Compile Data Set for Download or QSAR
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Found 59 with Last Name = 'funke' and Initial = 'u'
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Tours

Curated by ChEMBL
LigandPNGBDBM50218673(2-(2-((dimethylamino)methyl)-4-fluorophenylthio)-5...)
Affinity DataKi:  0.270nMAssay Description:Displacement of [3H]paroxetine from SERT in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Tours

Curated by ChEMBL
LigandPNGBDBM50218674(3-amino-4-(2-((dimethylamino)methyl)-4-fluoropheny...)
Affinity DataKi:  0.280nMAssay Description:Displacement of [3H]citalopram from SERT in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Tours

Curated by ChEMBL
LigandPNGBDBM50218670(5-chloro-2-(2-((dimethylamino)methyl)-4-fluorophen...)
Affinity DataKi:  0.350nMAssay Description:Displacement of [3H]paroxetine from SERT in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Institut FüR InterdisziplinäRe Isotopenforschung

Curated by ChEMBL
LigandPNGBDBM22416((3S,4R)-3-[(1,3-benzodioxol-5-yloxy)methyl]-4-(4-f...)
Affinity DataKi:  0.380nMAssay Description:Displacement of [3H]paroxetine from human SERT expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Institut FüR InterdisziplinäRe Isotopenforschung

Curated by ChEMBL
LigandPNGBDBM22416((3S,4R)-3-[(1,3-benzodioxol-5-yloxy)methyl]-4-(4-f...)
Affinity DataKi:  0.420nMAssay Description:Displacement of [3H]citalopram from human SERT expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Tours

Curated by ChEMBL
LigandPNGBDBM50110788(2-(2-((dimethylamino)methyl)phenylthio)-5-methylan...)
Affinity DataKi:  0.620nMAssay Description:Displacement of [3H]paroxetine from SERT in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Institut FüR InterdisziplinäRe Isotopenforschung

Curated by ChEMBL
LigandPNGBDBM50110788(2-(2-((dimethylamino)methyl)phenylthio)-5-methylan...)
Affinity DataKi:  0.730nMAssay Description:Displacement of [3H]citalopram from human SERT expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Institut FüR InterdisziplinäRe Isotopenforschung

Curated by ChEMBL
LigandPNGBDBM50110788(2-(2-((dimethylamino)methyl)phenylthio)-5-methylan...)
Affinity DataKi:  2.03nMAssay Description:Displacement of [3H]paroxetine from human SERT expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Tours

Curated by ChEMBL
LigandPNGBDBM50218671(2-(4-chloro-2-((dimethylamino)methyl)phenoxy)-5-fl...)
Affinity DataKi:  2.06nMAssay Description:Displacement of [3H]citalopram from SERT in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Tours

Curated by ChEMBL
LigandPNGBDBM50218675(3-amino-4-(2-((dimethylamino)methyl)-4-fluoropheno...)
Affinity DataKi:  2.91nMAssay Description:Displacement of [3H]paroxetine from SERT in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Institut FüR InterdisziplinäRe Isotopenforschung

Curated by ChEMBL
LigandPNGBDBM50102006(3-[4-(6-Methoxy-3,4-dihydro-1H-isoquinolin-2-yl)-c...)
Affinity DataKi:  4.10nMAssay Description:Displacement of [3H]citalopram from human SERT expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Institut FüR InterdisziplinäRe Isotopenforschung

Curated by ChEMBL
LigandPNGBDBM25870(1-[3-(dimethylamino)propyl]-1-(4-fluorophenyl)-1,3...)
Affinity DataKi:  4.38nMAssay Description:Displacement of [3H]citalopram from human SERT expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Institut FüR InterdisziplinäRe Isotopenforschung

Curated by ChEMBL
LigandPNGBDBM50102010(3-[4-(3,4-Dihydro-1H-isoquinolin-2-yl)-cyclohexyl]...)
Affinity DataKi:  4.51nMAssay Description:Displacement of [3H]citalopram from human SERT expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Institut FüR InterdisziplinäRe Isotopenforschung

