Found 5 Enz. Inhib. hit(s) with Target = 'Type-1 angiotensin II receptor A/Type-1 angiotensin II receptor B/Type-2 angiotensin II receptor' and Ligand = 'BDBM50003399'
TargetType-1 angiotensin II receptor A/Type-1 angiotensin II receptor B/Type-2 angiotensin II receptor(RAT)
Istituto Lusofarmaco
Curated by ChEMBL
Istituto Lusofarmaco
Curated by ChEMBL
Affinity DataKi: 350nMAssay Description:Tested for the binding affinity using radioligand [125I]-Sar1 Ile8-AII in the rat adrenal capsular membranes (adrenal cortex)More data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/Type-1 angiotensin II receptor B/Type-2 angiotensin II receptor(RAT)
Istituto Lusofarmaco
Curated by ChEMBL
Istituto Lusofarmaco
Curated by ChEMBL
Affinity DataIC50: 170nMAssay Description:Ability to displace [125I]-labeled angiotensin II from its receptor of a rat uterus membraneMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/Type-1 angiotensin II receptor B/Type-2 angiotensin II receptor(RAT)
Istituto Lusofarmaco
Curated by ChEMBL
Istituto Lusofarmaco
Curated by ChEMBL
Affinity DataIC50: 230nMAssay Description:Inhibition of radioligand [3H]angiotensin II binding to angiotensin II receptor of rat adrenal cortical membraneMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/Type-1 angiotensin II receptor B/Type-2 angiotensin II receptor(RAT)
Istituto Lusofarmaco
Curated by ChEMBL
Istituto Lusofarmaco
Curated by ChEMBL
Affinity DataIC50: 330nMAssay Description:Ability to displace [125I]-labeled angiotensin II from its receptor of a rat uterus membraneMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/Type-1 angiotensin II receptor B/Type-2 angiotensin II receptor(RAT)
Istituto Lusofarmaco
Curated by ChEMBL
Istituto Lusofarmaco
Curated by ChEMBL
Affinity DataIC50: 330nMAssay Description:Ability to displace [125I]-labeled angiotensin II from its receptor of a rat uterus membraneMore data for this Ligand-Target Pair