BindingDB PrimarySearch_ki

Found 180 with Last Name = 'bu' and Initial = 'jh'

Corticotropin-releasing factor receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL

PNG

BDBM50422737(CHEMBL380800)

IC50: 79nMAssay Description:In vitro inhibition of CRF-stimulated cAMP production in cell membranes expressing human CRF1 receptorMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD GoogleScholar

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Potassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Virginia Tech

Curated by ChEMBL

PNG

BDBM50582244(CHEMBL5070756)

IC50: 510nMAssay Description:Inhibition of human ERG expressed in HEK-293 cells by patch clamp methodMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Details Article PubMed

Runt-related transcription factor 1(Homo sapiens (Human))
University of Virginia At Charlottesville

PNG

BDBM31183(thiazol-2-amine, 14)

IC50: 700nMAssay Description:His6-CBFbeta (1-141) was expressed and purified with the exception of the protease cleavage step. Cerulean-Runt domain fusion protein (Runx1 41-190) ...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
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Core-binding factor subunit beta(Homo sapiens (Human))
University of Virginia Patent Foundation

US Patent

PNG

BDBM123672(US8748618, AI-4-49)

IC50: 700nMAssay Description:We have developed effective assays to monitor the inhibition of CBFβ-SMMHC binding to the Runt domain (as well as for CBFβ binding to the R...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
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Core-binding factor subunit beta(Homo sapiens (Human))
University of Virginia Patent Foundation

US Patent

PNG

BDBM123674(US8748618, AI-4-48)

IC50: 760nMAssay Description:We have developed effective assays to monitor the inhibition of CBFβ-SMMHC binding to the Runt domain (as well as for CBFβ binding to the R...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
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Core-binding factor subunit beta(Homo sapiens (Human))
University of Virginia Patent Foundation

US Patent

PNG

BDBM123684(US8748618, LD-2-101)

IC50: 1.00E+3nMAssay Description:We have developed effective assays to monitor the inhibition of CBFβ-SMMHC binding to the Runt domain (as well as for CBFβ binding to the R...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
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Core-binding factor subunit beta(Homo sapiens (Human))
University of Virginia Patent Foundation

US Patent

PNG

BDBM123675(US8748618, AI-10-3)

IC50: 1.00E+3nMAssay Description:We have developed effective assays to monitor the inhibition of CBFβ-SMMHC binding to the Runt domain (as well as for CBFβ binding to the R...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
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Core-binding factor subunit beta(Homo sapiens (Human))
University of Virginia Patent Foundation

US Patent

PNG

BDBM123665(US8748618, AI-10-47)

IC50: 1.00E+3nMAssay Description:We have developed effective assays to monitor the inhibition of CBFβ-SMMHC binding to the Runt domain (as well as for CBFβ binding to the R...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
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Runt-related transcription factor 1(Homo sapiens (Human))
University of Virginia At Charlottesville

PNG

BDBM31183(thiazol-2-amine, 14)

IC50: 1.10E+3nMpH: 7.5 T: 2°CAssay Description:For the FRET measurements, the Cerulean-Runt (Runx1 41-190) and Venus-CBFbeta (1-141) fusion proteins were dialyzed into FRET assay buffer. Protein c...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
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Core-binding factor subunit beta(Homo sapiens (Human))
University of Virginia Patent Foundation

US Patent

PNG

BDBM123673(US8748618, LD-2-23)

IC50: 1.10E+3nMAssay Description:We have developed effective assays to monitor the inhibition of CBFβ-SMMHC binding to the Runt domain (as well as for CBFβ binding to the R...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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CXXC-type zinc finger protein 4(Homo sapiens)
University Of Virginia

Curated by ChEMBL

PNG

BDBM50594525(CHEMBL5189434)

IC50: 1.20E+3nMAssay Description:Inhibition of GST-tagged human IDAX (130 to 181 residues) expressed in Escherichia coli BL21 cells incubated for 30 mins by fluorescence polarization...More data for this Ligand-Target Pair

PDB MMDB KEGG
UniProtKB/SwissProt
B.MOAD DrugBank GoogleScholar

Core-binding factor subunit beta(Homo sapiens (Human))
University of Virginia Patent Foundation

US Patent

PNG

BDBM123671(US8748618, AI-10-51)

