Report error Found 61 with Last Name = 'tradtrantip' and Initial = 'l'
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibition of wild type human CFTR chloride conductance expressed in forskolin-stimulated rat FRT cells by short-circuit current analysis in presence...More data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Inhibition of human wild-type CFTR expressed in FRT cells assessed as inhibition of forskolin-induced short-circuit current by voltage clamp electrop...More data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition of human wild-type CFTR expressed in FRT cells assessed as inhibition of forskolin-induced short-circuit current by voltage clamp electrop...More data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition of human wild-type CFTR expressed in FRT cells assessed as inhibition of forskolin-induced short-circuit current by voltage clamp electrop...More data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition of human wild-type CFTR expressed in FRT cells assessed as inhibition of forskolin-induced short-circuit current by voltage clamp electrop...More data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of human wild-type CFTR expressed in FRT cells coexpressing YFP-H148Q assessed as inhibition of cAMP agonist-induced iodide influx after 4...More data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of human wild-type CFTR expressed in FRT cells assessed as inhibition of forskolin-induced short-circuit current by voltage clamp electrop...More data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of human wild-type CFTR expressed in FRT cells coexpressing YFP-H148Q assessed as inhibition of cAMP agonist-induced iodide influx after 4...More data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 80nMAssay Description:Inhibition of human wild-type CFTR expressed in FRT cells coexpressing YFP-H148Q assessed as inhibition of cAMP agonist-induced iodide influx after 4...More data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 90nMAssay Description:Inhibition of human CFTR expressed in rat FRT cells assessed as inhibition of CPT-cAMP-induced apical membrane current in presence of transepithelial...More data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 90nMAssay Description:Inhibition of human wild-type CFTR expressed in FRT cells assessed as inhibition of forskolin-induced short-circuit current by voltage clamp electrop...More data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 90nMAssay Description:Inhibition of human wild-type CFTR expressed in FRT cells coexpressing YFP-H148Q assessed as inhibition of cAMP agonist-induced iodide influx after 4...More data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of human wild-type CFTR expressed in FRT cells assessed as inhibition of forskolin-induced short-circuit current by voltage clamp electrop...More data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of human wild-type CFTR expressed in FRT cells assessed as inhibition of forskolin-induced short-circuit current by voltage clamp electrop...More data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of human wild-type CFTR expressed in FRT cells coexpressing YFP-H148Q assessed as inhibition of cAMP agonist-induced iodide influx after 4...More data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:Inhibition of human wild-type CFTR expressed in FRT cells coexpressing YFP-H148Q assessed as inhibition of cAMP agonist-induced iodide influx after 4...More data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 150nMAssay Description:Inhibition of human wild-type CFTR expressed in FRT cells coexpressing YFP-H148Q assessed as inhibition of cAMP agonist-induced iodide influx after 4...More data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 150nMAssay Description:Inhibition of human wild-type CFTR expressed in FRT cells coexpressing YFP-H148Q assessed as inhibition of cAMP agonist-induced iodide influx after 4...More data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 170nMAssay Description:Inhibition of human wild-type CFTR expressed in FRT cells coexpressing YFP-H148Q assessed as inhibition of cAMP agonist-induced iodide influx after 4...More data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 170nMAssay Description:Inhibition of human wild-type CFTR expressed in FRT cells coexpressing YFP-H148Q assessed as inhibition of cAMP agonist-induced iodide influx after 4...More data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 170nMAssay Description:Inhibition of human wild-type CFTR expressed in FRT cells coexpressing YFP-H148Q assessed as inhibition of cAMP agonist-induced iodide influx after 4...More data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of human wild-type CFTR expressed in FRT cells coexpressing YFP-H148Q assessed as inhibition of cAMP agonist-induced iodide influx after 4...More data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 250nMAssay Description:Inhibition of human wild-type CFTR expressed in FRT cells coexpressing YFP-H148Q assessed as inhibition of cAMP agonist-induced iodide influx after 4...More data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inhibition of human wild-type CFTR expressed in FRT cells coexpressing YFP-H148Q