TargetType-1 angiotensin II receptor A(RAT)
Parke-Davis Pharmaceutical Research
Curated by PDSP Ki Database
Parke-Davis Pharmaceutical Research
Curated by PDSP Ki Database
TargetType-2 angiotensin II receptor(RAT)
Parke-Davis Pharmaceutical Research
Curated by PDSP Ki Database
Parke-Davis Pharmaceutical Research
Curated by PDSP Ki Database
TargetType-1 angiotensin II receptor A(RAT)
Parke-Davis Pharmaceutical Research
Curated by PDSP Ki Database
Parke-Davis Pharmaceutical Research
Curated by PDSP Ki Database
TargetType-1 angiotensin II receptor A(RAT)
Parke-Davis Pharmaceutical Research
Curated by PDSP Ki Database
Parke-Davis Pharmaceutical Research
Curated by PDSP Ki Database
TargetType-1 angiotensin II receptor A(RAT)
Parke-Davis Pharmaceutical Research
Curated by PDSP Ki Database
Parke-Davis Pharmaceutical Research
Curated by PDSP Ki Database
Affinity DataKi: 82nMAssay Description:Compound was tested for inhibitory activity against N-His (D381E) Interleukin -1 beta converting enzyme (resynthesized compound)More data for this Ligand-Target Pair
Affinity DataKi: 113nMAssay Description:Compound was tested for inhibitory activity against N-His (D381E) Interleukin -1 beta converting enzyme (resynthesized compound)More data for this Ligand-Target Pair
Affinity DataKi: 4.50E+3nMAssay Description:Compound was tested for binding affinity against N-His (D381E) Interleukin -1 beta converting enzymeMore data for this Ligand-Target Pair
TargetType-2 angiotensin II receptor(RAT)
Parke-Davis Pharmaceutical Research
Curated by PDSP Ki Database
Parke-Davis Pharmaceutical Research
Curated by PDSP Ki Database
TargetType-2 angiotensin II receptor(RAT)
Parke-Davis Pharmaceutical Research
Curated by PDSP Ki Database
Parke-Davis Pharmaceutical Research
Curated by PDSP Ki Database
TargetType-2 angiotensin II receptor(RAT)
Parke-Davis Pharmaceutical Research
Curated by PDSP Ki Database
Parke-Davis Pharmaceutical Research
Curated by PDSP Ki Database
TargetType-2 angiotensin II receptor(RAT)
Parke-Davis Pharmaceutical Research
Curated by PDSP Ki Database
Parke-Davis Pharmaceutical Research
Curated by PDSP Ki Database
TargetType-1 angiotensin II receptor A/Type-1 angiotensin II receptor B/Type-2 angiotensin II receptor(RAT)
Warner-Lambert
Curated by ChEMBL
Warner-Lambert
Curated by ChEMBL
Affinity DataIC50: 0.100nMAssay Description:Binding affinity for rat brain Angiotensin II receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:Inhibitory concentration against renin monkey plasmaMore data for this Ligand-Target Pair
Affinity DataIC50: 0.180nMAssay Description:Inhibition of monkey plasma reninMore data for this Ligand-Target Pair
Affinity DataIC50: 0.190nMAssay Description:Inhibition of monkey plasma reninMore data for this Ligand-Target Pair
Affinity DataIC50: 0.190nMAssay Description:Inhibition of monkey plasma reninMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Inhibition of monkey plasma reninMore data for this Ligand-Target Pair
Affinity DataIC50: 0.230nMAssay Description:Inhibition of monkey plasma reninMore data for this Ligand-Target Pair
Affinity DataIC50: 0.280nMAssay Description:Inhibitory concentration against renin monkey plasmaMore data for this Ligand-Target Pair
Affinity DataIC50: 0.280nMAssay Description:Inhibitory concentration against human reninMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/Type-1 angiotensin II receptor B/Type-2 angiotensin II receptor(RAT)
Warner-Lambert
Curated by ChEMBL
Warner-Lambert
Curated by ChEMBL
Affinity DataIC50: 0.350nMAssay Description:Binding affinity against Angiotensin II receptor, from rat adrenal glandMore data for this Ligand-Target Pair
Affinity DataIC50: 0.400nMAssay Description:Inhibitory concentration against renin monkey plasmaMore data for this Ligand-Target Pair
Affinity DataIC50: 0.410nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:Inhibitory activity against monkey plasma renin.More data for this Ligand-Target Pair
Affinity DataIC50: 0.580nMAssay Description:Inhibitory activity against angiotensin II type 2 (AT2) receptor in rabbit uterine membranes.More data for this Ligand-Target Pair
Affinity DataIC50: 0.580nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.680nMAssay Description:Inhibition of monkey plasma reninMore data for this Ligand-Target Pair
Affinity DataIC50: 0.75nMAssay Description:Inhibition of monkey plasma reninMore data for this Ligand-Target Pair
Affinity DataIC50: 0.790nMAssay Description:Inhibition of monkey plasma reninMore data for this Ligand-Target Pair
Affinity DataIC50: 0.800nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.820nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.830nMAssay Description:Inhibition of monkey plasma reninMore data for this Ligand-Target Pair
Affinity DataIC50: 0.840nMAssay Description:Inhibitory activity against angiotensin II type 2 (AT2) receptor in rabbit uterine membranes.More data for this Ligand-Target Pair
Affinity DataIC50: 0.840nMAssay Description:Inhibitory activity against angiotensin II type 2 (AT2) receptor in rabbit uterine membranes.More data for this Ligand-Target Pair
Affinity DataIC50: 0.890nMAssay Description:Inhibitory activity against angiotensin II type 2 (AT2) receptor in rabbit uterine membranes.More data for this Ligand-Target Pair
Affinity DataIC50: 0.900nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.950nMAssay Description:Inhibition of monkey plasma reninMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10nMAssay Description:Inhibitory activity against angiotensin II type 2 (AT2) receptor in rabbit uterine membranes.More data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/Type-1 angiotensin II receptor B/Type-2 angiotensin II receptor(RAT)
Warner-Lambert
Curated by ChEMBL
Warner-Lambert
Curated by ChEMBL
Affinity DataIC50: 1.30nMAssay Description:Binding affinity against Angiotensin II receptor, from rat adrenal glandMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40nMAssay Description:Inhibition of monkey plasma reninMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/Type-1 angiotensin II receptor B/Type-2 angiotensin II receptor(RAT)
Warner-Lambert
Curated by ChEMBL
Warner-Lambert
Curated by ChEMBL
Affinity DataIC50: 1.60nMAssay Description:Binding affinity against Angiotensin II receptor, from rat adrenal glandMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60nMAssay Description:Tested for inhibitory concentration against AT1 receptor binding affinity in rat liverMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70nMAssay Description:Inhibitory concentration against renin monkey plasmaMore data for this Ligand-Target Pair
Affinity DataIC50: 1.80nMAssay Description:Inhibitory concentration against [125I]angiotensin II(AII) induced contraction in rabbit aorta by 50%More data for this Ligand-Target Pair