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Found 648 with Last Name = 'bauzo' and Initial = 'rm'
TargetMelanocortin receptor 3(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50115373(2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propionyl...)
Affinity DataKi:  56nMAssay Description:Binding constant (Ki) at mouse Melanocortin-3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50115362(2-{2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propionyl...)
Affinity DataKi:  295nMAssay Description:Binding constant (Ki) at mouse Melanocortin-3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50114745(1N-{3-[1-[4-amino(imino)methylamino-1-[1-carbamoyl...)
Affinity DataKi:  2.50E+3nMAssay Description:Agonist activity of compound in mouse Melanocortin-3 receptor (mMC3R)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50144869(CHEMBL411775 | Tyr-c[Asp-His-DPhe-Arg-Trp-Asn-Ala-...)
Affinity DataIC50:  0.260nMAssay Description:Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]-hAGRP(82-132)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50144869(CHEMBL411775 | Tyr-c[Asp-His-DPhe-Arg-Trp-Asn-Ala-...)
Affinity DataIC50:  0.960nMAssay Description:Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]NDP-MSHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50144877(CHEMBL269274)
Affinity DataIC50:  1.46nMAssay Description:Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]NDP-MSHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50121900(Ac-Ser-Try-Ser-Nle-Glu-His-DPhe-Arg-Trp-Gly-Lys-Pr...)
Affinity DataIC50:  4.22nMAssay Description:Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]-NDP-MSH; ND = not determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50144877(CHEMBL269274)
Affinity DataIC50:  4.45nMAssay Description:Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]-hAGRP(82-132)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50144871(CHEMBL428134)
Affinity DataIC50:  4.74nMAssay Description:Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]-hAGRP(82-132)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50144882(CHEMBL266288)
Affinity DataIC50:  5.48nMAssay Description:Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]-hAGRP(82-132)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50155865(CHEMBL2373991 | CUDPUATUYCRFFNAFCYCRKL)
Affinity DataIC50:  10nMAssay Description:Displacement of [125I]-hAGRP(87-132) from mouse Melanocortin 4 ReceptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50144871(CHEMBL428134)
Affinity DataIC50:  29.8nMAssay Description:Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]NDP-MSHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50155865(CHEMBL2373991 | CUDPUATUYCRFFNAFCYCRKL)
Affinity DataIC50:  140nMAssay Description:Displacement of [125I]-hAGRP(87-132) from mouse Melanocortin 3 ReceptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50410195(CHEMBL2096710)
Affinity DataIC50:  275nMAssay Description:Displacement of [125I]-hAGRP(87-132) from mouse Melanocortin 4 ReceptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50144880(CHEMBL406032 | Tyr-c[Asp-His-Phe-Arg-Trp-Asn-Ala-P...)
Affinity DataIC50:  290nMAssay Description:Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]-hAGRP(82-132)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50144880(CHEMBL406032 | Tyr-c[Asp-His-Phe-Arg-Trp-Asn-Ala-P...)
Affinity DataIC50:  540nMAssay Description:Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]NDP-MSHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50144879(CHEMBL406550 | Tyr-c[Asp-DPhe-Arg-Trp-Asn-Ala-Phe-...)
Affinity DataIC50:  3.10E+3nMAssay Description:Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]-hAGRP(82-132)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50144878(CHEMBL402258 | Tyr-c[Asp-Arg-Phe-Phe-Asn-Ala-Phe-D...)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]-hAGRP(82-132)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50144874(CHEMBL440633 | Tyr-c[Asp-Phe-Arg-Trp-Asn-Ala-Phe-D...)
Affinity DataIC50:  4.10E+3nMAssay Description:Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]-hAGRP(82-132)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50144878(CHEMBL402258 | Tyr-c[Asp-Arg-Phe-Phe-Asn-Ala-Phe-D...)
Affinity DataIC50:  4.80E+3nMAssay Description:Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]NDP-MSHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50144879(CHEMBL406550 | Tyr-c[Asp-DPhe-Arg-Trp-Asn-Ala-Phe-...)
Affinity DataIC50:  6.80E+3nMAssay Description:Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]NDP-MSHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50144881(CHEMBL413465 | Tyr-c[Asp-Trp-Arg-Phe-Asn-Ala-Phe-D...)
