TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataKi: 0.0200nMAssay Description:Inhibition of matripase (unknown origin) using Boc-QAR-AMC as substrate incubated for 30 mins prior to substrate addition by fluorescence assayMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Consejo Superior De Investigaciones Cient�Ficas (Iqm-Csic)
Curated by ChEMBL
Consejo Superior De Investigaciones Cient�Ficas (Iqm-Csic)
Curated by ChEMBL
Affinity DataKi: 0.130nMAssay Description:Displacement of [125l]-lodomelatonin from human MT2 receptor expressed in CHO cells incubated for 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Consejo Superior De Investigaciones Cient�Ficas (Iqm-Csic)
Curated by ChEMBL
Consejo Superior De Investigaciones Cient�Ficas (Iqm-Csic)
Curated by ChEMBL
Affinity DataKi: 0.270nMAssay Description:Displacement of [125l]-lodomelatonin from human MT1 receptor expressed in CHO cells incubated for 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 0.530nMAssay Description:Inhibition of hepsin (unknown origin) using Boc-QAR-AMC as substrate after 30 mins prior to substrate addition by fluorescence assayMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Consejo Superior De Investigaciones Cient�Ficas (Iqm-Csic)
Curated by ChEMBL
Consejo Superior De Investigaciones Cient�Ficas (Iqm-Csic)
Curated by ChEMBL
Affinity DataKi: 4nMAssay Description:Displacement of [125l]-lodomelatonin from human MT2 receptor expressed in CHO cells incubated for 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataKi: 4.30nMAssay Description:Inhibition of matripase (unknown origin) using Boc-QAR-AMC as substrate incubated for 30 mins prior to substrate addition by fluorescence assayMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Consejo Superior De Investigaciones Cient�Ficas (Iqm-Csic)
Curated by ChEMBL
Consejo Superior De Investigaciones Cient�Ficas (Iqm-Csic)
Curated by ChEMBL
Affinity DataKi: 5.10nMAssay Description:Displacement of [125l]-lodomelatonin from human MT2 receptor expressed in CHO cells incubated for 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Consejo Superior De Investigaciones Cient�Ficas (Iqm-Csic)
Curated by ChEMBL
Consejo Superior De Investigaciones Cient�Ficas (Iqm-Csic)
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Displacement of [125l]-lodomelatonin from human MT2 receptor expressed in CHO cells incubated for 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Inhibition of human N-terminal His-tagged glycolate oxidase expressed in C41(D43) Escherichia coli using glycolate as substrate preincubated for 30 m...More data for this Ligand-Target Pair
TargetHepatocyte growth factor activator(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataKi: 25nMAssay Description:Inhibition of recombinant N-terminal His-tagged HGFA (unknown origin) expressed in baculovirus-infected Sf9 cells using Boc-QLR-AMC as substrate incu...More data for this Ligand-Target Pair
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Consejo Superior De Investigaciones Cient�Ficas (Iqm-Csic)
Curated by ChEMBL
Consejo Superior De Investigaciones Cient�Ficas (Iqm-Csic)
Curated by ChEMBL
Affinity DataKi: 35nMAssay Description:Displacement of [125l]-lodomelatonin from human MT1 receptor expressed in CHO cells incubated for 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 48nMAssay Description:Inhibition of hepsin (unknown origin) using Boc-QAR-AMC as substrate after 30 mins prior to substrate addition by fluorescence assayMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Consejo Superior De Investigaciones Cient�Ficas (Iqm-Csic)
Curated by ChEMBL
Consejo Superior De Investigaciones Cient�Ficas (Iqm-Csic)
Curated by ChEMBL
Affinity DataKi: 69nMAssay Description:Displacement of [125l]-lodomelatonin from human MT2 receptor expressed in CHO cells incubated for 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 90nMAssay Description:Non-competitive inhibition of human recombinant LDHA assessed as inhibition constant using varying concentration of pyruvate as substrate preincubate...More data for this Ligand-Target Pair
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Consejo Superior De Investigaciones Cient�Ficas (Iqm-Csic)
Curated by ChEMBL
Consejo Superior De Investigaciones Cient�Ficas (Iqm-Csic)
Curated by ChEMBL
Affinity DataKi: >100nMAssay Description:Displacement of [125l]-lodomelatonin from human MT1 receptor expressed in CHO cells incubated for 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Consejo Superior De Investigaciones Cient�Ficas (Iqm-Csic)
Curated by ChEMBL
Consejo Superior De Investigaciones Cient�Ficas (Iqm-Csic)
Curated by ChEMBL
Affinity DataKi: >100nMAssay Description:Displacement of [125l]-lodomelatonin from human MT2 receptor expressed in CHO cells incubated for 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Consejo Superior De Investigaciones Cient�Ficas (Iqm-Csic)
Curated by ChEMBL
Consejo Superior De Investigaciones Cient�Ficas (Iqm-Csic)
Curated by ChEMBL
Affinity DataKi: >100nMAssay Description:Displacement of [125l]-lodomelatonin from human MT2 receptor expressed in CHO cells incubated for 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Consejo Superior De Investigaciones Cient�Ficas (Iqm-Csic)
Curated by ChEMBL
Consejo Superior De Investigaciones Cient�Ficas (Iqm-Csic)
Curated by ChEMBL
Affinity DataKi: >100nMAssay Description:Displacement of [125l]-lodomelatonin from human MT2 receptor expressed in CHO cells incubated for 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Consejo Superior De Investigaciones Cient�Ficas (Iqm-Csic)
Curated by ChEMBL
Consejo Superior De Investigaciones Cient�Ficas (Iqm-Csic)
Curated by ChEMBL
Affinity DataKi: >100nMAssay Description:Displacement of [125l]-lodomelatonin from human MT2 receptor expressed in CHO cells incubated for 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Consejo Superior De Investigaciones Cient�Ficas (Iqm-Csic)
Curated by ChEMBL
Consejo Superior De Investigaciones Cient�Ficas (Iqm-Csic)
Curated by ChEMBL
Affinity DataKi: >100nMAssay Description:Displacement of [125l]-lodomelatonin from human MT1 receptor expressed in CHO cells incubated for 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Consejo Superior De Investigaciones Cient�Ficas (Iqm-Csic)
Curated by ChEMBL
Consejo Superior De Investigaciones Cient�Ficas (Iqm-Csic)
Curated by ChEMBL
Affinity DataKi: >100nMAssay Description:Displacement of [125l]-lodomelatonin from human MT1 receptor expressed in CHO cells incubated for 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Consejo Superior De Investigaciones Cient�Ficas (Iqm-Csic)
Curated by ChEMBL
Consejo Superior De Investigaciones Cient�Ficas (Iqm-Csic)
Curated by ChEMBL
Affinity DataKi: >100nMAssay Description:Displacement of [125l]-lodomelatonin from human MT1 receptor expressed in CHO cells incubated for 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Consejo Superior De Investigaciones Cient�Ficas (Iqm-Csic)
Curated by ChEMBL
Consejo Superior De Investigaciones Cient�Ficas (Iqm-Csic)
Curated by ChEMBL
Affinity DataKi: >100nMAssay Description:Displacement of [125l]-lodomelatonin from human MT1 receptor expressed in CHO cells incubated for 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Consejo Superior De Investigaciones Cient�Ficas (Iqm-Csic)
Curated by ChEMBL
Consejo Superior De Investigaciones Cient�Ficas (Iqm-Csic)
Curated by ChEMBL
Affinity DataKi: 110nMAssay Description:Displacement of [125l]-lodomelatonin from human MT2 receptor expressed in CHO cells incubated for 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataKi: 120nMAssay Description:Inhibition of matripase (unknown origin) using Boc-QAR-AMC as substrate incubated for 30 mins prior to substrate addition by fluorescence assayMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Consejo Superior De Investigaciones Cient�Ficas (Iqm-Csic)
Curated by ChEMBL
Consejo Superior De Investigaciones Cient�Ficas (Iqm-Csic)
Curated by ChEMBL
Affinity DataKi: 230nMAssay Description:Displacement of [125l]-lodomelatonin from human MT2 receptor expressed in CHO cells incubated for 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Consejo Superior De Investigaciones Cient�Ficas (Iqm-Csic)
Curated by ChEMBL
Consejo Superior De Investigaciones Cient�Ficas (Iqm-Csic)
Curated by ChEMBL
Affinity DataKi: 260nMAssay Description:Displacement of [125l]-lodomelatonin from human MT1 receptor expressed in CHO cells incubated for 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Consejo Superior De Investigaciones Cient�Ficas (Iqm-Csic)
Curated by ChEMBL
Consejo Superior De Investigaciones Cient�Ficas (Iqm-Csic)
Curated by ChEMBL
Affinity DataKi: 260nMAssay Description:Displacement of [125l]-lodomelatonin from human MT2 receptor expressed in CHO cells incubated for 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataKi: 300nMAssay Description:Inhibition of matripase (unknown origin) using Boc-QAR-AMC as substrate incubated for 30 mins prior to substrate addition by fluorescence assayMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Consejo Superior De Investigaciones Cient�Ficas (Iqm-Csic)
Curated by ChEMBL
Consejo Superior De Investigaciones Cient�Ficas (Iqm-Csic)
Curated by ChEMBL
Affinity DataKi: 300nMAssay Description:Displacement of [125l]-lodomelatonin from human MT2 receptor expressed in CHO cells incubated for 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Consejo Superior De Investigaciones Cient�Ficas (Iqm-Csic)
Curated by ChEMBL
Consejo Superior De Investigaciones Cient�Ficas (Iqm-Csic)
Curated by ChEMBL
Affinity DataKi: 320nMAssay Description:Displacement of [125l]-lodomelatonin from human MT2 receptor expressed in CHO cells incubated for 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Consejo Superior De Investigaciones Cient�Ficas (Iqm-Csic)
Curated by ChEMBL
Consejo Superior De Investigaciones Cient�Ficas (Iqm-Csic)
Curated by ChEMBL
Affinity DataKi: 390nMAssay Description:Displacement of [125l]-lodomelatonin from human MT2 receptor expressed in CHO cells incubated for 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataKi: 480nMAssay Description:Inhibition of matripase (unknown origin) using Boc-QAR-AMC as substrate incubated for 30 mins prior to substrate addition by fluorescence assayMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Consejo Superior De Investigaciones Cient�Ficas (Iqm-Csic)
Curated by ChEMBL
Consejo Superior De Investigaciones Cient�Ficas (Iqm-Csic)
Curated by ChEMBL
Affinity DataKi: 530nMAssay Description:Displacement of [125l]-lodomelatonin from human MT2 receptor expressed in CHO cells incubated for 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Consejo Superior De Investigaciones Cient�Ficas (Iqm-Csic)
Curated by ChEMBL
Consejo Superior De Investigaciones Cient�Ficas (Iqm-Csic)
Curated by ChEMBL
Affinity DataKi: 550nMAssay Description:Displacement of [125l]-lodomelatonin from human MT1 receptor expressed in CHO cells incubated for 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Consejo Superior De Investigaciones Cient�Ficas (Iqm-Csic)
Curated by ChEMBL
Consejo Superior De Investigaciones Cient�Ficas (Iqm-Csic)
Curated by ChEMBL
Affinity DataKi: 550nMAssay Description:Displacement of [125l]-lodomelatonin from human MT1 receptor expressed in CHO cells incubated for 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 553nMAssay Description:Inhibition of hepsin (unknown origin) using Boc-QAR-AMC as substrate after 30 mins prior to substrate addition by fluorescence assayMore data for this Ligand-Target Pair
TargetHepatocyte growth factor activator(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataKi: 590nMAssay Description:Inhibition of HGFA (unknown origin) after 40 mins by Eadie-Hofstee plot analysisMore data for this Ligand-Target Pair
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataKi: 620nMAssay Description:Inhibition of matripase (unknown origin) using Boc-QAR-AMC as substrate incubated for 30 mins prior to substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 670nMAssay Description:Inhibition of hepsin (unknown origin) using Boc-QAR-AMC as substrate after 30 mins prior to substrate addition by fluorescence assayMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Consejo Superior De Investigaciones Cient�Ficas (Iqm-Csic)
Curated by ChEMBL
Consejo Superior De Investigaciones Cient�Ficas (Iqm-Csic)
Curated by ChEMBL
Affinity DataKi: 690nMAssay Description:Displacement of [125l]-lodomelatonin from human MT1 receptor expressed in CHO cells incubated for 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 700nMAssay Description:Non-competitive inhibition of human recombinant LDHB assessed as inhibition constant using varying concentration of pyruvate as substrate preincubate...More data for this Ligand-Target Pair
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataKi: 760nMAssay Description:Inhibition of matripase (unknown origin) using Boc-QAR-AMC as substrate incubated for 30 mins prior to substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 835nMAssay Description:Inhibition of hepsin (unknown origin) using Boc-QAR-AMC as substrate after 30 mins prior to substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 900nMAssay Description:Non-competitive inhibition of human recombinant LDHA assessed as inhibition constant using varying concentration of pyruvate as substrate preincubate...More data for this Ligand-Target Pair
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Consejo Superior De Investigaciones Cient�Ficas (Iqm-Csic)
Curated by ChEMBL
Consejo Superior De Investigaciones Cient�Ficas (Iqm-Csic)
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [125l]-lodomelatonin from human MT1 receptor expressed in CHO cells incubated for 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+3nMAssay Description:Inhibition of hepsin (unknown origin) using Boc-QAR-AMC as substrate after 30 mins prior to substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.10E+3nMAssay Description:Non-competitive mixed inhibition of N-terminal His-tagged human recombinant glycolate oxidase expressed in Escherichia coli BL21 (DE3) cells assessed...More data for this Ligand-Target Pair
Affinity DataKi: 1.20E+3nMAssay Description:Inhibition of hepsin (unknown origin) using Boc-QAR-AMC as substrate after 30 mins prior to substrate addition by fluorescence assayMore data for this Ligand-Target Pair
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataKi: 1.20E+3nMAssay Description:Inhibition of matripase (unknown origin) using Boc-QAR-AMC as substrate incubated for 30 mins prior to substrate addition by fluorescence assayMore data for this Ligand-Target Pair