Compile Data Set for Download or QSAR
maximum 50k data
Found 73 with Last Name = 'bovy' and Initial = 'pr'
TargetAtrial natriuretic peptide receptor 2(Homo sapiens (Human))
G. D. Searle

Curated by ChEMBL
LigandPNGBDBM50228184(CHEMBL3349623)
Affinity DataIC50:  0.0540nMAssay Description:Inhibitory activity against guanylate cyclase coupled receptor binding site in rabbit lung by using [125I]-ANP-(103-126)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAtrial natriuretic peptide receptor 2(Homo sapiens (Human))
G. D. Searle

Curated by ChEMBL
LigandPNGBDBM50228174(CHEMBL413432)
Affinity DataIC50:  0.290nMAssay Description:Inhibitory activity against guanylate cyclase coupled receptor binding site in rabbit lung by using [125I]-ANP-(103-126)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Searle

Curated by ChEMBL
LigandPNGBDBM50046078(5-[4'-(3,5-Dibutyl-[1,2,4]triazol-1-ylmethyl)-biph...)
Affinity DataIC50:  6.5nMAssay Description:Activity against high affinity Angiotensin II receptor, type 1 was measured from the ability to inhibit [125I]-angiotensin II binding to rat uterine ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Searle

Curated by ChEMBL
LigandPNGBDBM50046079(CHEMBL12810 | {2-Butyl-5-chloro-3-[2'-(2H-tetrazol...)
Affinity DataIC50:  33nMAssay Description:Activity against high affinity Angiotensin II receptor, type 1 was measured from the ability to inhibit [125I]-angiotensin II binding to rat uterine ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAtrial natriuretic peptide receptor 2(Homo sapiens (Human))
G. D. Searle

Curated by ChEMBL
LigandPNGBDBM50228181(CHEMBL3349961)
Affinity DataIC50:  36nMAssay Description:Inhibitory activity against guanylate cyclase coupled receptor binding site in rabbit lung by using [125I]-ANP-(103-126)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Searle Research & Development

Curated by ChEMBL
LigandPNGBDBM50031555((S)-3-[3-(4-Carbamimidoyl-phenylcarbamoyl)-propion...)
Affinity DataIC50:  50nMAssay Description:Inhibition of collagen-induced canine platelet aggregation in vitro (blood is pooled from more than 2 dogs).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAtrial natriuretic peptide receptor 2(Homo sapiens (Human))
G. D. Searle

Curated by ChEMBL
LigandPNGBDBM50228182(CHEMBL3349622)
Affinity DataIC50:  52nMAssay Description:Inhibitory activity against guanylate cyclase coupled receptor binding site in rabbit lung by using [125I]-ANP-(103-126)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Searle

Curated by ChEMBL
LigandPNGBDBM50046076(CHEMBL276150 | {2-Butyl-5-chloro-3-[2'-(2H-tetrazo...)
Affinity DataIC50:  52nMAssay Description:Activity against high affinity Angiotensin II receptor, type 1 was measured from the ability to inhibit [125I]-angiotensin II binding to rat uterine ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Searle Research & Development

Curated by ChEMBL
LigandPNGBDBM50031545((S)-3-Benzo[1,3]dioxol-5-yl-3-[3-(4-carbamimidoyl-...)
Affinity DataIC50:  52nMAssay Description:Inhibition of collagen-induced canine platelet aggregation in vitro (blood is pooled from more than 2 dogs).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Searle Research & Development

Curated by ChEMBL
LigandPNGBDBM50031565((S)-3-[3-(4-Carbamimidoyl-phenylcarbamoyl)-propion...)
Affinity DataIC50:  67nMAssay Description:Inhibition of collagen-induced canine platelet aggregation in vitro (blood is pooled from more than 2 dogs).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Searle

Curated by ChEMBL
LigandPNGBDBM50046087(CHEMBL12693 | {2-Butyl-5-chloro-3-[2'-(2H-tetrazol...)
Affinity DataIC50:  72nMAssay Description:Activity against high affinity Angiotensin II receptor, type 1 was measured from the ability to inhibit [125I]-angiotensin II binding to rat uterine ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Searle

Curated by ChEMBL
LigandPNGBDBM50046085(CHEMBL12451 | {2-Butyl-5-chloro-3-[2'-(2H-tetrazol...)
Affinity DataIC50:  88nMAssay Description:Activity against high affinity Angiotensin II receptor, type 1 was measured from the ability to inhibit [125I]-angiotensin II binding to rat uterine ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Searle