IC50: 1.30E+3nMAssay Description:We have developed effective assays to monitor the inhibition of CBFβ-SMMHC binding to the Runt domain (as well as for CBFβ binding to the R...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
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Core-binding factor subunit beta(Homo sapiens (Human))
University of Virginia Patent Foundation

US Patent

PNG

BDBM123670(US8748618, LD-1-39)

IC50: 1.30E+3nMAssay Description:We have developed effective assays to monitor the inhibition of CBFβ-SMMHC binding to the Runt domain (as well as for CBFβ binding to the R...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
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Core-binding factor subunit beta(Homo sapiens (Human))
University of Virginia Patent Foundation

US Patent

PNG

BDBM123669(US8748618, AI-4-43)

IC50: 1.40E+3nMAssay Description:We have developed effective assays to monitor the inhibition of CBFβ-SMMHC binding to the Runt domain (as well as for CBFβ binding to the R...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
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Core-binding factor subunit beta(Homo sapiens (Human))
University of Virginia Patent Foundation

US Patent

PNG

BDBM123659(US8748618, AI-4-70 (or) LD-2-21)

IC50: 1.40E+3nMAssay Description:We have developed effective assays to monitor the inhibition of CBFβ-SMMHC binding to the Runt domain (as well as for CBFβ binding to the R...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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Core-binding factor subunit beta(Homo sapiens (Human))
University of Virginia Patent Foundation

US Patent

PNG

BDBM123657(US8748618, LD-1-29 (or) AI-10-54)

IC50: 1.50E+3nMAssay Description:We have developed effective assays to monitor the inhibition of CBFβ-SMMHC binding to the Runt domain (as well as for CBFβ binding to the R...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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Runt-related transcription factor 1(Homo sapiens (Human))
University of Virginia At Charlottesville

PNG

BDBM434071(US10562890, Compound Al-12-16)

IC50: 1.69E+3nMAssay Description:FRET assay can be used to effectively monitor the inhibition of CBF binding to the Runt domain of RUNX proteins (as well as for CBFβ-SMMHC bindi...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
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Runt-related transcription factor 1(Homo sapiens (Human))
University of Virginia At Charlottesville

PNG

BDBM434079(US10562890, Compound Al-14-72)

IC50: 1.72E+3nMAssay Description:FRET assay can be used to effectively monitor the inhibition of CBF binding to the Runt domain of RUNX proteins (as well as for CBFβ-SMMHC bindi...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
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Core-binding factor subunit beta(Homo sapiens (Human))
University of Virginia Patent Foundation

US Patent

PNG

BDBM123663(US8748618, AI-10-35)

IC50: 1.80E+3nMAssay Description:We have developed effective assays to monitor the inhibition of CBFβ-SMMHC binding to the Runt domain (as well as for CBFβ binding to the R...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
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F-box/LRR-repeat protein 19(Homo sapiens)
University Of Virginia

Curated by ChEMBL

PNG

BDBM50594520(CHEMBL5194845)

IC50: 1.80E+3nMAssay Description:Inhibition of GST-tagged human FBXL19 (31 to 86 residues) expressed in Escherichia coli BL21 cells incubated for 30 mins by fluorescence polarization...More data for this Ligand-Target Pair

PDB MMDB KEGG
UniProtKB/SwissProt
B.MOAD GoogleScholar

Core-binding factor subunit beta(Homo sapiens (Human))
University of Virginia Patent Foundation

US Patent

PNG

BDBM123678(US8748618, AI-10-96)

IC50: 2.00E+3nMAssay Description:We have developed effective assays to monitor the inhibition of CBFβ-SMMHC binding to the Runt domain (as well as for CBFβ binding to the R...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
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Core-binding factor subunit beta(Homo sapiens (Human))
University of Virginia Patent Foundation

US Patent

PNG

BDBM50180737(5,6-dimethyl-2-(pyridin-2-yl)-1H-benzo[d]imidazole...)

IC50: 2.00E+3nMAssay Description:We have developed effective assays to monitor the inhibition of CBFβ-SMMHC binding to the Runt domain (as well as for CBFβ binding to the R...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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Core-binding factor subunit beta(Homo sapiens (Human))
University of Virginia Patent Foundation

US Patent

PNG

BDBM123685(US8748618, AI-10-77)

IC50: 2.00E+3nMAssay Description:We have developed effective assays to monitor the inhibition of CBFβ-SMMHC binding to the Runt domain (as well as for CBFβ binding to the R...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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Core-binding factor subunit beta(Homo sapiens (Human))
University of Virginia Patent Foundation

US Patent

PNG

BDBM123654(US8748618, AI-4-57 (or) LD-1-11C | US8748618, LD-1...)

