Affinity DataKi: 0.230nM ΔG°: -55.0kJ/molepH: 7.5 T: 2°CAssay Description:The effectiveness of compounds against the activity of human recombinant caspase-1-8 was measured using fluorometric assays. Assays were carried out ...More data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Inhibition of rat 11beta-HSD1More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Binding affinity to mineralocorticoid receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 3.90nMAssay Description:Inhibition of rat 11beta-HSD1More data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Inhibition against human granzyme BMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Inhibition of rat 11beta-HSD1More data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Inhibition against human granzyme BMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Inhibition against human granzyme BMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Inhibition against human granzyme BMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Inhibition of rat 11beta-HSD1More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Inhibition against human granzyme BMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Inhibition against human granzyme BMore data for this Ligand-Target Pair
Affinity DataKi: 18nM ΔG°: -44.2kJ/molepH: 7.5 T: 2°CAssay Description:The effectiveness of compounds against the activity of human recombinant caspase-1-8 was measured using fluorometric assays. Assays were carried out ...More data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Compound was tested for its inhibition against Caspase-3More data for this Ligand-Target Pair
Affinity DataKi: 38nMAssay Description:Inhibition against human granzyme BMore data for this Ligand-Target Pair
Affinity DataKi: 71nMAssay Description:Compound was tested for its inhibition against Caspase-3More data for this Ligand-Target Pair
Affinity DataKi: 74nMAssay Description:Inhibition against human granzyme BMore data for this Ligand-Target Pair
Affinity DataKi: 75nMAssay Description:Inhibition against human granzyme BMore data for this Ligand-Target Pair
Affinity DataKi: 80nMAssay Description:Inhibition against human granzyme BMore data for this Ligand-Target Pair
Affinity DataKi: 85nMAssay Description:Inhibition against human granzyme BMore data for this Ligand-Target Pair
Affinity DataKi: 122nMAssay Description:Inhibition against human granzyme BMore data for this Ligand-Target Pair
Affinity DataKi: 133nMAssay Description:Inhibition against human granzyme BMore data for this Ligand-Target Pair
Affinity DataKi: 143nMAssay Description:Compound was tested for its inhibition against Caspase-3More data for this Ligand-Target Pair
Affinity DataKi: 202nMAssay Description:Compound was tested for its inhibition against Caspase-3More data for this Ligand-Target Pair
Affinity DataKi: 270nMAssay Description:Inhibition against human granzyme BMore data for this Ligand-Target Pair
Affinity DataKi: 350nMAssay Description:Compound was tested for its inhibition against Caspase-8More data for this Ligand-Target Pair
Affinity DataKi: 360nMAssay Description:Inhibition against human granzyme BMore data for this Ligand-Target Pair
Affinity DataKi: 580nMAssay Description:Inhibition against human granzyme BMore data for this Ligand-Target Pair
Affinity DataKi: 2.30E+3nMAssay Description:Inhibition against human granzyme BMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0390nMAssay Description:Inhibition of mouse recombinant PrCP using Mca-Ala-Pro-Lys(Dnp)-OH as substrate for 30 mins by continuous fluorimetric assayMore data for this Ligand-Target Pair
TargetLysosomal Pro-X carboxypeptidase(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 0.0790nMAssay Description:Inhibition of recombinant human PrCP using Mca-Ala-Pro-Lys(Dnp)-OH as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.110nMAssay Description:Inhibition of mouse PrCPMore data for this Ligand-Target Pair
TargetLysosomal Pro-X carboxypeptidase(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 0.170nMAssay Description:Inhibition of human recombinant PrCP using Mca-Ala-Pro-Lys(Dnp)-OH as substrate for 30 mins by continuous fluorimetric assayMore data for this Ligand-Target Pair
TargetLysosomal Pro-X carboxypeptidase(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 0.180nMAssay Description:Inhibition of recombinant human PrCP using Mca-Ala-Pro-Lys(Dnp)-OH as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.180nMAssay Description:Inhibition of mouse PrCPMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Inhibition of mouse PrCPMore data for this Ligand-Target Pair
TargetLysosomal Pro-X carboxypeptidase(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:Inhibition of human PrCPMore data for this Ligand-Target Pair
TargetLysosomal Pro-X carboxypeptidase(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:Inhibition of human PrCPMore data for this Ligand-Target Pair
TargetLysosomal Pro-X carboxypeptidase(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:Inhibition of human PrCPMore data for this Ligand-Target Pair
Affinity DataIC50: 0.280nMAssay Description:Inhibition of recombinant mouse PrCP using Mca-Ala-Pro-Lys(Dnp)-OH as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetLysosomal Pro-X carboxypeptidase(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 0.300nMAssay Description:Inhibition of human PrCPMore data for this Ligand-Target Pair
TargetLysosomal Pro-X carboxypeptidase(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 0.300nMAssay Description:Inhibition of recombinant human PrCP using Mca-Ala-Pro-Lys(Dnp)-OH as substrate measured for 30 mins by continuous fluorometric assayMore data for this Ligand-Target Pair
TargetLysosomal Pro-X carboxypeptidase(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 0.300nMAssay Description:Inhibition of human PrCPMore data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:Inhibition of mouse PrCPMore data for this Ligand-Target Pair
Affinity DataIC50: 0.310nMAssay Description:Inhibition of mouse PrCPMore data for this Ligand-Target Pair
TargetLysosomal Pro-X carboxypeptidase(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 0.370nMAssay Description:Inhibition of human recombinant PrCP using Mca-Ala-Pro-Lys(Dnp)-OH as substrate for 30 mins by continuous fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.380nMAssay Description:Inhibition of mouse PrCPMore data for this Ligand-Target Pair
Affinity DataIC50: 0.390nMAssay Description:Inhibition of mouse PrCPMore data for this Ligand-Target Pair
Affinity DataIC50: 0.400nMAssay Description:Inhibition of mouse PrCPMore data for this Ligand-Target Pair
Affinity DataIC50: 0.400nMAssay Description:Inhibition of mouse PrCPMore data for this Ligand-Target Pair