Curated by ChEMBL
LigandPNGBDBM50046080(CHEMBL12766 | {2-Butyl-5-chloro-3-[2'-(2H-tetrazol...)
Affinity DataIC50:  95nMAssay Description:Activity against high affinity Angiotensin II receptor, type 1 was measured from the ability to inhibit [125I]-angiotensin II binding to rat uterine ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAtrial natriuretic peptide receptor 2(Homo sapiens (Human))
G. D. Searle

Curated by ChEMBL
LigandPNGBDBM50228183(Drigaqsglgcnsfry)
Affinity DataIC50: >100nMAssay Description:Inhibitory activity against guanylate cyclase coupled receptor binding site in rabbit lung by using [125I]-ANP-(103-126)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAtrial natriuretic peptide receptor 2(Homo sapiens (Human))
G. D. Searle

Curated by ChEMBL
LigandPNGBDBM50228180(GRIDRIG)
Affinity DataIC50: >100nMAssay Description:Inhibitory activity against guanylate cyclase coupled receptor binding site in rabbit lung by using [125I]-ANP-(103-126)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAtrial natriuretic peptide receptor 2(Homo sapiens (Human))
G. D. Searle

Curated by ChEMBL
LigandPNGBDBM50228179(CHEMBL3349962)
Affinity DataIC50: >100nMAssay Description:Inhibitory activity against guanylate cyclase coupled receptor binding site in rabbit lung by using [125I]-ANP-(103-126)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAtrial natriuretic peptide receptor 2(Homo sapiens (Human))
G. D. Searle

Curated by ChEMBL
LigandPNGBDBM50228178(CHEMBL428843 | S-Fggridrigaqsglg-Nsfry)
Affinity DataIC50: >100nMAssay Description:Inhibitory activity against guanylate cyclase coupled receptor binding site in rabbit lung by using [125I]-ANP-(103-126)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAtrial natriuretic peptide receptor 2(Homo sapiens (Human))
G. D. Searle

Curated by ChEMBL
LigandPNGBDBM50228175(CHEMBL265243)
Affinity DataIC50: >100nMAssay Description:Inhibitory activity against guanylate cyclase coupled receptor binding site in rabbit lung by using [125I]-ANP-(103-126)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAtrial natriuretic peptide receptor 1/2/3(Homo sapiens (Human))
G. D. Searle

Curated by ChEMBL
LigandPNGBDBM50228173(CHEMBL2371607)
Affinity DataIC50: >100nMAssay Description:Inhibitory activity against guanylate cyclase coupled receptor binding site in rabbit lung by using [125I]-ANP-(103-126)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Searle Research & Development

Curated by ChEMBL
LigandPNGBDBM50031553(3-[3-(4-Carbamimidoyl-phenylcarbamoyl)-propionylam...)
Affinity DataIC50:  101nMAssay Description:Inhibition of collagen-induced canine platelet aggregation in vitro (blood is pooled from more than 2 dogs).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Searle Research & Development

Curated by ChEMBL
LigandPNGBDBM50031559(3-Benzo[1,3]dioxol-5-yl-3-[3-(4-carbamimidoyl-phen...)
Affinity DataIC50:  104nMAssay Description:Inhibition of collagen-induced canine platelet aggregation in vitro (blood is pooled from more than 2 dogs).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Searle Research & Development

Curated by ChEMBL
LigandPNGBDBM50031561(3-[3-(4-Carbamimidoyl-phenylcarbamoyl)-propionylam...)
Affinity DataIC50:  108nMAssay Description:Inhibition of collagen-induced canine platelet aggregation in vitro (blood is pooled from more than 2 dogs).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Searle Research & Development

Curated by ChEMBL
LigandPNGBDBM50031544(3-[3-(4-Carbamimidoyl-phenylcarbamoyl)-propionylam...)
Affinity DataIC50:  115nMAssay Description:Inhibition of collagen-induced canine platelet aggregation in vitro (blood is pooled from more than 2 dogs).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Searle Research & Development

Curated by ChEMBL
LigandPNGBDBM50031547(3-[3-(4-Carbamimidoyl-phenylcarbamoyl)-propionylam...)
Affinity DataIC50:  122nMAssay Description:Inhibition of collagen-induced canine platelet aggregation in vitro (blood is pooled from more than 2 dogs).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Searle Research & Development

