Compile Data Set for Download or QSAR
maximum 50k data
Found 68 with Last Name = 'sarkar-tyson' and Initial = 'm'
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50067004((S)-1-(3,3-Dimethyl-2-oxo-pentanoyl)-piperidine-2-...)
Affinity DataKi:  10nMAssay Description:Inhibition of recombinant human FKBP12 expressed in Escherichia coli using succinyl-Ala-Phe-Pro-Phe-4-nitroanilide as substrateMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50335225((S)-1-Phenylmethanesulfonyl-piperidine-2-carboxyli...)
Affinity DataKi:  230nMAssay Description:Inhibition of recombinant human FKBP12 expressed in Escherichia coli using succinyl-Ala-Phe-Pro-Phe-4-nitroanilide as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50565509(CHEMBL4790993)
Affinity DataIC50:  180nMAssay Description:Inhibition of human FKBP12 assessed as reduction in PPIase activity using succinyl-Ala-Leu-Pro-Phe-4-nitroanilide as substrate incubated for 4 mins b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50565511(CHEMBL4788177)
Affinity DataIC50:  190nMAssay Description:Inhibition of human FKBP12 assessed as reduction in PPIase activity using succinyl-Ala-Leu-Pro-Phe-4-nitroanilide as substrate incubated for 4 mins b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50565510(CHEMBL4794577)
Affinity DataIC50:  220nMAssay Description:Inhibition of human FKBP12 assessed as reduction in PPIase activity using succinyl-Ala-Leu-Pro-Phe-4-nitroanilide as substrate incubated for 4 mins b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50565512(CHEMBL4798300)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of human FKBP12 assessed as reduction in PPIase activity using succinyl-Ala-Leu-Pro-Phe-4-nitroanilide as substrate incubated for 4 mins b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Homo sapiens (Human))
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50437711(CHEMBL2409076)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of human Pin1 assessed as reduction in PPIase activity using Suc-Ala-Glu-Pro-Phe-MCA as substrate measured for 20 secs by fluorescence met...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOuter membrane protein MIP(Legionella pneumophila)
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50565509(CHEMBL4790993)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of Legionella pneumophila Mip assessed as reduction in PPIase activity using succinyl-Ala-Leu-Pro-Phe-4-nitroanilide as substrate incubate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOuter membrane protein MIP(Legionella pneumophila)
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50200286(CHEMBL3890138)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of Mip PPIase activity in Legionella pneumophilaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOuter membrane protein MIP(Legionella pneumophila)
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50200286(CHEMBL3890138)
Affinity DataIC50:  2.24E+3nMAssay Description:Inhibition of Mip PPIase activity in Legionella pneumophilaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOuter membrane protein MIP(Legionella pneumophila)
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50200320(CHEMBL3949202)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibition of Mip PPIase activity in Legionella pneumophilaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOuter membrane protein MIP(Legionella pneumophila)
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50200320(CHEMBL3949202)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibition of Mip PPIase activity in Legionella pneumophilaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOuter membrane protein MIP(Legionella pneumophila)
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50200285(CHEMBL3930292)
Affinity DataIC50:  2.57E+3nMAssay Description:Inhibition of Mip PPIase activity in Legionella pneumophilaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOuter membrane protein MIP(Legionella pneumophila)
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50200285(CHEMBL3930292)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of Mip PPIase activity in Legionella pneumophilaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOuter membrane protein MIP(Legionella pneumophila)
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50200317(CHEMBL3950488)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibition of Mip PPIase activity in Legionella pneumophilaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOuter membrane protein MIP(Legionella pneumophila)
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50200317(CHEMBL3950488)
Affinity DataIC50:  3.24E+3nMAssay Description:Inhibition of Mip PPIase activity in Legionella pneumophilaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOuter membrane protein MIP(Legionella pneumophila)
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50200298(CHEMBL3899080)
