Affinity DataKi: 0.650nMAssay Description:In vitro binding affinity measured by displacement of [3H]rauwolscine from alpha-2c adrenergic receptor expressed in CHO cells in presence of phentol...More data for this Ligand-Target Pair
Affinity DataKi: 0.880nMAssay Description:In vitro binding affinity measured by displacement of [3H]rauwolscine from alpha-2c adrenergic receptor expressed in CHO cells in presence of phentol...More data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:In vitro binding affinity measured by displacement of [3H]rauwolscine from alpha-2c adrenergic receptor expressed in CHO cells in presence of phentol...More data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:In vitro binding affinity towards alpha-2a adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.80nMAssay Description:In vitro binding affinity measured by displacement of [3H]rauwolscine from alpha-2c adrenergic receptor expressed in CHO cells in presence of phentol...More data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:In vitro binding affinity measured by displacement of [3H]rauwolscine from alpha-2c adrenergic receptor expressed in CHO cells in presence of phentol...More data for this Ligand-Target Pair
Affinity DataKi: 3.80nMAssay Description:Binding affinity towards human alpha-2C adrenergic receptor expressed in Chinese Hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataKi: 4.10nMAssay Description:Binding affinity towards alpha-1A adrenergic receptor expressed in human embryonic kidney (HEK293) cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.20nMAssay Description:Binding affinity towards human alpha-2A adrenergic receptor expressed in Chinese Hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.70nMAssay Description:Binding affinity towards human alpha-2A adrenergic receptor expressed in Chinese Hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5.20nMAssay Description:In vitro binding affinity measured by displacement of [3H]rauwolscine from alpha-2c adrenergic receptor expressed in CHO cells in presence of phentol...More data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataKi: 5.30nMAssay Description:Binding affinity towards alpha-1A adrenergic receptor expressed in human embryonic kidney (HEK293) cellsMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataKi: 5.30nMAssay Description:Binding affinity towards alpha-1A adrenergic receptor expressed in human embryonic kidney (HEK293) cellsMore data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:Binding affinity towards human alpha-2A adrenergic receptor expressed in Chinese Hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
Affinity DataKi: 7.10nMAssay Description:In vitro binding affinity towards alpha-2b adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 7.30nMAssay Description:Binding affinity towards human alpha-2B adrenergic receptor expressed in Chinese Hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:In vitro binding affinity measured by displacement of [3H]rauwolscine from alpha-2c adrenergic receptor expressed in CHO cells in presence of phentol...More data for this Ligand-Target Pair
Affinity DataKi: 8.5nMAssay Description:In vitro binding affinity measured by displacement of [3H]rauwolscine from alpha-2c adrenergic receptor expressed in CHO cells in presence of phentol...More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Binding affinity towards human alpha-2C adrenergic receptor expressed in Chinese Hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataKi: 18nMAssay Description:Binding affinity towards human alpha-1D adrenergic receptor expressed in Chinese Hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Binding affinity towards human alpha-2B adrenergic receptor expressed in Chinese Hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataKi: 19nMAssay Description:Binding affinity towards human alpha-1D adrenergic receptor expressed in Chinese Hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:In vitro binding affinity measured by displacement of [3H]rauwolscine from alpha-2c adrenergic receptor expressed in CHO cells in presence of phentol...More data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Binding affinity towards alpha-1A adrenergic receptor expressed in human embryonic kidney (HEK293) cellsMore data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Binding affinity towards human alpha-2A adrenergic receptor expressed in Chinese Hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataKi: 27nMAssay Description:Binding affinity towards alpha-1A adrenergic receptor expressed in human embryonic kidney (HEK293) cellsMore data for this Ligand-Target Pair
Affinity DataKi: 29nMAssay Description:In vitro binding affinity towards alpha-2a adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:In vitro binding affinity measured by displacement of [3H]rauwolscine from alpha-2c adrenergic receptor expressed in CHO cells in presence of phentol...More data for this Ligand-Target Pair
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataKi: 47nMAssay Description:Binding affinity towards human alpha-1B adrenergic receptor expressed in Chinese Hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
Affinity DataKi: 48nMAssay Description:Binding affinity towards human alpha-2B adrenergic receptor expressed in Chinese Hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataKi: 50nMAssay Description:Binding affinity towards human alpha-1D adrenergic receptor expressed in Chinese Hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
Affinity DataKi: 56nMAssay Description:Binding affinity towards human alpha-2A adrenergic receptor expressed in Chinese Hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
Affinity DataKi: 80nMAssay Description:Binding affinity towards human alpha-2C adrenergic receptor expressed in Chinese Hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataKi: 103nMAssay Description:Binding affinity towards human alpha-1B adrenergic receptor expressed in Chinese Hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Chungbuk National University
Curated by ChEMBL
Chungbuk National University
Curated by ChEMBL
Affinity DataKi: 843nMAssay Description:Binding affinity towards human alpha-1B adrenergic receptor expressed in Chinese Hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.30E+3nMAssay Description:In vitro binding affinity towards alpha-2b adrenergic receptorMore data for this Ligand-Target Pair