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Found 132 with Last Name = 'beresford' and Initial = 'ij'
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Glaxo Wellcome Research and Development

Curated by PDSP Ki Database
LigandPNGBDBM29611(2-Iodomelatonin | CHEMBL289233 | Melatonin,2-Iodo)
Affinity DataKi:  0.0100nMMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1A(GUINEA PIG)
Glaxo Wellcome Research and Development

Curated by PDSP Ki Database
LigandPNGBDBM29611(2-Iodomelatonin | CHEMBL289233 | Melatonin,2-Iodo)
Affinity DataKi:  0.0300nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Glaxo Wellcome Research and Development

Curated by PDSP Ki Database
LigandPNGBDBM29611(2-Iodomelatonin | CHEMBL289233 | Melatonin,2-Iodo)
Affinity DataKi:  0.0300nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Glaxo Wellcome Research and Development

Curated by PDSP Ki Database
LigandPNGBDBM50035179(Agomelatine | CHEMBL10878 | N-[2-(7-Methoxy-naphth...)
Affinity DataKi:  0.0300nMMore data for this Ligand-Target Pair
In DepthDetails PubMedDrugBank

TargetMelatonin receptor type 1A(GUINEA PIG)
Glaxo Wellcome Research and Development

Curated by PDSP Ki Database
LigandPNGBDBM29611(2-Iodomelatonin | CHEMBL289233 | Melatonin,2-Iodo)
Affinity DataKi:  0.0400nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Glaxo Wellcome Research and Development

Curated by PDSP Ki Database
LigandPNGBDBM50035179(Agomelatine | CHEMBL10878 | N-[2-(7-Methoxy-naphth...)
Affinity DataKi:  0.0400nMMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Glaxo Wellcome Research and Development

Curated by PDSP Ki Database
LigandPNGBDBM29611(2-Iodomelatonin | CHEMBL289233 | Melatonin,2-Iodo)
Affinity DataKi:  0.0500nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Glaxo Wellcome Research and Development

Curated by PDSP Ki Database
LigandPNGBDBM9019(CHEMBL45 | Melatonin | N-[2-(5-methoxy-1H-indol-3-...)
Affinity DataKi:  0.0800nMMore data for this Ligand-Target Pair
In DepthDetails PubMedDrugBank

TargetMelatonin receptor type 1A(GUINEA PIG)
Glaxo Wellcome Research and Development

Curated by PDSP Ki Database
LigandPNGBDBM50035179(Agomelatine | CHEMBL10878 | N-[2-(7-Methoxy-naphth...)
Affinity DataKi:  0.0900nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMelatonin receptor type 1A(GUINEA PIG)
Glaxo Wellcome Research and Development

Curated by PDSP Ki Database
LigandPNGBDBM50035179(Agomelatine | CHEMBL10878 | N-[2-(7-Methoxy-naphth...)
Affinity DataKi:  0.100nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Glaxo Wellcome Research and Development

Curated by PDSP Ki Database
LigandPNGBDBM85064(CAS_5311134 | GR 196429 | NSC_5311134)
Affinity DataKi:  0.140nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Glaxo Wellcome Research and Development

Curated by PDSP Ki Database
LigandPNGBDBM50043289(CHEMBL34730 | N-[2-(6-Chloro-5-methoxy-1H-indol-3-...)
Affinity DataKi:  0.140nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50444496(CHEMBL3092650)
Affinity DataKi:  0.148nMAssay Description:Displacement of [3H]-R-alpha-ethylhistamine from rat histamine H3 receptor expressed in HEK293 cells after 45 mins by liquid scintillation spectromet...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Glaxo Institute For Molecular Biology

Curated by ChEMBL
LigandPNGBDBM50469874(CHEMBL59780)
Affinity DataKi:  0.155nMAssay Description:Binding affinity against human NK2 receptors expressed in CHO cells using [3H]GR-100679 as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Glaxo Wellcome Research and Development

Curated by PDSP Ki Database
LigandPNGBDBM85064(CAS_5311134 | GR 196429 | NSC_5311134)
Affinity DataKi:  0.160nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Glaxo Wellcome Research and Development