Affinity DataIC50:  3.47E+3nMAssay Description:Inhibition of Mip PPIase activity in Legionella pneumophilaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOuter membrane protein MIP(Legionella pneumophila)
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50200298(CHEMBL3899080)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibition of Mip PPIase activity in Legionella pneumophilaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOuter membrane protein MIP(Legionella pneumophila)
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50200331(CHEMBL3941933)
Affinity DataIC50:  3.89E+3nMAssay Description:Inhibition of Mip PPIase activity in Legionella pneumophilaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOuter membrane protein MIP(Legionella pneumophila)
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50200331(CHEMBL3941933)
Affinity DataIC50:  3.90E+3nMAssay Description:Inhibition of Mip PPIase activity in Legionella pneumophilaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOuter membrane protein MIP(Legionella pneumophila)
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50565510(CHEMBL4794577)
Affinity DataIC50:  4.90E+3nMAssay Description:Inhibition of Legionella pneumophila Mip assessed as reduction in PPIase activity using succinyl-Ala-Leu-Pro-Phe-4-nitroanilide as substrate incubate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOuter membrane protein MIP(Legionella pneumophila)
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50565511(CHEMBL4788177)
Affinity DataIC50:  5.60E+3nMAssay Description:Inhibition of Legionella pneumophila Mip assessed as reduction in PPIase activity using succinyl-Ala-Leu-Pro-Phe-4-nitroanilide as substrate incubate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOuter membrane protein MIP(Legionella pneumophila)
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50200338(CHEMBL3970282)
Affinity DataIC50:  5.60E+3nMAssay Description:Inhibition of Mip PPIase activity in Legionella pneumophilaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOuter membrane protein MIP(Legionella pneumophila)
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50200338(CHEMBL3970282)
Affinity DataIC50:  5.62E+3nMAssay Description:Inhibition of Mip PPIase activity in Legionella pneumophilaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOuter membrane protein MIP(Legionella pneumophila)
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50200297(CHEMBL3939283)
Affinity DataIC50:  5.70E+3nMAssay Description:Inhibition of Mip PPIase activity in Legionella pneumophilaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOuter membrane protein MIP(Legionella pneumophila)
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50200283(CHEMBL3924013)
Affinity DataIC50:  5.75E+3nMAssay Description:Inhibition of Mip PPIase activity in Legionella pneumophilaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOuter membrane protein MIP(Legionella pneumophila)
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50200297(CHEMBL3939283)
Affinity DataIC50:  5.75E+3nMAssay Description:Inhibition of Mip PPIase activity in Legionella pneumophilaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOuter membrane protein MIP(Legionella pneumophila)
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50200283(CHEMBL3924013)
Affinity DataIC50:  5.80E+3nMAssay Description:Inhibition of Mip PPIase activity in Legionella pneumophilaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOuter membrane protein MIP(Legionella pneumophila)
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50200316(CHEMBL3970581)
Affinity DataIC50:  7.50E+3nMAssay Description:Inhibition of Mip PPIase activity in Legionella pneumophilaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOuter membrane protein MIP(Legionella pneumophila)
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50200316(CHEMBL3970581)
Affinity DataIC50:  7.59E+3nMAssay Description:Inhibition of Mip PPIase activity in Legionella pneumophilaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOuter membrane protein MIP(Legionella pneumophila)
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50200288(CHEMBL3921322)
Affinity DataIC50:  7.70E+3nMAssay Description:Inhibition of Mip PPIase activity in Legionella pneumophilaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOuter membrane protein MIP(Legionella pneumophila)
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50200288(CHEMBL3921322)
Affinity DataIC50:  7.76E+3nMAssay Description:Inhibition of Mip PPIase activity in Legionella pneumophilaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOuter membrane protein MIP(Legionella pneumophila)
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50200321(CHEMBL3911322)
Affinity DataIC50:  7.90E+3nMAssay Description:Inhibition of Mip PPIase activity in Legionella pneumophilaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOuter membrane protein MIP(Legionella pneumophila)
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50200321(CHEMBL3911322)
Affinity DataIC50:  7.94E+3nMAssay Description:Inhibition of Mip PPIase activity in Legionella pneumophilaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOuter membrane protein MIP(Legionella pneumophila)
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50200291(CHEMBL3893328)
Affinity DataIC50:  8.51E+3nMAssay Description:Inhibition of Mip PPIase activity in Legionella pneumophilaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOuter membrane protein MIP(Legionella pneumophila)
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50200291(CHEMBL3893328)
Affinity DataIC50:  8.60E+3nMAssay Description:Inhibition of Mip PPIase activity in Legionella pneumophilaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOuter membrane protein MIP(Legionella pneumophila)
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50200300(CHEMBL3922939)
Affinity DataIC50:  8.70E+3nMAssay Description:Inhibition of Mip PPIase activity in Legionella pneumophilaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOuter membrane protein MIP(Legionella pneumophila)
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50200300(CHEMBL3922939)
Affinity DataIC50:  8.71E+3nMAssay Description:Inhibition of Mip PPIase activity in Legionella pneumophilaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOuter membrane protein MIP(Legionella pneumophila)
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50200293(CHEMBL3896009)
Affinity DataIC50:  1.07E+4nMAssay Description:Inhibition of Mip PPIase activity in Legionella pneumophilaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOuter membrane protein MIP(Legionella pneumophila)
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50200293(CHEMBL3896009)
Affinity DataIC50:  1.07E+4nMAssay Description:Inhibition of Mip PPIase activity in Legionella pneumophilaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOuter membrane protein MIP(Legionella pneumophila)
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50200319(CHEMBL3902318)
Affinity DataIC50:  1.14E+4nMAssay Description:Inhibition of Mip PPIase activity in Legionella pneumophilaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOuter membrane protein MIP(Legionella pneumophila)
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50200319(CHEMBL3902318)
Affinity DataIC50:  1.15E+4nMAssay Description:Inhibition of Mip PPIase activity in Legionella pneumophilaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOuter membrane protein MIP(Legionella pneumophila)
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50200299(CHEMBL3920840)
Affinity DataIC50:  1.15E+4nMAssay Description:Inhibition of Mip PPIase activity in Legionella pneumophilaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOuter membrane protein MIP(Legionella pneumophila)
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50200299(CHEMBL3920840)
Affinity DataIC50:  1.15E+4nMAssay Description:Inhibition of Mip PPIase activity in Legionella pneumophilaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOuter membrane protein MIP(Legionella pneumophila)
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50200292(CHEMBL3936855)
Affinity DataIC50:  1.28E+4nMAssay Description:Inhibition of Mip PPIase activity in Legionella pneumophilaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOuter membrane protein MIP(Legionella pneumophila)
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50200292(CHEMBL3936855)
Affinity DataIC50:  1.29E+4nMAssay Description:Inhibition of Mip PPIase activity in Legionella pneumophilaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOuter membrane protein MIP(Legionella pneumophila)
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50200295(CHEMBL3963890)
Affinity DataIC50:  2.14E+4nMAssay Description:Inhibition of Mip PPIase activity in Legionella pneumophilaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOuter membrane protein MIP(Legionella pneumophila)
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50200295(CHEMBL3963890)
Affinity DataIC50:  2.14E+4nMAssay Description:Inhibition of Mip PPIase activity in Legionella pneumophilaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOuter membrane protein MIP(Legionella pneumophila)
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50565512(CHEMBL4798300)
Affinity DataIC50:  2.18E+4nMAssay Description:Inhibition of Legionella pneumophila Mip assessed as reduction in PPIase activity using succinyl-Ala-Leu-Pro-Phe-4-nitroanilide as substrate incubate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOuter membrane protein MIP(Legionella pneumophila)
University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50565513(CHEMBL4779246)
Affinity DataIC50:  3.17E+4nMAssay Description:Inhibition of Legionella pneumophila Mip assessed as reduction in PPIase activity using succinyl-Ala-Leu-Pro-Phe-4-nitroanilide as substrate incubate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 68 total ) | Next | Last >>
Jump to: