Found 55 with Last Name = 'bernardi' and Initial = 't' 
Affinity DataKi: 48nMAssay Description:Binding affinity to human NPSR by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 4.80E+4nMAssay Description:Inhibition of mouse B16-BL6 cells derived heparanase using [3H]HS as substrate after 6 hrs by size exclusion chromatography based liquid scintillatio...More data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Corvas International
Curated by ChEMBL
Corvas International
Curated by ChEMBL
Affinity DataIC50: 3.10nMAssay Description:The compound was tested in vitro for its inhibitory activity against human urokinase enzyme, activity expressed as IC50More data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Corvas International
Curated by ChEMBL
Corvas International
Curated by ChEMBL
Affinity DataIC50: 5.10nMAssay Description:The compound was tested in vitro for its inhibitory activity against human urokinase enzyme, activity expressed as IC50More data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Corvas International
Curated by ChEMBL
Corvas International
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:The compound was tested in vitro for its inhibitory activity against human urokinase enzyme, activity expressed as IC50More data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Corvas International
Curated by ChEMBL
Corvas International
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:The compound was tested in vitro for its inhibitory activity against human urokinase enzyme, activity expressed as IC50More data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Corvas International
Curated by ChEMBL
Corvas International
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:The compound was tested in vitro for its inhibitory activity against human urokinase enzyme, activity expressed as IC50More data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Corvas International
Curated by ChEMBL
Corvas International
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:The compound was tested in vitro for its inhibitory activity against human urokinase enzyme, activity expressed as IC50More data for this Ligand-Target Pair
Affinity DataIC50: 21nMAssay Description:Inhibition of FITC-geldanamycin binding to recombinant human HSP90alpha expressed in Escherichia coli by fluorescence anisotropy methodMore data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Corvas International
Curated by ChEMBL
Corvas International
Curated by ChEMBL
Affinity DataIC50: 23nMAssay Description:The compound was tested in vitro for its inhibitory activity against human urokinase enzyme, activity expressed as IC50More data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Corvas International
Curated by ChEMBL
Corvas International
Curated by ChEMBL
Affinity DataIC50: 101nMAssay Description:The compound was tested in vitro for its inhibitory activity against human urokinase enzyme, activity expressed as IC50More data for this Ligand-Target Pair
Affinity DataIC50: 125nMAssay Description:The compound was tested in vitro for its inhibitory activity against human Plasmin enzyme, activity expressed as IC50More data for this Ligand-Target Pair
TargetHeat shock protein 75 kDa, mitochondrial(Homo sapiens (Human))
University Of Ferrara
Curated by ChEMBL
University Of Ferrara
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged TRAP1 (60 to 704 residues) ATPase activity expressed in Escherichia coli BL21-CodonPlus-RIL af...More data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Corvas International
Curated by ChEMBL
Corvas International
Curated by ChEMBL
Affinity DataIC50: 261nMAssay Description:The compound was tested in vitro for its inhibitory activity against human urokinase enzyme, activity expressed as IC50More data for this Ligand-Target Pair
Affinity DataIC50: 275nMAssay Description:The compound was tested in vitro for its inhibitory activity against human Plasmin enzyme, activity expressed as IC50More data for this Ligand-Target Pair
Affinity DataIC50: 367nMAssay Description:The compound was tested in vitro for its inhibitory activity against human Plasmin enzyme, activity expressed as IC50More data for this Ligand-Target Pair
TargetHeat shock protein 75 kDa, mitochondrial(Homo sapiens (Human))
University Of Ferrara
Curated by ChEMBL
University Of Ferrara
Curated by ChEMBL
Affinity DataIC50: 400nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged TRAP1 (60 to 704 residues) ATPase activity expressed in Escherichia coli BL21-CodonPlus-RIL af...More data for this Ligand-Target Pair
Affinity DataIC50: 482nMAssay Description:The compound was tested in vitro for its inhibitory activity against human Plasmin enzyme, activity expressed as IC50More data for this Ligand-Target Pair
TargetHeat shock protein 75 kDa, mitochondrial(Homo sapiens (Human))
University Of Ferrara
Curated by ChEMBL
University Of Ferrara
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged TRAP1 (60 to 704 residues) ATPase activity expressed in Escherichia coli BL21-CodonPlus-RIL af...More data for this Ligand-Target Pair
TargetHeat shock protein 75 kDa, mitochondrial(Homo sapiens (Human))
University Of Ferrara
Curated by ChEMBL
University Of Ferrara
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged TRAP1 (60 to 704 residues) ATPase activity expressed in Escherichia coli BL21-CodonPlus-RIL af...More data for this Ligand-Target Pair
Affinity DataIC50: 660nMAssay Description:Inhibition of heparanase (unknown origin) assessed as reduction in AGA*IA cleavage after 3 hrs by WST1 dye based colorimetric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 699nMAssay Description:The compound was tested in vitro for its inhibitory activity against human Plasmin enzyme, activity expressed as IC50More data for this Ligand-Target Pair