Curated by ChEMBL
LigandPNGBDBM50031556((Aminobenzamidino)succinyl analogue | (S)-3-[3-(4-...)
Affinity DataIC50:  133nMAssay Description:Inhibition of collagen-induced canine platelet aggregation in vitro (blood is pooled from more than 2 dogs).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Searle Research & Development

Curated by ChEMBL
LigandPNGBDBM50031556((Aminobenzamidino)succinyl analogue | (S)-3-[3-(4-...)
Affinity DataIC50:  133nMAssay Description:Inhibition of collagen-induced canine platelet aggregation in vitro (blood is pooled from more than 2 dogs).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Searle Research & Development

Curated by ChEMBL
LigandPNGBDBM50031563(3-[3-(4-Carbamimidoyl-phenylcarbamoyl)-propionylam...)
Affinity DataIC50:  158nMAssay Description:Inhibition of collagen-induced canine platelet aggregation in vitro (blood is pooled from more than 2 dogs).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Searle Research & Development

Curated by ChEMBL
LigandPNGBDBM50031550(3-[3-(4-Carbamimidoyl-phenylcarbamoyl)-propionylam...)
Affinity DataIC50:  170nMAssay Description:Inhibition of collagen-induced canine platelet aggregation in vitro (blood is pooled from more than 2 dogs).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50003399(4'-(2-Butyl-4-chloro-5-hydroxymethyl-imidazol-1-yl...)
Affinity DataIC50:  170nMAssay Description:Ability to displace [125I]-labeled angiotensin II from its receptor of a rat uterus membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Searle Research & Development

Curated by ChEMBL
LigandPNGBDBM50031557(3-[3-(4-Carbamimidoyl-phenylcarbamoyl)-propionylam...)
Affinity DataIC50:  224nMAssay Description:Inhibition of collagen-induced canine platelet aggregation in vitro (blood is pooled from more than 2 dogs).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Searle Research & Development

Curated by ChEMBL
LigandPNGBDBM50031554(3-[3-(4-Carbamimidoyl-phenylcarbamoyl)-propionylam...)
Affinity DataIC50:  256nMAssay Description:Inhibition of collagen-induced canine platelet aggregation in vitro (blood is pooled from more than 2 dogs).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Searle

Curated by ChEMBL
LigandPNGBDBM50046086(CHEMBL12737 | {2-Butyl-5-chloro-3-[2'-(2H-tetrazol...)
Affinity DataIC50:  270nMAssay Description:Activity against high affinity Angiotensin II receptor, type 1 was measured from the ability to inhibit [125I]-angiotensin II binding to rat uterine ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Searle

Curated by ChEMBL
LigandPNGBDBM50046077(CHEMBL276381 | {2-Butyl-5-chloro-3-[2'-(2H-tetrazo...)
Affinity DataIC50:  290nMAssay Description:Activity against high affinity Angiotensin II receptor, type 1 was measured from the ability to inhibit [125I]-angiotensin II binding to rat uterine ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Searle Research & Development

Curated by ChEMBL
LigandPNGBDBM50031552(3-[3-(4-Carbamimidoyl-phenylcarbamoyl)-propionylam...)
Affinity DataIC50:  294nMAssay Description:Inhibition of collagen-induced canine platelet aggregation in vitro (blood is pooled from more than 2 dogs).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Searle Research & Development

Curated by ChEMBL
LigandPNGBDBM50031539(3-[3-(4-Carbamimidoyl-phenylcarbamoyl)-propionylam...)
Affinity DataIC50:  302nMAssay Description:Inhibition of collagen-induced canine platelet aggregation in vitro (blood is pooled from more than 2 dogs).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Searle Research & Development

Curated by ChEMBL
LigandPNGBDBM50031540(3-[3-(4-Carbamimidoyl-phenylcarbamoyl)-propionylam...)
Affinity DataIC50:  321nMAssay Description:Inhibition of collagen-induced canine platelet aggregation in vitro (blood is pooled from more than 2 dogs).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50003399(4'-(2-Butyl-4-chloro-5-hydroxymethyl-imidazol-1-yl...)
Affinity DataIC50:  330nMAssay Description:Ability to displace [125I]-labeled angiotensin II from its receptor of a rat uterus membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50003399(4'-(2-Butyl-4-chloro-5-hydroxymethyl-imidazol-1-yl...)
Affinity DataIC50:  330nMAssay Description:Ability to displace [125I]-labeled angiotensin II from its receptor of a rat uterus membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Searle

