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Found 80 with Last Name = 'brownell' and Initial = 'j'
TargetLactoylglutathione lyase(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50241121((S)-5-((R)-3-(4-bromobenzylthio)-1-(carboxymethyla...)
Affinity DataKi:  9.14E+3nMpH: 6.6Assay Description:Ability to inhibit yeast glyoxalase I enzyme in 0.05 M phosphate buffer, pH 6.6, 30 degree CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine deaminase(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50088426((1R,2S,3R,5R)-3-(6-amino-9H-purin-9-yl)-5-(hydroxy...)
Affinity DataKi:  9.90E+3nMAssay Description:Compound was evaluated for competitive inhibition of adenosine deaminase and expressed as KiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLactoylglutathione lyase(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50076046(2-Amino-3-{3-[2-(4-bromo-benzylsulfanyl)-1-(carbox...)
Affinity DataKi:  1.55E+4nMpH: 6.6Assay Description:Ability to inhibit yeast glyoxalase I enzyme in 0.05 M phosphate buffer, pH 6.6, 30 degree CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUbiquitin-like modifier-activating enzyme 1 [957-994](Homo sapiens (Human))
Millennium Pharmaceuticals

LigandPNGBDBM92475(Compound I)
Affinity DataIC50:  10.2nMAssay Description:Inhibition assay using ubiquitin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUbiquitin-like modifier-activating enzyme ATG7(Homo sapiens (Human))
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM475984(US10865208, Compound I-42 | {(2R,3S,4R,5R)-5-[4-am...)
Affinity DataIC50:  14nMAssay Description:Inhibition of recombinant His-tagged human ATG7 incubated for 105 mins in presence of GST-tagged ATG3 and Flag-tagged Gabarap and measured after 2 hr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUbiquitin-like modifier-activating enzyme ATG7(Homo sapiens (Human))
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM475978(US10865208, Compound I-36 | {(2R,3S,4R,5R)-5-[4-am...)
Affinity DataIC50:  16nMAssay Description:Inhibition of recombinant His-tagged human ATG7 incubated for 105 mins in presence of GST-tagged ATG3 and Flag-tagged Gabarap and measured after 2 hr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUbiquitin-like modifier-activating enzyme ATG7(Homo sapiens (Human))
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM476001(US10865208, Compound I-58 | {(2R,3S,4R,5R)-5-[4-am...)
Affinity DataIC50:  17nMAssay Description:Inhibition of recombinant His-tagged human ATG7 incubated for 105 mins in presence of GST-tagged ATG3 and Flag-tagged Gabarap and measured after 2 hr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUbiquitin-like modifier-activating enzyme ATG7(Homo sapiens (Human))
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM476012(US10865208, Compound I-69 | [(2R,3S,4R,5R)-5-{4-am...)
Affinity DataIC50:  18nMAssay Description:Inhibition of recombinant His-tagged human ATG7 incubated for 105 mins in presence of GST-tagged ATG3 and Flag-tagged Gabarap and measured after 2 hr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUbiquitin-like modifier-activating enzyme ATG7(Homo sapiens (Human))
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM476084(US10865208, Compound I-139 | {(2R,3R,4S,5R)-5-[4-a...)
Affinity DataIC50:  20nMAssay Description:Inhibition of recombinant His-tagged human ATG7 incubated for 105 mins in presence of GST-tagged ATG3 and Flag-tagged Gabarap and measured after 2 hr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUbiquitin-like modifier-activating enzyme ATG7(Homo sapiens (Human))
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM475993(US10865208, Compound I-51 | {(2R,3S,4R,5R)-5-[4-am...)
Affinity DataIC50:  22nMAssay Description:Inhibition of recombinant His-tagged human ATG7 incubated for 105 mins in presence of GST-tagged ATG3 and Flag-tagged Gabarap and measured after 2 hr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUbiquitin-like modifier-activating enzyme ATG7(Homo sapiens (Human))
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM475994(US10865208, Compound I-52 | {(2R,3S,4R,5R)-5-[4-am...)
Affinity DataIC50:  23nMAssay Description:Inhibition of recombinant His-tagged human ATG7 incubated for 105 mins in presence of GST-tagged ATG3 and Flag-tagged Gabarap and measured after 2 hr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUbiquitin-like modifier-activating enzyme ATG7(Homo sapiens (Human))
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM476126(US10865208, Compound I-181 | {(2R,3S,5R)-5-[4-amin...)
Affinity DataIC50:  27nMAssay Description:Inhibition of recombinant His-tagged human ATG7 incubated for 105 mins in presence of GST-tagged ATG3 and Flag-tagged Gabarap and measured after 2 hr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUbiquitin-like modifier-activating enzyme ATG7(Homo sapiens (Human))
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM475969(US10865208, Compound I-27 | {(2R,3S,4R,5R)-5-[4-am...)
Affinity DataIC50:  29nMAssay Description:Inhibition of recombinant His-tagged human ATG7 incubated for 105 mins in presence of GST-tagged ATG3 and Flag-tagged Gabarap and measured after 2 hr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUbiquitin-like modifier-activating enzyme ATG7(Homo sapiens (Human))
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM476025(US10865208, Compound I-82 | {(2R,3S,4R,5R)-5-[4-am...)
Affinity DataIC50:  29nMAssay Description:Inhibition of recombinant His-tagged human ATG7 incubated for 105 mins in presence of GST-tagged ATG3 and Flag-tagged Gabarap and measured after 2 hr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUbiquitin-like modifier-activating enzyme ATG7(Homo sapiens (Human))
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM476049(US10865208, Compound I-106 | [(2R,3R,4S,5R)-5-{4-a...)
Affinity DataIC50:  31nMAssay Description:Inhibition of recombinant His-tagged human ATG7 incubated for 105 mins in presence of GST-tagged ATG3 and Flag-tagged Gabarap and measured after 2 hr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUbiquitin-like modifier-activating enzyme ATG7(Homo sapiens (Human))
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM476086(US10865208, Compound I-141 | [(2R,3R,4S,5R)-5-{4-a...)
Affinity DataIC50:  35nMAssay Description:Inhibition of recombinant His-tagged human ATG7 incubated for 105 mins in presence of GST-tagged ATG3 and Flag-tagged Gabarap and measured after 2 hr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUbiquitin-like modifier-activating enzyme ATG7(Homo sapiens (Human))
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM476058(US10865208, Compound I-115 | {(2R,3R,4S,5R)-5-[4-a...)
Affinity DataIC50:  41nMAssay Description:Inhibition of recombinant His-tagged human ATG7 incubated for 105 mins in presence of GST-tagged ATG3 and Flag-tagged Gabarap and measured after 2 hr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUbiquitin-like modifier-activating enzyme ATG7(Homo sapiens (Human))
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM476042(US10865208, Compound I-99 | {(2R,3R,4S,5R)-5-[4-am...)
Affinity DataIC50:  43nMAssay Description:Inhibition of recombinant His-tagged human ATG7 incubated for 105 mins in presence of GST-tagged ATG3 and Flag-tagged Gabarap and measured after 2 hr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUbiquitin-like modifier-activating enzyme ATG7(Homo sapiens (Human))
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM476058(US10865208, Compound I-115 | {(2R,3R,4S,5R)-5-[4-a...)
Affinity DataIC50:  47nMAssay Description:Inhibition of ATG7 in human 293HEK cells assessed as inhibition of ATG7:ATG8 thioester formation after 8 hrs by Western blot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUbiquitin-like modifier-activating enzyme ATG7(Homo sapiens (Human))
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM476145(US10865208, Compound I-200 | {(2R,3S,5R)-5-[4-amin...)
Affinity DataIC50:  48nMAssay Description:Inhibition of recombinant His-tagged human ATG7 incubated for 105 mins in presence of GST-tagged ATG3 and Flag-tagged Gabarap and measured after 2 hr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUbiquitin-like modifier-activating enzyme ATG7(Homo sapiens (Human))
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM476086(US10865208, Compound I-141 | [(2R,3R,4S,5R)-5-{4-a...)
Affinity DataIC50:  51nMAssay Description:Inhibition of ATG7 in human 293HEK cells assessed as inhibition of ATG7:ATG8 thioester formation after 8 hrs by Western blot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUbiquitin-like modifier-activating enzyme ATG7(Homo sapiens (Human))
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM476117(US10865208, Compound I-172 | {(2R,3S,5R)-5-[4-amin...)
Affinity DataIC50:  52nMAssay Description:Inhibition of recombinant His-tagged human ATG7 incubated for 105 mins in presence of GST-tagged ATG3 and Flag-tagged Gabarap and measured after 2 hr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUbiquitin-like modifier-activating enzyme ATG7(Homo sapiens (Human))
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM476049(US10865208, Compound I-106 | [(2R,3R,4S,5R)-5-{4-a...)
Affinity DataIC50:  56nMAssay Description:Inhibition of ATG7 in human 293HEK cells assessed as inhibition of ATG7:ATG8 thioester formation after 8 hrs by Western blot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUbiquitin-like modifier-activating enzyme ATG7(Homo sapiens (Human))
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM476084(US10865208, Compound I-139 | {(2R,3R,4S,5R)-5-[4-a...)
Affinity DataIC50:  56nMAssay Description:Inhibition of ATG7 in human 293HEK cells assessed as inhibition of ATG7:ATG8 thioester formation after 8 hrs by Western blot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUbiquitin-like modifier-activating enzyme ATG7(Homo sapiens (Human))
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM476165(US10865208, Compound I-220 | {(2S,3S,5R)-5-[4-amin...)
Affinity DataIC50:  57nMAssay Description:Inhibition of recombinant His-tagged human ATG7 incubated for 105 mins in presence of GST-tagged ATG3 and Flag-tagged Gabarap and measured after 2 hr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUbiquitin-like modifier-activating enzyme ATG7(Homo sapiens (Human))
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM50561267(CHEMBL4754045)
Affinity DataIC50:  62nMAssay Description:Inhibition of recombinant His-tagged human ATG7 incubated for 105 mins in presence of GST-tagged ATG3 and Flag-tagged Gabarap and measured after 2 hr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUbiquitin-like modifier-activating enzyme ATG7(Homo sapiens (Human))
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM476105(US10865208, Compound I-160 | {(2R,3S,5R)-5-[4-amin...)
Affinity DataIC50:  66nMAssay Description:Inhibition of recombinant His-tagged human ATG7 incubated for 105 mins in presence of GST-tagged ATG3 and Flag-tagged Gabarap and measured after 2 hr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUbiquitin-like modifier-activating enzyme ATG7(Homo sapiens (Human))
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM476106(US10865208, Compound I-161 | US10865208, Compound ...)
Affinity DataIC50:  80nMAssay Description:Inhibition of recombinant His-tagged human ATG7 incubated for 105 mins in presence of GST-tagged ATG3 and Flag-tagged Gabarap and measured after 2 hr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUbiquitin-like modifier-activating enzyme ATG7(Homo sapiens (Human))
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM475984(US10865208, Compound I-42 | {(2R,3S,4R,5R)-5-[4-am...)
Affinity DataIC50:  83nMAssay Description:Inhibition of ATG7 in human 293HEK cells assessed as inhibition of ATG7:ATG8 thioester formation after 8 hrs by Western blot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUbiquitin-like modifier-activating enzyme ATG7(Homo sapiens (Human))
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM50561266(CHEMBL4740719)
Affinity DataIC50:  84nMAssay Description:Inhibition of recombinant His-tagged human ATG7 incubated for 105 mins in presence of GST-tagged ATG3 and Flag-tagged Gabarap and measured after 2 hr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUbiquitin-like modifier-activating enzyme ATG7(Homo sapiens (Human))
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM476145(US10865208, Compound I-200 | {(2R,3S,5R)-5-[4-amin...)
