Affinity DataKi: 0.00480nMAssay Description:Inhibition of Human cathepsin KMore data for this Ligand-Target Pair
Affinity DataKi: 0.0800nMAssay Description:Inhibition of type-2 human steroid 5-alpha-reductase.More data for this Ligand-Target Pair
Affinity DataKi: 0.160nMAssay Description:Inhibition of Human cathepsin KMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Apparent inhibition constant towards human Steroid 5-alpha-reductase type 2More data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Inhibition of type-2 human steroid 5-alpha-reductase.More data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Inhibition of type-2 human steroid 5-alpha-reductase.More data for this Ligand-Target Pair
Affinity DataKi: 0.490nMAssay Description:Inhibitory activity of the compound against Human cathepsin LMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Inhibition of cathepsin KMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals
Smithkline Beecham Pharmaceuticals
Affinity DataKi: 0.600nM EC50: 1nMAssay Description:FKBP12 assay using rapamycin analogs.More data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Binding affinity for rat uterine oxytocin receptor (rOTr)More data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Relative binding affinity was measured for Cathepsin KMore data for this Ligand-Target Pair
Affinity DataKi: 0.710nMAssay Description:Binding affinity for rat uterine oxytocin receptor (rOTr)More data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Relative binding affinity was measured for Cathepsin KMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Apparent inhibition constant towards human Steroid 5-alpha-reductase type 2More data for this Ligand-Target Pair
Affinity DataKi: 0.860nMAssay Description:Binding affinity for human oxytocin receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.890nMAssay Description:Inhibition of type-2 human steroid 5-alpha-reductase.More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals
Smithkline Beecham Pharmaceuticals
Affinity DataKi: 1nM EC50: 4nMAssay Description:FKBP12 assay using rapamycin analogs.More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity for human oxytocin receptorMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals
Smithkline Beecham Pharmaceuticals
Affinity DataKi: 1nM EC50: 45nMAssay Description:FKBP12 assay using rapamycin analogs.More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals
Smithkline Beecham Pharmaceuticals
Affinity DataKi: 1nM EC50: 2nMAssay Description:FKBP12 assay using rapamycin analogs.More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals
Smithkline Beecham Pharmaceuticals
Affinity DataKi: 1nM EC50: 4nMAssay Description:FKBP12 assay using rapamycin analogs.More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals
Smithkline Beecham Pharmaceuticals
Affinity DataKi: 1nM EC50: 30nMAssay Description:FKBP12 assay using rapamycin analogs.More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Relative binding affinity was measured for Cathepsin KMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nM IC50: 2.5nMAssay Description:The substrate peptides terminating in AMC/AFC are processed by caspases with or without inhibitors, and the accumulation of AMC/AFC was assessed with...More data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Binding affinity for rat uterine oxytocin receptor (rOTr)More data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Inhibition of type-2 human steroid 5-alpha-reductase.More data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Binding affinity for human oxytocin receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Binding affinity for human oxytocin receptorMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals
Smithkline Beecham Pharmaceuticals
Affinity DataKi: 1.5nM EC50: 70nMAssay Description:FKBP12 assay using rapamycin analogs.More data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Inhibition of Human cathepsin KMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Binding affinity towards rat liver Vasopressin V1a receptor by using functional assayMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Inhibition of type-2 human steroid 5-alpha-reductase.More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Inhibition of Human cathepsin KMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Apparent inhibition constant towards human Steroid 5-alpha-reductase type 2More data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Binding affinity for rat uterine oxytocin receptor (rOTr)More data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Inhibitory activity of the compound against Human cathepsin LMore data for this Ligand-Target Pair
Affinity DataKi: 2.30nMAssay Description:Inhibition of cathepsin KMore data for this Ligand-Target Pair
Affinity DataKi: 2.30nMAssay Description:Inhibition of Human cathepsin KMore data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:Binding affinity for human oxytocin receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.60nMAssay Description:Inhibition of Human cathepsin KMore data for this Ligand-Target Pair
Affinity DataKi: 2.60nMAssay Description:Inhibition of cathepsin KMore data for this Ligand-Target Pair
Affinity DataKi: 2.80nMAssay Description:Binding affinity for rat uterine oxytocin receptor (rOTr)More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals
Smithkline Beecham Pharmaceuticals
Affinity DataKi: 3nM EC50: 20nMAssay Description:FKBP12 assay using rapamycin analogs.More data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Inhibition of type-1 human steroid 5-alpha-reductaseMore data for this Ligand-Target Pair
Affinity DataKi: 3.40nMAssay Description:Relative binding affinity was measured for Cathepsin KMore data for this Ligand-Target Pair
Affinity DataKi: 3.5nMAssay Description:Inhibition of cathepsin KMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals
Smithkline Beecham Pharmaceuticals
Affinity DataKi: 3.5nM EC50: 10nMAssay Description:FKBP12 assay using rapamycin analogs.More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals
Smithkline Beecham Pharmaceuticals
Affinity DataKi: 3.70nM EC50: 2.50E+3nMAssay Description:FKBP12 assay using rapamycin analogs.More data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Inhibitory activity of the compound against Human cathepsin SMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:In vitro inhibition of recombinant human Steroid 5-alpha-reductase type IMore data for this Ligand-Target Pair
![](/img/powered_by_small.gif)