Affinity DataIC50:  7.30E+3nMAssay Description:Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]-hAGRP(82-132)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50144874(CHEMBL440633 | Tyr-c[Asp-Phe-Arg-Trp-Asn-Ala-Phe-D...)
Affinity DataIC50:  9.20E+3nMAssay Description:Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]NDP-MSHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50144870(CHEMBL410091 | Tyr-c[Asp-Trp-Arg-DPhe-Asn-Ala-Phe-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]-hAGRP(82-132)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50144870(CHEMBL410091 | Tyr-c[Asp-Trp-Arg-DPhe-Asn-Ala-Phe-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]NDP-MSHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50144881(CHEMBL413465 | Tyr-c[Asp-Trp-Arg-Phe-Asn-Ala-Phe-D...)
Affinity DataIC50:  1.03E+4nMAssay Description:Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]NDP-MSHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50410195(CHEMBL2096710)
Affinity DataIC50:  1.17E+4nMAssay Description:Displacement of [125I]-hAGRP(87-132) from mouse Melanocortin 3 ReceptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50422954(CHEMBL2304247)
Affinity DataEC50:  6.20nMAssay Description:Displacement of MT2 from mouse MC3R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50422955(CHEMBL2304248)
Affinity DataEC50:  8.30E+3nMAssay Description:Agonist activity at mouse MC4R expressed in HEK293 cells by beta-galactosidase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50422956(CHEMBL2304249)
Affinity DataEC50:  6.24E+3nMAssay Description:Agonist activity at mouse MC4R expressed in HEK293 cells by beta-galactosidase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50422955(CHEMBL2304248)
Affinity DataEC50:  1.75E+3nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cells by beta-galactosidase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50422954(CHEMBL2304247)
Affinity DataEC50:  6.10nMAssay Description:Displacement of MT2 from mouse MC3R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50422954(CHEMBL2304247)
Affinity DataEC50:  93nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cells by beta-galactosidase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50422957(CHEMBL2304250)
Affinity DataEC50:  3.77E+4nMAssay Description:Agonist activity at mouse MC4R expressed in HEK293 cells by beta-galactosidase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50422956(CHEMBL2304249)
Affinity DataEC50:  1.14E+4nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells by beta-galactosidase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50422954(CHEMBL2304247)
Affinity DataEC50:  1.41E+3nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells by beta-galactosidase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50422954(CHEMBL2304247)
Affinity DataEC50: >100nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells by beta-galactosidase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50422956(CHEMBL2304249)
Affinity DataEC50:  120nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cells by beta-galactosidase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50422954(CHEMBL2304247)
Affinity DataEC50:  6.90nMAssay Description:Displacement of MT2 from mouse MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50422958(CHEMBL2304246)
Affinity DataEC50:  5.27E+3nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cells by beta-galactosidase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50422957(CHEMBL2304250)
Affinity DataEC50:  1.98E+4nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells by beta-galactosidase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50422954(CHEMBL2304247)
Affinity DataEC50:  93nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cells by beta-galactosidase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50422958(CHEMBL2304246)
Affinity DataEC50:  8.33E+3nMAssay Description:Agonist activity at mouse MC4R expressed in HEK293 cells by beta-galactosidase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50422955(CHEMBL2304248)
Affinity DataEC50:  4.60E+3nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells by beta-galactosidase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50422958(CHEMBL2304246)
Affinity DataEC50:  2.26E+4nMAssay Description:Agonist activity at mouse MC3R expressed in HEK293 cells by beta-galactosidase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50422957(CHEMBL2304250)
Affinity DataEC50:  6.33E+3nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cells by beta-galactosidase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50422956(CHEMBL2304249)
Affinity DataEC50:  3.70E+3nMAssay Description:Agonist activity at mouse MC4R expressed in HEK293 cells by beta-galactosidase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50422956(CHEMBL2304249)
Affinity DataEC50:  6.33E+4nMAssay Description:Agonist activity at mouse MC3R expressed in HEK293 cells by beta-galactosidase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50422957(CHEMBL2304250)
Affinity DataEC50:  1.83E+4nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells by beta-galactosidase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50422956(CHEMBL2304249)
Affinity DataEC50:  2.22E+3nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells by beta-galactosidase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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