Found 72 with Last Name = 'bretner' and Initial = 'm' 
Affinity DataKi: 10nMAssay Description:Apparent Ki value of the compound was measured by competitive inhibition of Thymidylate Synthases from Ehrlich Carcinoma cells of mouseMore data for this Ligand-Target Pair
3D Structure (crystal)Affinity DataKi: 20nMAssay Description:Time-independent inhibition of thymidylate synthase from parenteral L1210 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Apparent Ki value of the compound was measured by competitive inhibition of Thymidylate Synthases from L1210 cells of mouseMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Time-independent inhibition of thymidylate synthase from FdUrd-resistant L1210 cellsMore data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Warsaw University Of Technology
Curated by ChEMBL
Warsaw University Of Technology
Curated by ChEMBL
Affinity DataKi: 40nMAssay Description:Binding affinity to CK2alpha (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 70nMAssay Description:Apparent Ki value of the compound was measured by competitive inhibition of Thymidylate Synthase from L1210 cells of mouseMore data for this Ligand-Target Pair
Affinity DataKi: 140nMAssay Description:Apparent Ki value of the compound was measured by competitive inhibition of Thymidylate Synthase from Ehrlich Carcinoma cells of mouseMore data for this Ligand-Target Pair
Affinity DataKi: 150nMAssay Description:Time-independent inhibition of thymidylate synthase from FdUrd-resistant L1210 cellsMore data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Warsaw University Of Technology
Curated by ChEMBL
Warsaw University Of Technology
Curated by ChEMBL
Affinity DataKi: 270nMAssay Description:The activity of CK2α was tested using P81 filter isotopic assay, as it was described earlier [Łukowska-Chojnacka et al., Bioorg. Med. Chem....More data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:Time-independent inhibition of thymidylate synthase from parenteral L1210 cellsMore data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Warsaw University Of Technology
Curated by ChEMBL
Warsaw University Of Technology
Curated by ChEMBL
Affinity DataKi: 400nMAssay Description:Binding affinity to CK2alpha (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 460nMAssay Description:Time-independent inhibition of thymidylate synthase from FdUrd-resistant L1210 cellsMore data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Warsaw University Of Technology
Curated by ChEMBL
Warsaw University Of Technology
Curated by ChEMBL
Affinity DataKi: 680nMAssay Description:The activity of CK2α was tested using P81 filter isotopic assay, as it was described earlier [Łukowska-Chojnacka et al., Bioorg. Med. Chem....More data for this Ligand-Target Pair
Affinity DataKi: 800nMAssay Description:Time-independent inhibition of thymidylate synthase from parenteral L1210 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 900nMAssay Description:Time-independent inhibition of thymidylate synthase from FdUrd-resistant L1210 cellsMore data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Warsaw University Of Technology
Curated by ChEMBL
Warsaw University Of Technology
Curated by ChEMBL
Affinity DataKi: 910nMAssay Description:The activity of CK2α was tested using P81 filter isotopic assay, as it was described earlier [Łukowska-Chojnacka et al., Bioorg. Med. Chem....More data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Warsaw University Of Technology
Curated by ChEMBL
Warsaw University Of Technology
Curated by ChEMBL
Affinity DataKi: 1.03E+3nMAssay Description:Inhibition of recombinant human CK2alpha using RRRDDDSDDD substrate peptide by scintillation counter in presence of [32P]ATPMore data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Warsaw University Of Technology
Curated by ChEMBL
Warsaw University Of Technology
Curated by ChEMBL
Affinity DataKi: 1.11E+3nMAssay Description:Inhibition of recombinant human CK2alpha using RRRDDDSDDD substrate peptide by scintillation counter in presence of [32P]ATPMore data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Warsaw University Of Technology
Curated by ChEMBL
Warsaw University Of Technology
Curated by ChEMBL
Affinity DataKi: 1.27E+3nMAssay Description:Inhibition of recombinant human CK2alpha using RRRDDDSDDD substrate peptide by scintillation counter in presence of [32P]ATPMore data for this Ligand-Target Pair
Affinity DataKi: 1.40E+3nMAssay Description:Time-independent inhibition of thymidylate synthase from FdUrd-resistant L1210 cellsMore data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Warsaw University Of Technology
Curated by ChEMBL
Warsaw University Of Technology
Curated by ChEMBL
Affinity DataKi: 1.42E+3nMAssay Description:Inhibition of recombinant human CK2alpha using RRRDDDSDDD substrate peptide by scintillation counter in presence of [32P]ATPMore data for this Ligand-Target Pair
Affinity DataKi: 1.50E+3nMAssay Description:Time-independent inhibition of thymidylate synthase from parenteral L1210 cellsMore data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Warsaw University Of Technology
Curated by ChEMBL
Warsaw University Of Technology
Curated by ChEMBL
Affinity DataKi: 1.63E+3nMAssay Description:Inhibition of recombinant human CK2alpha using RRRDDDSDDD substrate peptide by scintillation counter in presence of [32P]ATPMore data for this Ligand-Target Pair
Affinity DataKi: 1.70E+3nMAssay Description:Time-independent inhibition of thymidylate synthase from parenteral L1210 cellsMore data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Warsaw University Of Technology
Curated by ChEMBL
Warsaw University Of Technology
Curated by ChEMBL
Affinity DataKi: 1.78E+3nMAssay Description:The activity of CK2α was tested using P81 filter isotopic assay, as it was described earlier [Łukowska-Chojnacka et al., Bioorg. Med. Chem....More data for this Ligand-Target Pair
Affinity DataKi: 1.91E+3nMAssay Description:Time-independent inhibition of thymidylate synthase from parenteral L1210 cellsMore data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Warsaw University Of Technology
