Compile Data Set for Download or QSAR
maximum 50k data
Found 66 with Last Name = 'goel' and Initial = 'a'
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50198352(1-(5-acetyl-6,6'-dihydroxy-2',3'-dihydro-[2,3']-bi...)
Affinity DataKi:  2.75E+4nMAssay Description:Inhibition of PTP1B in presence of 0.01% Triton X-100More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50198349(7-(4-methoxy-phenyl)-furo[3,2-g]chromen-5-one | CH...)
Affinity DataKi:  3.00E+4nMAssay Description:Inhibition of PTP1BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50198352(1-(5-acetyl-6,6'-dihydroxy-2',3'-dihydro-[2,3']-bi...)
Affinity DataKi:  3.50E+4nMAssay Description:Inhibition of PTP1BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50198349(7-(4-methoxy-phenyl)-furo[3,2-g]chromen-5-one | CH...)
Affinity DataKi:  3.60E+4nMAssay Description:Inhibition of PTP1B in presence of 0.01% Triton X-100More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50198350(1-(5-acetyl-4,4'-dihydroxy-2',3'-dihydro-[2,3']bib...)
Affinity DataKi:  3.70E+4nMAssay Description:Inhibition of PTP1BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50198348(7-phenyl-furo[3,2-g]chromen-5-one | CHEMBL388814)
Affinity DataKi:  4.50E+4nMAssay Description:Inhibition of PTP1B in presence of 0.01% Triton X-100More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50198351(1-(7'-acetyl-6,6'-dihydroxy-2',3'-dihydro-[2,3']bi...)
Affinity DataKi:  5.40E+4nMAssay Description:Inhibition of PTP1B in presence of 0.01% Triton X-100More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50198348(7-phenyl-furo[3,2-g]chromen-5-one | CHEMBL388814)
Affinity DataKi:  5.70E+4nMAssay Description:Inhibition of PTP1BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50198350(1-(5-acetyl-4,4'-dihydroxy-2',3'-dihydro-[2,3']bib...)
Affinity DataKi:  6.10E+4nMAssay Description:Inhibition of PTP1B in presence of 0.01% Triton X-100More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50198351(1-(7'-acetyl-6,6'-dihydroxy-2',3'-dihydro-[2,3']bi...)
Affinity DataKi:  6.40E+4nMAssay Description:Inhibition of PTP1BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50198351(1-(7'-acetyl-6,6'-dihydroxy-2',3'-dihydro-[2,3']bi...)
Affinity DataIC50:  5.63E+4nMAssay Description:Inhibition of PTP1B in presence of 0.01% Triton X-100More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50277785(4'-Amino-6'-methylsulfanyl-[1,1';2',1'']terphenyl-...)
Affinity DataIC50:  5.80E+4nMAssay Description:Inhibition of PTP1B (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50198352(1-(5-acetyl-6,6'-dihydroxy-2',3'-dihydro-[2,3']-bi...)
Affinity DataIC50:  5.88E+4nMAssay Description:Inhibition of PTP1B in presence of 0.01% Triton X-100More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50198348(7-phenyl-furo[3,2-g]chromen-5-one | CHEMBL388814)
Affinity DataIC50:  6.13E+4nMAssay Description:Inhibition of PTP1B in presence of 0.01% Triton X-100More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50198349(7-(4-methoxy-phenyl)-furo[3,2-g]chromen-5-one | CH...)
Affinity DataIC50:  6.88E+4nMAssay Description:Inhibition of PTP1B in presence of 0.01% Triton X-100More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50277825(4'-Amino-4,4''-dimethoxy-6'-methylsulfanyl-[1,1';2...)
Affinity DataIC50:  7.20E+4nMAssay Description:Inhibition of PTP1B (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50198349(7-(4-methoxy-phenyl)-furo[3,2-g]chromen-5-one | CH...)
Affinity DataIC50:  7.25E+4nMAssay Description:Inhibition of PTP1BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50198351(1-(7'-acetyl-6,6'-dihydroxy-2',3'-dihydro-[2,3']bi...)
Affinity DataIC50:  7.50E+4nMAssay Description:Inhibition of PTP1BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-6-phosphatase catalytic subunit 1(Homo sapiens (Human))
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50277824(4'-Amino-4-fluoro-2'',4''-dimethoxy-6'-methylsulfa...)
Affinity DataIC50:  7.90E+4nMAssay Description:Inhibition of glucose-6-phosphatase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50198350(1-(5-acetyl-4,4'-dihydroxy-2',3'-dihydro-[2,3']bib...)
