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Found 162 with Last Name = 'debiton' and Initial = 'e'
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50299249(1,10-Dihydropyrrolo[2,3-a]carbazole-3-carbaldehyde...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human Pim3 using RSRHSSYPAGT as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£

Curated by ChEMBL
LigandPNGBDBM50347798(CHEMBL1802410)
Affinity DataIC50:  26nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£

Curated by ChEMBL
LigandPNGBDBM50347802(CHEMBL1802406)
Affinity DataIC50:  30nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£

Curated by ChEMBL
LigandPNGBDBM50347793(CHEMBL1802966)
Affinity DataIC50:  32nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50347793(CHEMBL1802966)
Affinity DataIC50:  34nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50347792(CHEMBL1802967)
Affinity DataIC50:  39nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£

Curated by ChEMBL
LigandPNGBDBM50347815(CHEMBL1802405)
Affinity DataIC50:  41nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50385115(CHEMBL2036116)
Affinity DataIC50:  41nMAssay Description:Inhibition of Pim-3 using RSRHSSYPAGT as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£

Curated by ChEMBL
LigandPNGBDBM50347792(CHEMBL1802967)
Affinity DataIC50:  42nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Clermont Universit£

Curated by ChEMBL
LigandPNGBDBM50385115(CHEMBL2036116)
Affinity DataIC50:  46nMAssay Description:Inhibition of Pim-1 using RSRHSSYPAGT as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£

Curated by ChEMBL
LigandPNGBDBM50347796(CHEMBL1802963)
Affinity DataIC50:  65nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50347802(CHEMBL1802406)
Affinity DataIC50:  66nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£

Curated by ChEMBL
LigandPNGBDBM50347803(CHEMBL1802404)
Affinity DataIC50:  67nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50347796(CHEMBL1802963)
Affinity DataIC50:  68nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£

Curated by ChEMBL
LigandPNGBDBM50347806(CHEMBL1802401)
Affinity DataIC50:  70nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Clermont Universit£

Curated by ChEMBL
LigandPNGBDBM50385117(CHEMBL2036118)
Affinity DataIC50:  75nMAssay Description:Inhibition of Pim-1 using RSRHSSYPAGT as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£

Curated by ChEMBL
LigandPNGBDBM50347799(CHEMBL1802409)
Affinity DataIC50:  80nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50385117(CHEMBL2036118)
Affinity DataIC50:  80nMAssay Description:Inhibition of Pim-3 using RSRHSSYPAGT as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50347806(CHEMBL1802401)
Affinity DataIC50:  85nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£

Curated by ChEMBL
LigandPNGBDBM50347814(CHEMBL1802391)
Affinity DataIC50:  87nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50347803(CHEMBL1802404)
Affinity DataIC50:  95nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50347798(CHEMBL1802410)
Affinity DataIC50:  110nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£

Curated by ChEMBL
LigandPNGBDBM50347804(CHEMBL1802403)
Affinity DataIC50:  120nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£

Curated by ChEMBL
LigandPNGBDBM10841(4-(6-bromo-1H-indol-3-yl)pyrimidin-2-amine | Merid...)
Affinity DataIC50:  120nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Clermont Universit£

Curated by ChEMBL
LigandPNGBDBM50299249(1,10-Dihydropyrrolo[2,3-a]carbazole-3-carbaldehyde...)
Affinity DataIC50:  120nMAssay Description:Inhibition of human Pim1 using RSRHSSYPAGT as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM10841(4-(6-bromo-1H-indol-3-yl)pyrimidin-2-amine | Merid...)
Affinity DataIC50:  130nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£

Curated by ChEMBL
LigandPNGBDBM50347794(CHEMBL1802965)
Affinity DataIC50:  180nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50347814(CHEMBL1802391)
Affinity DataIC50:  190nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50385116(CHEMBL2036117)
Affinity DataIC50:  200nMAssay Description:Inhibition of Pim-3 using RSRHSSYPAGT as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50347799(CHEMBL1802409)
Affinity DataIC50:  220nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£

Curated by ChEMBL
LigandPNGBDBM10840(4-(5-bromo-1H-indol-3-yl)pyrimidin-2-amine | Merid...)
Affinity DataIC50:  220nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50347804(CHEMBL1802403)
Affinity DataIC50:  250nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50347788(CHEMBL1802971)
Affinity DataIC50:  290nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50347794(CHEMBL1802965)
Affinity DataIC50:  330nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM10840(4-(5-bromo-1H-indol-3-yl)pyrimidin-2-amine | Merid...)
Affinity DataIC50:  330nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£

Curated by ChEMBL
LigandPNGBDBM50347788(CHEMBL1802971)
Affinity DataIC50:  380nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£

Curated by ChEMBL
LigandPNGBDBM50347807(CHEMBL1802400)
Affinity DataIC50:  380nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50295872(5-Iodo-4-(1-Methyl-1H-indol-3-yl)pyrimidin-2-amine...)
Affinity DataIC50:  400nMAssay Description:Inhibition of rat recombinant DYRK1A expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50420295(CHEMBL2088998)
Affinity DataIC50:  410nMAssay Description:Inhibition of human Pim3 using RSRHSSYPAGT as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50347815(CHEMBL1802405)
Affinity DataIC50:  460nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Clermont Universit£

Curated by ChEMBL
LigandPNGBDBM50385116(CHEMBL2036117)
Affinity DataIC50:  470nMAssay Description:Inhibition of Pim-1 using RSRHSSYPAGT as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50420296(CHEMBL2089000)
Affinity DataIC50:  500nMAssay Description:Inhibition of human Pim3 using RSRHSSYPAGT as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50299249(1,10-Dihydropyrrolo[2,3-a]carbazole-3-carbaldehyde...)
Affinity DataIC50:  510nMAssay Description:Inhibition of human Pim2 using RSRHSSYPAGT as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£

Curated by ChEMBL
LigandPNGBDBM50347785(CHEMBL1802390)
Affinity DataIC50:  530nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£

Curated by ChEMBL
LigandPNGBDBM10844(4-(1H-indol-3-yl)pyrimidin-2-amine | Meridianin G)
Affinity DataIC50:  530nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 1(Rattus norvegicus (rat))
Clermont Universit£

Curated by ChEMBL
LigandPNGBDBM50295874(4-(1H-indol-3-yl)-5-(4-(trifluoromethyl)phenyl)pyr...)
Affinity DataIC50:  580nMAssay Description:Inhibition of rat recombinant Erk2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50295873(4-[2-Amino-4-(1H-indol-3-yl)pyrimidin-5-yl]benzami...)
Affinity DataIC50:  580nMAssay Description:Inhibition of rat recombinant DYRK1A expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50295875(4-(1H-Indol-3-yl)-5-(3-methoxyphenyl)pyrimidin-2-a...)
Affinity DataIC50:  600nMAssay Description:Inhibition of rat recombinant DYRK1A expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£

Curated by ChEMBL
LigandPNGBDBM50347800(CHEMBL1802408)
Affinity DataIC50:  610nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50295876(4-(1H-Indol-3-yl)-5-(3-aminophenyl)pyrimidin-2-ami...)
Affinity DataIC50:  640nMAssay Description:Inhibition of rat recombinant DYRK1A expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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