Affinity DataKi: 1.40nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cells incubated for 90 mins by liquid scintillation spectrophotometry relative ...More data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in CHO cells incubated for 90 mins by liquid scintillation spectrophotometry relative ...More data for this Ligand-Target Pair
Affinity DataKi: 2.90nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cells incubated for 90 mins by liquid scintillation spectrophotometry relative ...More data for this Ligand-Target Pair
Affinity DataKi: 4.90nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cells incubated for 90 mins by liquid scintillation spectrophotometry relative ...More data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in CHO cells incubated for 90 mins by liquid scintillation spectrophotometry relative ...More data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cells incubated for 90 mins by liquid scintillation spectrophotometry relative ...More data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cells incubated for 90 mins by liquid scintillation spectrophotometry relative ...More data for this Ligand-Target Pair
Affinity DataKi: 39nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in CHO cells incubated for 90 mins by liquid scintillation spectrophotometry relative ...More data for this Ligand-Target Pair
Affinity DataKi: 63nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cells incubated for 90 mins by liquid scintillation spectrophotometry relative ...More data for this Ligand-Target Pair
Affinity DataKi: 130nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cells incubated for 90 mins by liquid scintillation spectrophotometry relative ...More data for this Ligand-Target Pair
Affinity DataKi: 152nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in CHO cells incubated for 90 mins by liquid scintillation spectrophotometry relative ...More data for this Ligand-Target Pair
Affinity DataKi: 325nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in CHO cells incubated for 90 mins by liquid scintillation spectrophotometry relative ...More data for this Ligand-Target Pair
Affinity DataKi: 1.90E+3nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in CHO cells incubated for 90 mins by liquid scintillation spectrophotometry relative ...More data for this Ligand-Target Pair
Affinity DataKi: 2.56E+3nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in CHO cells incubated for 90 mins by liquid scintillation spectrophotometry relative ...More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase F(Homo sapiens (Human))
University of Utah
Curated by ChEMBL
University of Utah
Curated by ChEMBL
Affinity DataKi: 1.30E+5nMAssay Description:Non-covalent inhibition of LAR (unknown origin) using DiFMUP as substrate incubated for 15 to 120 mins followed by substrate addition at pH 6.5 by st...More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase F(Homo sapiens (Human))
University of Utah
Curated by ChEMBL
University of Utah
Curated by ChEMBL
Affinity DataKi: 1.30E+5nMAssay Description:Non-covalent inhibition of LAR (unknown origin) using DiFMUP as substrate incubated for 15 to 120 mins followed by substrate addition at pH 6.5 by st...More data for this Ligand-Target Pair
Affinity DataIC50: 1.80E+3nMAssay Description:Antagonist activity at human CB2 receptor expressed in CHO cell membrane assessed as reduction in CP55940-induced [35S]GTPgammaS binding by liquid sc...More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase F(Homo sapiens (Human))
University of Utah
Curated by ChEMBL
University of Utah
Curated by ChEMBL
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of LAR (unknown origin) using DiFMUP as substrate incubated for 30 mins followed by substrate addition at pH 6.5 by standard phosphatase a...More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase F(Homo sapiens (Human))
University of Utah
Curated by ChEMBL
University of Utah
Curated by ChEMBL
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of LAR (unknown origin) using DiFMUP as substrate incubated for 30 mins followed by substrate addition at pH 6.5 by standard phosphatase a...More data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
West Virginia University
Curated by ChEMBL
West Virginia University
Curated by ChEMBL
Affinity DataIC50: 4.16E+3nMAssay Description:Inhibition of recombinant human LSD1 using ARTK(diMethyl)QTARKSTGGKAPRKQLAPRKQLA as substrate measured after 30 mins by ADHP/horseradish peroxidase c...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
West Virginia University
Curated by ChEMBL
West Virginia University
Curated by ChEMBL