Affinity DataIC50:  8.00E+4nMAssay Description:Inhibition of PTP1BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50277823(4'-Amino-4''-methoxy-6'-methylsulfanyl-[1,1';2',1'...)
Affinity DataIC50:  8.60E+4nMAssay Description:Inhibition of PTP1B (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50198352(1-(5-acetyl-6,6'-dihydroxy-2',3'-dihydro-[2,3']-bi...)
Affinity DataIC50:  8.70E+4nMAssay Description:Inhibition of PTP1BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50198350(1-(5-acetyl-4,4'-dihydroxy-2',3'-dihydro-[2,3']bib...)
Affinity DataIC50:  9.13E+4nMAssay Description:Inhibition of PTP1B in presence of 0.01% Triton X-100More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50198348(7-phenyl-furo[3,2-g]chromen-5-one | CHEMBL388814)
Affinity DataIC50:  9.40E+4nMAssay Description:Inhibition of PTP1BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50261701(2-Methyl-c-5-[4-(5-methyl-2-phenyloxazol-4-ylmetho...)
Affinity DataEC50:  1.09nMAssay Description:Agonist activity at PPARalpha (unknown origin) expressed in human HepG2 cells assessed as induction of receptor transactivation by reporter gene assa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50261880(CHEMBL512789 | c-5-[4-{2-(2-tert-Butyl-5-methyloxa...)
Affinity DataEC50:  4.20nMAssay Description:Agonist activity at PPARalpha (unknown origin) expressed in human HepG2 cells assessed as induction of receptor transactivation by reporter gene assa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50261879(2-Methyl-c-5-{4-[2-(5-methyl-2-(5-methylthiophen-2...)
Affinity DataEC50:  0.0300nMAssay Description:Agonist activity at PPARalpha (unknown origin) expressed in human HepG2 cells assessed as induction of receptor transactivation by reporter gene assa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50261878(2-Methyl-c-5-{4-[5-methyl-2-(5-methylthiophen-2-yl...)
Affinity DataEC50:  0.600nMAssay Description:Agonist activity at PPARalpha (unknown origin) expressed in human HepG2 cells assessed as induction of receptor transactivation by reporter gene assa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50261703(2-Methyl-c-5-{4-[2-(5-methyl-2-(4-methylphenyl)oxa...)
Affinity DataEC50:  0.0890nMAssay Description:Agonist activity at PPARalpha (unknown origin) expressed in human HepG2 cells assessed as induction of receptor transactivation by reporter gene assa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50261702(2-Methyl-c-5-[4-{2-(5-methyl-2-phenyloxazol-4-yl)e...)
Affinity DataEC50:  0.272nMAssay Description:Agonist activity at PPARalpha (unknown origin) expressed in human HepG2 cells assessed as induction of receptor transactivation by reporter gene assa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50256109((2s,5s)-2-methyl-5-(4-((5-methyl-2-p-tolyloxazol-4...)
Affinity DataEC50:  0.0720nMAssay Description:Agonist activity at PPARalpha (unknown origin) expressed in human HepG2 cells assessed as induction of receptor transactivation by reporter gene assa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50261880(CHEMBL512789 | c-5-[4-{2-(2-tert-Butyl-5-methyloxa...)
Affinity DataEC50:  5.01E+3nMAssay Description:Agonist activity at PPARgamma (unknown origin) expressed in human HepG2 cells assessed as induction of receptor transactivation by reporter gene assa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50261879(2-Methyl-c-5-{4-[2-(5-methyl-2-(5-methylthiophen-2...)
Affinity DataEC50:  239nMAssay Description:Agonist activity at PPARgamma (unknown origin) expressed in human HepG2 cells assessed as induction of receptor transactivation by reporter gene assa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50261878(2-Methyl-c-5-{4-[5-methyl-2-(5-methylthiophen-2-yl...)
Affinity DataEC50:  19.8nMAssay Description:Agonist activity at PPARgamma (unknown origin) expressed in human HepG2 cells assessed as induction of receptor transactivation by reporter gene assa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50261703(2-Methyl-c-5-{4-[2-(5-methyl-2-(4-methylphenyl)oxa...)
Affinity DataEC50:  1.39E+3nMAssay Description:Agonist activity at PPARgamma (unknown origin) expressed in human HepG2 cells assessed as induction of receptor transactivation by reporter gene assa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50261702(2-Methyl-c-5-[4-{2-(5-methyl-2-phenyloxazol-4-yl)e...)
Affinity DataEC50:  4.10E+3nMAssay Description:Agonist activity at PPARgamma (unknown origin) expressed in human HepG2 cells assessed as induction of receptor transactivation by reporter gene assa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50256109((2s,5s)-2-methyl-5-(4-((5-methyl-2-p-tolyloxazol-4...)
Affinity DataEC50:  15nMAssay Description:Agonist activity at PPARgamma (unknown origin) expressed in human HepG2 cells assessed as induction of receptor transactivation by reporter gene assa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM28681(5-[(4-{2-[methyl(pyridin-2-yl)amino]ethoxy}phenyl)...)
Affinity DataEC50:  50nMAssay Description:Agonist activity at PPARgamma (unknown origin) expressed in human HepG2 cells assessed as induction of receptor transactivation by reporter gene assa...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM24566(2-({4-chloro-6-[(2,3-dimethylphenyl)amino]pyrimidi...)
Affinity DataEC50:  4.80E+3nMAssay Description:Agonist activity at PPARalpha (unknown origin) expressed in human HepG2 cells assessed as induction of receptor transactivation by reporter gene assa...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50261701(2-Methyl-c-5-[4-(5-methyl-2-phenyloxazol-4-ylmetho...)
Affinity DataEC50:  96nMAssay Description:Agonist activity at PPARgamma (unknown origin) expressed in human HepG2 cells assessed as induction of receptor transactivation by reporter gene assa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50225835((2s,5s)-2-methyl-5-(4-(5-methyl-2-p-tolyloxazol-4-...)
Affinity DataEC50:  7.00E+3nMAssay Description:Agonist activity at human PPARgamma ligand binding domain expressed in human HepG2 cells cotransfected with PPRE3-TK-luc assessed as induction of bet...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50275488(CHEMBL487561 | cis-2-methyl-5-(4-(4-(methylsulfony...)
Affinity DataEC50:  2.00E+4nMAssay Description:Agonist activity at human PPARalpha ligand binding domain expressed in human HepG2 cells cotransfected with PPRE3-TK-luc assessed as induction of bet...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM28798((2S)-2-ethoxy-3-(4-{2-[4-(methanesulfonyloxy)pheny...)
Affinity DataEC50:  820nMAssay Description:Agonist activity at human PPARalpha ligand binding domain expressed in human HepG2 cells cotransfected with PPRE3-TK-luc assessed as induction of bet...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50225835((2s,5s)-2-methyl-5-(4-(5-methyl-2-p-tolyloxazol-4-...)
Affinity DataEC50:  7.00E+3nMAssay Description:Agonist activity at human PPARalpha ligand binding domain expressed in human HepG2 cells cotransfected with PPRE3-TK-luc assessed as induction of bet...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50275537(CHEMBL520856 | cis-2-methyl-5-(6-(4-(methylsulfony...)
Affinity DataEC50:  1.50E+4nMAssay Description:Agonist activity at human PPARalpha ligand binding domain expressed in human HepG2 cells cotransfected with PPRE3-TK-luc assessed as induction of bet...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50275536(CHEMBL485942 | cis-2-methyl-5-(5-(4-(methylsulfony...)
Affinity DataEC50:  2.50E+3nMAssay Description:Agonist activity at human PPARalpha ligand binding domain expressed in human HepG2 cells cotransfected with PPRE3-TK-luc assessed as induction of bet...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM28798((2S)-2-ethoxy-3-(4-{2-[4-(methanesulfonyloxy)pheny...)
Affinity DataEC50:  13nMAssay Description:Agonist activity at human PPARgamma ligand binding domain expressed in human HepG2 cells cotransfected with PPRE3-TK-luc assessed as induction of bet...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50275537(CHEMBL520856 | cis-2-methyl-5-(6-(4-(methylsulfony...)
Affinity DataEC50:  1.50E+4nMAssay Description:Agonist activity at human PPARgamma ligand binding domain expressed in human HepG2 cells cotransfected with PPRE3-TK-luc assessed as induction of bet...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50256064(2-(((4-methoxyphenoxy)carbonyl)(5-(2-p-tolyloxazol...)
Affinity DataEC50:  44nMAssay Description:Agonist activity at human PPARalpha transactivation expressed in human HePG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50256065(2-(((4-methoxyphenoxy)carbonyl)(6-(5-methyl-2-p-to...)
Affinity DataEC50:  34nMAssay Description:Agonist activity at human PPARalpha transactivation expressed in human HePG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 66 total ) | Next | Last >>
Jump to: