Affinity DataIC50: 0.0400nMAssay Description:Inhibition of ATM (unknown origin) using p53 as substrate preincubated for 30 mins followed by substrate addition and measured after 2 hrs by HTRF as...More data for this Ligand-Target Pair
Affinity DataIC50: 0.170nMAssay Description:Inhibition of ATM autophosphorylation at Ser1981 in human HT29 cells preincubated for 1 hr followed by X ray irradiation and measured after 1 hr by H...More data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Inhibition of ATM autophosphorylation at Ser1981 in human HT29 cells preincubated for 1 hr followed by X ray irradiation and measured after 1 hr by H...More data for this Ligand-Target Pair
Affinity DataIC50: 0.240nMAssay Description:Inhibition of ATM autophosphorylation at Ser1981 in human HT29 cells preincubated for 1 hr followed by X ray irradiation and measured after 1 hr by H...More data for this Ligand-Target Pair
Affinity DataIC50: 0.25nMAssay Description:Inhibition of ATM autophosphorylation at Ser1981 in human HT29 cells preincubated for 1 hr followed by X ray irradiation and measured after 1 hr by H...More data for this Ligand-Target Pair
Affinity DataIC50: 0.25nMAssay Description:Inhibition of ATM autophosphorylation at Ser1981 in human HT29 cells preincubated for 1 hr followed by X ray irradiation and measured after 1 hr by H...More data for this Ligand-Target Pair
Affinity DataIC50: 0.290nMAssay Description:Inhibition of ATM autophosphorylation at Ser1981 in human HT29 cells preincubated for 1 hr followed by X ray irradiation and measured after 1 hr by H...More data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:Antagonist activity at integrin alphavbeta3 in human A375M cells assessed as inhibition of cell adhesion to fibrinogen in presence of Mg2+More data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:Antagonist activity at integrin alphaVbeta3 in human A375M cells assessed as cell adhesion to fibrinogen in presence of Mg2+More data for this Ligand-Target Pair
Affinity DataIC50: 0.330nMAssay Description:Inhibition of ATM autophosphorylation at Ser1981 in human HT29 cells preincubated for 1 hr followed by X ray irradiation and measured after 1 hr by H...More data for this Ligand-Target Pair
Affinity DataIC50: 0.570nMAssay Description:Inhibition of ATM autophosphorylation at Ser1981 in human HT29 cells preincubated for 1 hr followed by X ray irradiation and measured after 1 hr by H...More data for this Ligand-Target Pair
Affinity DataIC50: 0.760nMAssay Description:Inhibition of ATM autophosphorylation at Ser1981 in human HT29 cells preincubated for 1 hr followed by X ray irradiation and measured after 1 hr by H...More data for this Ligand-Target Pair
Affinity DataIC50: 0.780nMAssay Description:Inhibition of ATM autophosphorylation at Ser1981 in human HT29 cells preincubated for 1 hr followed by X ray irradiation and measured after 1 hr by H...More data for this Ligand-Target Pair
Affinity DataIC50: 0.940nMAssay Description:Inhibition of ATM autophosphorylation at Ser1981 in human HT29 cells preincubated for 1 hr followed by X ray irradiation and measured after 1 hr by H...More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Binding affinity to integrin alpha5beta1More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Binding affinity to integrin alpha5beta1More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Binding affinity to integrin alpha5beta1More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Binding affinity to integrin alpha5beta1More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Antagonist activity at integrin alphavbeta3 in human A375M cells assessed as inhibition of cell adhesion to fibrinogen in presence of Mg2+More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Binding affinity to integrin alpha5beta1More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Binding affinity to integrin alpha5beta1More data for this Ligand-Target Pair
Affinity DataIC50: 1.10nMAssay Description:Inhibition of ATM autophosphorylation at Ser1981 in human HT29 cells preincubated for 1 hr followed by X ray irradiation and measured after 1 hr by H...More data for this Ligand-Target Pair
Affinity DataIC50: 1.10nMAssay Description:Inhibition of ATM autophosphorylation at Ser1981 in human HT29 cells preincubated for 1 hr followed by X ray irradiation and measured after 1 hr by H...More data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Inhibition of ATM autophosphorylation at Ser1981 in human HT29 cells preincubated for 1 hr followed by X ray irradiation and measured after 1 hr by H...More data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:Inhibition of ATM autophosphorylation at Ser1981 in human HT29 cells preincubated for 1 hr followed by X ray irradiation and measured after 1 hr by H...More data for this Ligand-Target Pair
Affinity DataIC50: 1.70nMAssay Description:Inhibition of ATM autophosphorylation at Ser1981 in human HT29 cells preincubated for 1 hr followed by X ray irradiation and measured after 1 hr by H...More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Binding affinity to integrin alpha5beta1More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Binding affinity to integrin alpha5beta1More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Antagonist activity at integrin alpha5beta1 in human A375M cells assessed as inhibition of cell adhesion to fibronectin in presence of Mg2+ and MK-04...More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Binding affinity to integrin alpha5beta1More data for this Ligand-Target Pair
Affinity DataIC50: 2.60nMAssay Description:Inhibition of ATM autophosphorylation at Ser1981 in human HT29 cells preincubated for 1 hr followed by X ray irradiation and measured after 1 hr by H...More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Binding affinity to integrin alpha5beta1More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of ATM derived from human HeLa cell nuclear extract using glutathione S-transferase p53N66 as substrate preincubated for 10 mins followed ...More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Binding affinity to integrin alpha5beta1More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Binding affinity to integrin alpha5beta1More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Binding affinity to integrin alpha5beta1More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Binding affinity to integrin alpha5beta1More data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Binding affinity to integrin alpha5beta1More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Binding affinity to integrin alpha5beta1More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Binding affinity to integrin alpha5beta1More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibition of ATM autophosphorylation at Ser1981 in human HT29 cells preincubated for 1 hr followed by X ray irradiation and measured after 1 hr by H...More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Binding affinity to integrin alpha5beta1More data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Binding affinity to integrin alpha5beta1More data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition of ATM autophosphorylation at Ser1981 in human HT29 cells preincubated for 1 hr followed by X ray irradiation and measured after 1 hr by H...More data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Antagonist activity at integrin alphavbeta3 in human A375M cells assessed as inhibition of cell adhesion to fibrinogen in presence of Mg2+More data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Antagonist activity at integrin alpha5beta1 in human K562 cells assessed as inhibition of cell adhesionMore data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Antagonist activity at integrin alpha5beta1 in human K562 cells assessed as inhibition of cell adhesionMore data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Binding affinity to integrin alpha5beta1More data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Binding affinity to integrin alpha5beta1More data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Binding affinity to integrin alpha5beta1More data for this Ligand-Target Pair