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Found 54 with Last Name = 'bertolasi' and Initial = 'v'
TargetTranslocator protein(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50029750(CHEMBL288551 | Dimethyl-carbamic acid 5-phenyl-6-t...)
Affinity DataKi:  9nMAssay Description:Binding affinity constant for peripheral (mitochondrial) Benzodiazepine receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50029751(CHEMBL284371 | Nicotinic acid 5-(4-methoxy-phenyl)...)
Affinity DataKi: >10nMAssay Description:Binding affinity constant for peripheral (mitochondrial) Benzodiazepine receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50029756(3,4,5-Trimethoxy-benzoic acid 9-chloro-5-(4-methox...)
Affinity DataKi: >10nMAssay Description:Binding affinity constant for peripheral (mitochondrial) Benzodiazepine receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50029755(Acetic acid 5-(4-chloro-phenyl)-6-thia-10b-aza-ben...)
Affinity DataKi:  30nMAssay Description:Binding affinity constant for peripheral (mitochondrial) Benzodiazepine receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50029754(CHEMBL286909 | Methanesulfonic acid 5-(4-methoxy-p...)
Affinity DataKi:  95nMAssay Description:Binding affinity constant for peripheral (mitochondrial) Benzodiazepine receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50029752(5-Phenyl-6-thia-10b-aza-benzo[e]azulene | CHEMBL35...)
Affinity DataKi:  3.15E+3nMAssay Description:Binding affinity constant for peripheral (mitochondrial) Benzodiazepine receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50029753(4-Methoxy-5-phenyl-6-thia-10b-aza-benzo[e]azulene ...)
Affinity DataKi:  7.00E+3nMAssay Description:Binding affinity constant for peripheral (mitochondrial) Benzodiazepine receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50084717((+)-(1R,2R,3S,5S)-methyl 3-(benzoyloxy)-8-methyl-8...)
Affinity DataIC50:  0.5nMAssay Description:Displacement of [3H]paroxetine from Serotonin transporter of rat caudate putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50166145((3S,6R)-3-[Bis-(4-fluoro-phenyl)-methoxy]-6-methox...)
Affinity DataIC50:  10nMAssay Description:Displacement of [3H]WIN-35428 from Dopamine transporter of rat caudate putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50166146((3S,6S)-3-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl...)
Affinity DataIC50:  12nMAssay Description:Displacement of [3H]WIN-35428 from Dopamine transporter of rat caudate putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50166135((3S,6S)-3-[Bis-(4-fluoro-phenyl)-methoxy]-6-methox...)
Affinity DataIC50:  25nMAssay Description:Displacement of [3H]WIN-35428 from Dopamine transporter of rat caudate putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50166141((3S,6S)-3-[(4-Chloro-phenyl)-phenyl-methoxy]-6-met...)
Affinity DataIC50:  32nMAssay Description:Displacement of [3H]WIN-35428 from Dopamine transporter of rat caudate putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50366775(BENZTROPINE | Benzatropine)
Affinity DataIC50:  118nMAssay Description:Displacement of [3H]WIN-35428 from Dopamine transporter of rat caudate putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50166147((3S,6R)-3-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl...)
Affinity DataIC50:  140nMAssay Description:Displacement of [3H]WIN-35428 from Dopamine transporter of rat caudate putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50084717((+)-(1R,2R,3S,5S)-methyl 3-(benzoyloxy)-8-methyl-8...)
Affinity DataIC50:  150nMAssay Description:Displacement of [3H]WIN-35428 from Dopamine transporter of rat caudate putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50166151((3S,6S)-3-Benzhydryloxy-6-methoxy-8-methyl-8-aza-b...)
Affinity DataIC50:  276nMAssay Description:Displacement of [3H]WIN-35428 from Dopamine transporter of rat caudate putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50166145((3S,6R)-3-[Bis-(4-fluoro-phenyl)-methoxy]-6-methox...)
Affinity DataIC50:  280nMAssay Description:Displacement of [3H]paroxetine from Serotonin transporter of rat caudate putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50166150((3S,6S)-3-[Bis-(4-fluoro-phenyl)-methoxy]-6-methox...)
Affinity DataIC50:  340nMAssay Description:Displacement of [3H]WIN-35428 from Dopamine transporter of rat caudate putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50166143((3S,6S)-3-[(4-Chloro-phenyl)-phenyl-methoxy]-6-met...)
Affinity DataIC50:  400nMAssay Description:Displacement of [3H]WIN-35428 from Dopamine transporter of rat caudate putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50166144((3S,6S)-3-[(4-Chloro-phenyl)-phenyl-methoxy]-8-met...)
Affinity DataIC50:  600nMAssay Description:Displacement of [3H]WIN-35428 from Dopamine transporter of rat caudate putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50051065(CHEMBL3318073)
Affinity DataIC50:  750nMAssay Description:Inhibition of bovine brain tubulin polymerization by turbidimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50166136((R)-6-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl-8-a...)
Affinity DataIC50:  900nMAssay Description:Displacement of [3H]WIN-35428 from Dopamine transporter of rat caudate putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50166140((S)-6-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl-8-a...)