Curated by ChEMBL
LigandPNGBDBM50262513(CHEMBL449277 | cis-3-(4-(6-(3-fluoropropoxy)-3,4-d...)
Affinity DataKi:  6.16nMAssay Description:Displacement of [3H]citalopram from human SERT expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Tours

Curated by ChEMBL
LigandPNGBDBM50218672(2-(2-((dimethylamino)methyl)-4-fluorophenoxy)-5-me...)
Affinity DataKi:  7.01nMAssay Description:Displacement of [3H]paroxetine from SERT in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Tours

Curated by ChEMBL
LigandPNGBDBM50218676(2-(2-((dimethylamino)methyl)phenoxy)-5-fluorobenze...)
Affinity DataKi:  13.4nMAssay Description:Displacement of [3H]paroxetine from SERT in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Institut FüR InterdisziplinäRe Isotopenforschung

Curated by ChEMBL
LigandPNGBDBM25870(1-[3-(dimethylamino)propyl]-1-(4-fluorophenyl)-1,3...)
Affinity DataKi:  32.8nMAssay Description:Displacement of [3H]paroxetine from human SERT expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Institut FüR InterdisziplinäRe Isotopenforschung

Curated by ChEMBL
LigandPNGBDBM50102008(3-[4-(6-Methoxy-3,4-dihydro-1H-isoquinolin-2-yl)-c...)
Affinity DataKi:  73.7nMAssay Description:Displacement of [3H]citalopram from human SERT expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Institut FüR InterdisziplinäRe Isotopenforschung

Curated by ChEMBL
LigandPNGBDBM50102019(3-[4-(3,4-Dihydro-1H-isoquinolin-2-yl)-cyclohexyl]...)
Affinity DataKi:  90.7nMAssay Description:Displacement of [3H]citalopram from human SERT expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Institut FüR InterdisziplinäRe Isotopenforschung

Curated by ChEMBL
LigandPNGBDBM50102008(3-[4-(6-Methoxy-3,4-dihydro-1H-isoquinolin-2-yl)-c...)
Affinity DataKi:  96.7nMAssay Description:Displacement of [3H]nisoxetine from human NET expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Institut FüR InterdisziplinäRe Isotopenforschung

Curated by ChEMBL
LigandPNGBDBM50262514(CHEMBL477587 | trans-3-(4-(6-(3-fluoropropoxy)-3,4...)
Affinity DataKi:  102nMAssay Description:Displacement of [3H]nisoxetine from human NET expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Institut FüR InterdisziplinäRe Isotopenforschung

Curated by ChEMBL
LigandPNGBDBM50102006(3-[4-(6-Methoxy-3,4-dihydro-1H-isoquinolin-2-yl)-c...)
Affinity DataKi:  165nMAssay Description:Displacement of [3H]paroxetine from human SERT expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Institut FüR InterdisziplinäRe Isotopenforschung

Curated by ChEMBL
LigandPNGBDBM50102019(3-[4-(3,4-Dihydro-1H-isoquinolin-2-yl)-cyclohexyl]...)
Affinity DataKi:  184nMAssay Description:Displacement of [3H]nisoxetine from human NET expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Institut FüR InterdisziplinäRe Isotopenforschung

Curated by ChEMBL
LigandPNGBDBM50102010(3-[4-(3,4-Dihydro-1H-isoquinolin-2-yl)-cyclohexyl]...)
Affinity DataKi:  189nMAssay Description:Displacement of [3H]paroxetine from human SERT expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Institut FüR InterdisziplinäRe Isotopenforschung

Curated by ChEMBL
LigandPNGBDBM50102008(3-[4-(6-Methoxy-3,4-dihydro-1H-isoquinolin-2-yl)-c...)
Affinity DataKi:  267nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Institut FüR InterdisziplinäRe Isotopenforschung

Curated by ChEMBL
LigandPNGBDBM50102019(3-[4-(3,4-Dihydro-1H-isoquinolin-2-yl)-cyclohexyl]...)
Affinity DataKi:  286nMAssay Description:Displacement of [3H]paroxetine from human SERT expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Institut FüR InterdisziplinäRe Isotopenforschung

Curated by ChEMBL
LigandPNGBDBM50102019(3-[4-(3,4-Dihydro-1H-isoquinolin-2-yl)-cyclohexyl]...)
Affinity DataKi:  309nMAssay Description:Displacement of [3H]WIN35428 from human DAT expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Institut FüR InterdisziplinäRe Isotopenforschung

Curated by ChEMBL
LigandPNGBDBM50262514(CHEMBL477587 | trans-3-(4-(6-(3-fluoropropoxy)-3,4...)
Affinity DataKi:  327nMAssay Description:Displacement of [3H]citalopram from human SERT expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Institut FüR InterdisziplinäRe Isotopenforschung

Curated by ChEMBL
LigandPNGBDBM50262514(CHEMBL477587 | trans-3-(4-(6-(3-fluoropropoxy)-3,4...)
Affinity DataKi:  343nMAssay Description:Displacement of [3H]WIN35428 from human DAT expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Institut FüR InterdisziplinäRe Isotopenforschung

Curated by ChEMBL
LigandPNGBDBM50262513(CHEMBL449277 | cis-3-(4-(6-(3-fluoropropoxy)-3,4-d...)
Affinity DataKi:  366nMAssay Description:Displacement of [3H]WIN35428 from human DAT expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Institut FüR InterdisziplinäRe Isotopenforschung

Curated by ChEMBL
LigandPNGBDBM50102006(3-[4-(6-Methoxy-3,4-dihydro-1H-isoquinolin-2-yl)-c...)
Affinity DataKi:  370nMAssay Description:Displacement of [3H]WIN35428 from human DAT expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Institut FüR InterdisziplinäRe Isotopenforschung

Curated by ChEMBL
LigandPNGBDBM50102010(3-[4-(3,4-Dihydro-1H-isoquinolin-2-yl)-cyclohexyl]...)
Affinity DataKi:  424nMAssay Description:Displacement of [3H]WIN35428 from human DAT expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Institut FüR InterdisziplinäRe Isotopenforschung

Curated by ChEMBL
LigandPNGBDBM50102008(3-[4-(6-Methoxy-3,4-dihydro-1H-isoquinolin-2-yl)-c...)
Affinity DataKi:  462nMAssay Description:Displacement of [3H]WIN35428 from human DAT expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
University Of Tours

Curated by ChEMBL
LigandPNGBDBM50218672(2-(2-((dimethylamino)methyl)-4-fluorophenoxy)-5-me...)
Affinity DataKi:  518nMAssay Description:Displacement of [3H]nisoxetine from NET in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Institut FüR InterdisziplinäRe Isotopenforschung

Curated by ChEMBL
LigandPNGBDBM50102008(3-[4-(6-Methoxy-3,4-dihydro-1H-isoquinolin-2-yl)-c...)
Affinity DataKi:  518nMAssay Description:Displacement of [3H]paroxetine from human SERT expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Institut FüR InterdisziplinäRe Isotopenforschung

Curated by ChEMBL
LigandPNGBDBM50262513(CHEMBL449277 | cis-3-(4-(6-(3-fluoropropoxy)-3,4-d...)
Affinity DataKi:  772nMAssay Description:Displacement of [3H]nisoxetine from human NET expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Institut FüR InterdisziplinäRe Isotopenforschung

Curated by ChEMBL
LigandPNGBDBM50262513(CHEMBL449277 | cis-3-(4-(6-(3-fluoropropoxy)-3,4-d...)
Affinity DataKi:  914nMAssay Description:Displacement of [3H]paroxetine from human SERT expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
University Of Tours

