Affinity DataIC50: 0.5nMAssay Description:Inhibition of N-terminal His-tagged human B-Raf kinase domain (448 to 723 residues) expressed in Escherichia coli BL21 (DE3) by Lanthascreen assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70nMAssay Description:Inhibition of N-terminal His-tagged human recombinant B-Raf V600E mutant (448 to 723 residues) expressed in Escherichia coli BL21 (DE3) by Lanthascre...More data for this Ligand-Target Pair
Affinity DataIC50: 1.70nMAssay Description:Inhibition of N-terminal His-tagged human recombinant B-Raf V600E mutant (448 to 723 residues) expressed in Escherichia coli BL21 (DE3) by Lanthascre...More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibition of N-terminal His-tagged human recombinant B-Raf V600E mutant (448 to 723 residues) expressed in Escherichia coli BL21 (DE3) by Lanthascre...More data for this Ligand-Target Pair
Affinity DataIC50: 2.10nMAssay Description:Inhibition of N-terminal His-tagged human recombinant B-Raf V600E mutant (448 to 723 residues) expressed in Escherichia coli BL21 (DE3) by Lanthascre...More data for this Ligand-Target Pair
Affinity DataIC50: 3.60nMAssay Description:Inhibition of N-terminal His-tagged human recombinant B-Raf V600E mutant (448 to 723 residues) expressed in Escherichia coli BL21 (DE3) by Lanthascre...More data for this Ligand-Target Pair
Affinity DataIC50: 4.40nMAssay Description:Inhibition of N-terminal His-tagged human recombinant B-Raf V600E mutant (448 to 723 residues) expressed in Escherichia coli BL21 (DE3) by Lanthascre...More data for this Ligand-Target Pair
Affinity DataIC50: 4.5nMAssay Description:Inhibition of N-terminal His-tagged human recombinant B-Raf V600E mutant (448 to 723 residues) expressed in Escherichia coli BL21 (DE3) by Lanthascre...More data for this Ligand-Target Pair
Affinity DataIC50: 5.90nMAssay Description:Inhibition of N-terminal His-tagged human recombinant B-Raf V600E mutant (448 to 723 residues) expressed in Escherichia coli BL21 (DE3) by Lanthascre...More data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition of N-terminal His-tagged human recombinant B-Raf V600E mutant (448 to 723 residues) expressed in Escherichia coli BL21 (DE3) by Lanthascre...More data for this Ligand-Target Pair
Affinity DataIC50: 6.30nMAssay Description:Inhibition of N-terminal His-tagged human recombinant B-Raf V600E mutant (448 to 723 residues) expressed in Escherichia coli BL21 (DE3) by Lanthascre...More data for this Ligand-Target Pair
Affinity DataIC50: 7.60nMAssay Description:Inhibition of N-terminal His-tagged human recombinant B-Raf V600E mutant (448 to 723 residues) expressed in Escherichia coli BL21 (DE3) by Lanthascre...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Aix Marseille University
Curated by ChEMBL
Aix Marseille University
Curated by ChEMBL
Affinity DataIC50: 7.70nMAssay Description:Agonist activity at PPARg-LBD (unknown origin) expressed in HEK293 cells assessed as displacement of SMRT incubated for 16 hrs by luciferase reporter...More data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inhibition of N-terminal His-tagged human B-Raf kinase domain (448 to 723 residues) expressed in Escherichia coli BL21 (DE3) by Lanthascreen assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Aix Marseille University
Curated by ChEMBL
Aix Marseille University
Curated by ChEMBL
Affinity DataIC50: 88nMAssay Description:Agonist activity at PPARg-LBD (unknown origin) expressed in HEK293 cells assessed as displacement of NCoR incubated for 16 hrs by luciferase reporter...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Aix Marseille University
Curated by ChEMBL
Aix Marseille University
Curated by ChEMBL
Affinity DataIC50: 956nMAssay Description:Agonist activity at PPARg-LBD (unknown origin) expressed in HEK293 cells assessed as displacement of NCoR incubated for 16 hrs by luciferase reporter...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Aix Marseille University
Curated by ChEMBL
Aix Marseille University
Curated by ChEMBL
Affinity DataIC50: 2.25E+3nMAssay Description:Agonist activity at PPARg-LBD (unknown origin) expressed in HEK293 cells assessed as displacement of SMRT incubated for 16 hrs by luciferase reporter...More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataEC50: 49nMAssay Description:Agonist activity at human pregnane X receptor expressed in HGPXR reporter cellsMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataEC50: 55nMAssay Description:Agonist activity at human pregnane X receptor expressed in HGPXR reporter cellsMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataEC50: 385nMAssay Description:Agonist activity at human pregnane X receptor expressed in HGPXR reporter cellsMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataEC50: 13nMAssay Description:Agonist activity at human pregnane X receptor expressed in HGPXR reporter cellsMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataEC50: 55nMAssay Description:Agonist activity at human pregnane X receptor expressed in HGPXR reporter cellsMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataEC50: 52nMAssay Description:Agonist activity at human pregnane X receptor expressed in HGPXR reporter cellsMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataEC50: 42nMAssay Description:Agonist activity at human pregnane X receptor expressed in HGPXR reporter cellsMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataEC50: 0.700nMAssay Description:Agonist activity at human pregnane X receptor expressed in HGPXR reporter cellsMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataEC50: 1.5nMAssay Description:Agonist activity at human pregnane X receptor expressed in HGPXR reporter cellsMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataEC50: 33nMAssay Description:Agonist activity at human pregnane X receptor expressed in HGPXR reporter cellsMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataEC50: 45nMAssay Description:Agonist activity at human pregnane X receptor expressed in HGPXR reporter cellsMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataEC50: 388nMAssay Description:Agonist activity at human pregnane X receptor expressed in HGPXR reporter cellsMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataEC50: 51nMAssay Description:Agonist activity at human pregnane X receptor expressed in HGPXR reporter cellsMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataEC50: 20nMAssay Description:Agonist activity at human pregnane X receptor expressed in HGPXR reporter cellsMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataEC50: 336nMAssay Description:Agonist activity at human pregnane X receptor expressed in HGPXR reporter cellsMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataEC50: 271nMAssay Description:Agonist activity at human pregnane X receptor expressed in HGPXR reporter cellsMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataEC50: 101nMAssay Description:Agonist activity at human pregnane X receptor expressed in HGPXR reporter cellsMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataEC50: 20nMAssay Description:Agonist activity at human pregnane X receptor expressed in HGPXR reporter cellsMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataEC50: >5.00E+3nMAssay Description:Agonist activity at human pregnane X receptor expressed in HGPXR reporter cellsMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataEC50: 217nMAssay Description:Agonist activity at human pregnane X receptor expressed in HGPXR reporter cellsMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataEC50: 515nMAssay Description:Agonist activity at human pregnane X receptor expressed in HGPXR reporter cellsMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataEC50: >5.00E+3nMAssay Description:Agonist activity at human pregnane X receptor expressed in HGPXR reporter cellsMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataEC50: >5.00E+3nMAssay Description:Agonist activity at human pregnane X receptor expressed in HGPXR reporter cellsMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataEC50: 1.46E+3nMAssay Description:Agonist activity at human pregnane X receptor expressed in HGPXR reporter cellsMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataEC50: 197nMAssay Description:Agonist activity at human pregnane X receptor expressed in HGPXR reporter cellsMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataEC50: 340nMAssay Description:Agonist activity at human pregnane X receptor expressed in HGPXR reporter cellsMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataEC50: 376nMAssay Description:Agonist activity at human pregnane X receptor expressed in HGPXR reporter cellsMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataEC50: 23nMAssay Description:Agonist activity at human pregnane X receptor expressed in HGPXR reporter cellsMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataEC50: 428nMAssay Description:Agonist activity at human pregnane X receptor expressed in HGPXR reporter cellsMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataEC50: 176nMAssay Description:Agonist activity at human pregnane X receptor expressed in HGPXR reporter cellsMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataEC50: 809nMAssay Description:Protection of human pregnane X receptor against proteolytic digestion in presence of trypsinMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataEC50: 8.04nMAssay Description:Protection of human pregnane X receptor against proteolytic digestion in presence of trypsinMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataEC50: 8.05nMAssay Description:Protection of human pregnane X receptor against proteolytic digestion in presence of trypsinMore data for this Ligand-Target Pair