Affinity DataKi: 0.794nMAssay Description:Displacement of 3H-oxytocin from human recombinant oxytocin receptor expressed in CHO cells by filtration binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.794nMAssay Description:Antagonist activity at human oxytocin receptor expressed in CHO cells by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.26nMAssay Description:Displacement of [3H]oxytocin from human oxytocin receptor expressed in CHO cells by filtration binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.58nMAssay Description:Binding affinity to human recombinant oxytocin receptor expressed in CHO cells by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Antagonist activity at human CCR2 receptor expressed in CHO cells assessed as inhibition of MCP1-induced [35S]-GTPgammaS binding after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Antagonist activity at human NPY Y2 receptor in KAN-TS cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Antagonist activity at human recombinant oxytocin receptor expressed in CHO cells by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.51nMAssay Description:Binding affinity to human recombinant oxytocin receptor expressed in CHO cells by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.51nMAssay Description:Antagonist activity at human neuropeptide Y2 receptor in KAN-TS cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Antagonist activity at human CCR2 receptor expressed in CHO cells assessed as inhibition of MCP1-induced [35S]-GTPgammaS binding after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 3.16nMAssay Description:Antagonist activity at human oxytocin receptor expressed in CHO cells by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataKi: 3.16nMAssay Description:Antagonist activity at human recombinant oxytocin receptor expressed in CHO cells by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataKi: 3.16nMAssay Description:Antagonist activity at human oxytocin receptor expressed in CHO cells by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataKi: 3.98nMAssay Description:Antagonist activity at human neuropeptide Y2 receptor in KAN-TS cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
Affinity DataKi: 3.98nMAssay Description:Binding affinity to human recombinant oxytocin receptor expressed in CHO cells by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Antagonist activity at human CCR2 receptor expressed in CHO cells assessed as inhibition of MCP1-induced [35S]-GTPgammaS binding after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 5.01nMAssay Description:Antagonist activity at human neuropeptide Y2 receptor in KAN-TS cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Antagonist activity at human CCR2 receptor expressed in CHO cells assessed as inhibition of MCP1-induced [35S]-GTPgammaS binding after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 6.31nMAssay Description:Antagonist activity at human recombinant oxytocin receptor expressed in CHO cells by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataKi: 6.31nMAssay Description:Binding affinity to human recombinant oxytocin receptor expressed in CHO cells by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 6.31nMAssay Description:Antagonist activity at human neuropeptide Y2 receptor in KAN-TS cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
Affinity DataKi: 6.31nMAssay Description:Binding affinity to human recombinant oxytocin receptor expressed in CHO cells by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 6.80nMAssay Description:Binding affinity to oxytocin receptorMore data for this Ligand-Target Pair
Affinity DataKi: 7.94nMAssay Description:Antagonist activity at human oxytocin receptor expressed in CHO cells by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataKi: 7.94nMAssay Description:Antagonist activity at human recombinant oxytocin receptor expressed in CHO cells by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataKi: 7.94nMAssay Description:Binding affinity to human recombinant oxytocin receptor expressed in CHO cells by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Antagonist activity at human CCR2 receptor expressed in CHO cells assessed as inhibition of MCP1-induced [35S]-GTPgammaS binding after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Antagonist activity at human CCR2 receptor expressed in CHO cells assessed as inhibition of MCP1-induced [35S]-GTPgammaS binding after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Antagonist activity at human CCR2 receptor expressed in CHO cells assessed as inhibition of MCP1-induced [35S]-GTPgammaS binding after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Antagonist activity at human neuropeptide Y2 receptor in KAN-TS cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Antagonist activity at human CCR2 receptor expressed in CHO cells assessed as inhibition of MCP1-induced [35S]-GTPgammaS binding after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity to human recombinant oxytocin receptor expressed in CHO cells by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity to human CCR2More data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity to human recombinant oxytocin receptor expressed in CHO cells by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity to CCR2 by 35S-gamma-GTP membrane assayMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity to CCR2 by 35S-gamma-GTP membrane assayMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity to CCR2 by 35S-gamma-GTP membrane assayMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Antagonist activity at human CCR2 receptor expressed in CHO cells assessed as inhibition of MCP1-induced [35S]-GTPgammaS binding after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity to CCR2 by 35S-gamma-GTP membrane assayMore data for this Ligand-Target Pair
Affinity DataKi: 12.6nMAssay Description:Binding affinity to CCR2 by 35S-gamma-GTP membrane assayMore data for this Ligand-Target Pair
Affinity DataKi: 12.6nMAssay Description:Binding affinity to CCR2 by 35S-gamma-GTP membrane assayMore data for this Ligand-Target Pair
Affinity DataKi: 12.6nMAssay Description:Binding affinity to human recombinant oxytocin receptor expressed in CHO cells by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 12.6nMAssay Description:Binding affinity to human recombinant oxytocin receptor expressed in CHO cells by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 12.6nMAssay Description:Binding affinity to human recombinant oxytocin receptor expressed in CHO cells by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 12.6nMAssay Description:Binding affinity to human recombinant oxytocin receptor expressed in CHO cells by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 12.6nMAssay Description:Binding affinity to human recombinant oxytocin receptor expressed in CHO cells by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 12.6nMAssay Description:Antagonist activity at human neuropeptide Y2 receptor in KAN-TS cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
Affinity DataKi: 12.6nMAssay Description:Antagonist activity at human neuropeptide Y2 receptor in KAN-TS cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
Affinity DataKi: 12.6nMAssay Description:Binding affinity to human recombinant oxytocin receptor expressed in CHO cells by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Antagonist activity at human CCR2 receptor expressed in CHO cells assessed as inhibition of MCP1-induced [35S]-GTPgammaS binding after 3 hrsMore data for this Ligand-Target Pair