM-1 binding interaction using a protein ELISA formatMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50060213((3R,8R)-3-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propio...)
Affinity DataIC50:  31nMAssay Description:Inhibition of purified alpha-4 beta-1 binding to VCAM-1 was determined in an ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50060227((4R,7S,10S,13R)-13-[(S)-2-Amino-3-(4-hydroxy-pheny...)
Affinity DataIC50:  34nMAssay Description:Inhibition of purified alpha-4 beta-1 binding to VCAM-1 was determined in an ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50119097((S)-3-(4-Allylcarbamoyloxy-phenyl)-2-(2-chloro-ben...)
Affinity DataIC50:  35nMAssay Description:Inhibitory activity against alpha4-beta1 integrin (vascular cell adhesion molecule) in ELISA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50060236((4R,12R)-12-[(S)-2-Amino-3-(4-hydroxy-phenyl)-prop...)
Affinity DataIC50:  38nMAssay Description:Inhibition of purified alpha-4 beta-1 binding to VCAM-1 was determined in an ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50060211(8-(2-{2-[2-(2-Amino-3-phenyl-propionylamino)-3-mer...)
Affinity DataIC50:  40nMAssay Description:Inhibition of purified alpha-4 beta-1 binding to VCAM-1 was determined in an ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-7(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50119085((S)-2-(2-Chloro-benzoylamino)-3-(4-propylcarbamoyl...)
Affinity DataIC50:  40nMAssay Description:Inhibitory activity against alpha4-beta1 integrin (vascular cell adhesion molecule) in ELISA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50060239((5S,8R,13R,15aS)-8-[(S)-2-Amino-3-(4-hydroxy-pheny...)
Affinity DataIC50:  40nMAssay Description:Inhibition of purified alpha-4 beta-1 binding to VCAM-1 was determined in an ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50060197((5S,8R,13R,15aS)-8-{(S)-2-[(S)-2-Amino-3-(4-hydrox...)
Affinity DataIC50:  40nMAssay Description:Inhibition of purified alpha-4 beta-1 binding to VCAM-1 was determined in an ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50060172((4R,11R)-11-[(S)-2-Amino-3-(4-hydroxy-phenyl)-prop...)
Affinity DataIC50:  47nMAssay Description:Inhibition of purified alpha-4 beta-1 binding to VCAM-1 was determined in an ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50119088((S)-2-(2-Chloro-benzoylamino)-3-(3'-{[2-(4-hydroxy...)
Affinity DataIC50:  48nMAssay Description:Inhibitory activity against alpha4-beta1 integrin (vascular cell adhesion molecule) in ELISA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-7(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50119090((S)-2-(2-Chloro-benzoylamino)-3-[2'-(phenethylamin...)
Affinity DataIC50:  48nMAssay Description:Inhibitory activity against alpha4-beta7/ MAdCAM integrin (mucosal addressin cell adhesion molecule) in ELISA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-7(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50119095((S)-2-(2-Chloro-benzoylamino)-3-{2'-[(3-methyl-but...)
Affinity DataIC50:  50nMAssay Description:Inhibitory activity against alpha4-beta7/ MAdCAM integrin (mucosal addressin cell adhesion molecule) in ELISA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50060209((5S,8R,13R,15aS)-8-{(S)-2-[(S)-2-Amino-3-(4-hydrox...)
Affinity DataIC50:  50nMAssay Description:Inhibition of purified alpha-4 beta-1 binding to VCAM-1 was determined in an ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50116479(CHEMBL331024 | [22-Amino-19-benzyl-4-carbamoyl-10-...)
Affinity DataIC50:  50nMAssay Description:Inhibitory concentration affording 50% inhibition of alpha4-beta1 integrin binding to VCAM-1, using ELISA assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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