Affinity DataKi: 240nMAssay Description:In vitro inhibitory activity against human neutrophil leukotriene B4 (LTB4)More data for this Ligand-Target Pair
Affinity DataKi: 280nMAssay Description:In vitro antagonist activity against leukotriene B4 (LTB4) receptor in [3H]-LTB4 human neutrophil receptor binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 330nMAssay Description:In vitro inhibitory activity against human neutrophil leukotriene B4 (LTB4)More data for this Ligand-Target Pair
Affinity DataKi: 650nMAssay Description:Inhibition of [3H]-LTD4 binding to LTD4 receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+3nMAssay Description:In vitro inhibitory activity against leukotriene D4 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.30E+3nMAssay Description:In vitro inhibitory activity against leukotriene D4 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.50E+3nMAssay Description:Inhibition of [3H]-LTD4 binding to LTD4 receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.60E+3nMAssay Description:In vitro inhibitory activity against human leukotriene D4 (LTD4)More data for this Ligand-Target Pair
Affinity DataKi: 1.90E+3nMAssay Description:In vitro inhibitory activity against human neutrophil leukotriene B4 (LTB4)More data for this Ligand-Target Pair
Affinity DataKi: 3.30E+3nMAssay Description:In vitro inhibitory activity against human neutrophil leukotriene B4 (LTB4)More data for this Ligand-Target Pair
Affinity DataKi: 4.10E+3nMAssay Description:In vitro inhibitory activity against leukotriene D4 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5.20E+3nMAssay Description:In vitro inhibitory activity against human neutrophil leukotriene B4 (LTB4)More data for this Ligand-Target Pair
Affinity DataKi: 6.80E+3nMAssay Description:Inhibition of [3H]-LTD4 binding to LTD4 receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 8.00E+3nMAssay Description:Inhibition of [3H]-LTD4 binding to LTD4 receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.60E+4nMAssay Description:In vitro inhibitory activity against human neutrophil leukotriene B4 (LTB4)More data for this Ligand-Target Pair
Affinity DataKi: 2.40E+4nMAssay Description:Inhibition of [3H]-LTD4 binding to LTD4 receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 3.80E+4nMAssay Description:In vitro inhibitory activity against human neutrophil leukotriene B4 (LTB4)More data for this Ligand-Target Pair
Affinity DataKi: 3.80E+4nMAssay Description:In vitro inhibitory activity against human neutrophil leukotriene B4 (LTB4)More data for this Ligand-Target Pair
Affinity DataKi: 3.90E+4nMAssay Description:In vitro inhibitory activity was evaluated against leukotriene B4 (LTB4) in guinea pig binding assayMore data for this Ligand-Target Pair
Affinity DataKi: >5.00E+4nMAssay Description:In vitro inhibitory activity against leukotriene D4 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >5.00E+4nMAssay Description:In vitro inhibitory activity against leukotriene D4 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >5.00E+4nMAssay Description:In vitro inhibitory activity against leukotriene D4 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >5.00E+4nMAssay Description:In vitro inhibitory activity against leukotriene D4 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >5.00E+4nMAssay Description:In vitro inhibitory activity against leukotriene D4 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 5.60nMAssay Description:Tested for binding activity against [3H]-LTB4 to whole human neutrophil with halh maximal inhibitionMore data for this Ligand-Target Pair
Affinity DataIC50: 9.70nMAssay Description:Tested for antagonistic activity against LTB4 receptor in guinea pig spleen membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 30.3nMAssay Description:Tested for antagonistic activity in mouse spleen membrane against LTB4 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 140nMAssay Description:In vitro inhibitory activity against human neutrophil leukotriene B4 (LTB4) induced ChemotaxisMore data for this Ligand-Target Pair
Affinity DataIC50: 150nMAssay Description:Inhibition of 5-Lipoxygenase (5-LO) in rat basophilic leukemic cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 220nMAssay Description:In vitro inhibitory activity against human neutrophil leukotriene B4 (LTB4) induced ChemotaxisMore data for this Ligand-Target Pair
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of 5-Lipoxygenase (5-LO) in rat basophilic leukemia cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 3.40E+3nMAssay Description:In vitro inhibitory activity against human neutrophil leukotriene B4 (LTB4) induced ChemotaxisMore data for this Ligand-Target Pair
Affinity DataIC50: 6.10E+3nMAssay Description:In vitro inhibitory activity against human neutrophil leukotriene B4 (LTB4) induced ChemotaxisMore data for this Ligand-Target Pair
Affinity DataIC50: 8.10E+3nMAssay Description:Inhibition of 5-Lipoxygenase (5-LO) in rat basophilic leukemia cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+4nMAssay Description:In vitro inhibitory activity against human neutrophil leukotriene B4 (LTB4) induced ChemotaxisMore data for this Ligand-Target Pair
Affinity DataIC50: 3.80E+4nMAssay Description:In vitro inhibitory activity against human neutrophil leukotriene B4 (LTB4) induced ChemotaxisMore data for this Ligand-Target Pair