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Found 42 with Last Name = 'beshr' and Initial = 'ea'
TargetHistone deacetylase 1(Homo sapiens (Human))
Minia University

Curated by ChEMBL
LigandPNGBDBM50292317(CHEMBL4172557)
Affinity DataIC50:  27nMAssay Description:Inhibition of HDAC1 in human HeLa cells after 72 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Minia University

Curated by ChEMBL
LigandPNGBDBM19149(CHEMBL98 | N-hydroxy-N'-phenyloctanediamide | SAHA...)
Affinity DataIC50:  31nMAssay Description:Inhibition of HDAC1 in human HeLa cells after 72 hrs by ELISAMore data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
Minia University

Curated by ChEMBL
LigandPNGBDBM19149(CHEMBL98 | N-hydroxy-N'-phenyloctanediamide | SAHA...)
Affinity DataIC50:  33nMAssay Description:Inhibition of HDAC6 in human HeLa cells after 72 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetHistone deacetylase 1(Homo sapiens (Human))
Minia University

Curated by ChEMBL
LigandPNGBDBM50292331(CHEMBL4168150)
Affinity DataIC50:  38nMAssay Description:Inhibition of HDAC1 in human HeLa cells after 72 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Minia University

Curated by ChEMBL
LigandPNGBDBM50292318(CHEMBL4174925)
Affinity DataIC50:  58nMAssay Description:Inhibition of HDAC1 in human HeLa cells after 72 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Minia University

LigandPNGBDBM13065(5-(4-chlorophenyl)-1-(4-methoxyphenyl)-3-(trifluor...)
Affinity DataIC50:  66nMpH: 8.0 T: 2°CAssay Description:COX fluorescent inhibitor screening assay kit (catalog number 700100, Cayman chemical, Ann Arbour, MI, USA) has been employed to investigate the isoz...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Minia University

LigandPNGBDBM50029600(5-Bromo-2-(4-fluoro-phenyl)-3-(4-methanesulfonyl-p...)
Affinity DataIC50:  70nMpH: 8.0 T: 2°CAssay Description:COX fluorescent inhibitor screening assay kit (catalog number 700100, Cayman chemical, Ann Arbour, MI, USA) has been employed to investigate the isoz...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Minia University

Curated by ChEMBL
LigandPNGBDBM19149(CHEMBL98 | N-hydroxy-N'-phenyloctanediamide | SAHA...)
Affinity DataIC50:  81nMAssay Description:Inhibition of VLA-4 from HL60 lysate in a protein-based ligand binding assay.More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Minia University

Curated by ChEMBL
LigandPNGBDBM19149(CHEMBL98 | N-hydroxy-N'-phenyloctanediamide | SAHA...)
Affinity DataIC50:  91nMAssay Description:Inhibition of HDAC4 in human HeLa cells after 72 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 4(Homo sapiens (Human))
Minia University

Curated by ChEMBL
LigandPNGBDBM50292317(CHEMBL4172557)
Affinity DataIC50:  99nMAssay Description:Inhibition of HDAC4 in human HeLa cells after 72 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Minia University

Curated by ChEMBL
LigandPNGBDBM50292317(CHEMBL4172557)
Affinity DataIC50:  114nMAssay Description:Inhibition of HDAC2 in human HeLa cells after 72 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 4(Homo sapiens (Human))
Minia University

Curated by ChEMBL
LigandPNGBDBM50292331(CHEMBL4168150)
Affinity DataIC50:  180nMAssay Description:Inhibition of HDAC4 in human HeLa cells after 72 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 4(Homo sapiens (Human))
Minia University

Curated by ChEMBL
LigandPNGBDBM50292318(CHEMBL4174925)
Affinity DataIC50:  198nMAssay Description:Inhibition of HDAC4 in human HeLa cells after 72 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Minia University

Curated by ChEMBL
LigandPNGBDBM50292331(CHEMBL4168150)
Affinity DataIC50:  232nMAssay Description:Inhibition of HDAC2 in human HeLa cells after 72 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Minia University

Curated by ChEMBL
LigandPNGBDBM50292317(CHEMBL4172557)
Affinity DataIC50:  261nMAssay Description:Inhibition of HDAC6 in human HeLa cells after 72 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Minia University

Curated by ChEMBL
LigandPNGBDBM50292318(CHEMBL4174925)
Affinity DataIC50:  263nMAssay Description:Inhibition of HDAC2 in human HeLa cells after 72 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Minia University

Curated by ChEMBL
LigandPNGBDBM50292331(CHEMBL4168150)
Affinity DataIC50:  276nMAssay Description:Inhibition of HDAC6 in human HeLa cells after 72 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Minia University

Curated by ChEMBL
LigandPNGBDBM50292318(CHEMBL4174925)
Affinity DataIC50:  290nMAssay Description:Inhibition of HDAC6 in human HeLa cells after 72 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Minia University

LigandPNGBDBM17638(2-{1-[(4-chlorophenyl)carbonyl]-5-methoxy-2-methyl...)
Affinity DataIC50:  600nMAssay Description:Inhibition of ovine COX1 assessed as prostaglandin F2alpha levelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Minia University

LigandPNGBDBM202550(N-{4-[(1Z)-1-(hydroxyimino)ethyl]phenyl}-2-{[5-(3,...)
Affinity DataIC50:  750nMpH: 8.0 T: 2°CAssay Description:COX fluorescent inhibitor screening assay kit (catalog number 700100, Cayman chemical, Ann Arbour, MI, USA) has been employed to investigate the isoz...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Minia University

LigandPNGBDBM202549(N-{4-[(1Z)-1-(hydroxyimino)ethyl]phenyl}-2-{[5-(4-...)
Affinity DataIC50:  980nMpH: 8.0 T: 2°CAssay Description:COX fluorescent inhibitor screening assay kit (catalog number 700100, Cayman chemical, Ann Arbour, MI, USA) has been employed to investigate the isoz...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Minia University

LigandPNGBDBM202547(N-(4-acetylphenyl)-2-[(5-phenyl-1,3,4-oxadiazol-2-...)
Affinity DataIC50:  1.20E+3nMpH: 8.0 T: 2°CAssay Description:COX fluorescent inhibitor screening assay kit (catalog number 700100, Cayman chemical, Ann Arbour, MI, USA) has been employed to investigate the isoz...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Minia University

LigandPNGBDBM50029593(CHEMBL7162 | N-(2-(cyclohexyloxy)-4-nitrophenyl)me...)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of human recombinant COX2 assessed as prostaglandin F2alpha levelMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Minia University

LigandPNGBDBM202550(N-{4-[(1Z)-1-(hydroxyimino)ethyl]phenyl}-2-{[5-(3,...)
Affinity DataIC50:  2.12E+3nMpH: 8.0 T: 2°CAssay Description:COX fluorescent inhibitor screening assay kit (catalog number 700100, Cayman chemical, Ann Arbour, MI, USA) has been employed to investigate the isoz...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Minia University

LigandPNGBDBM202549(N-{4-[(1Z)-1-(hydroxyimino)ethyl]phenyl}-2-{[5-(4-...)
Affinity DataIC50:  3.30E+3nMpH: 8.0 T: 2°CAssay Description:COX fluorescent inhibitor screening assay kit (catalog number 700100, Cayman chemical, Ann Arbour, MI, USA) has been employed to investigate the isoz...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Minia University

LigandPNGBDBM202547(N-(4-acetylphenyl)-2-[(5-phenyl-1,3,4-oxadiazol-2-...)
Affinity DataIC50:  7.10E+3nMpH: 8.0 T: 2°CAssay Description:COX fluorescent inhibitor screening assay kit (catalog number 700100, Cayman chemical, Ann Arbour, MI, USA) has been employed to investigate the isoz...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Minia University