Affinity DataIC50:  86nMAssay Description:Inhibition of ATG7 in human 293HEK cells assessed as inhibition of ATG7:ATG8 thioester formation after 8 hrs by Western blot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUbiquitin-like modifier-activating enzyme ATG7(Homo sapiens (Human))
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM475937(US10865208, Compound I-1 | [(2R,3S,4R,5R)-5-(4-ami...)
Affinity DataIC50:  89nMAssay Description:Inhibition of recombinant His-tagged human ATG7 incubated for 105 mins in presence of GST-tagged ATG3 and Flag-tagged Gabarap and measured after 2 hr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUbiquitin-like modifier-activating enzyme 1 [957-994](Homo sapiens (Human))
Millennium Pharmaceuticals

LigandPNGBDBM92475(Compound I)
Affinity DataIC50:  90.8nMAssay Description:Inhibition assay using ubiquitin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUbiquitin-like modifier-activating enzyme ATG7(Homo sapiens (Human))
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM476150(US10865208, Compound I-205 | [(2R,3S,5R)-5-{4-amin...)
Affinity DataIC50:  95nMAssay Description:Inhibition of recombinant His-tagged human ATG7 incubated for 105 mins in presence of GST-tagged ATG3 and Flag-tagged Gabarap and measured after 2 hr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUbiquitin-like modifier-activating enzyme ATG7(Homo sapiens (Human))
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM476140(US10865208, Compound I-195 | {(2R,3S,5R)-5-[4-amin...)
Affinity DataIC50:  100nMAssay Description:Inhibition of recombinant His-tagged human ATG7 incubated for 105 mins in presence of GST-tagged ATG3 and Flag-tagged Gabarap and measured after 2 hr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUbiquitin-like modifier-activating enzyme ATG7(Homo sapiens (Human))
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM476124(US10865208, Compound I-179 | [(2R,3S,5R)-5-{4-amin...)
Affinity DataIC50:  104nMAssay Description:Inhibition of recombinant His-tagged human ATG7 incubated for 105 mins in presence of GST-tagged ATG3 and Flag-tagged Gabarap and measured after 2 hr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUbiquitin-like modifier-activating enzyme ATG7(Homo sapiens (Human))
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM476164(US10865208, Compound I-219 | {(2S,3S,5R)-5-[4-amin...)
Affinity DataIC50:  124nMAssay Description:Inhibition of recombinant His-tagged human ATG7 incubated for 105 mins in presence of GST-tagged ATG3 and Flag-tagged Gabarap and measured after 2 hr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUbiquitin-like modifier-activating enzyme ATG7(Homo sapiens (Human))
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM476038(US10865208, Compound I-95 | {(2S,3S,4R,5R)-5-[4-am...)
Affinity DataIC50:  129nMAssay Description:Inhibition of recombinant His-tagged human ATG7 incubated for 105 mins in presence of GST-tagged ATG3 and Flag-tagged Gabarap and measured after 2 hr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUbiquitin-like modifier-activating enzyme ATG7(Homo sapiens (Human))
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM476086(US10865208, Compound I-141 | [(2R,3R,4S,5R)-5-{4-a...)
Affinity DataIC50:  140nMAssay Description:Inhibition of ATG7 in human 293HEK cells assessed as inhibition of ATG7:ATG8 thioester formation after 4 hrs by Western blot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUbiquitin-like modifier-activating enzyme ATG7(Homo sapiens (Human))
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM476039(US10865208, Compound I-96 | {(2S,3R,4S,5R)-5-[4-am...)
Affinity DataIC50:  145nMAssay Description:Inhibition of recombinant His-tagged human ATG7 incubated for 105 mins in presence of GST-tagged ATG3 and Flag-tagged Gabarap and measured after 2 hr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUbiquitin-like modifier-activating enzyme ATG7(Homo sapiens (Human))
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM476126(US10865208, Compound I-181 | {(2R,3S,5R)-5-[4-amin...)
