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Found 298 with Last Name = 'anderson' and Initial = 'mo'
TargetFalcilysin(Plasmodium falciparum (isolate 3D7))
California State University

Curated by ChEMBL
LigandPNGBDBM50552265(CHEMBL4799253)
Affinity DataKi:  220nMAssay Description:Inhibition of Plasmodium falciparum FLNMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcilysin(Plasmodium falciparum (isolate 3D7))
California State University

Curated by ChEMBL
LigandPNGBDBM50552271(CHEMBL4743280)
Affinity DataKi:  600nMAssay Description:Inhibition of Plasmodium falciparum FLNMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcilysin(Plasmodium falciparum (isolate 3D7))
California State University

Curated by ChEMBL
LigandPNGBDBM50552264(CHEMBL4782486)
Affinity DataKi:  900nMAssay Description:Inhibition of Plasmodium falciparum FLNMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcilysin(Plasmodium falciparum (isolate 3D7))
California State University

Curated by ChEMBL
LigandPNGBDBM50552268(CHEMBL4799260)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of Plasmodium falciparum FLNMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcilysin(Plasmodium falciparum (isolate 3D7))
California State University

Curated by ChEMBL
LigandPNGBDBM50552275(CHEMBL4797916)
Affinity DataKi:  1.10E+3nMAssay Description:Inhibition of Plasmodium falciparum FLNMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcilysin(Plasmodium falciparum (isolate 3D7))
California State University

Curated by ChEMBL
LigandPNGBDBM50552272(CHEMBL4794156)
Affinity DataKi:  1.40E+3nMAssay Description:Inhibition of Plasmodium falciparum FLNMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcilysin(Plasmodium falciparum (isolate 3D7))
California State University

Curated by ChEMBL
LigandPNGBDBM50552263(CHEMBL4749474)
Affinity DataKi:  1.40E+3nMAssay Description:Inhibition of Plasmodium falciparum FLNMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcilysin(Plasmodium falciparum (isolate 3D7))
California State University

Curated by ChEMBL
LigandPNGBDBM50552269(CHEMBL4785958)
Affinity DataKi:  1.70E+3nMAssay Description:Inhibition of Plasmodium falciparum FLNMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcilysin(Plasmodium falciparum (isolate 3D7))
California State University

Curated by ChEMBL
LigandPNGBDBM50552270(CHEMBL4741390)
Affinity DataKi:  2.50E+3nMAssay Description:Inhibition of Plasmodium falciparum FLNMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcilysin(Plasmodium falciparum (isolate 3D7))
California State University

Curated by ChEMBL
LigandPNGBDBM50552266(CHEMBL4753948)
Affinity DataKi:  2.50E+3nMAssay Description:Inhibition of Plasmodium falciparum FLNMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcilysin(Plasmodium falciparum (isolate 3D7))
California State University

Curated by ChEMBL
LigandPNGBDBM50552273(CHEMBL4763576)
Affinity DataKi:  2.60E+3nMAssay Description:Inhibition of Plasmodium falciparum FLNMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcilysin(Plasmodium falciparum (isolate 3D7))
California State University

Curated by ChEMBL
LigandPNGBDBM50461717(CHEMBL4225532)
Affinity DataKi:  3.00E+3nMAssay Description:Inhibition of Plasmodium falciparum FLNMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcilysin(Plasmodium falciparum (isolate 3D7))
California State University

Curated by ChEMBL
LigandPNGBDBM50552258(CHEMBL4759772)
Affinity DataKi:  3.50E+3nMAssay Description:Inhibition of Plasmodium falciparum FLNMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcilysin(Plasmodium falciparum (isolate 3D7))
California State University

Curated by ChEMBL
LigandPNGBDBM50552261(CHEMBL4797275)
Affinity DataKi:  4.00E+3nMAssay Description:Inhibition of Plasmodium falciparum FLNMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcilysin(Plasmodium falciparum (isolate 3D7))
California State University

Curated by ChEMBL
LigandPNGBDBM50552252(CHEMBL4787612)
Affinity DataKi:  4.00E+3nMAssay Description:Inhibition of Plasmodium falciparum FLNMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcilysin(Plasmodium falciparum (isolate 3D7))
California State University