Curated by ChEMBL
Warsaw University Of Technology
Curated by ChEMBL
Affinity DataKi: 1.96E+3nMAssay Description:The activity of CK2α was tested using P81 filter isotopic assay, as it was described earlier [Łukowska-Chojnacka et al., Bioorg. Med. Chem....More data for this Ligand-Target Pair
Affinity DataKi: 2.18E+3nMAssay Description:Time-independent inhibition of thymidylate synthase from FdUrd-resistant L1210 cellsMore data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Warsaw University Of Technology
Curated by ChEMBL
Warsaw University Of Technology
Curated by ChEMBL
Affinity DataKi: 2.26E+3nMAssay Description:The activity of CK2α was tested using P81 filter isotopic assay, as it was described earlier [Łukowska-Chojnacka et al., Bioorg. Med. Chem....More data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Warsaw University Of Technology
Curated by ChEMBL
Warsaw University Of Technology
Curated by ChEMBL
Affinity DataKi: 2.34E+3nMAssay Description:The activity of CK2α was tested using P81 filter isotopic assay, as it was described earlier [Łukowska-Chojnacka et al., Bioorg. Med. Chem....More data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Warsaw University Of Technology
Curated by ChEMBL
Warsaw University Of Technology
Curated by ChEMBL
Affinity DataKi: 2.37E+3nMAssay Description:The activity of CK2α was tested using P81 filter isotopic assay, as it was described earlier [Łukowska-Chojnacka et al., Bioorg. Med. Chem....More data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Warsaw University Of Technology
Curated by ChEMBL
Warsaw University Of Technology
Curated by ChEMBL
Affinity DataKi: 2.42E+3nMAssay Description:Inhibition of recombinant human CK2alpha using RRRDDDSDDD substrate peptide by scintillation counter in presence of [32P]ATPMore data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Warsaw University Of Technology
Curated by ChEMBL
Warsaw University Of Technology
Curated by ChEMBL
Affinity DataKi: 2.47E+3nMAssay Description:The activity of CK2α was tested using P81 filter isotopic assay, as it was described earlier [Łukowska-Chojnacka et al., Bioorg. Med. Chem....More data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Warsaw University Of Technology
Curated by ChEMBL
Warsaw University Of Technology
Curated by ChEMBL
Affinity DataKi: 2.49E+3nMAssay Description:Inhibition of recombinant human CK2alpha using RRRDDDSDDD substrate peptide by scintillation counter in presence of [32P]ATPMore data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Warsaw University Of Technology
Curated by ChEMBL
Warsaw University Of Technology
Curated by ChEMBL
Affinity DataKi: 2.51E+3nMAssay Description:Inhibition of recombinant human CK2alpha using RRRDDDSDDD substrate peptide by scintillation counter in presence of [32P]ATPMore data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Warsaw University Of Technology
Curated by ChEMBL
Warsaw University Of Technology
Curated by ChEMBL
Affinity DataKi: 2.77E+3nMAssay Description:Inhibition of recombinant human CK2alpha using RRRDDDSDDD substrate peptide by scintillation counter in presence of [32P]ATPMore data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Warsaw University Of Technology
Curated by ChEMBL
Warsaw University Of Technology
Curated by ChEMBL
Affinity DataKi: 3.16E+3nMAssay Description:The activity of CK2α was tested using P81 filter isotopic assay, as it was described earlier [Łukowska-Chojnacka et al., Bioorg. Med. Chem....More data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Warsaw University Of Technology
Curated by ChEMBL
Warsaw University Of Technology
Curated by ChEMBL
Affinity DataKi: 3.28E+3nMAssay Description:The activity of CK2α was tested using P81 filter isotopic assay, as it was described earlier [Łukowska-Chojnacka et al., Bioorg. Med. Chem....More data for this Ligand-Target Pair
Affinity DataKi: 3.70E+3nMAssay Description:Time-independent inhibition of thymidylate synthase from parenteral L1210 cellsMore data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Warsaw University Of Technology
Curated by ChEMBL
Warsaw University Of Technology
Curated by ChEMBL
Affinity DataKi: 5.03E+3nMAssay Description:Inhibition of recombinant human CK2alpha using RRRDDDSDDD substrate peptide by scintillation counter in presence of [32P]ATPMore data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Homo sapiens (Human))
Warsaw University Of Technology
Curated by ChEMBL
Warsaw University Of Technology
Curated by ChEMBL
Affinity DataKi: 5.37E+3nMAssay Description:The activity of CK2α was tested using P81 filter isotopic assay, as it was described earlier [Łukowska-Chojnacka et al., Bioorg. Med. Chem....More data for this Ligand-Target Pair
Affinity DataKi: 5.70E+3nMAssay Description:Time-independent inhibition of thymidylate synthase from FdUrd-resistant L1210 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 6.99E+3nMAssay Description:Time-independent inhibition of thymidylate synthase from FdUrd-resistant L1210 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 7.30E+3nMAssay Description:Time-independent inhibition of thymidylate synthase from parenteral L1210 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 7.46E+3nMAssay Description:Time-independent inhibition of thymidylate synthase from parenteral L1210 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 7.68E+3nMAssay Description:Time-independent inhibition of thymidylate synthase from parenteral L1210 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 8.40E+3nMAssay Description:Time-independent inhibition of thymidylate synthase from FdUrd-resistant L1210 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 8.50E+3nMAssay Description:Time-independent inhibition of thymidylate synthase from parenteral L1210 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 9.30E+3nMAssay Description:Time-independent inhibition of thymidylate synthase from FdUrd-resistant L1210 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.21E+4nMAssay Description:Time-independent inhibition of thymidylate synthase from parenteral L1210 cellsMore data for this Ligand-Target Pair