Curated by PDSP Ki Database
LigandPNGBDBM9019(CHEMBL45 | Melatonin | N-[2-(5-methoxy-1H-indol-3-...)
Affinity DataKi:  0.190nMMore data for this Ligand-Target Pair
In DepthDetails PubMedDrugBank

TargetHistamine H3 receptor(Rattus norvegicus (rat))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50444491(CHEMBL3092823)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]-R-alpha-ethylhistamine from histamine H3 receptor in rat cerebral cortical tissue membranes after 45 mins by liquid scintillatio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(GUINEA PIG)
Glaxo Wellcome Research and Development

Curated by PDSP Ki Database
LigandPNGBDBM9019(CHEMBL45 | Melatonin | N-[2-(5-methoxy-1H-indol-3-...)
Affinity DataKi:  0.240nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMelatonin receptor type 1A(GUINEA PIG)
Glaxo Wellcome Research and Development

Curated by PDSP Ki Database
LigandPNGBDBM9019(CHEMBL45 | Melatonin | N-[2-(5-methoxy-1H-indol-3-...)
Affinity DataKi:  0.25nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMelatonin receptor type 1A(GUINEA PIG)
Glaxo Wellcome Research and Development

Curated by PDSP Ki Database
LigandPNGBDBM85064(CAS_5311134 | GR 196429 | NSC_5311134)
Affinity DataKi:  0.330nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50444496(CHEMBL3092650)
Affinity DataKi:  0.363nMAssay Description:Displacement of [3H]-R-alpha-ethylhistamine from histamine H3 receptor in rat cerebral cortical tissue membranes after 45 mins by liquid scintillatio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Glaxo Wellcome Research and Development

Curated by PDSP Ki Database
LigandPNGBDBM9019(CHEMBL45 | Melatonin | N-[2-(5-methoxy-1H-indol-3-...)
Affinity DataKi:  0.380nMMore data for this Ligand-Target Pair
In DepthDetails PubMedDrugBank

TargetMelatonin receptor type 1B(Homo sapiens (Human))
Glaxo Wellcome Research and Development

Curated by PDSP Ki Database
LigandPNGBDBM50035179(Agomelatine | CHEMBL10878 | N-[2-(7-Methoxy-naphth...)
Affinity DataKi:  0.410nMMore data for this Ligand-Target Pair
In DepthDetails PubMedDrugBank

TargetMelatonin receptor type 1A(GUINEA PIG)
Glaxo Wellcome Research and Development

Curated by PDSP Ki Database
LigandPNGBDBM50043289(CHEMBL34730 | N-[2-(6-Chloro-5-methoxy-1H-indol-3-...)
Affinity DataKi:  0.460nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50444500(CHEMBL3092834)
Affinity DataKi:  0.501nMAssay Description:Displacement of [3H]-R-alpha-ethylhistamine from histamine H3 receptor in rat cerebral cortical tissue membranes after 45 mins by liquid scintillatio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Glaxo Wellcome Research and Development

Curated by PDSP Ki Database
LigandPNGBDBM82509(Melatonin,6-Hydroxy | melatonin, 6-Hydroxy)
Affinity DataKi:  0.540nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMelatonin receptor type 1A(GUINEA PIG)
Glaxo Wellcome Research and Development

Curated by PDSP Ki Database
LigandPNGBDBM85064(CAS_5311134 | GR 196429 | NSC_5311134)
Affinity DataKi:  0.610nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50444507(CHEMBL3092826)
Affinity DataKi:  0.631nMAssay Description:Displacement of [3H]-R-alpha-ethylhistamine from histamine H3 receptor in rat cerebral cortical tissue membranes after 45 mins by liquid scintillatio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50444505(CHEMBL3092828)
Affinity DataKi:  0.631nMAssay Description:Displacement of [3H]-R-alpha-ethylhistamine from histamine H3 receptor in rat cerebral cortical tissue membranes after 45 mins by liquid scintillatio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50444509(CHEMBL3092840)
Affinity DataKi:  0.631nMAssay Description:Displacement of [3H]-R-alpha-ethylhistamine from histamine H3 receptor in rat cerebral cortical tissue membranes after 45 mins by liquid scintillatio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Glaxo Wellcome Research and Development