IC50: 2.00E+3nMAssay Description:We have developed effective assays to monitor the inhibition of CBFβ-SMMHC binding to the Runt domain (as well as for CBFβ binding to the R...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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Runt-related transcription factor 1(Homo sapiens (Human))
University of Virginia At Charlottesville

PNG

BDBM434076(US10562890, Compound Al-14-100)

IC50: 2.16E+3nMAssay Description:FRET assay can be used to effectively monitor the inhibition of CBF binding to the Runt domain of RUNX proteins (as well as for CBFβ-SMMHC bindi...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
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CXXC-type zinc finger protein 4(Homo sapiens)
University Of Virginia

Curated by ChEMBL

PNG

BDBM50594530(CHEMBL5181110)

IC50: 2.20E+3nMAssay Description:Inhibition of GST-tagged human IDAX (130 to 181 residues) expressed in Escherichia coli BL21 cells incubated for 30 mins by fluorescence polarization...More data for this Ligand-Target Pair

PDB MMDB KEGG
UniProtKB/SwissProt
B.MOAD DrugBank GoogleScholar

Core-binding factor subunit beta(Homo sapiens (Human))
University of Virginia Patent Foundation

US Patent

PNG

BDBM123681(US8748618, AI-10-87)

IC50: 2.30E+3nMAssay Description:We have developed effective assays to monitor the inhibition of CBFβ-SMMHC binding to the Runt domain (as well as for CBFβ binding to the R...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
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Core-binding factor subunit beta(Homo sapiens (Human))
University of Virginia Patent Foundation

US Patent

PNG

BDBM123680(US8748618, AI-10-11)

IC50: 2.30E+3nMAssay Description:We have developed effective assays to monitor the inhibition of CBFβ-SMMHC binding to the Runt domain (as well as for CBFβ binding to the R...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
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Core-binding factor subunit beta(Homo sapiens (Human))
University of Virginia Patent Foundation

US Patent

PNG

BDBM50180732(5-Chloro-2-pyridin-2-yl-1H-benzoimidazole | 5-chlo...)

IC50: 2.30E+3nMAssay Description:We have developed effective assays to monitor the inhibition of CBFβ-SMMHC binding to the Runt domain (as well as for CBFβ binding to the R...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
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CXXC-type zinc finger protein 4(Homo sapiens)
University Of Virginia

Curated by ChEMBL

PNG

BDBM50594527(CHEMBL5177921)

IC50: 2.40E+3nMAssay Description:Inhibition of GST-tagged human IDAX (130 to 181 residues) expressed in Escherichia coli BL21 cells incubated for 30 mins by fluorescence polarization...More data for this Ligand-Target Pair

PDB MMDB KEGG
UniProtKB/SwissProt
B.MOAD DrugBank GoogleScholar

F-box/LRR-repeat protein 19(Homo sapiens)
University Of Virginia

Curated by ChEMBL

PNG

BDBM50594525(CHEMBL5189434)

IC50: 2.40E+3nMAssay Description:Inhibition of GST-tagged human FBXL19 (31 to 86 residues) expressed in Escherichia coli BL21 cells incubated for 30 mins by fluorescence polarization...More data for this Ligand-Target Pair

PDB MMDB KEGG
UniProtKB/SwissProt
B.MOAD GoogleScholar

Core-binding factor subunit beta(Homo sapiens (Human))
University of Virginia Patent Foundation

US Patent

PNG

BDBM123679(US8748618, AI-4-61 (or) AI-10-52)

IC50: 2.50E+3nMAssay Description:We have developed effective assays to monitor the inhibition of CBFβ-SMMHC binding to the Runt domain (as well as for CBFβ binding to the R...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
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Core-binding factor subunit beta(Homo sapiens (Human))
University of Virginia Patent Foundation

US Patent

PNG

BDBM123661(US8748618, AI-10-61)

IC50: 2.50E+3nMAssay Description:We have developed effective assays to monitor the inhibition of CBFβ-SMMHC binding to the Runt domain (as well as for CBFβ binding to the R...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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Core-binding factor subunit beta(Homo sapiens (Human))
University of Virginia Patent Foundation

US Patent

PNG

BDBM50180735(5-fluoro-2-(pyridin-2-yl)-1H-benzo[d]imidazole | 5...)