Curated by ChEMBL
LigandPNGBDBM50552274(CHEMBL4747594)
Affinity DataKi:  4.00E+3nMAssay Description:Inhibition of Plasmodium falciparum FLNMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcilysin(Plasmodium falciparum (isolate 3D7))
California State University

Curated by ChEMBL
LigandPNGBDBM50552267(CHEMBL4749198)
Affinity DataKi:  4.00E+3nMAssay Description:Inhibition of Plasmodium falciparum FLNMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcilysin(Plasmodium falciparum (isolate 3D7))
California State University

Curated by ChEMBL
LigandPNGBDBM50552262(CHEMBL4746210)
Affinity DataKi:  4.90E+3nMAssay Description:Inhibition of Plasmodium falciparum FLNMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcilysin(Plasmodium falciparum (isolate 3D7))
California State University

Curated by ChEMBL
LigandPNGBDBM50552260(CHEMBL4786923)
Affinity DataKi:  5.00E+3nMAssay Description:Inhibition of Plasmodium falciparum FLNMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcilysin(Plasmodium falciparum (isolate 3D7))
California State University

Curated by ChEMBL
LigandPNGBDBM50552257(CHEMBL4744749)
Affinity DataKi:  9.00E+3nMAssay Description:Inhibition of Plasmodium falciparum FLNMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcilysin(Plasmodium falciparum (isolate 3D7))
California State University

Curated by ChEMBL
LigandPNGBDBM50552253(CHEMBL4748768)
Affinity DataKi:  1.00E+4nMAssay Description:Inhibition of Plasmodium falciparum FLNMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcilysin(Plasmodium falciparum (isolate 3D7))
California State University

Curated by ChEMBL
LigandPNGBDBM50552254(CHEMBL4760331)
Affinity DataKi:  1.10E+4nMAssay Description:Inhibition of Plasmodium falciparum FLNMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcilysin(Plasmodium falciparum (isolate 3D7))
California State University

Curated by ChEMBL
LigandPNGBDBM50552256(CHEMBL4743581)
Affinity DataKi: >2.50E+4nMAssay Description:Inhibition of Plasmodium falciparum FLNMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcilysin(Plasmodium falciparum (isolate 3D7))
California State University

Curated by ChEMBL
LigandPNGBDBM50552276(CHEMBL4779972)
Affinity DataKi: >2.50E+4nMAssay Description:Inhibition of Plasmodium falciparum FLNMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcilysin(Plasmodium falciparum (isolate 3D7))
California State University

Curated by ChEMBL
LigandPNGBDBM50552277(CHEMBL4795927)
Affinity DataKi: >2.50E+4nMAssay Description:Inhibition of Plasmodium falciparum FLNMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcilysin(Plasmodium falciparum (isolate 3D7))
California State University

Curated by ChEMBL
LigandPNGBDBM50552259(CHEMBL4793336)
Affinity DataKi: >2.50E+4nMAssay Description:Inhibition of Plasmodium falciparum FLNMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFalcilysin(Plasmodium falciparum (isolate 3D7))
California State University