LigandPNGBDBM202548(N-(4-acetylphenyl)-2-{[5-(4-chlorophenyl)-1,3,4-ox...)
Affinity DataIC50:  8.90E+3nMpH: 8.0 T: 2°CAssay Description:COX fluorescent inhibitor screening assay kit (catalog number 700100, Cayman chemical, Ann Arbour, MI, USA) has been employed to investigate the isoz...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Minia University

LigandPNGBDBM202548(N-(4-acetylphenyl)-2-{[5-(4-chlorophenyl)-1,3,4-ox...)
Affinity DataIC50:  1.03E+4nMpH: 8.0 T: 2°CAssay Description:COX fluorescent inhibitor screening assay kit (catalog number 700100, Cayman chemical, Ann Arbour, MI, USA) has been employed to investigate the isoz...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Minia University

LigandPNGBDBM17638(2-{1-[(4-chlorophenyl)carbonyl]-5-methoxy-2-methyl...)
Affinity DataIC50:  1.85E+4nMAssay Description:Inhibition of human recombinant COX2 assessed as prostaglandin F2alpha levelMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Minia University

LigandPNGBDBM50001297(CHEMBL3237075)
Affinity DataIC50:  3.98E+4nMAssay Description:Inhibition of ovine COX1 assessed as prostaglandin F2alpha levelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Minia University

LigandPNGBDBM50001252(CHEMBL3236777)
Affinity DataIC50:  4.59E+4nMAssay Description:Inhibition of ovine COX1 assessed as prostaglandin F2alpha levelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Minia University

LigandPNGBDBM50001297(CHEMBL3237075)
Affinity DataIC50:  4.63E+4nMAssay Description:Inhibition of human recombinant COX2 assessed as prostaglandin F2alpha levelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Minia University

LigandPNGBDBM50001252(CHEMBL3236777)
Affinity DataIC50:  6.82E+4nMAssay Description:Inhibition of human recombinant COX2 assessed as prostaglandin F2alpha levelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Minia University

LigandPNGBDBM202551(N-(4-acetylphenyl)-2-[(5-{1-[4-(2-methylpropyl)phe...)
Affinity DataIC50:  7.03E+4nMpH: 8.0 T: 2°CAssay Description:COX fluorescent inhibitor screening assay kit (catalog number 700100, Cayman chemical, Ann Arbour, MI, USA) has been employed to investigate the isoz...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Minia University

LigandPNGBDBM202551(N-(4-acetylphenyl)-2-[(5-{1-[4-(2-methylpropyl)phe...)
Affinity DataIC50:  7.05E+4nMpH: 8.0 T: 2°CAssay Description:COX fluorescent inhibitor screening assay kit (catalog number 700100, Cayman chemical, Ann Arbour, MI, USA) has been employed to investigate the isoz...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Minia University

LigandPNGBDBM50001261(CHEMBL3237067)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of ovine COX1 assessed as prostaglandin F2alpha levelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Minia University

LigandPNGBDBM50001292(CHEMBL3237068)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of ovine COX1 assessed as prostaglandin F2alpha levelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Minia University

LigandPNGBDBM50001261(CHEMBL3237067)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant COX2 assessed as prostaglandin F2alpha levelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Minia University

LigandPNGBDBM50001292(CHEMBL3237068)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant COX2 assessed as prostaglandin F2alpha levelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Minia University

LigandPNGBDBM50001294(CHEMBL3237071)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant COX2 assessed as prostaglandin F2alpha levelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Minia University

LigandPNGBDBM50001294(CHEMBL3237071)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of ovine COX1 assessed as prostaglandin F2alpha levelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Minia University

LigandPNGBDBM50029593(CHEMBL7162 | N-(2-(cyclohexyloxy)-4-nitrophenyl)me...)
Affinity DataIC50:  2.13E+5nMAssay Description:Inhibition of ovine COX1 assessed as prostaglandin F2alpha levelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed