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Found 363 with Last Name = 'gomez-monterrey' and Initial = 'i'
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50048691(CHEMBL3315139)
Affinity DataKi:  0.200nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50413761(CHEMBL390094)
Affinity DataKi:  0.200nMAssay Description:Displacement of [125I]urotensin-2 from human UT2 receptor expressed in CHO-K1 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50413760(CHEMBL426020)
Affinity DataKi:  0.251nMAssay Description:Displacement of [125I]urotensin-2 from human UT2 receptor expressed in CHO-K1 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50320463(CHEMBL218994 | D[CFWKYC]V | H-Asp-Cys-Phe-Trp-Lys-...)
Affinity DataKi:  0.251nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50413764(CHEMBL504097)
Affinity DataKi:  0.282nMAssay Description:Displacement of [125I]urotensin-2 from human UT2 receptor expressed in CHO-K1 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50048696(CHEMBL3315142)
Affinity DataKi:  0.398nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50048695(CHEMBL3315141)
Affinity DataKi:  0.724nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50048701(CHEMBL3315148)
Affinity DataKi:  0.776nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50378580(CHEMBL437430)
Affinity DataKi:  0.794nMAssay Description:Displacement of [125I]urotensin-2 from human UT2 receptor expressed in CHO-K1 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50413762(CHEMBL509604)
Affinity DataKi:  0.794nMAssay Description:Displacement of [125I]urotensin-2 from human UT2 receptor expressed in CHO-K1 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50413784(UROTENSIN-II)
Affinity DataKi:  0.794nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50413766(CHEMBL510618)
Affinity DataKi:  0.891nMAssay Description:Displacement of [125I]urotensin-2 from human UT2 receptor expressed in CHO-K1 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50048700(CHEMBL3315147)
Affinity DataKi:  1nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50048699(CHEMBL3315146)
Affinity DataKi:  1.20nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50413763(CHEMBL448403)
Affinity DataKi:  1.66nMAssay Description:Displacement of [125I]urotensin-2 from human UT2 receptor expressed in CHO-K1 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50048697(CHEMBL3315144)
Affinity DataKi:  1.70nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50048703(CHEMBL3315150)
Affinity DataKi:  1.80nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50048705(CHEMBL3315152)
Affinity DataKi:  1.80nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeprilysin(Oryctolagus cuniculus (rabbit))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50024102(((S)-2-Mercaptomethyl-3-phenyl-propionylamino)-ace...)
Affinity DataKi:  1.90nMAssay Description:Tested for binding affinity against neutral endopeptidase (NEP)More data for this Ligand-Target Pair
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50048692(CHEMBL3315140)
Affinity DataKi:  2nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50048702(CHEMBL3315149)
Affinity DataKi:  2.20nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50413777(CHEMBL524855)
Affinity DataKi:  2.63nMAssay Description:Displacement of [125I]urotensin-2 from human UT2 receptor expressed in CHO-K1 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50413769(CHEMBL507406)
Affinity DataKi:  3.89nMAssay Description:Displacement of [125I]urotensin-2 from human UT2 receptor expressed in CHO-K1 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50411333(URANTIDE)
Affinity DataKi:  5nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50411333(URANTIDE)
Affinity DataKi:  5.01nMAssay Description:Displacement of [125I]urotensin-2 from human UT2 receptor expressed in CHO-K1 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50413770(CHEMBL452403)
Affinity DataKi:  6.46nMAssay Description:Displacement of [125I]urotensin-2 from human UT2 receptor expressed in CHO-K1 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50048690(CHEMBL3315143)
Affinity DataKi:  6.5nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50413775(CHEMBL501794)
Affinity DataKi:  9.33nMAssay Description:Displacement of [125I]urotensin-2 from human UT2 receptor expressed in CHO-K1 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50413774(CHEMBL509009)
Affinity DataKi:  9.33nMAssay Description:Displacement of [125I]urotensin-2 from human UT2 receptor expressed in CHO-K1 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50413767(CHEMBL504723)
Affinity DataKi:  9.55nMAssay Description:Displacement of [125I]urotensin-2 from human UT2 receptor expressed in CHO-K1 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeprilysin(Oryctolagus cuniculus (rabbit))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50084679(2-[1-(2-Carboxy-2-hydroxy-ethylcarbamoyl)-2-phenyl...)
Affinity DataKi:  11nMAssay Description:Tested for binding affinity against neutral endopeptidase (NEP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50413771(CHEMBL509042)
Affinity DataKi:  11.8nMAssay Description:Displacement of [125I]urotensin-2 from human UT2 receptor expressed in CHO-K1 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50048704(CHEMBL3315151)
Affinity DataKi:  12nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50048698(CHEMBL3315145)
Affinity DataKi:  13nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50413772(CHEMBL508811)
Affinity DataKi:  13.5nMAssay Description:Displacement of [125I]urotensin-2 from human UT2 receptor expressed in CHO-K1 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50413773(CHEMBL500949)
Affinity DataKi:  15.8nMAssay Description:Displacement of [125I]urotensin-2 from human UT2 receptor expressed in CHO-K1 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50048706(CHEMBL3315153)
Affinity DataKi:  17nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50413765(CHEMBL501579)
Affinity DataKi:  19.5nMAssay Description:Displacement of [125I]urotensin-2 from human UT2 receptor expressed in CHO-K1 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50413768(CHEMBL505358)
Affinity DataKi:  26.3nMAssay Description:Displacement of [125I]urotensin-2 from human UT2 receptor expressed in CHO-K1 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThermolysin(Bacillus thermoproteolyticus)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50422014(CHEMBL319299)
Affinity DataKi:  50nMAssay Description:Tested for binding affinity against ThermolysinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50413776(CHEMBL505288)
Affinity DataKi:  219nMAssay Description:Displacement of [125I]urotensin-2 from human UT2 receptor expressed in CHO-K1 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThermolysin(Bacillus thermoproteolyticus)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50024102(((S)-2-Mercaptomethyl-3-phenyl-propionylamino)-ace...)
Affinity DataKi:  1.80E+3nMAssay Description:Tested for binding against ThermolysinMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50166018(2-[(R)-1-Amino-2-((S)-4-hydroxy-phenyl)-ethyl]-thi...)
Affinity DataKi:  3.10E+3nMAssay Description:Inhibition of [3H]-DAMGO binding to rat whole brain Opioid receptor muMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily M member 8(Rattus norvegicus (Rat))
University Of Salerno

Curated by ChEMBL
LigandPNGBDBM50465610(CHEMBL4295040)
Affinity DataIC50:  0.200nMAssay Description:Antagonist activity at rat TRPM8 expressed in HEK293 cells assessed as reduction in menthol-induced channel currents by whole cell patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeprilysin(Oryctolagus cuniculus (rabbit))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50024102(((S)-2-Mercaptomethyl-3-phenyl-propionylamino)-ace...)
Affinity DataIC50:  1.90nMAssay Description:Tested for inhibition against neutral endopeptidase (NEP)More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Rattus norvegicus (Rat))
University Of Salerno

Curated by ChEMBL
LigandPNGBDBM50465611(CHEMBL4284808)
Affinity DataIC50:  3.5nMAssay Description:Antagonist activity at rat TRPM8 expressed in HEK293 cells assessed as reduction in menthol-induced channel currents by whole cell patch clamp methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeprilysin(Oryctolagus cuniculus (rabbit))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50406747(CHEMBL2110347)
Affinity DataIC50:  3.60nMAssay Description:Inhibitory concentration was evaluated by Inhibiting 50% of Neutral endopeptidase enzyme (NEP) activity using 20 nM [3H]-D-Ala2-Leu-enkephalin as sub...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeprilysin(Oryctolagus cuniculus (rabbit))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50038623(2-(2-Benzyl-3-mercapto-5-methyl-hexanoylamino)-pro...)
Affinity DataIC50:  3.60nMAssay Description:Tested for inhibitory potency against neutral endopeptidase (NEP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeprilysin(Oryctolagus cuniculus (rabbit))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM21641(2-(2-benzyl-3-sulfanylpropanamido)acetic acid | CH...)
Affinity DataIC50:  4nMAssay Description:Inhibitory concentration was evaluated by Inhibiting 50% of Neutral endopeptidase enzyme (NEP) activity using 20 nM [3H]-D-Ala2-Leu-enkephalin as sub...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Homo sapiens (Human))
University Of Salerno

Curated by ChEMBL
LigandPNGBDBM50544523(CHEMBL4647674)
Affinity DataIC50:  4.10nMAssay Description:Antagonist activity at human TRPM8 expressed in HEK-293/TRPM8 exon1 K3 cells assessed as inhibition of menthol-induced current response by whole-cell...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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