Affinity DataKi: 5.90nMAssay Description:Binding affinity for Adenosine A1 receptor of rat cortical membrane by displacing [3H]DPCPX More data for this Ligand-Target Pair
Affinity DataKi: 6.40nMAssay Description:In vitro binding affinity towards human adenosine A1 receptor by [3H]DPCPX displacement.More data for this Ligand-Target Pair
Affinity DataKi: 9.80nMAssay Description:Binding affinity for Adenosine A3 receptor expressed in HEK 293 cells by displacing i[125I]-ABMECAMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Inhibition of [125 I]-IABMECA binding to human adenosine A3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:In vitro binding affinity towards human adenosine A1 receptor by [3H]DPCPX displacement.More data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Binding affinity for Adenosine A3 receptor expressed in HEK 293 cells by displacing i[125I]-ABMECAMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:In vitro binding affinity towards human adenosine A1 receptor by [3H]DPCPX displacement.More data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Binding affinity for Adenosine A3 receptor expressed in HEK 293 cells by displacing i[125I]-ABMECAMore data for this Ligand-Target Pair
Affinity DataKi: 36nMAssay Description:Binding affinity for Adenosine A3 receptor expressed in HEK 293 cells by displacing i[125I]-ABMECAMore data for this Ligand-Target Pair
Affinity DataKi: 47nMAssay Description:Binding affinity for Adenosine A1 receptor of rat cortical membrane by displacing [3H]DPCPX More data for this Ligand-Target Pair
Affinity DataKi: 53nMAssay Description:Binding affinity for Adenosine A1 receptor of rat cortical membrane by displacing [3H]DPCPX More data for this Ligand-Target Pair
Affinity DataKi: 59nMAssay Description:Binding affinity for human Adenosine A3 receptor using [125 I]-IABMECAMore data for this Ligand-Target Pair
Affinity DataKi: 60nMAssay Description:Tested for binding affinity towards human adenosine A2A receptor using [3H]ZM-241385 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 79nMAssay Description:Binding affinity for Adenosine A1 receptor of rat cortical membrane by displacing [3H]DPCPX More data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Binding affinity for Adenosine A1 receptor of rat cortical membrane by displacing [3H]DPCPX More data for this Ligand-Target Pair
Affinity DataKi: 110nMAssay Description:Binding affinity for Adenosine A1 receptor of rat cortical membrane by displacing [3H]DPCPX More data for this Ligand-Target Pair
Affinity DataKi: 120nMAssay Description:Binding affinity for Adenosine A3 receptor expressed in HEK 293 cells by displacing i[125I]-ABMECAMore data for this Ligand-Target Pair
Affinity DataKi: 138nMAssay Description:Binding affinity for Adenosine A1 receptor of rat cortical membrane by displacing [3H]DPCPX More data for this Ligand-Target Pair
Affinity DataKi: 163nMAssay Description:Binding affinity for Adenosine A3 receptor expressed in HEK 293 cells by displacing i[125I]-ABMECAMore data for this Ligand-Target Pair
Affinity DataKi: 202nMAssay Description:Binding affinity for Adenosine A3 receptor expressed in HEK 293 cells by displacing i[125I]-ABMECAMore data for this Ligand-Target Pair
Affinity DataKi: 208nMAssay Description:Binding affinity for adenosine A2A receptor of rat striatal membrane by displacing [3H]-ZM 241385More data for this Ligand-Target Pair
Affinity DataKi: 216nMAssay Description:Binding affinity for Adenosine A3 receptor expressed in HEK 293 cells by displacing i[125I]-ABMECAMore data for this Ligand-Target Pair
Affinity DataKi: 222nMAssay Description:Binding affinity for Adenosine A3 receptor expressed in HEK 293 cells by displacing i[125I]-ABMECAMore data for this Ligand-Target Pair
Affinity DataKi: 281nMAssay Description:Inhibition of [125 I]-IABMECA binding to human adenosine A3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 286nMAssay Description:Binding affinity for adenosine A2A receptor of rat striatal membrane by displacing [3H]-ZM 241385More data for this Ligand-Target Pair
Affinity DataKi: 340nMAssay Description:Binding affinity for adenosine A2A receptor of rat striatal membrane by displacing [3H]-ZM 241385More data for this Ligand-Target Pair
Affinity DataKi: 340nMAssay Description:Binding affinity for Adenosine A3 receptor expressed in HEK 293 cells by displacing i[125I]-ABMECAMore data for this Ligand-Target Pair
Affinity DataKi: 344nMAssay Description:Binding affinity for Adenosine A1 receptor of rat cortical membrane by displacing [3H]DPCPX More data for this Ligand-Target Pair
Affinity DataKi: 437nMAssay Description:Binding affinity for adenosine A2A receptor of rat striatal membrane by displacing [3H]-ZM 241385More data for this Ligand-Target Pair
Affinity DataKi: 577nMAssay Description:Inhibition of [125 I]-IABMECA binding to human adenosine A3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 580nMAssay Description:Binding affinity for adenosine A2A receptor of rat striatal membrane by displacing [3H]-ZM 241385More data for this Ligand-Target Pair
Affinity DataKi: 639nMAssay Description:Tested for binding affinity towards human adenosine A2A receptor using [3H]ZM-241385 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 646nMAssay Description:Binding affinity for Adenosine A1 receptor of rat cortical membrane by displacing [3H]DPCPX More data for this Ligand-Target Pair
Affinity DataKi: 1.16E+3nMAssay Description:Binding affinity for Adenosine A1 receptor of rat cortical membrane by displacing [3H]DPCPX More data for this Ligand-Target Pair
Affinity DataKi: 1.42E+3nMAssay Description:Binding affinity for Adenosine A1 receptor of rat cortical membrane by displacing [3H]DPCPX More data for this Ligand-Target Pair
Affinity DataKi: 1.44E+3nMAssay Description:Binding affinity for adenosine A2A receptor of rat striatal membrane by displacing [3H]-ZM 241385More data for this Ligand-Target Pair
Affinity DataKi: 3.51E+3nMAssay Description:Binding affinity for adenosine A2A receptor of rat striatal membrane by displacing [3H]-ZM 241385More data for this Ligand-Target Pair
Affinity DataKi: 1.01E+4nMAssay Description:Binding affinity for adenosine A2A receptor of rat striatal membrane by displacing [3H]-ZM 241385More data for this Ligand-Target Pair
Affinity DataIC50: 1.30nMAssay Description:Inhibition of cAMP formation in CHO cells expressing adenosine A1 receptorMore data for this Ligand-Target Pair