Affinity DataKi: 0.400nMAssay Description:Displacement of [125I]RTI-55 from DATMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Displacement of [125I]RTI-55 from DATMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Institute Of Biomolecular Chemistry
Curated by ChEMBL
Institute Of Biomolecular Chemistry
Curated by ChEMBL
Affinity DataKi: 0.700nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Displacement of [125I]RTI-55 from DATMore data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Displacement of [125I]RTI-55 from DATMore data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Displacement of [125I]RTI-55 from DATMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Displacement of [125I]RTI-55 from DATMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Displacement of [125I]RTI-55 from DATMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Inhibition of [3H]DA uptakeMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Displacement of [125I]RTI-55 from DATMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Displacement of [125I]RTI-55 from DATMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Displacement of [125I]RTI-55 from DATMore data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Inhibition of [3H]DA uptakeMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Displacement of [125I]RTI-55 from DATMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Institute Of Biomolecular Chemistry
Curated by ChEMBL
Institute Of Biomolecular Chemistry
Curated by ChEMBL
Affinity DataKi: 2nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Inhibition of [3H]DA uptakeMore data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Displacement of [125I]RTI-55 from DATMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Institute Of Biomolecular Chemistry
Curated by ChEMBL
Institute Of Biomolecular Chemistry
Curated by ChEMBL
Affinity DataKi: 2.10nMAssay Description:Displacement of [3H]CP55940 from human recombinant CB2 receptor expressed in HEK293 cells after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Displacement of [125I]RTI-55 from DATMore data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Displacement of [125I]RTI-55 from DATMore data for this Ligand-Target Pair
Affinity DataKi: 3.80nMAssay Description:Inhibition of [3H]DA uptakeMore data for this Ligand-Target Pair
Affinity DataKi: 5.10nMAssay Description:Displacement of [125I]RTI-55 from DATMore data for this Ligand-Target Pair
Affinity DataKi: 5.40nMAssay Description:Inhibitory activity against monoamine oxidase A in isolated bovine brain mitochondriaMore data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:Displacement of [125I]RTI-55 from DATMore data for this Ligand-Target Pair
Affinity DataKi: 6.90nMAssay Description:Displacement of [125I]RTI-55 from DATMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Displacement of [125I]RTI-55 from DATMore data for this Ligand-Target Pair
Affinity DataKi: 9.20nMAssay Description:Displacement of [3H]CP55940 from human recombinant CB1 receptor expressed in HEK293 cells after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Displacement of [125I]RTI-55 from DATMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Inhibition of [3H]DA uptakeMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Displacement of [125I]RTI-55 from SERTMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Displacement of [125I]RTI-55 from SERTMore data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Inhibition of [3H]DA uptakeMore data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Inhibition of [3H]5HT uptakeMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Inhibitory activity against monoamine oxidase B in isolated bovine brain mitochondriaMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Inhibitory activity against monoamine oxidase B in isolated bovine brain mitochondriaMore data for this Ligand-Target Pair
Affinity DataKi: 21nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Displacement of [125I]RTI-55 from SERTMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Displacement of [125I]RTI-55 from SERTMore data for this Ligand-Target Pair
Affinity DataKi: 38nMAssay Description:Displacement of [125I]RTI-55 from SERTMore data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Inhibition of [3H]NE uptakeMore data for this Ligand-Target Pair
Affinity DataKi: 41nMAssay Description:Inhibition of [3H]5HT uptakeMore data for this Ligand-Target Pair
Affinity DataKi: 43nMAssay Description:Displacement of [3H]nisoxetine from NETMore data for this Ligand-Target Pair
Affinity DataKi: 43nMAssay Description:Displacement of [125I]RTI-55 from SERTMore data for this Ligand-Target Pair
Affinity DataKi: 53nMAssay Description:Displacement of [125I]RTI-55 from SERTMore data for this Ligand-Target Pair
Affinity DataKi: 54nMAssay Description:Inhibitory activity against monoamine oxidase A in isolated bovine brain mitochondriaMore data for this Ligand-Target Pair
Affinity DataKi: 58nMAssay Description:Displacement of [125I]RTI-55 from SERTMore data for this Ligand-Target Pair
Affinity DataKi: 68nMAssay Description:Displacement of [125I]RTI-55 from SERTMore data for this Ligand-Target Pair
Affinity DataKi: 72nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 75nMAssay Description:Inhibitory activity against monoamine oxidase A in isolated bovine brain mitochondriaMore data for this Ligand-Target Pair