IC50: 2.50E+3nMAssay Description:We have developed effective assays to monitor the inhibition of CBFβ-SMMHC binding to the Runt domain (as well as for CBFβ binding to the R...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
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Core-binding factor subunit beta(Homo sapiens (Human))
University of Virginia Patent Foundation

US Patent

PNG

BDBM123668(US8748618, LD-1-33)

IC50: 2.50E+3nMAssay Description:We have developed effective assays to monitor the inhibition of CBFβ-SMMHC binding to the Runt domain (as well as for CBFβ binding to the R...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
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Core-binding factor subunit beta(Homo sapiens (Human))
University of Virginia Patent Foundation

US Patent

PNG

BDBM123654(US8748618, AI-4-57 (or) LD-1-11C | US8748618, LD-1...)

IC50: 2.60E+3nMAssay Description:We have developed effective assays to monitor the inhibition of CBFβ-SMMHC binding to the Runt domain (as well as for CBFβ binding to the R...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
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F-box/LRR-repeat protein 19(Homo sapiens)
University Of Virginia

Curated by ChEMBL

PNG

BDBM50594530(CHEMBL5181110)

IC50: 2.60E+3nMAssay Description:Inhibition of GST-tagged human FBXL19 (31 to 86 residues) expressed in Escherichia coli BL21 cells incubated for 30 mins by fluorescence polarization...More data for this Ligand-Target Pair

PDB MMDB KEGG
UniProtKB/SwissProt
B.MOAD GoogleScholar

Runt-related transcription factor 1(Homo sapiens (Human))
University of Virginia At Charlottesville

PNG

BDBM434075(US10562890, Compound Al-14-95)

IC50: 2.65E+3nMAssay Description:FRET assay can be used to effectively monitor the inhibition of CBF binding to the Runt domain of RUNX proteins (as well as for CBFβ-SMMHC bindi...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
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Runt-related transcription factor 1(Homo sapiens (Human))
University of Virginia At Charlottesville

PNG

BDBM434070(US10562890, Compound Al-10-104)

IC50: 2.65E+3nMAssay Description:FRET assay can be used to effectively monitor the inhibition of CBF binding to the Runt domain of RUNX proteins (as well as for CBFβ-SMMHC bindi...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
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Core-binding factor subunit beta(Homo sapiens (Human))
University of Virginia Patent Foundation

US Patent

PNG

BDBM50180733(5-Methyl-2-pyridin-2-yl-1H-benzoimidazole | 5-meth...)

IC50: 2.90E+3nMAssay Description:We have developed effective assays to monitor the inhibition of CBFβ-SMMHC binding to the Runt domain (as well as for CBFβ binding to the R...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
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Runt-related transcription factor 1(Homo sapiens (Human))
University of Virginia At Charlottesville

PNG

BDBM434074(US10562890, Compound Al-14-91)

IC50: 2.97E+3nMAssay Description:FRET assay can be used to effectively monitor the inhibition of CBF binding to the Runt domain of RUNX proteins (as well as for CBFβ-SMMHC bindi...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
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Runt-related transcription factor 1(Homo sapiens (Human))
University of Virginia At Charlottesville

PNG

BDBM31175(thiazol-2-amine, 5)

IC50: 3.00E+3nMAssay Description:His6-CBFbeta (1-141) was expressed and purified with the exception of the protease cleavage step. Cerulean-Runt domain fusion protein (Runx1 41-190) ...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
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Core-binding factor subunit beta(Homo sapiens (Human))
University of Virginia Patent Foundation

US Patent

PNG

BDBM123682(US8748618, AI-10-53)

IC50: 3.00E+3nMAssay Description:We have developed effective assays to monitor the inhibition of CBFβ-SMMHC binding to the Runt domain (as well as for CBFβ binding to the R...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
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F-box/LRR-repeat protein 19(Homo sapiens)
University Of Virginia

Curated by ChEMBL

PNG

BDBM50594527(CHEMBL5177921)