Curated by ChEMBL
LigandPNGBDBM50046084(CHEMBL12548 | {2-Butyl-5-chloro-3-[2'-(2H-tetrazol...)
Affinity DataIC50:  480nMAssay Description:Activity against high affinity Angiotensin II receptor, type 1 was measured from the ability to inhibit [125I]-angiotensin II binding to rat uterine ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Searle Research & Development

Curated by ChEMBL
LigandPNGBDBM50031558(3-[3-(4-Carbamimidoyl-phenylcarbamoyl)-propionylam...)
Affinity DataIC50:  491nMAssay Description:Inhibition of collagen-induced canine platelet aggregation in vitro (blood is pooled from more than 2 dogs).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Searle Research & Development

Curated by ChEMBL
LigandPNGBDBM50031566(3-[3-(4-Carbamimidoyl-phenylcarbamoyl)-propionylam...)
Affinity DataIC50:  580nMAssay Description:Inhibition of collagen-induced canine platelet aggregation in vitro (blood is pooled from more than 2 dogs).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Searle Research & Development

Curated by ChEMBL
LigandPNGBDBM50031551(3-[5-(4-Carbamimidoyl-phenyl)-pent-4-enoylamino]-p...)
Affinity DataIC50:  904nMAssay Description:Inhibition of collagen-induced canine platelet aggregation in vitro (blood is pooled from more than 2 dogs).More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Searle Research & Development

Curated by ChEMBL
LigandPNGBDBM50031564(3-[3-(4-Carbamimidoyl-phenylcarbamoyl)-propionylam...)
Affinity DataIC50:  1.09E+3nMAssay Description:Inhibition of collagen-induced canine platelet aggregation in vitro (blood is pooled from more than 2 dogs).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Searle

Curated by ChEMBL
LigandPNGBDBM50046083(CHEMBL267547 | {2-Butyl-5-chloro-3-[2'-(2H-tetrazo...)
Affinity DataIC50:  1.10E+3nMAssay Description:Activity against high affinity Angiotensin II receptor, type 1 was measured from the ability to inhibit [125I]-angiotensin II binding to rat uterine ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Searle Research & Development

Curated by ChEMBL
LigandPNGBDBM50031546(3-[3-(4-Carbamimidoyl-phenylcarbamoyl)-propionylam...)
Affinity DataIC50:  1.17E+3nMAssay Description:Inhibition of collagen-induced canine platelet aggregation in vitro (blood is pooled from more than 2 dogs).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Searle Research & Development

Curated by ChEMBL
LigandPNGBDBM50031548((Aminobenzamidino)succinyl analogue | {amino[4-(3-...)
Affinity DataIC50:  1.24E+3nMAssay Description:Inhibition of collagen-induced canine platelet aggregation in vitro (blood is pooled from more than 2 dogs).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Searle

Curated by ChEMBL
LigandPNGBDBM50046082(CHEMBL13071 | {2-Butyl-5-chloro-3-[2'-(2H-tetrazol...)
Affinity DataIC50:  2.00E+3nMAssay Description:Activity against high affinity Angiotensin II receptor, type 1 was measured from the ability to inhibit [125I]-angiotensin II binding to rat uterine ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Searle Research & Development

Curated by ChEMBL
LigandPNGBDBM50031538(3-[5-(4-Carbamimidoyl-phenyl)-pentanoylamino]-buty...)
Affinity DataIC50:  2.87E+3nMAssay Description:Inhibition of collagen-induced canine platelet aggregation in vitro (blood is pooled from more than 2 dogs).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(RAT)
Searle

Curated by ChEMBL
LigandPNGBDBM50003399(4'-(2-Butyl-4-chloro-5-hydroxymethyl-imidazol-1-yl...)
Affinity DataIC50:  3.30E+3nMAssay Description:Activity against low affinity Angiotensin II receptor, type 2 was measured from the ability to inhibit [125I]-angiotensin II binding to rat uterine m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor B(RAT)
Searle

Curated by ChEMBL
LigandPNGBDBM50009474(2-[4-(2-Butyl-4-chloro-5-hydroxymethyl-imidazol-1-...)
Affinity DataIC50:  4.20E+3nMAssay Description:Activity against high affinity Angiotensin II receptor, type 1 was measured from the ability to inhibit [125I]-angiotensin II binding to rat uterine ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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