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Found 607 with Last Name = 'desjardins' and Initial = 'r'
TargetProprotein convertase subtilisin/kexin type 6(Homo sapiens (Human))
University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50264960(CHEMBL4089819)
Affinity DataKi:  0.200nMAssay Description:Inhibition of recombinant human PACE4 expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuroendocrine convertase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50446944(CHEMBL3115771)
Affinity DataKi:  0.240nMAssay Description:Inhibition of human PC2 expressed in drosophila schneider 2 cells using pyroGlu-Arg-Thr-Lys-Arg-AMC as substrate after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProprotein convertase subtilisin/kexin type 6(Homo sapiens (Human))
University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50264892(CHEMBL4065072)
Affinity DataKi:  0.300nMAssay Description:Inhibition of recombinant human PACE4 expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProprotein convertase subtilisin/kexin type 6(Homo sapiens (Human))
University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50399749(CHEMBL2179430)
Affinity DataKi:  0.340nMpH: 6.5Assay Description:Competitive inhibition of human recombinant PACE4 expressed in Drosophila S2 cells using pyroGlu-Arg-Val-Lys-Arg-methyl-coumaryl-7-amide as substrate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProprotein convertase subtilisin/kexin type 6(Homo sapiens (Human))
University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50399753(CHEMBL2179835)
Affinity DataKi:  0.400nMpH: 6.5Assay Description:Competitive inhibition of human recombinant PACE4 expressed in Drosophila S2 cells using pyroGlu-Arg-Val-Lys-Arg-methyl-coumaryl-7-amide as substrate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProprotein convertase subtilisin/kexin type 6(Homo sapiens (Human))
University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50264931(CHEMBL4084457)
Affinity DataKi:  0.400nMAssay Description:Inhibition of recombinant human PACE4 expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50264892(CHEMBL4065072)
Affinity DataKi:  0.400nMAssay Description:Inhibition of recombinant human furin expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProprotein convertase subtilisin/kexin type 6(Homo sapiens (Human))
University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50265119(CHEMBL4091099)
Affinity DataKi:  0.400nMAssay Description:Inhibition of recombinant human PACE4 expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProprotein convertase subtilisin/kexin type 6(Homo sapiens (Human))
University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50265083(CHEMBL4100996)
Affinity DataKi:  0.5nMAssay Description:Inhibition of recombinant human PACE4 expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50265344(CHEMBL4070237)
Affinity DataKi:  0.5nMAssay Description:Inhibition of recombinant human furin expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50265119(CHEMBL4091099)
Affinity DataKi:  0.5nMAssay Description:Inhibition of recombinant human furin expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProprotein convertase subtilisin/kexin type 6(Homo sapiens (Human))
University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50265384(CHEMBL4104777)
Affinity DataKi:  0.600nMAssay Description:Inhibition of recombinant human PACE4 expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50265083(CHEMBL4100996)
Affinity DataKi:  0.600nMAssay Description:Inhibition of recombinant human furin expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50264960(CHEMBL4089819)
Affinity DataKi:  0.700nMAssay Description:Inhibition of recombinant human furin expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProprotein convertase subtilisin/kexin type 6(Homo sapiens (Human))
University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50265344(CHEMBL4070237)
Affinity DataKi:  0.900nMAssay Description:Inhibition of recombinant human PACE4 expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50264941(CHEMBL4063327)
Affinity DataKi:  0.900nMAssay Description:Inhibition of recombinant human furin expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50264931(CHEMBL4084457)
Affinity DataKi:  0.900nMAssay Description:Inhibition of recombinant human furin expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50265090(CHEMBL4101304)
Affinity DataKi:  1nMAssay Description:Inhibition of recombinant human furin expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProprotein convertase subtilisin/kexin type 6(Homo sapiens (Human))
University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50265130(CHEMBL4064275)
Affinity DataKi:  1nMAssay Description:Inhibition of recombinant human PACE4 expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProprotein convertase subtilisin/kexin type 6(Homo sapiens (Human))
University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50265091(CHEMBL4083310)
Affinity DataKi:  1nMAssay Description:Inhibition of recombinant human PACE4 expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50265384(CHEMBL4104777)
Affinity DataKi:  1.10nMAssay Description:Inhibition of recombinant human furin expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50264971(CHEMBL4089913)
Affinity DataKi:  1.10nMAssay Description:Inhibition of recombinant human furin expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProprotein convertase subtilisin/kexin type 6(Homo sapiens (Human))
University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50399754(CHEMBL2179836)
Affinity DataKi:  1.10nMpH: 6.5Assay Description:Competitive inhibition of human recombinant PACE4 expressed in Drosophila S2 cells using pyroGlu-Arg-Val-Lys-Arg-methyl-coumaryl-7-amide as substrate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProprotein convertase subtilisin/kexin type 6(Homo sapiens (Human))
University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50265145(CHEMBL4073661)
Affinity DataKi:  1.30nMAssay Description:Inhibition of recombinant human PACE4 expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProprotein convertase subtilisin/kexin type 6(Homo sapiens (Human))
University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50399752(CHEMBL2179429)