Curated by ChEMBL
LigandPNGBDBM50218670(5-chloro-2-(2-((dimethylamino)methyl)-4-fluorophen...)
Affinity DataKi:  919nMAssay Description:Displacement of [3H]nisoxetine from NET in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Institut FüR InterdisziplinäRe Isotopenforschung

Curated by ChEMBL
LigandPNGBDBM50102010(3-[4-(3,4-Dihydro-1H-isoquinolin-2-yl)-cyclohexyl]...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Institut FüR InterdisziplinäRe Isotopenforschung

Curated by ChEMBL
LigandPNGBDBM50102006(3-[4-(6-Methoxy-3,4-dihydro-1H-isoquinolin-2-yl)-c...)
Affinity DataKi:  1.02E+3nMAssay Description:Displacement of [3H]nisoxetine from human NET expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
University Of Tours

Curated by ChEMBL
LigandPNGBDBM50218673(2-(2-((dimethylamino)methyl)-4-fluorophenylthio)-5...)
Affinity DataKi:  1.04E+3nMAssay Description:Displacement of [3H]nisoxetine from NET in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
University Of Tours

Curated by ChEMBL
LigandPNGBDBM50218676(2-(2-((dimethylamino)methyl)phenoxy)-5-fluorobenze...)
Affinity DataKi:  1.08E+3nMAssay Description:Displacement of [3H]nisoxetine from NET in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Institut FüR InterdisziplinäRe Isotopenforschung

Curated by ChEMBL
LigandPNGBDBM50102010(3-[4-(3,4-Dihydro-1H-isoquinolin-2-yl)-cyclohexyl]...)
Affinity DataKi:  1.43E+3nMAssay Description:Displacement of [3H]nisoxetine from human NET expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Tours

Curated by ChEMBL
LigandPNGBDBM50218670(5-chloro-2-(2-((dimethylamino)methyl)-4-fluorophen...)
Affinity DataKi:  1.84E+3nMAssay Description:Displacement of [3H]WIN35428 from DAT in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Institut FüR InterdisziplinäRe Isotopenforschung

Curated by ChEMBL
LigandPNGBDBM50262514(CHEMBL477587 | trans-3-(4-(6-(3-fluoropropoxy)-3,4...)
Affinity DataKi:  2.31E+3nMAssay Description:Displacement of [3H]paroxetine from human SERT expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Institut FüR InterdisziplinäRe Isotopenforschung

Curated by ChEMBL
LigandPNGBDBM50102019(3-[4-(3,4-Dihydro-1H-isoquinolin-2-yl)-cyclohexyl]...)
Affinity DataKi:  2.53E+3nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Tours

Curated by ChEMBL
LigandPNGBDBM50218671(2-(4-chloro-2-((dimethylamino)methyl)phenoxy)-5-fl...)
Affinity DataKi:  2.53E+3nMAssay Description:Displacement of [3H]WIN35428 from DAT in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
University Of Tours

Curated by ChEMBL
LigandPNGBDBM50218671(2-(4-chloro-2-((dimethylamino)methyl)phenoxy)-5-fl...)
Affinity DataKi:  2.74E+3nMAssay Description:Displacement of [3H]nisoxetine from NET in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Tours

Curated by ChEMBL
LigandPNGBDBM50218672(2-(2-((dimethylamino)methyl)-4-fluorophenoxy)-5-me...)
Affinity DataKi:  2.79E+3nMAssay Description:Displacement of [3H]WIN35428 from DAT in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Institut FüR InterdisziplinäRe Isotopenforschung

Curated by ChEMBL
LigandPNGBDBM50262514(CHEMBL477587 | trans-3-(4-(6-(3-fluoropropoxy)-3,4...)
Affinity DataKi: >2.86E+3nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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