assessed as inhibition of cAMP agonist-induced iodide influx after 4...More data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 350nMAssay Description:Inhibition of human wild-type CFTR expressed in FRT cells coexpressing YFP-H148Q assessed as inhibition of cAMP agonist-induced iodide influx after 4...More data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 370nMAssay Description:Inhibition of human wild-type CFTR expressed in FRT cells coexpressing YFP-H148Q assessed as inhibition of cAMP agonist-induced iodide influx after 4...More data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibition of human wild-type CFTR expressed in FRT cells coexpressing YFP-H148Q assessed as inhibition of cAMP agonist-induced iodide influx after 4...More data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 600nMAssay Description:Inhibition of human wild-type CFTR expressed in FRT cells coexpressing YFP-H148Q assessed as inhibition of cAMP agonist-induced iodide influx after 4...More data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 700nMAssay Description:Inhibition of human CFTR expressed in rat FRT cells coexpressing halide indicator YFP-H148Q assessed as inhibition of halide influx preincubated for ...More data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:Inhibition of human CFTR expressed in rat FRT cells coexpressing halide indicator YFP-H148Q assessed as inhibition of halide influx preincubated for ...More data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:Inhibition of human CFTR expressed in rat FRT cells coexpressing halide indicator YFP-H148Q assessed as inhibition of halide influx preincubated for ...More data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:Inhibition of human CFTR expressed in rat FRT cells coexpressing halide indicator YFP-H148Q assessed as inhibition of halide influx preincubated for ...More data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: <1.00E+3nMAssay Description:Inhibition of CFTR in nonpermeabilized human T84 cells assessed as inhibition of forskolin and IBMX-induced chloride current by short-circuit current...More data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human wild-type CFTR expressed in FRT cells coexpressing YFP-H148Q assessed as inhibition of cAMP agonist-induced iodide influx after 4...More data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: <1.00E+3nMAssay Description:Inhibition of CFTR in nonpermeabilized human bronchial epithelial cells assessed as inhibition of forskolin and IBMX-induced chloride current at by s...More data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of human CFTR expressed in rat FRT cells coexpressing halide indicator YFP-H148Q assessed as inhibition of halide influx preincubated for ...More data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of human CFTR expressed in rat FRT cells coexpressing halide indicator YFP-H148Q assessed as inhibition of halide influx preincubated for ...More data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of human CFTR expressed in rat FRT cells coexpressing halide indicator YFP-H148Q assessed as inhibition of halide influx preincubated for ...More data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of human CFTR expressed in rat FRT cells coexpressing halide indicator YFP-H148Q assessed as inhibition of halide influx preincubated for ...More data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of human wild-type CFTR expressed in FRT cells coexpressing YFP-H148Q assessed as inhibition of cAMP agonist-induced iodide influx after 4...More data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of human wild-type CFTR expressed in FRT cells coexpressing YFP-H148Q assessed as inhibition of cAMP agonist-induced iodide influx after 4...More data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of human CFTR expressed in rat FRT cells coexpressing halide indicator YFP-H148Q assessed as inhibition of halide influx preincubated for ...More data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of human CFTR expressed in rat FRT cells coexpressing halide indicator YFP-H148Q assessed as inhibition of halide influx preincubated for ...More data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of human CFTR expressed in rat FRT cells coexpressing halide indicator YFP-H148Q assessed as inhibition of halide influx preincubated for ...More data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human wild-type CFTR expressed in FRT cells coexpressing YFP-H148Q assessed as inhibition of cAMP agonist-induced iodide influx after 4...More data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human CFTR expressed in rat FRT cells coexpressing halide indicator YFP-H148Q assessed as inhibition of halide influx preincubated for ...More data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human CFTR expressed in rat FRT cells coexpressing halide indicator YFP-H148Q assessed as inhibition of halide influx preincubated for ...More data for this Ligand-Target Pair
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human CFTR expressed in rat FRT cells coexpressing halide indicator YFP-H148Q assessed as inhibition of halide influx preincubated for ...More data for this Ligand-Target Pair