Affinity DataKi:  1.30nMpH: 6.5Assay Description:Competitive inhibition of human recombinant PACE4 expressed in Drosophila S2 cells using pyroGlu-Arg-Val-Lys-Arg-methyl-coumaryl-7-amide as substrate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50399754(CHEMBL2179836)
Affinity DataKi:  1.40nMpH: 7.5Assay Description:Competitive inhibition of human recombinant furin expressed in Drosophila S2 cells using pyroGlu-Arg-Val-Lys-Arg-methyl-coumaryl-7-amide as substrate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50265185(CHEMBL4092088)
Affinity DataKi:  1.40nMAssay Description:Inhibition of recombinant human furin expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProprotein convertase subtilisin/kexin type 6(Homo sapiens (Human))
University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50265141(CHEMBL4094478)
Affinity DataKi:  1.5nMAssay Description:Inhibition of recombinant human PACE4 expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50265091(CHEMBL4083310)
Affinity DataKi:  1.5nMAssay Description:Inhibition of recombinant human furin expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50265328(CHEMBL4087970)
Affinity DataKi:  1.5nMAssay Description:Inhibition of recombinant human furin expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50399753(CHEMBL2179835)
Affinity DataKi:  1.70nMpH: 7.5Assay Description:Competitive inhibition of human recombinant furin expressed in Drosophila S2 cells using pyroGlu-Arg-Val-Lys-Arg-methyl-coumaryl-7-amide as substrate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProprotein convertase subtilisin/kexin type 6(Homo sapiens (Human))
University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50264955(CHEMBL4099961)
Affinity DataKi:  1.70nMAssay Description:Inhibition of recombinant human PACE4 expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50265130(CHEMBL4064275)
Affinity DataKi:  1.70nMAssay Description:Inhibition of recombinant human furin expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuroendocrine convertase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50446945(CHEMBL3115770)
Affinity DataKi:  1.70nMAssay Description:Inhibition of human PC2 expressed in drosophila schneider 2 cells using pyroGlu-Arg-Thr-Lys-Arg-AMC as substrate after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50265145(CHEMBL4073661)
Affinity DataKi:  1.80nMAssay Description:Inhibition of recombinant human furin expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProprotein convertase subtilisin/kexin type 6(Homo sapiens (Human))
University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50265045(CHEMBL4097940)
Affinity DataKi:  1.80nMAssay Description:Inhibition of recombinant human PACE4 expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50448473(CHEMBL3126399)
Affinity DataKi:  1.90nMAssay Description:Competitive inhibition of recombinant furin (unknown origin) using as substrate after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50265048(CHEMBL4065627)
Affinity DataKi:  2nMAssay Description:Inhibition of recombinant human furin expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProprotein convertase subtilisin/kexin type 6(Homo sapiens (Human))
University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50265331(CHEMBL4103443)
Affinity DataKi:  2nMAssay Description:Inhibition of recombinant human PACE4 expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProprotein convertase subtilisin/kexin type 6(Homo sapiens (Human))
University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50264941(CHEMBL4063327)
Affinity DataKi:  2nMAssay Description:Inhibition of recombinant human PACE4 expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50265131(CHEMBL4093570)
Affinity DataKi:  2nMAssay Description:Inhibition of recombinant human furin expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProprotein convertase subtilisin/kexin type 6(Homo sapiens (Human))
University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50399751(CHEMBL2179431)
Affinity DataKi:  2nMpH: 6.5Assay Description:Competitive inhibition of human recombinant PACE4 expressed in Drosophila S2 cells using pyroGlu-Arg-Val-Lys-Arg-methyl-coumaryl-7-amide as substrate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProprotein convertase subtilisin/kexin type 6(Homo sapiens (Human))
University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50265129(CHEMBL4085824)
Affinity DataKi:  2nMAssay Description:Inhibition of recombinant human PACE4 expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProprotein convertase subtilisin/kexin type 6(Homo sapiens (Human))
University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50264969(CHEMBL4096348)
Affinity DataKi:  2nMAssay Description:Inhibition of recombinant human PACE4 expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProprotein convertase subtilisin/kexin type 6(Homo sapiens (Human))
University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50265131(CHEMBL4093570)
Affinity DataKi:  2nMAssay Description:Inhibition of recombinant human PACE4 expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProprotein convertase subtilisin/kexin type 6(Homo sapiens (Human))
University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50265000(CHEMBL4101342)
Affinity DataKi:  2nMAssay Description:Inhibition of recombinant human PACE4 expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProprotein convertase subtilisin/kexin type 6(Homo sapiens (Human))
University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50265328(CHEMBL4087970)
Affinity DataKi:  2nMAssay Description:Inhibition of recombinant human PACE4 expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProprotein convertase subtilisin/kexin type 6(Homo sapiens (Human))
University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50265170(CHEMBL4075692)
Affinity DataKi:  2.10nMAssay Description:Inhibition of recombinant human PACE4 expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProprotein convertase subtilisin/kexin type 6(Homo sapiens (Human))
University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50265047(CHEMBL4072949)
Affinity DataKi:  2.20nMAssay Description:Inhibition of recombinant human PACE4 expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50265092(CHEMBL4063219)
Affinity DataKi:  2.30nMAssay Description:Inhibition of recombinant human furin expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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