Affinity DataIC50:  150nMAssay Description:Inhibition of ATG7 in human 293HEK cells assessed as inhibition of ATG7:ATG8 thioester formation after 8 hrs by Western blot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUbiquitin-like modifier-activating enzyme ATG7(Homo sapiens (Human))
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM476161(US10865208, Compound I-216 | {(2S,3S,5R)-5-[4-amin...)
Affinity DataIC50:  156nMAssay Description:Inhibition of recombinant His-tagged human ATG7 incubated for 105 mins in presence of GST-tagged ATG3 and Flag-tagged Gabarap and measured after 2 hr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUbiquitin-like modifier-activating enzyme ATG7(Homo sapiens (Human))
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM475993(US10865208, Compound I-51 | {(2R,3S,4R,5R)-5-[4-am...)
Affinity DataIC50:  160nMAssay Description:Inhibition of ATG7 in human 293HEK cells assessed as inhibition of ATG7:ATG8 thioester formation after 8 hrs by Western blot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUbiquitin-like modifier-activating enzyme ATG7(Homo sapiens (Human))
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM475969(US10865208, Compound I-27 | {(2R,3S,4R,5R)-5-[4-am...)
Affinity DataIC50:  162nMAssay Description:Inhibition of ATG7 in human 293HEK cells assessed as inhibition of ATG7:ATG8 thioester formation after 8 hrs by Western blot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUbiquitin-like modifier-activating enzyme ATG7(Homo sapiens (Human))
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM476048(US10865208, Compound I-105 | [(2R,3R,4S,5R)-5-(4-a...)
Affinity DataIC50:  177nMAssay Description:Inhibition of recombinant His-tagged human ATG7 incubated for 105 mins in presence of GST-tagged ATG3 and Flag-tagged Gabarap and measured after 2 hr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUbiquitin-like modifier-activating enzyme ATG7(Homo sapiens (Human))
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM476012(US10865208, Compound I-69 | [(2R,3S,4R,5R)-5-{4-am...)
Affinity DataIC50:  178nMAssay Description:Inhibition of ATG7 in human 293HEK cells assessed as inhibition of ATG7:ATG8 thioester formation after 8 hrs by Western blot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUbiquitin-like modifier-activating enzyme ATG7(Homo sapiens (Human))
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM476169(US10865208, Compound I-224 | [(2S,3S,5R)-5-{4-amin...)
Affinity DataIC50:  190nMAssay Description:Inhibition of recombinant His-tagged human ATG7 incubated for 105 mins in presence of GST-tagged ATG3 and Flag-tagged Gabarap and measured after 2 hr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUbiquitin-like modifier-activating enzyme ATG7(Homo sapiens (Human))
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM476049(US10865208, Compound I-106 | [(2R,3R,4S,5R)-5-{4-a...)
Affinity DataIC50:  198nMAssay Description:Inhibition of ATG7 in human 293HEK cells assessed as inhibition of ATG7:ATG8 thioester formation after 4 hrs by Western blot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUbiquitin-like modifier-activating enzyme ATG7(Homo sapiens (Human))
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM476084(US10865208, Compound I-139 | {(2R,3R,4S,5R)-5-[4-a...)
Affinity DataIC50:  199nMAssay Description:Inhibition of ATG7 in human 293HEK cells assessed as inhibition of ATG7:ATG8 thioester formation after 4 hrs by Western blot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUbiquitin-like modifier-activating enzyme ATG7(Homo sapiens (Human))
Takeda Pharmaceuticals International

Curated by ChEMBL
LigandPNGBDBM476025(US10865208, Compound I-82 | {(2R,3S,4R,5R)-5-[4-am...)
Affinity DataIC50:  201nMAssay Description:Inhibition of ATG7 in human 293HEK cells assessed as inhibition of ATG7:ATG8 thioester formation after 8 hrs by Western blot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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