Affinity DataIC50: 7.91E+3nMAssay Description:Inhibition of MAOA (unknown origin) using kynuramine as substrateMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase C(Homo sapiens (Human))
University of Utah
Curated by ChEMBL
University of Utah
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CD45 (unknown origin) using DiFMUP as substrate incubated for 30 mins followed by substrate addition at pH 6.5 by standard phosphatase ...More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase C(Homo sapiens (Human))
University of Utah
Curated by ChEMBL
University of Utah
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CD45 (unknown origin) using DiFMUP as substrate incubated for 30 mins followed by substrate addition at pH 6.5 by standard phosphatase ...More data for this Ligand-Target Pair
Affinity DataIC50: 1.22E+4nMAssay Description:Inhibition of recombinant human Ero1Lalpha C104A/C131A/C166A triple mutant (22 to 468 residues) expressed in Escherichia coli BL21(DE3)-RIL measured ...More data for this Ligand-Target Pair
Affinity DataIC50: 1.27E+4nMAssay Description:Inhibition of recombinant human Ero1Lalpha C104A/C131A/C166A triple mutant (22 to 468 residues) expressed in Escherichia coli BL21(DE3)-RIL measured ...More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase mu(Homo sapiens (Human))
University of Utah
Curated by ChEMBL
University of Utah
Curated by ChEMBL
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of PTPmu (unknown origin) using DiFMUP as substrate incubated for 30 mins followed by substrate addition at pH 6.5 by standard phosphatase...More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase mu(Homo sapiens (Human))
University of Utah
Curated by ChEMBL
University of Utah
Curated by ChEMBL
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of PTPmu (unknown origin) using DiFMUP as substrate incubated for 30 mins followed by substrate addition at pH 6.5 by standard phosphatase...More data for this Ligand-Target Pair
Affinity DataIC50: 2.21E+4nMAssay Description:Inhibition of recombinant human Ero1Lalpha C104A/C131A/C166A triple mutant (22 to 468 residues) expressed in Escherichia coli BL21(DE3)-RIL using hum...More data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 11(Homo sapiens (Human))
University of Utah
Curated by ChEMBL
University of Utah
Curated by ChEMBL
Affinity DataIC50: 2.90E+4nMAssay Description:Inhibition of SHP2 (unknown origin) using DiFMUP as substrate incubated for 30 mins followed by substrate addition at pH 6.5 by standard phosphatase ...More data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 11(Homo sapiens (Human))
University of Utah
Curated by ChEMBL
University of Utah
Curated by ChEMBL
Affinity DataIC50: 2.90E+4nMAssay Description:Inhibition of SHP2 (unknown origin) using DiFMUP as substrate incubated for 30 mins followed by substrate addition at pH 6.5 by standard phosphatase ...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
West Virginia University
Curated by ChEMBL
West Virginia University
Curated by ChEMBL
Affinity DataIC50: 3.06E+4nMAssay Description:Inhibition of MAOB (unknown origin) using kynuramine as substrateMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase F(Homo sapiens (Human))
University of Utah
Curated by ChEMBL
University of Utah
Curated by ChEMBL
Affinity DataIC50: 5.50E+4nMAssay Description:Inhibition of LAR (unknown origin) using DiFMUP as substrate incubated for 30 mins followed by substrate addition at pH 6.5 by standard phosphatase a...More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase F(Homo sapiens (Human))
University of Utah
Curated by ChEMBL
University of Utah
Curated by ChEMBL
Affinity DataIC50: 5.50E+4nMAssay Description:Inhibition of LAR (unknown origin) using DiFMUP as substrate incubated for 30 mins followed by substrate addition at pH 6.5 by standard phosphatase a...More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase epsilon(Homo sapiens (Human))
University of Utah
Curated by ChEMBL
University of Utah
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of PTPep (unknown origin) using DiFMUP as substrate incubated for 30 mins followed by substrate addition at pH 6.5 by standard phosphatase...More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase C(Homo sapiens (Human))
University of Utah
Curated by ChEMBL
University of Utah
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of CD45 (unknown origin) using DiFMUP as substrate incubated for 30 mins followed by substrate addition at pH 6.5 by standard phosphatase ...More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
University of Utah
Curated by ChEMBL
University of Utah
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of LMWPTP (unknown origin) using DiFMUP as substrate incubated for 30 mins followed by substrate addition at pH 6.5 by standard phosphatas...More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
University of Utah
Curated by ChEMBL
University of Utah
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of LMWPTP (unknown origin) using DiFMUP as substrate incubated for 30 mins followed by substrate addition at pH 6.5 by standard phosphatas...More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase C(Homo sapiens (Human))
University of Utah
Curated by ChEMBL
University of Utah
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of CD45 (unknown origin) using DiFMUP as substrate incubated for 30 mins followed by substrate addition at pH 6.5 by standard phosphatase ...More data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 7(Homo sapiens (Human))
University of Utah
Curated by ChEMBL
University of Utah
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of HePTP (unknown origin) using DiFMUP as substrate incubated for 30 mins followed by substrate addition at pH 6.5 by standard phosphatase...More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 3(Homo sapiens (Human))
University of Utah
Curated by ChEMBL
University of Utah
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of VHR (unknown origin) using DiFMUP as substrate incubated for 30 mins followed by substrate addition at pH 6.5 by standard phosphatase a...More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase epsilon(Homo sapiens (Human))
University of Utah
Curated by ChEMBL
University of Utah
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of PTPep (unknown origin) using DiFMUP as substrate incubated for 30 mins followed by substrate addition at pH 6.5 by standard phosphatase...More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase epsilon(Homo sapiens (Human))
University of Utah
Curated by ChEMBL
University of Utah
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of PTPep (unknown origin) using DiFMUP as substrate incubated for 30 mins followed by substrate addition at pH 6.5 by standard phosphatase...More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 3(Homo sapiens (Human))
University of Utah
Curated by ChEMBL
University of Utah
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of VHR (unknown origin) using DiFMUP as substrate incubated for 30 mins followed by substrate addition at pH 6.5 by standard phosphatase a...More data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 2(Homo sapiens (Human))
University of Utah
Curated by ChEMBL
University of Utah
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of TCPTP (unknown origin) using DiFMUP as substrate incubated for 30 mins followed by substrate addition at pH 6.5 by standard phosphatase...More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 3(Homo sapiens (Human))
University of Utah
Curated by ChEMBL
University of Utah
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of VHR (unknown origin) using DiFMUP as substrate incubated for 30 mins followed by substrate addition at pH 6.5 by standard phosphatase a...More data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 2(Homo sapiens (Human))
University of Utah
Curated by ChEMBL
University of Utah
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of TCPTP (unknown origin) using DiFMUP as substrate incubated for 30 mins followed by substrate addition at pH 6.5 by standard phosphatase...More data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 11(Homo sapiens (Human))
University of Utah
Curated by ChEMBL
University of Utah
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of SHP2 (unknown origin) using DiFMUP as substrate incubated for 30 mins followed by substrate addition at pH 6.5 by standard phosphatase ...More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase mu(Homo sapiens (Human))
University of Utah
Curated by ChEMBL
University of Utah
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of PTPmu (unknown origin) using DiFMUP as substrate incubated for 30 mins followed by substrate addition at pH 6.5 by standard phosphatase...More data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 7(Homo sapiens (Human))
University of Utah
Curated by ChEMBL
University of Utah
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of HePTP (unknown origin) using DiFMUP as substrate incubated for 30 mins followed by substrate addition at pH 6.5 by standard phosphatase...More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein phosphatase epsilon(Homo sapiens (Human))
University of Utah
Curated by ChEMBL
University of Utah
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of PTPep (unknown origin) using DiFMUP as substrate incubated for 30 mins followed by substrate addition at pH 6.5 by standard phosphatase...More data for this Ligand-Target Pair