TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Kyoto Pharmaceutical University
Curated by ChEMBL
Kyoto Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 0.00240nMAssay Description:Inhibition of HIV1 recombinant protease after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Kyoto Pharmaceutical University
Curated by ChEMBL
Kyoto Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 0.0310nMAssay Description:Inhibition of HIV1 recombinant protease after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Inhibition of influenza B/Memphis/3/89 neuraminidaseMore data for this Ligand-Target Pair
Affinity DataKi: 0.140nMAssay Description:Inhibition of influenza B/Memphis/3/89 neuraminidaseMore data for this Ligand-Target Pair
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Kyoto Pharmaceutical University
Curated by ChEMBL
Kyoto Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 0.190nMAssay Description:Inhibition of HIV1 recombinant protease after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Inhibition of influenza B/Memphis/3/89 neuraminidaseMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Inhibition of influenza B/Memphis/3/89 neuraminidaseMore data for this Ligand-Target Pair
Affinity DataKi: 0.670nMAssay Description:Inhibition of influenza B/Memphis/3/89 neuraminidaseMore data for this Ligand-Target Pair
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Kyoto Pharmaceutical University
Curated by ChEMBL
Kyoto Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 0.830nMAssay Description:Inhibition of HIV1 recombinant protease after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.840nMAssay Description:Displacement of [3H]nisoxetine from NET in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Inhibition of influenza B/Memphis/3/89 neuraminidaseMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Inhibition of influenza B/Memphis/3/89 neuraminidaseMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Inhibition of influenza B/Memphis/3/89 neuraminidaseMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Inhibition of influenza B/Memphis/3/89 neuraminidaseMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Inhibition of influenza B/Memphis/3/89 neuraminidaseMore data for this Ligand-Target Pair
Affinity DataKi: 2.47nMAssay Description:Displacement of [3H]nisoxetine from NET in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2.80nMAssay Description:Inhibition of influenza B/Memphis/3/89 neuraminidaseMore data for this Ligand-Target Pair
Affinity DataKi: 4.80nMAssay Description:Inhibition of influenza B/Memphis/3/89 neuraminidaseMore data for this Ligand-Target Pair
Affinity DataKi: 6.5nMAssay Description:Inhibition of influenza B/Memphis/3/89 neuraminidaseMore data for this Ligand-Target Pair
Affinity DataKi: 9.30nMAssay Description:Inhibition of influenza B/Memphis/3/89 neuraminidaseMore data for this Ligand-Target Pair
Affinity DataKi: 10.3nMAssay Description:Inhibition of influenza B/Memphis/3/89 neuraminidaseMore data for this Ligand-Target Pair
Affinity DataKi: 10.6nMAssay Description:Inhibition of influenza B/Memphis/3/89 neuraminidaseMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Inhibition of influenza B/Memphis/3/89 neuraminidaseMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Institute For Degenerative Diseases
Curated by ChEMBL
Institute For Degenerative Diseases
Curated by ChEMBL
Affinity DataKi: 14.2nMAssay Description:Displacement of [3H]GBR from DAT in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 15.4nMAssay Description:Displacement of [3H]nisoxetine from NET in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 17.5nMAssay Description:Inhibition of influenza B/Memphis/3/89 neuraminidaseMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:A fluorogenic assay was used to measure influenza virus neuraminidase activity. The substrate, 4-methylumbelliferyl-N-acetylneuraminic acid, is cleav...More data for this Ligand-Target Pair
Affinity DataKi: 21nMAssay Description:Inhibition of influenza B/Memphis/3/89 neuraminidaseMore data for this Ligand-Target Pair
Affinity DataKi: 24.2nMAssay Description:Inhibition of influenza B/Memphis/3/89 neuraminidaseMore data for this Ligand-Target Pair
Affinity DataKi: 27.6nMAssay Description:Displacement of [3H]nisoxetine from NET in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Inhibition of influenza B/Memphis/3/89 neuraminidaseMore data for this Ligand-Target Pair
Affinity DataKi: 28.5nMAssay Description:Displacement of [3H]nisoxetine from NET in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 29nMAssay Description:Inhibition of influenza B/Memphis/3/89 neuraminidaseMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:A fluorogenic assay was used to measure influenza virus neuraminidase activity. The substrate, 4-methylumbelliferyl-N-acetylneuraminic acid, is cleav...More data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Inhibition of influenza B/Memphis/3/89 neuraminidaseMore data for this Ligand-Target Pair
Affinity DataKi: 38nMAssay Description:Inhibition of influenza B/Memphis/3/89 neuraminidaseMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Institute For Degenerative Diseases
Curated by ChEMBL
Institute For Degenerative Diseases
Curated by ChEMBL
Affinity DataKi: 40.4nMAssay Description:Displacement of [3H]paroxetine from SERT in brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 45nM ΔG°: -41.5kJ/molepH: 7.5 T: 2°CAssay Description:A fluorogenic assay was used to measure influenza virus neuraminidase activity. The substrate, 4-methylumbelliferyl-N-acetylneuraminic acid, is cleav...More data for this Ligand-Target Pair
Affinity DataKi: 46nMAssay Description:Inhibition of influenza B/Memphis/3/89 neuraminidaseMore data for this Ligand-Target Pair
Affinity DataKi: 49nMAssay Description:Inhibition of influenza B/Memphis/3/89 neuraminidaseMore data for this Ligand-Target Pair
Affinity DataKi: 57nM ΔG°: -40.9kJ/molepH: 7.5 T: 2°CAssay Description:A fluorogenic assay was used to measure influenza virus neuraminidase activity. The substrate, 4-methylumbelliferyl-N-acetylneuraminic acid, is cleav...More data for this Ligand-Target Pair
Affinity DataKi: 70.4nMAssay Description:Displacement of [3H]nisoxetine from NET in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 71.9nMAssay Description:Displacement of [3H]nisoxetine from NET in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 73.8nMAssay Description:Displacement of [3H]nisoxetine from NET in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 79nMAssay Description:A fluorogenic assay was used to measure influenza virus neuraminidase activity. The substrate, 4-methylumbelliferyl-N-acetylneuraminic acid, is cleav...More data for this Ligand-Target Pair
Affinity DataKi: 79.6nMAssay Description:Displacement of [3H]nisoxetine from NET in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 85nMAssay Description:Inhibition of influenza B/Memphis/3/89 neuraminidaseMore data for this Ligand-Target Pair
Affinity DataKi: 86nMAssay Description:Inhibition of influenza B/Memphis/3/89 neuraminidaseMore data for this Ligand-Target Pair
Affinity DataKi: 101nMAssay Description:Displacement of [3H]nisoxetine from NET in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 110nMAssay Description:Inhibition of influenza B/Memphis/3/89 neuraminidaseMore data for this Ligand-Target Pair