TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Affinity DataKi: 50nMAssay Description:Competitive inhibition of recombinant glucocerebrosidaseMore data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Affinity DataKi: 50nMAssay Description:Competitive inhibition of recombinant glucocerebrosidaseMore data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Affinity DataKi: 60nMpH: 5.2Assay Description:Competitive inhibition of beta-glucocerebrosidase at pH 5.2 by Lineweaver-Burke plot analysisMore data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Affinity DataKi: 80nMpH: 5.2Assay Description:Competitive inhibition of beta-glucocerebrosidase at pH 5.2 by Lineweaver-Burke plot analysisMore data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Affinity DataKi: 90nMpH: 5.2Assay Description:Competitive inhibition of beta-glucocerebrosidase at pH 5.2 by Lineweaver-Burke plot analysisMore data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Affinity DataKi: 290nMAssay Description:Competitive inhibition of recombinant glucocerebrosidaseMore data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Affinity DataKi: 300nMAssay Description:Competitive inhibition of recombinant glucocerebrosidaseMore data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Affinity DataKi: 300nMAssay Description:Competitive inhibition of recombinant glucocerebrosidaseMore data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Affinity DataKi: 300nMpH: 5.2Assay Description:Competitive inhibition of beta-glucocerebrosidase at pH 5.2 by Lineweaver-Burke plot analysisMore data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Affinity DataKi: 300nMpH: 5.2Assay Description:Competitive inhibition of beta-glucocerebrosidase at pH 5.2 by Lineweaver-Burke plot analysisMore data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Affinity DataKi: 330nMpH: 5.2Assay Description:Competitive inhibition of beta-glucocerebrosidase at pH 5.2 by Lineweaver-Burke plot analysisMore data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Affinity DataKi: 770nMAssay Description:Competitive inhibition of recombinant glucocerebrosidaseMore data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Affinity DataKi: 890nMAssay Description:Competitive inhibition of recombinant glucocerebrosidaseMore data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Affinity DataKi: 1.05E+3nMAssay Description:Competitive inhibition of recombinant glucocerebrosidaseMore data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Affinity DataKi: 1.80E+3nMpH: 5.2Assay Description:Competitive inhibition of beta-glucocerebrosidase at pH 5.2 by Lineweaver-Burke plot analysisMore data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Affinity DataKi: 2.40E+3nMpH: 5.2Assay Description:Competitive inhibition of beta-glucocerebrosidase at pH 5.2 by Lineweaver-Burke plot analysisMore data for this Ligand-Target Pair
TargetSphingosine-1-phosphate lyase 1(Rattus norvegicus)
Spanish National Research Council (Csic)
Curated by ChEMBL
Spanish National Research Council (Csic)
Curated by ChEMBL
Affinity DataKi: 5.00E+3nMAssay Description:Competitive inhibition of rat liver microsomal S1PL using varying levels of [3-3H]-D(+) erythro-sphinganine-1-phosphate as substrate incubated for 15...More data for this Ligand-Target Pair
TargetSphingosine-1-phosphate lyase 1(Rattus norvegicus)
Spanish National Research Council (Csic)
Curated by ChEMBL
Spanish National Research Council (Csic)
Curated by ChEMBL
Affinity DataKi: 5.00E+3nMAssay Description:Competitive inhibition of rat S1PL in presence of D(+)-erythro-sphinganine-1-phosphate measured after 15 mins by Dixon plot analysisMore data for this Ligand-Target Pair
TargetSphingosine-1-phosphate lyase 1(Homo sapiens (Human))
Spanish National Research Council (Csic)
Curated by ChEMBL
Spanish National Research Council (Csic)
Curated by ChEMBL
Affinity DataKi: 5.60E+3nMAssay Description:Competitive inhibition of human S1PL using varying levels of RBM13 as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
TargetSphingosine-1-phosphate lyase 1(Homo sapiens (Human))
Spanish National Research Council (Csic)
Curated by ChEMBL
Spanish National Research Council (Csic)
Curated by ChEMBL
Affinity DataKi: 6.30E+3nMAssay Description:Competitive inhibition of human S1PL using varying levels of RBM13 as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Affinity DataKi: 7.60E+3nMpH: 5.2Assay Description:Competitive inhibition of beta-glucocerebrosidase at pH 5.2 by Lineweaver-Burke plot analysisMore data for this Ligand-Target Pair
TargetSphingosine-1-phosphate lyase 1(Homo sapiens (Human))
Spanish National Research Council (Csic)
Curated by ChEMBL
Spanish National Research Council (Csic)
Curated by ChEMBL
Affinity DataKi: 9.10E+3nMAssay Description:Competitive inhibition of human S1PL using varying levels of RBM13 as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
TargetSphingosine-1-phosphate lyase 1(Homo sapiens (Human))
Spanish National Research Council (Csic)
Curated by ChEMBL
Spanish National Research Council (Csic)
Curated by ChEMBL
Affinity DataKi: 1.64E+4nMAssay Description:Competitive inhibition of human S1PL using varying levels of RBM13 as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
TargetSphingosine-1-phosphate lyase 1(Homo sapiens (Human))
Spanish National Research Council (Csic)
Curated by ChEMBL
Spanish National Research Council (Csic)
Curated by ChEMBL
Affinity DataKi: 1.75E+4nMAssay Description:Competitive inhibition of human S1PL using varying levels of RBM13 as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
TargetSphingosine-1-phosphate lyase 1(Homo sapiens (Human))
Spanish National Research Council (Csic)
Curated by ChEMBL
Spanish National Research Council (Csic)
Curated by ChEMBL