Affinity DataIC50: 860nMAssay Description:Inhibition of heparanase (unknown origin) assessed as reduction in AGA*IA cleavage after 3 hrs by WST1 dye based colorimetric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 904nMAssay Description:The compound was tested in vitro for its inhibitory activity against human Plasmin enzyme, activity expressed as IC50More data for this Ligand-Target Pair
Affinity DataIC50: 1.17E+3nMAssay Description:The compound was tested in vitro for its inhibitory activity against human Plasmin enzyme, activity expressed as IC50More data for this Ligand-Target Pair
Affinity DataIC50: 1.46E+3nMAssay Description:The compound was tested in vitro for its inhibitory activity against human Plasmin enzyme, activity expressed as IC50More data for this Ligand-Target Pair
Affinity DataIC50: 1.48E+3nMAssay Description:Inhibition of heparanase (unknown origin) assessed as reduction in AGA*IA cleavage after 3 hrs by WST1 dye based colorimetric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.72E+3nMAssay Description:Inhibition of heparanase (unknown origin) assessed as reduction in AGA*IA cleavage after 3 hrs by WST1 dye based colorimetric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of heparanase (unknown origin) assessed as reduction in AGA*IA cleavage after 3 hrs by WST1 dye based colorimetric assayMore data for this Ligand-Target Pair
Affinity DataIC50: >2.50E+3nMAssay Description:The compound was tested in vitro for its inhibitory activity against human t-PA enzyme, activity expressed as IC50More data for this Ligand-Target Pair
Affinity DataIC50: >2.50E+3nMAssay Description:The compound was tested in vitro for its inhibitory activity against human t-PA enzyme, activity expressed as IC50More data for this Ligand-Target Pair
Affinity DataIC50: >2.50E+3nMAssay Description:The compound was tested in vitro for its inhibitory activity against human t-PA enzyme, activity expressed as IC50More data for this Ligand-Target Pair
Affinity DataIC50: >2.50E+3nMAssay Description:The compound was tested in vitro for its inhibitory activity against human t-PA enzyme, activity expressed as IC50More data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Corvas International
Curated by ChEMBL
Corvas International
Curated by ChEMBL
Affinity DataIC50: >2.50E+3nMAssay Description:The compound was tested in vitro for its inhibitory activity against human urokinase enzyme, activity expressed as IC50More data for this Ligand-Target Pair
Affinity DataIC50: >2.50E+3nMAssay Description:The compound was tested in vitro for its inhibitory activity against human t-PA enzyme, activity expressed as IC50More data for this Ligand-Target Pair
Affinity DataIC50: >2.50E+3nMAssay Description:The compound was tested in vitro for its inhibitory activity against human t-PA enzyme, activity expressed as IC50More data for this Ligand-Target Pair
Affinity DataIC50: >2.50E+3nMAssay Description:The compound was tested in vitro for its inhibitory activity against human Plasmin enzyme, activity expressed as IC50More data for this Ligand-Target Pair
Affinity DataIC50: >2.50E+3nMAssay Description:The compound was tested in vitro for its inhibitory activity against human t-PA enzyme, activity expressed as IC50More data for this Ligand-Target Pair
Affinity DataIC50: >2.50E+3nMAssay Description:The compound was tested in vitro for its inhibitory activity against human Plasmin enzyme, activity expressed as IC50More data for this Ligand-Target Pair
Affinity DataIC50: >2.50E+3nMAssay Description:The compound was tested in vitro for its inhibitory activity against human t-PA enzyme, activity expressed as IC50More data for this Ligand-Target Pair
Affinity DataIC50: >2.50E+3nMAssay Description:The compound was tested in vitro for its inhibitory activity against human t-PA enzyme, activity expressed as IC50More data for this Ligand-Target Pair
Affinity DataIC50: >2.50E+3nMAssay Description:The compound was tested in vitro for its inhibitory activity against human t-PA enzyme, activity expressed as IC50More data for this Ligand-Target Pair
Affinity DataIC50: >2.50E+3nMAssay Description:The compound was tested in vitro for its inhibitory activity against human t-PA enzyme, activity expressed as IC50More data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Corvas International
Curated by ChEMBL
Corvas International
Curated by ChEMBL
Affinity DataIC50: >2.50E+3nMAssay Description:The compound was tested in vitro for its inhibitory activity against human urokinase enzyme, activity expressed as IC50More data for this Ligand-Target Pair
TargetHeat shock protein 75 kDa, mitochondrial(Homo sapiens (Human))
University Of Ferrara
Curated by ChEMBL
University Of Ferrara
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged TRAP1 (60 to 704 residues) ATPase activity expressed in Escherichia coli BL21-CodonPlus-RIL af...More data for this Ligand-Target Pair
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of heparanase (unknown origin) assessed as reduction in AGA*IA cleavage after 3 hrs by WST1 dye based colorimetric assayMore data for this Ligand-Target Pair
TargetHeat shock protein 75 kDa, mitochondrial(Homo sapiens (Human))
University Of Ferrara
Curated by ChEMBL
University Of Ferrara
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged TRAP1 (60 to 704 residues) ATPase activity expressed in Escherichia coli BL21-CodonPlus-RIL af...More data for this Ligand-Target Pair
Affinity DataIC50: 5.64E+3nMAssay Description:Inhibition of heparanase (unknown origin) assessed as reduction in AGA*IA cleavage after 3 hrs by WST1 dye based colorimetric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 8.53E+3nMAssay Description:Inhibition of heparanase (unknown origin) assessed as reduction in AGA*IA cleavage after 3 hrs by WST1 dye based colorimetric assayMore data for this Ligand-Target Pair
TargetHeat shock protein 75 kDa, mitochondrial(Homo sapiens (Human))
University Of Ferrara
Curated by ChEMBL
University Of Ferrara
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human N-terminal His6-tagged TRAP1 (60 to 704 residues) ATPase activity expressed in Escherichia coli BL21-CodonPlus-RIL af...More data for this Ligand-Target Pair