IC50: 3.10E+3nMAssay Description:Inhibition of GST-tagged human FBXL19 (31 to 86 residues) expressed in Escherichia coli BL21 cells incubated for 30 mins by fluorescence polarization...More data for this Ligand-Target Pair

PDB MMDB KEGG
UniProtKB/SwissProt
B.MOAD GoogleScholar

Runt-related transcription factor 1(Homo sapiens (Human))
University of Virginia At Charlottesville

PNG

BDBM434069(US10562890, Compound Al-10-47)

IC50: 3.19E+3nMAssay Description:FRET assay can be used to effectively monitor the inhibition of CBF binding to the Runt domain of RUNX proteins (as well as for CBFβ-SMMHC bindi...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
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Runt-related transcription factor 1(Homo sapiens (Human))
University of Virginia At Charlottesville

PNG

BDBM31185(thiazol-2-amine, 17)

IC50: 3.20E+3nMpH: 7.5 T: 2°CAssay Description:For the FRET measurements, the Cerulean-Runt (Runx1 41-190) and Venus-CBFbeta (1-141) fusion proteins were dialyzed into FRET assay buffer. Protein c...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
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Runt-related transcription factor 1(Homo sapiens (Human))
University of Virginia At Charlottesville

PNG

BDBM31186(thiazol-2-amine, 18)

IC50: 3.20E+3nMAssay Description:His6-CBFbeta (1-141) was expressed and purified with the exception of the protease cleavage step. Cerulean-Runt domain fusion protein (Runx1 41-190) ...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
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Histone-lysine N-methyltransferase 2A(Homo sapiens (Human))
University Of Virginia

Curated by ChEMBL

PNG

BDBM50594525(CHEMBL5189434)

IC50: 3.30E+3nMAssay Description:Inhibition of GST-tagged human MLL1 (1147 to 1203 residues) expressed in Escherichia coli BL21 cells incubated for 30 mins by fluorescence polarizati...More data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
GoogleScholar

Core-binding factor subunit beta(Homo sapiens (Human))
University of Virginia Patent Foundation

US Patent

PNG

BDBM123664(US8748618, AI-10-37)

IC50: 3.30E+3nMAssay Description:We have developed effective assays to monitor the inhibition of CBFβ-SMMHC binding to the Runt domain (as well as for CBFβ binding to the R...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
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Runt-related transcription factor 1(Homo sapiens (Human))
University of Virginia At Charlottesville

PNG

BDBM31182(thiazol-2-amine, 13)

IC50: 3.30E+3nMAssay Description:His6-CBFbeta (1-141) was expressed and purified with the exception of the protease cleavage step. Cerulean-Runt domain fusion protein (Runx1 41-190) ...More data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
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Displayed 1 to 50 (of 180 total ) | Next | Last >>

Filter my 180 hits

Targets 13▿
- Runt-related transcription factor 1 54
- Core-binding factor subunit beta 36
- Histone-lysine N-methyltransferase 2A 17
- CXXC-type zinc finger protein 5 9
- F-box/LRR-repeat protein 19 9
- Methylcytosine dioxygenase TET3 9
- Lysine-specific demethylase 2B 9
- Methylcytosine dioxygenase TET1 9
- CXXC-type zinc finger protein 4 9
- Lysine-specific demethylase 2A 9
- Disulfide bond formation protein B 8
- Corticotropin-releasing factor receptor 1 1
- Potassium voltage-gated channel subfamily H member 2 1
- ...
Publications 7▿
- ACS Med Chem Lett 13: 1363-1369 (2022) 80
- Chem Biol 14: 1186-97 (2007) 38
- US Patent US8748618 (2014) 36
- US Patent US10562890 (2020) 16
- Chem Biol 17: 881-91 (2010) 8
- ACS Med Chem Lett 13: 365-370 (2022) 1
- J Med Chem 48: 5780-93 (2005) 1
Institutions 6▿
- University Of Virginia 80
- University of Virginia Patent Foundation 52
- University of Virginia At Charlottesville 38
- Leiden University 8
- Virginia Tech 1
- Neurocrine Biosciences 1
Affinity: 79 to 1.0E+6 nM▿
- IC50 174
- Affinity ≤ nM
Xtal structures: 0
Docked structures: 0
Catalog Cmpds: 45