Curated by ChEMBL
LigandPNGBDBM50552255(CHEMBL4783383)
Affinity DataKi: >2.50E+4nMAssay Description:Inhibition of Plasmodium falciparum FLNMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50222546(CHEMBL241779 | tetralithium (2S)-2-(phosphonatoami...)
Affinity DataIC50:  0.860nMAssay Description:Inhibition of PSMAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50222549((S)-2-phosphonoamino-pentanedioic acid | CHEMBL238...)
Affinity DataIC50:  2.30nMAssay Description:Inhibition of PSMAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Homo sapiens (Human))
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50394962(CHEMBL1394231)
Affinity DataIC50:  11nMAssay Description:Inhibition of UT-B in human erythrocytes assessed as increase of hypotonic lysisMore data for this Ligand-Target Pair
TargetUrea transporter 1(Mus musculus)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50394962(CHEMBL1394231)
Affinity DataIC50:  11nMAssay Description:Inhibition of UT-B in mouse acetamide-loaded erythrocyte assessed as increase of hypotonic lysisMore data for this Ligand-Target Pair
TargetUrea transporter 1(Mus musculus)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50394962(CHEMBL1394231)
Affinity DataIC50:  11nMAssay Description:Inhibition of UT-B in wild type CD1 mouse erythrocyte assessed as hemolysis after 10 minsMore data for this Ligand-Target Pair
TargetUrea transporter 1(Mus musculus)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50394961(CHEMBL2165788)
Affinity DataIC50:  14nMAssay Description:Inhibition of UT-B in mouse acetamide-loaded erythrocyte assessed as increase of hypotonic lysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Mus musculus)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50394961(CHEMBL2165788)
Affinity DataIC50:  14nMAssay Description:Inhibition of UT-B in wild type CD1 mouse erythrocyte assessed as hemolysis after 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50222551(CHEMBL241780 | tetralithium (2S)-2-(phosphonatooxy...)
Affinity DataIC50:  15nMAssay Description:Inhibition of PSMAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Mus musculus)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50394961(CHEMBL2165788)
Affinity DataIC50:  23nMAssay Description:Inhibition of UT-B-mediated urea transport in wild type CD1 mouse erythrocytes incubated for 10 mins prior to urea addition by Stopped-flow light sca...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Mus musculus)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50394962(CHEMBL1394231)
Affinity DataIC50:  25.1nMAssay Description:Reversible inhibition of mouse UT-B-mediated urea transportMore data for this Ligand-Target Pair
TargetAnoctamin-1(Homo sapiens (Human))
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239459(CHEMBL4074929)
Affinity DataIC50:  30nMAssay Description:In vitro inhibition of [3H]norepinephrine uptake in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Mus musculus)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50394964(CHEMBL1590659)
Affinity DataIC50:  32nMAssay Description:Inhibition of UT-B in wild type CD1 mouse erythrocyte assessed as hemolysis after 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50222550(CHEMBL239882 | tetrapotassium (3S,8S)-6-oxido-1-ox...)
Affinity DataIC50:  35nMAssay Description:Inhibition of PSMAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Mus musculus)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50435308(CHEMBL2391344)
Affinity DataIC50:  38nMAssay Description:Inhibition of UT-B in mouse acetamide-loaded erythrocyte assessed as increase of hypotonic lysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Mus musculus)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50435309(CHEMBL2391345)
Affinity DataIC50:  43nMAssay Description:Inhibition of UT-B in mouse acetamide-loaded erythrocyte assessed as increase of hypotonic lysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50222542(CHEMBL238831 | tetrapotassium (3S,8S)-2-methyl-6-o...)
Affinity DataIC50:  55nMAssay Description:Inhibition of PSMAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnoctamin-1(Homo sapiens (Human))
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239465(CHEMBL4080525 | US11274074, Control [Ani9])
Affinity DataIC50:  77nMAssay Description:Inhibition of human TMEM16A expressed in FRT cells assessed as reduction of ATP-induced in chloride conductance preincubated for 20 mins followed by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnoctamin-1(Homo sapiens (Human))
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239467(CHEMBL4086165)
Affinity DataIC50:  80nMAssay Description:Inhibition of TMEM16A (unknown origin) expressed in Xenopus laevis oocytes at -60 mV holding potential by voltage-clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnoctamin-1(Homo sapiens (Human))
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239459(CHEMBL4074929)
Affinity DataIC50:  83nMAssay Description:Inhibition of human TMEM16A expressed in FRT cells co-expressing iodide sensitive fluorescent protein YFP-H148Q/I152L/F46L assessed as reduction in A...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Mus musculus)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50394967(CHEMBL2165784)
Affinity DataIC50:  104nMAssay Description:Inhibition of UT-B in wild type CD1 mouse erythrocyte assessed as hemolysis after 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnoctamin-1(Homo sapiens (Human))
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239465(CHEMBL4080525 | US11274074, Control [Ani9])
Affinity DataIC50:  110nMAssay Description:Inhibition of human TMEM16A expressed in FRT cells assessed as reduction of ATP-induced in chloride conductance preincubated for 5 mins followed by A...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Homo sapiens (Human))
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50372201(CHEMBL270610)
Affinity DataIC50:  125nMAssay Description:Inhibition of human PSMAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAnoctamin-1(Homo sapiens (Human))
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50239433(CHEMBL3134585)
Affinity DataIC50:  130nMAssay Description:Inhibition of human TMEM16A expressed in FRT cells assessed as reduction of ATP-induced in chloride conductance preincubated for 5 mins followed by A...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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