Affinity DataKi: 100nMAssay Description:Binding affinity against penicillopepsinMore data for this Ligand-Target Pair
Affinity DataKi: 190nMpH: 3.5Assay Description:Binding affinity against penicillopepsin at pH 3.5More data for this Ligand-Target Pair
Affinity DataKi: 374nMAssay Description:Binding affinity against human thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 400nMAssay Description:Binding affinity against saccharopepsinMore data for this Ligand-Target Pair
Affinity DataKi: 430nMAssay Description:Binding affinity against bovine trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 850nMAssay Description:Compound was tested for binding affinity against Glutamine synthetaseMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+3nMAssay Description:Binding affinity against penicillopepsinMore data for this Ligand-Target Pair
Affinity DataKi: 1.17E+3nMAssay Description:Binding affinity against bovine trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 1.20E+3nMAssay Description:Binding affinity against bovine trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 1.24E+3nMAssay Description:Binding affinity against human thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 1.24E+3nMAssay Description:Binding affinity against human thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 1.30E+3nMAssay Description:Binding affinity against bovine ThrombinMore data for this Ligand-Target Pair
Affinity DataKi: 2.70E+3nMpH: 4.5Assay Description:Binding affinity against penicillopepsin at pH 4.5More data for this Ligand-Target Pair
Affinity DataKi: 2.80E+3nMAssay Description:Binding affinity against penicillopepsinMore data for this Ligand-Target Pair
Affinity DataKi: 3.74E+3nMAssay Description:Binding affinity against saccharopepsinMore data for this Ligand-Target Pair
Affinity DataKi: 3.80E+3nMAssay Description:Compound was tested for binding affinity against CathepsinMore data for this Ligand-Target Pair
Affinity DataKi: 6.00E+3nMAssay Description:Binding affinity against bovine ThrombinMore data for this Ligand-Target Pair
Affinity DataKi: 9.00E+3nMAssay Description:Binding affinity against human thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+4nMAssay Description:Binding affinity against penicillopepsinMore data for this Ligand-Target Pair
Affinity DataKi: 1.10E+4nMAssay Description:Binding affinity against bovine trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 1.33E+4nMAssay Description:Binding affinity against bovine trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 1.40E+4nMAssay Description:Binding affinity against saccharopepsinMore data for this Ligand-Target Pair
Affinity DataKi: 1.50E+4nMAssay Description:Binding affinity against Triosephosphate isomeraseMore data for this Ligand-Target Pair
Affinity DataKi: 1.84E+4nMAssay Description:Binding affinity against bovine trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 1.84E+4nMAssay Description:Binding affinity against bovine trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 1.90E+4nMAssay Description:Binding affinity against bovine ThrombinMore data for this Ligand-Target Pair
Affinity DataKi: 2.00E+4nMAssay Description:Binding affinity against bovine trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 2.00E+4nMAssay Description:Binding affinity against penicillopepsinMore data for this Ligand-Target Pair
Affinity DataKi: 2.30E+4nMAssay Description:Binding affinity against bovine ThrombinMore data for this Ligand-Target Pair
Affinity DataKi: 3.25E+4nMAssay Description:Binding affinity against bovine trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 4.20E+4nMAssay Description:Binding affinity against penicillopepsinMore data for this Ligand-Target Pair
Affinity DataKi: 5.90E+4nMAssay Description:Inhibition of human recombinant serine racemase expressed in Escherichia coli Rosetta 2 (DE3) cells using L-serine as substrate by horseradish peroxi...More data for this Ligand-Target Pair
Affinity DataKi: 6.60E+4nMAssay Description:Inhibition of hexa-His-tagged purified human recombinant serine racemase expressed in Escherichia coli BL21 Codonplus (DE3)-RIL cells assessed as red...More data for this Ligand-Target Pair
Affinity DataKi: 1.07E+5nMpH: 5.5Assay Description:Binding affinity against penicillopepsin at pH 5.5More data for this Ligand-Target Pair
Affinity DataKi: 1.30E+6nMAssay Description:Inhibition of hexa-His-tagged purified human recombinant serine racemase expressed in Escherichia coli BL21 Codonplus (DE3)-RIL cells assessed as red...More data for this Ligand-Target Pair
Affinity DataKi: 1.50E+6nMAssay Description:Inhibition of hexa-His-tagged purified human recombinant serine racemase expressed in Escherichia coli BL21 Codonplus (DE3)-RIL cells assessed as red...More data for this Ligand-Target Pair
Affinity DataKi: 1.50E+6nMAssay Description:Inhibition of hexa-His-tagged purified human recombinant serine racemase expressed in Escherichia coli BL21 Codonplus (DE3)-RIL cells assessed as red...More data for this Ligand-Target Pair
Affinity DataKi: 1.70E+6nMAssay Description:Inhibition of hexa-His-tagged purified human recombinant serine racemase expressed in Escherichia coli BL21 Codonplus (DE3)-RIL cells assessed as red...More data for this Ligand-Target Pair
Affinity DataKi: 4.50E+6nMAssay Description:Inhibition of hexa-His-tagged purified human recombinant serine racemase expressed in Escherichia coli BL21 Codonplus (DE3)-RIL cells assessed as red...More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+7nMAssay Description:Inhibition of hexa-His-tagged purified human recombinant serine racemase expressed in Escherichia coli BL21 Codonplus (DE3)-RIL cells assessed as red...More data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Tested for 50% inhibition of generation of Human Ha-ras polymerase chain reaction(PCR) productsMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Tested for 50% inhibition of generation of Human Ha-ras polymerase chain reaction(PCR) productsMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Tested for 50% inhibition of generation of Human Ha-ras polymerase chain reaction(PCR) productsMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Inhibitory activity against alphaV-beta3 integrinMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Tested for 50% inhibition of generation of Human Ha-ras polymerase chain reaction(PCR) productsMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Tested for 50% inhibition of generation of Human Ha-ras polymerase chain reaction(PCR) productsMore data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Inhibitory activity against alphaV-beta3 integrinMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibitory activity against alpha IIb beta3 integrinMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:In vitro thromboxane-A2 receptor binding affinity to displace by 50% [3H]-SQ 29548 binding from washed human plateletsMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:In vitro inhibition of thromboxane-A2 synthase in rat whole blood during clotting at 37 degrees centigradeMore data for this Ligand-Target Pair