Affinity DataIC50:  1.13E+3nMAssay Description:Displacement of [3H]WIN-35428 from Dopamine transporter of rat caudate putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50051067(CHEMBL3318075)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of bovine brain tubulin polymerization by turbidimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50005480((-)-combretastatin | (Z)-3'-hydroxy-3,4,4',5-tetra...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of bovine brain tubulin polymerization by turbidimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50166139((3S,6S)-3-Benzhydryloxy-8-methyl-8-aza-bicyclo[3.2...)
Affinity DataIC50:  1.30E+3nMAssay Description:Displacement of [3H]WIN-35428 from Dopamine transporter of rat caudate putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50051068(CHEMBL3318076)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of bovine brain tubulin polymerization by turbidimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50051066(CHEMBL3318074)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of bovine brain tubulin polymerization by turbidimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50166140((S)-6-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl-8-a...)
Affinity DataIC50: >2.00E+3nMAssay Description:Displacement of [3H]paroxetine from Serotonin transporter of rat caudate putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50051072(CHEMBL3318084)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of bovine brain tubulin polymerization by turbidimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50166137((3S,6R)-3-[Bis-(4-fluoro-phenyl)-methoxy]-6-methox...)
Affinity DataIC50:  2.50E+3nMAssay Description:Displacement of [3H]WIN-35428 from Dopamine transporter of rat caudate putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50051071(CHEMBL3318080)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of bovine brain tubulin polymerization by turbidimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50166137((3S,6R)-3-[Bis-(4-fluoro-phenyl)-methoxy]-6-methox...)
Affinity DataIC50:  3.50E+3nMAssay Description:Displacement of [3H]paroxetine from Serotonin transporter of rat caudate putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50051070(CHEMBL3318079)
Affinity DataIC50:  3.70E+3nMAssay Description:Inhibition of bovine brain tubulin polymerization by turbidimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50166142((3S,6S)-3-Benzhydryloxy-6-methoxymethoxy-8-methyl-...)
Affinity DataIC50:  4.50E+3nMAssay Description:Displacement of [3H]WIN-35428 from Dopamine transporter of rat caudate putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50166146((3S,6S)-3-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl...)
Affinity DataIC50:  1.10E+4nMAssay Description:Displacement of [3H]paroxetine from Serotonin transporter of rat caudate putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50051069(CHEMBL3318077)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of bovine brain tubulin polymerization by turbidimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50166141((3S,6S)-3-[(4-Chloro-phenyl)-phenyl-methoxy]-6-met...)
Affinity DataIC50: >1.00E+5nMAssay Description:Displacement of [3H]paroxetine from Serotonin transporter of rat caudate putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50166150((3S,6S)-3-[Bis-(4-fluoro-phenyl)-methoxy]-6-methox...)
Affinity DataIC50: >1.00E+5nMAssay Description:Displacement of [3H]paroxetine from Serotonin transporter of rat caudate putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50166136((R)-6-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl-8-a...)
Affinity DataIC50: >1.00E+5nMAssay Description:Displacement of [3H]paroxetine from Serotonin transporter of rat caudate putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50166147((3S,6R)-3-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl...)
Affinity DataIC50: >1.00E+5nMAssay Description:Displacement of [3H]paroxetine from Serotonin transporter of rat caudate putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50166142((3S,6S)-3-Benzhydryloxy-6-methoxymethoxy-8-methyl-...)
Affinity DataIC50: >1.00E+5nMAssay Description:Displacement of [3H]paroxetine from Serotonin transporter of rat caudate putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50166139((3S,6S)-3-Benzhydryloxy-8-methyl-8-aza-bicyclo[3.2...)
Affinity DataIC50: >1.00E+5nMAssay Description:Displacement of [3H]paroxetine from Serotonin transporter of rat caudate putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50166143((3S,6S)-3-[(4-Chloro-phenyl)-phenyl-methoxy]-6-met...)
Affinity DataIC50: >1.00E+5nMAssay Description:Displacement of [3H]paroxetine from Serotonin transporter of rat caudate putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50166135((3S,6S)-3-[Bis-(4-fluoro-phenyl)-methoxy]-6-methox...)
Affinity DataIC50: >1.00E+5nMAssay Description:Displacement of [3H]paroxetine from Serotonin transporter of rat caudate putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50166144((3S,6S)-3-[(4-Chloro-phenyl)-phenyl-methoxy]-8-met...)
Affinity DataIC50: >1.00E+5nMAssay Description:Displacement of [3H]paroxetine from Serotonin transporter of rat caudate putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50166151((3S,6S)-3-Benzhydryloxy-6-methoxy-8-methyl-8-aza-b...)
Affinity DataIC50: >1.00E+5nMAssay Description:Displacement of [3H]paroxetine from Serotonin transporter of rat caudate putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50021058(7-Chloro-1-methyl-5-phenyl-2,3-dihydro-1H-benzo[e]...)
Affinity DataKd: >10nMAssay Description:Binding affinity constant for peripheral (mitochondrial) Benzodiazepine receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide S receptor(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50412707(CHEMBL230333)
Affinity DataEC50:  0.676nMAssay Description:Agonist activity at human NPSR Ile107 expressed in HEK293 cells assessed as induction of calcium mobilization after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM22032(1-(2-chlorophenyl)-N-methyl-N-(1-methylpropyl)isoq...)
Affinity DataKd:  2nMAssay Description:Binding affinity constant for peripheral (mitochondrial) Benzodiazepine receptorMore data for this Ligand-Target Pair
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