Curated by PDSP Ki Database
LigandPNGBDBM50043289(CHEMBL34730 | N-[2-(6-Chloro-5-methoxy-1H-indol-3-...)
Affinity DataKi:  0.670nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50247054(6-(3-cyclobutyl-2,3,4,5-tetrahydro-1H-benzo[d]azep...)
Affinity DataKi:  0.676nMAssay Description:Displacement of [3H]-R-alpha-ethylhistamine from rat histamine H3 receptor expressed in HEK293 cells after 45 mins by liquid scintillation spectromet...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(GUINEA PIG)
Glaxo Wellcome Research and Development

Curated by PDSP Ki Database
LigandPNGBDBM50043289(CHEMBL34730 | N-[2-(6-Chloro-5-methoxy-1H-indol-3-...)
Affinity DataKi:  0.740nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50444489(CHEMBL3092825)
Affinity DataKi:  0.794nMAssay Description:Displacement of [3H]-R-alpha-ethylhistamine from histamine H3 receptor in rat cerebral cortical tissue membranes after 45 mins by liquid scintillatio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50444495(CHEMBL3092651)
Affinity DataKi:  0.794nMAssay Description:Displacement of [3H]-R-alpha-ethylhistamine from histamine H3 receptor in rat cerebral cortical tissue membranes after 45 mins by liquid scintillatio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50346209(5-(3-cyclobutyl-2,3,4,5-tetrahydro-1H-benzo[d]azep...)
Affinity DataKi:  0.832nMAssay Description:Displacement of [3H]-R-alpha-ethylhistamine from histamine H3 receptor in rat cerebral cortical tissue membranes after 45 mins by liquid scintillatio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470598(CHEMBL126050)
Affinity DataKi:  1nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50444506(CHEMBL3092827)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]-R-alpha-ethylhistamine from histamine H3 receptor in rat cerebral cortical tissue membranes after 45 mins by liquid scintillatio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50444494(CHEMBL3092820)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]-R-alpha-ethylhistamine from histamine H3 receptor in rat cerebral cortical tissue membranes after 45 mins by liquid scintillatio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50346209(5-(3-cyclobutyl-2,3,4,5-tetrahydro-1H-benzo[d]azep...)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]-R-alpha-ethylhistamine from rat histamine H3 receptor expressed in HEK293 cells after 45 mins by liquid scintillation spectromet...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470604(CHEMBL338825)
Affinity DataKi:  1.30nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470590(CHEMBL341357)
Affinity DataKi:  1.30nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470591(CHEMBL124208)
Affinity DataKi:  1.30nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Glaxo Institute For Molecular Biology

Curated by ChEMBL
LigandPNGBDBM50469872(CHEMBL413650)
Affinity DataKi:  1.30nMAssay Description:Binding affinity against human NK2 receptors expressed in CHO cells using [3H]GR-100679 as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Glaxo Institute For Molecular Biology

Curated by ChEMBL
LigandPNGBDBM50469869(CHEMBL217548)
Affinity DataKi:  1.40nMAssay Description:Binding affinity against human NK2 receptors expressed in CHO cells using [3H]GR-100679 as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Glaxo Institute For Molecular Biology

Curated by ChEMBL
LigandPNGBDBM50469867(CHEMBL268783)
Affinity DataKi:  1.5nMAssay Description:Binding affinity against human NK2 receptors expressed in CHO cells using [3H]GR-100679 as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50444493(CHEMBL3092821)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]-R-alpha-ethylhistamine from histamine H3 receptor in rat cerebral cortical tissue membranes after 45 mins by liquid scintillatio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470583(CHEMBL125696)
Affinity DataKi:  1.60nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50470596(CHEMBL125310)
Affinity DataKi:  1.60nMAssay Description:Binding affinity against tachykinin receptor 2 from rat colon.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Glaxo Wellcome Research and Development

Curated by PDSP Ki Database
LigandPNGBDBM82509(Melatonin,6-Hydroxy | melatonin, 6-Hydroxy)
Affinity DataKi:  1.69nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
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