Affinity DataKi: 1.90E+4nMAssay Description:Competitive inhibition of human S1PL using varying levels of RBM13 as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Affinity DataKi: 1.91E+4nMpH: 5.2Assay Description:Competitive inhibition of beta-glucocerebrosidase at pH 5.2 by Lineweaver-Burke plot analysisMore data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Affinity DataKi: 1.99E+4nMpH: 5.2Assay Description:Competitive inhibition of beta-glucocerebrosidase at pH 5.2 by Lineweaver-Burke plot analysisMore data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Affinity DataKi: 2.02E+4nMpH: 5.2Assay Description:Competitive inhibition of beta-glucocerebrosidase at pH 5.2 by Lineweaver-Burke plot analysisMore data for this Ligand-Target Pair
TargetSphingosine-1-phosphate lyase 1(Homo sapiens (Human))
Spanish National Research Council (Csic)
Curated by ChEMBL
Spanish National Research Council (Csic)
Curated by ChEMBL
Affinity DataKi: 2.04E+4nMAssay Description:Competitive inhibition of human S1PL using varying levels of RBM13 as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
TargetSphingosine-1-phosphate lyase 1(Homo sapiens (Human))
Spanish National Research Council (Csic)
Curated by ChEMBL
Spanish National Research Council (Csic)
Curated by ChEMBL
Affinity DataKi: 3.67E+4nMAssay Description:Competitive inhibition of human S1PL using varying levels of RBM13 as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Affinity DataIC50: 30nMpH: 5.2Assay Description:Inhibition of recombinant beta-glucocerebrosidase at pH 5.2 after 10 mins by fluorimetryMore data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Affinity DataIC50: 30.2nMAssay Description:Inhibition of recombinant beta-glucocerebrosidase after 10 mins by fluorimetryMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institut De Qu£Mica Avan£Ada De Catalunya
Curated by ChEMBL
Institut De Qu£Mica Avan£Ada De Catalunya
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Antagonist activity at rat TRPV1 expressed in Xenopus laevis oocytes assessed as blockage of capsaicin-induced current at holding potential -60 mV by...More data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Affinity DataIC50: 50nMpH: 5.2Assay Description:Inhibition of recombinant glucocerebrosidase in McIlvaine buffer at pH 5.2 after 10 mins by fluorometric analysisMore data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Affinity DataIC50: 60nMpH: 7.4Assay Description:Inhibition of recombinant beta-glucocerebrosidase at pH 7.4 after 10 mins by fluorimetryMore data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Affinity DataIC50: 60nMpH: 5.2Assay Description:Inhibition of recombinant glucocerebrosidase in McIlvaine buffer at pH 5.2 after 10 mins by fluorometric analysisMore data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Affinity DataIC50: 60nMpH: 7.4Assay Description:Inhibition of recombinant glucocerebrosidase in McIlvaine buffer at pH 7.4 after 10 mins by fluorometric analysisMore data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Affinity DataIC50: 89.1nMAssay Description:Inhibition of recombinant beta-glucocerebrosidase after 10 mins by fluorimetryMore data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Affinity DataIC50: 90nMpH: 5.2Assay Description:Inhibition of recombinant beta-glucocerebrosidase at pH 5.2 after 10 mins by fluorimetryMore data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Affinity DataIC50: 90nMpH: 7.4Assay Description:Inhibition of recombinant beta-glucocerebrosidase at pH 7.4 after 10 mins by fluorimetryMore data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Affinity DataIC50: 93.3nMAssay Description:Inhibition of recombinant beta-glucocerebrosidase after 10 mins by fluorimetryMore data for this Ligand-Target Pair
TargetSphingosine-1-phosphate lyase 1(Homo sapiens (Human))
Spanish National Research Council (Csic)
Curated by ChEMBL
Spanish National Research Council (Csic)
Curated by ChEMBL
Affinity DataIC50: 94nMAssay Description:Inhibition of human S1PL using RBM13 as substrate measured after 1 hr by fluorogenic assayMore data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Affinity DataIC50: 100nMpH: 5.2Assay Description:Inhibition of recombinant beta-glucocerebrosidase at pH 5.2 after 10 mins by fluorimetryMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Institut De Qu£Mica Avan£Ada De Catalunya
Curated by ChEMBL
Institut De Qu£Mica Avan£Ada De Catalunya
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Antagonist activity at rat TRPV1 expressed in Xenopus laevis oocytes assessed as blockage of capsaicin-induced current at holding potential -60 mV by...More data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Affinity DataIC50: 100nMpH: 7.4Assay Description:Inhibition of recombinant beta-glucocerebrosidase at pH 7.4 after 10 mins by fluorimetryMore data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Affinity DataIC50: 100nMpH: 7.4Assay Description:Inhibition of recombinant glucocerebrosidase in McIlvaine buffer at pH 7.4 after 10 mins by fluorometric analysisMore data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Affinity DataIC50: 150nMpH: 5.2Assay Description:Inhibition of recombinant glucocerebrosidase in McIlvaine buffer at pH 5.2 after 10 mins by fluorometric analysisMore data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Affinity DataIC50: 200nMpH: 7.4Assay Description:Inhibition of recombinant beta-glucocerebrosidase at pH 7.4 after 10 mins by fluorimetryMore data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Affinity DataIC50: 200nMpH: 5.2Assay Description:Inhibition of recombinant beta-glucocerebrosidase at pH 5.2 after 10 mins by fluorimetryMore data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Spanish National Research Council (Consejo Superior De Investigaciones Cienti£?Ficas)
Curated by ChEMBL
Affinity DataIC50: 224nMAssay Description:Inhibition of recombinant beta-glucocerebrosidase after 10 mins by fluorimetryMore data for this Ligand-Target Pair